SK20099A3 - Treatment of upper airway allergic responses with a combination of histamine receptor antagonists - Google Patents

Treatment of upper airway allergic responses with a combination of histamine receptor antagonists Download PDF

Info

Publication number: SK20099A3
Authority: SK; Slovakia
Prior art keywords: receptor antagonist; receptor; treatment; receptor antagonists; histamine
Prior art date: 1996-08-16

Application number

SK200-99A

Other languages

English (en)

Slovak (sk)

Inventor

William Kreutner

John A Hey

Original Assignee

Schering Corp

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1996-08-16

Filing date

1997-08-13

Publication date

2000-08-14

1997-08-13 Application filed by Schering Corp filed Critical Schering Corp

2000-08-14 Publication of SK20099A3 publication Critical patent/SK20099A3/sk

Links

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239000003765 sweetening agent Substances 0.000 description 1
230000008961 swelling Effects 0.000 description 1
210000002820 sympathetic nervous system Anatomy 0.000 description 1
230000001975 sympathomimetic effect Effects 0.000 description 1
229960000351 terfenadine Drugs 0.000 description 1
229940126585 therapeutic drug Drugs 0.000 description 1
239000002562 thickening agent Substances 0.000 description 1
210000003437 trachea Anatomy 0.000 description 1
229960003223 tripelennamine Drugs 0.000 description 1
229960001128 triprolidine Drugs 0.000 description 1
CBEQULMOCCWAQT-WOJGMQOQSA-N triprolidine Chemical compound C1=CC(C)=CC=C1C(\C=1N=CC=CC=1)=C/CN1CCCC1 CBEQULMOCCWAQT-WOJGMQOQSA-N 0.000 description 1
230000024883 vasodilation Effects 0.000 description 1
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Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/02—Nasal agents, e.g. decongestants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/16—Otologicals
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

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Health & Medical Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Veterinary Medicine (AREA)
Chemical & Material Sciences (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
Animal Behavior & Ethology (AREA)
Life Sciences & Earth Sciences (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Engineering & Computer Science (AREA)
Chemical Kinetics & Catalysis (AREA)
Bioinformatics & Cheminformatics (AREA)
Organic Chemistry (AREA)
Pulmonology (AREA)
Epidemiology (AREA)
Immunology (AREA)
Otolaryngology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Medicinal Preparation (AREA)

SK200-99A 1996-08-16 1997-08-13 Treatment of upper airway allergic responses with a combination of histamine receptor antagonists SK20099A3 (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US68995196A	1996-08-16	1996-08-16
PCT/US1997/013903 WO1998006394A1 (en)	1996-08-16	1997-08-13	Treatment of upper airway allergic responses with a combination of histamine receptor antagonists

Publications (1)

Publication Number	Publication Date
SK20099A3 true SK20099A3 (en)	2000-08-14

Family

ID=24770500

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
SK200-99A SK20099A3 (en)	1996-08-16	1997-08-13	Treatment of upper airway allergic responses with a combination of histamine receptor antagonists

Country Status (25)

Country	Link
EP (1)	EP0920315B1 (cs)
JP (2)	JP3638289B2 (cs)
KR (1)	KR20000029975A (cs)
CN (1)	CN1152682C (cs)
AR (1)	AR008293A1 (cs)
AT (1)	ATE314071T1 (cs)
AU (1)	AU722040B2 (cs)
BR (1)	BR9711149A (cs)
CA (1)	CA2263163A1 (cs)
CO (1)	CO4910138A1 (cs)
CZ (1)	CZ43299A3 (cs)
DE (1)	DE69734984D1 (cs)
HU (1)	HUP9904362A3 (cs)
ID (1)	ID17871A (cs)
IL (1)	IL128573A0 (cs)
MY (1)	MY116130A (cs)
NO (1)	NO990706D0 (cs)
NZ (1)	NZ334063A (cs)
PE (1)	PE100298A1 (cs)
PL (1)	PL191073B1 (cs)
SK (1)	SK20099A3 (cs)
TR (1)	TR199900326T2 (cs)
TW (2)	TWI221768B (cs)
WO (1)	WO1998006394A1 (cs)
ZA (1)	ZA977263B (cs)

