SK13352003A3 - Use of azithromycin for the manufacture of a medicament for treatment of non-infective inflammatory diseases - Google Patents

Use of azithromycin for the manufacture of a medicament for treatment of non-infective inflammatory diseases Download PDF

Info

Publication number: SK13352003A3
Authority: SK; Slovakia
Prior art keywords: acid; azithromycin; agents; use according; pharmaceutical compositions
Prior art date: 2001-04-27

Application number

SK13352003A

Other languages

English (en)

Slovak (sk)

Inventor

Ognjen Culic

Michael Parnham

Vesna Erakovic

Original Assignee

Pliva D D

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2001-04-27

Filing date

2002-04-10

Publication date

2004-10-05

2002-04-10 Application filed by Pliva D D filed Critical Pliva D D

2004-10-05 Publication of SK13352003A3 publication Critical patent/SK13352003A3/sk

Links

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239000006228 supernatant Substances 0.000 description 1
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239000003765 sweetening agent Substances 0.000 description 1
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210000002437 synoviocyte Anatomy 0.000 description 1
238000003786 synthesis reaction Methods 0.000 description 1
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238000012360 testing method Methods 0.000 description 1
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RZWIIPASKMUIAC-VQTJNVASSA-N thromboxane Chemical compound CCCCCCCC[C@H]1OCCC[C@@H]1CCCCCCC RZWIIPASKMUIAC-VQTJNVASSA-N 0.000 description 1
AOBORMOPSGHCAX-DGHZZKTQSA-N tocofersolan Chemical compound OCCOC(=O)CCC(=O)OC1=C(C)C(C)=C2O[C@](CCC[C@H](C)CCC[C@H](C)CCCC(C)C)(C)CCC2=C1C AOBORMOPSGHCAX-DGHZZKTQSA-N 0.000 description 1
229960000984 tocofersolan Drugs 0.000 description 1
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230000002588 toxic effect Effects 0.000 description 1
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230000032258 transport Effects 0.000 description 1
231100000397 ulcer Toxicity 0.000 description 1
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NQPDZGIKBAWPEJ-UHFFFAOYSA-N valeric acid Chemical compound CCCCC(O)=O NQPDZGIKBAWPEJ-UHFFFAOYSA-N 0.000 description 1
210000003462 vein Anatomy 0.000 description 1
235000019154 vitamin C Nutrition 0.000 description 1
239000011718 vitamin C Substances 0.000 description 1
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239000011709 vitamin E Substances 0.000 description 1
238000005303 weighing Methods 0.000 description 1
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239000002076 α-tocopherol Substances 0.000 description 1
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- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
- A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
- A61K31/7048—Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
- A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
- A61K31/7052—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/12—Drugs for disorders of the urinary system of the kidneys
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/06—Antipsoriatics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators

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Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Public Health (AREA)
Pharmacology & Pharmacy (AREA)
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Veterinary Medicine (AREA)
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Medicinal Chemistry (AREA)
Animal Behavior & Ethology (AREA)
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Organic Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
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Epidemiology (AREA)
Molecular Biology (AREA)
Immunology (AREA)
Rheumatology (AREA)
Dermatology (AREA)
Urology & Nephrology (AREA)
Pulmonology (AREA)
Orthopedic Medicine & Surgery (AREA)
Physical Education & Sports Medicine (AREA)
Pain & Pain Management (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Saccharide Compounds (AREA)
Medicinal Preparation (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

SK13352003A 2001-04-27 2002-04-10 Use of azithromycin for the manufacture of a medicament for treatment of non-infective inflammatory diseases SK13352003A3 (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
HR20010301A HRP20010301A2 (en)	2001-04-27	2001-04-27	New therapeutic indication for azithromycin in the treatment of non-infective inflammatory diseases
PCT/EP2002/003984 WO2002087596A2 (en)	2001-04-27	2002-04-10	Use of azithromycin for the manufacture of a medicament for treatment of non-infective inflammatory diseases

Publications (1)

Publication Number	Publication Date
SK13352003A3 true SK13352003A3 (en)	2004-10-05

Family

ID=10947306

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
SK13352003A SK13352003A3 (en)	2001-04-27	2002-04-10	Use of azithromycin for the manufacture of a medicament for treatment of non-infective inflammatory diseases

Country Status (19)

