SK15532003A3 - Prípravok inzulínu na pľúcne podávanie - Google Patents

Prípravok inzulínu na pľúcne podávanie Download PDF

Info

Publication number: SK15532003A3
Authority: SK; Slovakia
Prior art keywords: insulin; peg; polyethylene glycol; composition; administration
Prior art date: 2001-05-21

Application number

SK1553-2003A

Other languages

English (en)

Slovak (sk)

Inventor

John S. Patton

Mei-Chang Kuo

J. Milton Harris

Chester Leach

Kimberly Perkins

Blaine Bueche

Original Assignee

Nektar Therapeutics

Nektar Therapeutics Al, Corporation

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2001-05-21

Filing date

2002-05-21

Publication date

2004-06-08

2002-05-21 Application filed by Nektar Therapeutics, Nektar Therapeutics Al, Corporation filed Critical Nektar Therapeutics

2004-06-08 Publication of SK15532003A3 publication Critical patent/SK15532003A3/sk

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Classifications

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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/50—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- A61K38/22—Hormones
- A61K38/28—Insulins
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/50—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
- A61K47/51—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent
- A61K47/56—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic macromolecular compound, e.g. an oligomeric, polymeric or dendrimeric molecule
- A61K47/59—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic macromolecular compound, e.g. an oligomeric, polymeric or dendrimeric molecule obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyureas or polyurethanes
- A61K47/60—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic macromolecular compound, e.g. an oligomeric, polymeric or dendrimeric molecule obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyureas or polyurethanes the organic macromolecular compound being a polyoxyalkylene oligomer, polymer or dendrimer, e.g. PEG, PPG, PEO or polyglycerol
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/48—Drugs for disorders of the endocrine system of the pancreatic hormones
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/48—Drugs for disorders of the endocrine system of the pancreatic hormones
- A61P5/50—Drugs for disorders of the endocrine system of the pancreatic hormones for increasing or potentiating the activity of insulin

Landscapes

Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Diabetes (AREA)
Chemical & Material Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Bioinformatics & Cheminformatics (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Engineering & Computer Science (AREA)
Medicinal Chemistry (AREA)
Animal Behavior & Ethology (AREA)
Endocrinology (AREA)
Epidemiology (AREA)
General Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Obesity (AREA)
Hematology (AREA)
Emergency Medicine (AREA)
Zoology (AREA)
Gastroenterology & Hepatology (AREA)
Immunology (AREA)
Proteomics, Peptides & Aminoacids (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Peptides Or Proteins (AREA)
Medicinal Preparation (AREA)

SK1553-2003A 2001-05-21 2002-05-21 Prípravok inzulínu na pľúcne podávanie SK15532003A3 (sk)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US29242301P	2001-05-21	2001-05-21
PCT/US2002/016464 WO2002094200A2 (en)	2001-05-21	2002-05-21	Pulmonary administration of chemically modified insulin

Publications (1)

Publication Number	Publication Date
SK15532003A3 true SK15532003A3 (sk)	2004-06-08

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ID=23124608

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SK1553-2003A SK15532003A3 (sk)	2001-05-21	2002-05-21	Prípravok inzulínu na pľúcne podávanie

Country Status (35)