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JP4344405B2 (ja) *	1997-08-26	2009-10-14	アベンティス・ファーマスーティカルズ・インコーポレイテッド	ピペリジノアルカノール−鬱血除去剤の組合せ用医薬組成物
US5990147A (en) *	1997-11-07	1999-11-23	Schering Corporation	H3 receptor ligands of the phenyl-alkyl-imidazoles type
US6034251A (en) *	1997-11-07	2000-03-07	Schering Corporation	Phenyl-alkyl-imidazoles
EP1028948B1 (en) *	1997-11-07	2003-01-29	Schering Corporation	Phenyl-alkyl-imidazoles as h3 receptor antagonists
EP1028956A1 (en) *	1997-11-07	2000-08-23	Schering Corporation	Imidazoylalkyl substituted with a five, six or seven membered heterocyclic ring containing one nitrogen atom
IL135729A0 (en) *	1997-11-07	2001-05-20	Schering Corp	H3 receptor ligands of the phenyl-alkyl-imidazoles type
US6384038B1 (en) *	1998-04-14	2002-05-07	Sepracor Inc.	Methods and compositions using cetirizine in combination with leukotriene inhibitors or decongestants
JP2002527381A (ja) *	1998-10-09	2002-08-27	シェーリングコーポレイション	アレルギー性疾患を処置するための組成物および方法
US6100279A (en) *	1998-11-05	2000-08-08	Schering Corporation	Imidazoylalkyl substituted with a five, six or seven membered heterocyclic ring containing one nitrogen atom
CA2383214A1 (en) *	1999-09-22	2001-03-29	Schering Corporation	Treating allergic and inflammatory conditions
HK1046367A1 (zh)	2000-02-03	2003-01-10	Schering Corporation	治疗过敏和炎症症状
PE20020507A1 (es)	2000-10-17	2002-06-25	Schering Corp	Compuestos no-imidazoles como antagonistas del receptor histamina h3
GB2373186A (en) *	2001-02-23	2002-09-18	Astrazeneca Ab	Pharmaceutical combinations of a CCR3 antagonist and a compound which is usefulreatment of asthma, allergic disease or inflammation
MXPA03008356A (es)	2001-03-13	2003-12-11	Schering Corp	Compuestos del tipo no imidazol como antagonistas de histamina h3.
US7105505B2 (en)	2002-04-18	2006-09-12	Schering Corporation	Benzimidazole derivatives useful as histamine H3 antagonists
US7220735B2 (en)	2002-04-18	2007-05-22	Schering Corporation	Benzimidazolone histamine H3 antagonists
IL165863A0 (en)	2002-06-24	2006-01-15	Schering Corp	Indole derivatives useful as histamine H3 antagonists
WO2004066960A2 (en) *	2003-01-28	2004-08-12	Schering Corporation	Combination of h1, h3 and h4 receptor antagonists for treatment of allergic and non-allergic pulmonary inflammation, congestion and allergic rhinitis
TW200738676A (en)	2005-06-20	2007-10-16	Schering Corp	Heteroatom-linked substituted piperidines and derivatives thereof useful as histamine H3 antagonists
EP2318388A2 (en)	2008-07-23	2011-05-11	Schering Corporation	Tricyclic spirocycle derivatives and methods of use thereof
AU2009303444A1 (en)	2008-10-16	2010-04-22	Schering Corporation	Azine derivatives and methods of use thereof
US20110245267A1 (en)	2008-12-19	2011-10-06	Schering Plough Corporation	Piperidine and piperazine derivatives and methods of use thereof
WO2010071819A1 (en)	2008-12-19	2010-06-24	Schering Corporation	Bicyclic heterocyclic derivatives and methods of use thereof
EP2408453B1 (en)	2009-03-17	2022-01-05	Nicox Ophthalmics, Inc.	Ophthalmic formulations of cetirizine and methods of use
US8569273B2 (en)	2009-03-17	2013-10-29	Aciex Therapeutics, Inc.	Ophthalmic formulations of cetirizine and methods of use
US9399032B2 (en) *	2009-05-14	2016-07-26	The General Hospital Corporation	Methods and compositions for treating degenerative and ischemic disorders
US8759357B2 (en)	2009-10-08	2014-06-24	Merck Sharp & Dohme Corp.	Inhibitors of fatty acid binding protein (FABP)
WO2013151982A1 (en)	2012-04-03	2013-10-10	Arena Pharmaceuticals, Inc.	Methods and compounds useful in treating pruritus, and methods for identifying such compounds
RU2685277C1 (ru) *	2018-05-24	2019-04-17	Общество с ограниченной ответственностью "Фарминтерпрайсез Аллерджи"	Применение бисамидного производного малоновой кислоты для лечения аллергических и других заболеваний человека и животных