Country	Link
US (1)	US20050054587A1 (cs)
EP (1)	EP1392327A2 (cs)
JP (1)	JP2004531539A (cs)
CN (1)	CN1582158A (cs)
AR (1)	AR034223A1 (cs)
BG (1)	BG108286A (cs)
BR (1)	BR0209276A (cs)
CA (1)	CA2443381A1 (cs)
CZ (1)	CZ20032932A3 (cs)
EA (1)	EA200301187A1 (cs)
HR (1)	HRP20010301A2 (cs)
HU (1)	HUP0303988A2 (cs)
IL (1)	IL158236A0 (cs)
MX (1)	MXPA03009849A (cs)
PL (1)	PL364086A1 (cs)
SK (1)	SK13352003A3 (cs)
WO (1)	WO2002087596A2 (cs)
YU (1)	YU84503A (cs)
ZA (1)	ZA200308933B (cs)

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HRP20020231A2 (en)	2002-03-18	2003-12-31	Pliva D D	ISOSTRUCTURAL PSEUDOPOLYMORPHS OF 9-DEOXO-9a-AZA-9a-METHYL-9a-HOMOERYTHROMYCIN A
HRP20020614A2 (en)	2002-07-22	2004-06-30	PLIVA-ISTRAŽIVAČKI INSTITUT d.o.o.	Rhombic pseudopolymorph of 9-deoxo-9a-aza-9a-methyl-9a-homoerythromycin a
GB0315671D0 (en)	2003-07-04	2003-08-13	Chelsea And Westminster Nhs Tr	Improvements in or relating to organic compounds
JP2007516951A (ja) *	2003-12-30	2007-06-28	アステラス製薬株式会社	気道閉塞症の治療または予防のためのマクロライドの使用
US7468428B2 (en)	2004-03-17	2008-12-23	App Pharmaceuticals, Llc	Lyophilized azithromycin formulation
WO2006115494A1 (en) *	2005-04-26	2006-11-02	American Pharmaceutical Partners, Inc.	Lyophilized azithromycin formulation
JP3933683B2 (ja)	2004-07-02	2007-06-20	わかもと製薬株式会社	アジスロマイシン含有水性医薬組成物及びその調製方法
WO2006097849A1 (en) *	2005-01-14	2006-09-21	Glaxosmithkline Istrazivacki Centar Zagreb D.O.O.	9a-carbamoyl and thiocarbamoyl azalides with anti-inflammatory activity
US20060293261A1 (en)	2005-06-24	2006-12-28	Taisho Pharmaceutical Co., Ltd.	Clarithromycin or a salt thereof for the treatment or prevention of pulmonary disorders caused by the destruction of pulmonary alveoli
EP2010153A2 (en) *	2006-04-03	2009-01-07	Teva Pharmaceutical Industries Limited	Drug microparticles
RU2455308C2 (ru)	2006-05-01	2012-07-10	Тайсо Фармасьютикал Ко., Лтд.	Макролидные производные
US7704959B2 (en) *	2006-10-03	2010-04-27	Dow Pharmaceutical Sciences	Azithromycin for the treatment of nodular acne
JP2011527709A (ja) *	2008-07-10	2011-11-04	インスパイアーファーマシューティカルズ，インコーポレイティド	眼瞼炎の治療方法
WO2010062787A1 (en)	2008-11-03	2010-06-03	Washington University	Bioluminescence imaging of myeloperoxidase activity in vivo, methods, compositions and apparatuses therefor
EP2393355A4 (en) *	2009-01-23	2012-07-25	Inspire Pharmaceuticals Inc	METHOD FOR TREATING A DRY EYE WITH AZITHROMYCIN
CN102378763A (zh)	2009-01-30	2012-03-14	葛兰素集团有限公司	消炎的大环内酯
WO2011116312A1 (en) *	2010-03-19	2011-09-22	Catabasis Pharmaceuticals, Inc.	Fatty acid macrolide derivatives and their uses
WO2017010382A1 (ja) *	2015-07-14	2017-01-19	国立大学法人大阪大学	筋強直性ジストロフィー治療薬
CN113209084A (zh) *	2021-05-18	2021-08-06	南开大学	化合物cp0119在制备用于治疗炎性肠病的药物中的应用
WO2025235305A1 (en)	2024-05-06	2025-11-13	Baxter International Inc.	Azithromycin premix formulation and product, methods of preparing same, and methods of using same