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US (3)	US6838076B2 (is)
EP (1)	EP1395294A4 (is)
JP (1)	JP2004535401A (is)
KR (1)	KR20030097876A (is)
CN (2)	CN1314445C (is)
AP (1)	AP1763A (is)
AR (1)	AR033903A1 (is)
AU (1)	AU2002303869B2 (is)
BG (1)	BG108494A (is)
BR (1)	BR0209896A (is)
CA (1)	CA2447236A1 (is)
CO (1)	CO5540371A2 (is)
CZ (1)	CZ20033182A3 (is)
EA (1)	EA007408B1 (is)
EC (1)	ECSP034855A (is)
GE (1)	GEP20063917B (is)
HR (1)	HRP20030949A2 (is)
HU (1)	HUP0400442A2 (is)
IL (2)	IL158862A0 (is)
IS (1)	IS7043A (is)
LT (1)	LT5153B (is)
LV (1)	LV13197B (is)
MA (1)	MA26185A1 (is)
MX (1)	MXPA03010649A (is)
MY (1)	MY137181A (is)
NO (1)	NO20035157D0 (is)
NZ (1)	NZ529572A (is)
OA (1)	OA13136A (is)
PL (1)	PL366911A1 (is)
SK (1)	SK15532003A3 (is)
TN (1)	TNSN03116A1 (is)
TR (1)	TR200400295T2 (is)
WO (1)	WO2002094200A2 (is)
YU (1)	YU98503A (is)
ZA (1)	ZA200309085B (is)

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JP2008528549A (ja) *	2005-01-27	2008-07-31	ノボノルディスクアクティーゼルスカブ	構造的に充分に定義された分岐ポリマーと接合されたインスリン誘導体
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US20080171695A1 (en)	2005-02-02	2008-07-17	Novo Nordisk A/S	Insulin Derivatives
JP2008533100A (ja) *	2005-03-18	2008-08-21	ノボノルディスクアクティーゼルスカブ	Ｐｅｇ化された単鎖インスリン
US20060271011A1 (en) *	2005-05-25	2006-11-30	Mock Bradley D	Methods and apparatus for indicating when a disposable component of a drug delivery system needs to be replaced
CN104324362B (zh)	2005-09-14	2018-04-24	曼金德公司	以提高活性试剂对结晶微粒表面的亲和力为基础的药物配制方法
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US8000981B2 (en)	2005-11-30	2011-08-16	The Invention Science Fund I, Llc	Methods and systems related to receiving nutraceutical associated information
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Publication number	Publication date
LV13197B (en)	2004-10-20
TR200400295T2 (tr)	2005-04-21
CN1314445C (zh)	2007-05-09
AR033903A1 (es)	2004-01-07
ECSP034855A (es)	2004-03-23
EP1395294A2 (en)	2004-03-10
AU2002303869B2 (en)	2007-08-16
AP1763A (en)	2007-08-02
MXPA03010649A (es)	2005-10-05
NO20035157D0 (no)	2003-11-20
OA13136A (en)	2006-12-13
YU98503A (sh)	2006-05-25
TNSN03116A1 (en)	2005-12-23
AP2003002918A0 (en)	2003-12-31
IS7043A (is)	2003-11-19
MA26185A1 (fr)	2004-07-01
HRP20030949A2 (en)	2005-04-30
HUP0400442A2 (hu)	2005-03-29
MY137181A (en)	2009-01-30
IL158862A (en)	2008-07-08
WO2002094200A2 (en)	2002-11-28
IL158862A0 (en)	2004-05-12
JP2004535401A (ja)	2004-11-25
WO2002094200A3 (en)	2003-02-20
EP1395294A4 (en)	2006-01-11
US6890518B2 (en)	2005-05-10
US20030118510A1 (en)	2003-06-26
CZ20033182A3 (cs)	2004-09-15
EA200301222A1 (ru)	2004-08-26
KR20030097876A (ko)	2003-12-31
NZ529572A (en)	2006-02-24
PL366911A1 (en)	2005-02-07
CO5540371A2 (es)	2005-07-29
BG108494A (en)	2004-07-30
CA2447236A1 (en)	2002-11-28
LT2003107A (en)	2004-05-25
EA007408B1 (ru)	2006-10-27
GEP20063917B (en)	2006-09-11
US20030216542A1 (en)	2003-11-20
US6838076B2 (en)	2005-01-04
US20050152848A1 (en)	2005-07-14
LT5153B (lt)	2004-08-25
CN101045166A (zh)	2007-10-03
ZA200309085B (en)	2004-11-22
CN1582171A (zh)	2005-02-16
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