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1997
- 1997-08-13 KR KR1019997001226A patent/KR20000029975A/ko not_active Abandoned
- 1997-08-13 TR TR1999/00326T patent/TR199900326T2/xx unknown
- 1997-08-13 WO PCT/US1997/013903 patent/WO1998006394A1/en not_active Ceased
- 1997-08-13 TW TW086111627A patent/TWI221768B/zh not_active IP Right Cessation
- 1997-08-13 JP JP50985998A patent/JP3638289B2/ja not_active Expired - Fee Related
- 1997-08-13 CZ CZ99432A patent/CZ43299A3/cs unknown
- 1997-08-13 BR BR9711149A patent/BR9711149A/pt not_active Application Discontinuation
- 1997-08-13 HU HU9904362A patent/HUP9904362A3/hu unknown
- 1997-08-13 TW TW093112764A patent/TW200427450A/zh unknown
- 1997-08-13 IL IL12857397A patent/IL128573A0/xx unknown
- 1997-08-13 AT AT97937153T patent/ATE314071T1/de not_active IP Right Cessation
- 1997-08-13 SK SK200-99A patent/SK20099A3/sk unknown
- 1997-08-13 AR ARP970103693A patent/AR008293A1/es unknown
- 1997-08-13 NZ NZ334063A patent/NZ334063A/xx unknown
- 1997-08-13 ZA ZA9707263A patent/ZA977263B/xx unknown
- 1997-08-13 CA CA002263163A patent/CA2263163A1/en not_active Abandoned
- 1997-08-13 EP EP97937153A patent/EP0920315B1/en not_active Expired - Lifetime
- 1997-08-13 PE PE1997000705A patent/PE100298A1/es not_active Application Discontinuation
- 1997-08-13 AU AU39733/97A patent/AU722040B2/en not_active Ceased
- 1997-08-13 CN CNB971987130A patent/CN1152682C/zh not_active Expired - Fee Related
- 1997-08-13 PL PL331617A patent/PL191073B1/pl not_active IP Right Cessation
- 1997-08-13 MY MYPI97003708A patent/MY116130A/en unknown
- 1997-08-13 DE DE69734984T patent/DE69734984D1/de not_active Expired - Lifetime
- 1997-08-14 CO CO97046887A patent/CO4910138A1/es unknown
- 1997-08-14 ID IDP972837A patent/ID17871A/id unknown
1999
- 1999-02-15 NO NO990706A patent/NO990706D0/no unknown
2002
- 2002-07-30 JP JP2002222138A patent/JP2003095979A/ja not_active Withdrawn

Also Published As

Publication number	Publication date
JP3638289B2 (ja)	2005-04-13
NZ334063A (en)	2000-09-29
JP2003095979A (ja)	2003-04-03
TR199900326T2 (xx)	1999-05-21
PL331617A1 (en)	1999-08-02
CN1233179A (zh)	1999-10-27
CA2263163A1 (en)	1998-02-19
NO990706L (no)	1999-02-15
ATE314071T1 (de)	2006-01-15
HUP9904362A3 (en)	2000-12-28
HUP9904362A2 (hu)	2000-11-28
CO4910138A1 (es)	2000-04-24
BR9711149A (pt)	1999-08-17
ID17871A (id)	1998-02-05
CN1152682C (zh)	2004-06-09
MY116130A (en)	2003-11-28
AR008293A1 (es)	1999-12-29
PE100298A1 (es)	1999-01-11
DE69734984D1 (de)	2006-02-02
IL128573A0 (en)	2000-01-31
NO990706D0 (no)	1999-02-15
AU722040B2 (en)	2000-07-20
EP0920315B1 (en)	2005-12-28
JP2000505094A (ja)	2000-04-25
TW200427450A (en)	2004-12-16
AU3973397A (en)	1998-03-06
ZA977263B (en)	1998-02-16
PL191073B1 (pl)	2006-03-31
WO1998006394A1 (en)	1998-02-19
TWI221768B (en)	2004-10-11
EP0920315A1 (en)	1999-06-09
CZ43299A3 (cs)	1999-07-14
KR20000029975A (ko)	2000-05-25

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SK20099A3 (en)	2000-08-14	Treatment of upper airway allergic responses with a combination of histamine receptor antagonists
US5869479A (en)	1999-02-09	Treatment of upper airway allergic responses
US6936601B2 (en)	2005-08-30	Compositions for treating pain
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