SK282914B6 - Sertralínová dávkovacia forma - Google Patents

Sertralínová dávkovacia forma Download PDF

Info

Publication number: SK282914B6
Authority: SK; Slovakia
Prior art keywords: sertraline; dosage form; mga; oil; vehicle
Prior art date: 1997-07-01

Application number

SK1805-99A

Other languages

English (en)

Slovak (sk)

Other versions

SK180599A3 (en

Inventor

William John Curatolo

Ravi Mysore Shanker

Original Assignee

Pfizer Products Inc.

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1997-07-01

Filing date

1998-06-16

Publication date

2003-01-09

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=21971076&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SK282914(B6) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

1998-06-16 Application filed by Pfizer Products Inc. filed Critical Pfizer Products Inc.

2001-01-18 Publication of SK180599A3 publication Critical patent/SK180599A3/sk

2003-01-09 Publication of SK282914B6 publication Critical patent/SK282914B6/sk

Links

VGKDLMBJGBXTGI-SJCJKPOMSA-N sertraline Chemical compound C1([C@@H]2CC[C@@H](C3=CC=CC=C32)NC)=CC=C(Cl)C(Cl)=C1 VGKDLMBJGBXTGI-SJCJKPOMSA-N 0.000 title claims abstract description 224
229960002073 sertraline Drugs 0.000 title claims abstract description 215
239000002552 dosage form Substances 0.000 title claims abstract description 70
229920000159 gelatin Polymers 0.000 title claims description 21
235000019322 gelatine Nutrition 0.000 title claims description 21
239000001828 Gelatine Substances 0.000 title 1
238000001556 precipitation Methods 0.000 claims abstract description 27
VEXZGXHMUGYJMC-UHFFFAOYSA-M Chloride anion Chemical compound [Cl-] VEXZGXHMUGYJMC-UHFFFAOYSA-M 0.000 claims abstract description 22
239000003981 vehicle Substances 0.000 claims description 83
239000000244 polyoxyethylene sorbitan monooleate Substances 0.000 claims description 22
235000010482 polyoxyethylene sorbitan monooleate Nutrition 0.000 claims description 22
229940068968 polysorbate 80 Drugs 0.000 claims description 22
229920000053 polysorbate 80 Polymers 0.000 claims description 22
108010010803 Gelatin Proteins 0.000 claims description 20
239000008273 gelatin Substances 0.000 claims description 20
235000011852 gelatine desserts Nutrition 0.000 claims description 20
DNIAPMSPPWPWGF-UHFFFAOYSA-N Propylene glycol Chemical group CC(O)CO DNIAPMSPPWPWGF-UHFFFAOYSA-N 0.000 claims description 18
150000003839 salts Chemical class 0.000 claims description 18
239000000203 mixture Substances 0.000 claims description 16
WWZKQHOCKIZLMA-UHFFFAOYSA-N octanoic acid Chemical compound CCCCCCCC(O)=O WWZKQHOCKIZLMA-UHFFFAOYSA-N 0.000 claims description 14
235000019485 Safflower oil Nutrition 0.000 claims description 12
GHVNFZFCNZKVNT-UHFFFAOYSA-N decanoic acid Chemical compound CCCCCCCCCC(O)=O GHVNFZFCNZKVNT-UHFFFAOYSA-N 0.000 claims description 12
239000003813 safflower oil Substances 0.000 claims description 12
235000005713 safflower oil Nutrition 0.000 claims description 12
LFQSCWFLJHTTHZ-UHFFFAOYSA-N Ethanol Chemical compound CCO LFQSCWFLJHTTHZ-UHFFFAOYSA-N 0.000 claims description 11
239000007788 liquid Substances 0.000 claims description 10
239000004006 olive oil Substances 0.000 claims description 9
235000008390 olive oil Nutrition 0.000 claims description 9
PEDCQBHIVMGVHV-UHFFFAOYSA-N glycerol Substances OCC(O)CO PEDCQBHIVMGVHV-UHFFFAOYSA-N 0.000 claims description 8
239000004094 surface-active agent Substances 0.000 claims description 8
WRIDQFICGBMAFQ-UHFFFAOYSA-N (E)-8-Octadecenoic acid Natural products CCCCCCCCCC=CCCCCCCC(O)=O WRIDQFICGBMAFQ-UHFFFAOYSA-N 0.000 claims description 6
LQJBNNIYVWPHFW-UHFFFAOYSA-N 20:1omega9c fatty acid Natural products CCCCCCCCCCC=CCCCCCCCC(O)=O LQJBNNIYVWPHFW-UHFFFAOYSA-N 0.000 claims description 6
QSBYPNXLFMSGKH-UHFFFAOYSA-N 9-Heptadecensaeure Natural products CCCCCCCC=CCCCCCCCC(O)=O QSBYPNXLFMSGKH-UHFFFAOYSA-N 0.000 claims description 6
239000005642 Oleic acid Substances 0.000 claims description 6
ZQPPMHVWECSIRJ-UHFFFAOYSA-N Oleic acid Natural products CCCCCCCCC=CCCCCCCCC(O)=O ZQPPMHVWECSIRJ-UHFFFAOYSA-N 0.000 claims description 6
235000005687 corn oil Nutrition 0.000 claims description 6
239000002285 corn oil Substances 0.000 claims description 6
235000014113 dietary fatty acids Nutrition 0.000 claims description 6