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YU43116B (en) *	1979-04-02	1989-04-30	Pliva Pharm & Chem Works	Process for preparing 11-aza-4-o-cladinosyl-6-o-desosaminyl-15-ethyl-7,13,14-trihydroxy-3,5,7,9,12,14-hexamethyl-oxacyclopentadecane-2-one(11-aza-10-deox
SI8110592A8 (en) *	1981-03-06	1996-06-30	Pliva Pharm & Chem Works	Process for preparing of n-methyl-11-aza-10-deoxo-10-dihydroerythromycine a and derivatives thereof
YU45590A (sh) *	1990-03-07	1992-07-20	PLIVA FARMACEVTSKA, KEMIJSKA, PREHRAMBENA I KOZMETIČKA INDUSTRIJA s.p.o.	Novi kompleksi odnosno helati antibiotika s dvovalentnim i/ili trovalentnim metalima i postupci za njihovo dobijanje
SI9011409A (en) *	1990-07-18	1995-10-31	Pliva Pharm & Chem Works	O-methyl azitromycin derivates, methods and intermediates for their preparation and methods for preparation of pharmaceuticals products which comprise them
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GB9723669D0 (en) *	1997-11-07	1998-01-07	Univ Aberdeen	Skin penetration enhancing components
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IT1313610B1 (it) *	1999-08-09	2002-09-09	S I F I Societa Ind Farmaceuti	Processo per la preparazione di formulazioni acquose per uso oftalmico
IL141438A0 (en) *	2000-02-23	2002-03-10	Pfizer Prod Inc	Method of increasing the bioavailability and tissue penetration of azithromycin

2001
- 2001-04-27 HR HR20010301A patent/HRP20010301A2/hr not_active Application Discontinuation
2002
- 2002-04-10 SK SK13352003A patent/SK13352003A3/sk not_active Application Discontinuation
- 2002-04-10 CN CNA028089162A patent/CN1582158A/zh active Pending
- 2002-04-10 EA EA200301187A patent/EA200301187A1/ru unknown
- 2002-04-10 YU YU84503A patent/YU84503A/sh unknown
- 2002-04-10 PL PL02364086A patent/PL364086A1/xx not_active Application Discontinuation
- 2002-04-10 MX MXPA03009849A patent/MXPA03009849A/es unknown
- 2002-04-10 US US10/476,377 patent/US20050054587A1/en not_active Abandoned
- 2002-04-10 HU HU0303988A patent/HUP0303988A2/hu unknown
- 2002-04-10 WO PCT/EP2002/003984 patent/WO2002087596A2/en not_active Ceased
- 2002-04-10 JP JP2002584941A patent/JP2004531539A/ja active Pending
- 2002-04-10 CZ CZ20032932A patent/CZ20032932A3/cs unknown
- 2002-04-10 EP EP02737939A patent/EP1392327A2/en not_active Withdrawn
- 2002-04-10 IL IL15823602A patent/IL158236A0/xx unknown
- 2002-04-10 CA CA002443381A patent/CA2443381A1/en not_active Abandoned
- 2002-04-10 BR BR0209276-0A patent/BR0209276A/pt not_active IP Right Cessation
- 2002-04-26 AR ARP020101524A patent/AR034223A1/es unknown
2003
- 2003-10-23 BG BG108286A patent/BG108286A/bg unknown
- 2003-11-17 ZA ZA200308933A patent/ZA200308933B/en unknown

Also Published As

Publication number	Publication date
CA2443381A1 (en)	2002-11-07
YU84503A (sh)	2006-08-17
IL158236A0 (en)	2004-05-12
WO2002087596A2 (en)	2002-11-07
PL364086A1 (en)	2004-12-13
CN1582158A (zh)	2005-02-16
WO2002087596A3 (en)	2003-01-03
JP2004531539A (ja)	2004-10-14
EA200301187A1 (ru)	2004-04-29
EP1392327A2 (en)	2004-03-03
ZA200308933B (en)	2004-11-17
HRP20010301A2 (en)	2001-12-31
BR0209276A (pt)	2004-06-15
MXPA03009849A (es)	2004-05-24
BG108286A (bg)	2004-09-30
HUP0303988A2 (hu)	2004-04-28
US20050054587A1 (en)	2005-03-10
AR034223A1 (es)	2004-02-04
CZ20032932A3 (cs)	2004-08-18

Legal Events

Date	Code	Title	Description
2011-03-04	FC9A	Refused patent application

Publication	Publication Date	Title
SK13352003A3 (en)	2004-10-05	Use of azithromycin for the manufacture of a medicament for treatment of non-infective inflammatory diseases
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