239000003995 emulsifying agent Substances 0.000 claims description 6
239000000194 fatty acid Substances 0.000 claims description 6
229930195729 fatty acid Natural products 0.000 claims description 6
150000004665 fatty acids Chemical class 0.000 claims description 6
QXJSBBXBKPUZAA-UHFFFAOYSA-N isooleic acid Natural products CCCCCCCC=CCCCCCCCCC(O)=O QXJSBBXBKPUZAA-UHFFFAOYSA-N 0.000 claims description 6
ZQPPMHVWECSIRJ-KTKRTIGZSA-N oleic acid Chemical compound CCCCCCCC\C=C/CCCCCCCC(O)=O ZQPPMHVWECSIRJ-KTKRTIGZSA-N 0.000 claims description 6
235000015112 vegetable and seed oil Nutrition 0.000 claims description 6
239000008158 vegetable oil Substances 0.000 claims description 6
239000008159 sesame oil Substances 0.000 claims description 5
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UFTFJSFQGQCHQW-UHFFFAOYSA-N triformin Chemical compound O=COCC(OC=O)COC=O UFTFJSFQGQCHQW-UHFFFAOYSA-N 0.000 claims description 5
239000005632 Capric acid (CAS 334-48-5) Substances 0.000 claims description 4
239000005635 Caprylic acid (CAS 124-07-2) Substances 0.000 claims description 4
125000002252 acyl group Chemical group 0.000 claims description 4
125000004432 carbon atom Chemical group C* 0.000 claims description 4
POULHZVOKOAJMA-UHFFFAOYSA-N dodecanoic acid Chemical compound CCCCCCCCCCCC(O)=O POULHZVOKOAJMA-UHFFFAOYSA-N 0.000 claims description 4
239000008136 water-miscible vehicle Substances 0.000 claims description 4
OYHQOLUKZRVURQ-HZJYTTRNSA-N Linoleic acid Chemical compound CCCCC\C=C/C\C=C/CCCCCCCC(O)=O OYHQOLUKZRVURQ-HZJYTTRNSA-N 0.000 claims description 3
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YHAIUSTWZPMYGG-UHFFFAOYSA-L disodium;2,2-dioctyl-3-sulfobutanedioate Chemical compound [Na+].[Na+].CCCCCCCCC(C([O-])=O)(C(C([O-])=O)S(O)(=O)=O)CCCCCCCC YHAIUSTWZPMYGG-UHFFFAOYSA-L 0.000 claims description 2
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OYHQOLUKZRVURQ-IXWMQOLASA-N linoleic acid Natural products CCCCC\C=C/C\C=C\CCCCCCCC(O)=O OYHQOLUKZRVURQ-IXWMQOLASA-N 0.000 claims description 2
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239000002775 capsule Substances 0.000 description 14
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238000010521 absorption reaction Methods 0.000 description 13
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FAPWRFPIFSIZLT-UHFFFAOYSA-M Sodium chloride Chemical compound [Na+].[Cl-] FAPWRFPIFSIZLT-UHFFFAOYSA-M 0.000 description 12
239000012729 immediate-release (IR) formulation Substances 0.000 description 12
150000003626 triacylglycerols Chemical class 0.000 description 12
LOKCTEFSRHRXRJ-UHFFFAOYSA-I dipotassium trisodium dihydrogen phosphate hydrogen phosphate dichloride Chemical compound P(=O)(O)(O)[O-].[K+].P(=O)(O)([O-])[O-].[Na+].[Na+].[Cl-].[K+].[Cl-].[Na+] LOKCTEFSRHRXRJ-UHFFFAOYSA-I 0.000 description 11
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JVTAAEKCZFNVCJ-UHFFFAOYSA-M Lactate Chemical compound CC(O)C([O-])=O JVTAAEKCZFNVCJ-UHFFFAOYSA-M 0.000 description 9
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GLQPTZAAUROJMO-UHFFFAOYSA-N 4-(3,4-dimethoxyphenyl)benzaldehyde Chemical compound C1=C(OC)C(OC)=CC=C1C1=CC=C(C=O)C=C1 GLQPTZAAUROJMO-UHFFFAOYSA-N 0.000 description 7
238000004128 high performance liquid chromatography Methods 0.000 description 7
239000000693 micelle Substances 0.000 description 7
210000000813 small intestine Anatomy 0.000 description 7
ZMANZCXQSJIPKH-UHFFFAOYSA-N Triethylamine Chemical compound CCN(CC)CC ZMANZCXQSJIPKH-UHFFFAOYSA-N 0.000 description 6
239000008280 blood Substances 0.000 description 6
210000004369 blood Anatomy 0.000 description 6
238000009472 formulation Methods 0.000 description 6
239000002609 medium Substances 0.000 description 6
238000000034 method Methods 0.000 description 6
229960003660 sertraline hydrochloride Drugs 0.000 description 6
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QTBSBXVTEAMEQO-UHFFFAOYSA-M Acetate Chemical compound CC([O-])=O QTBSBXVTEAMEQO-UHFFFAOYSA-M 0.000 description 5
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CKLJMWTZIZZHCS-REOHCLBHSA-N L-aspartic acid Chemical compound OC(=O)[C@@H](N)CC(O)=O CKLJMWTZIZZHCS-REOHCLBHSA-N 0.000 description 4
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GHBFNMLVSPCDGN-UHFFFAOYSA-N rac-1-monooctanoylglycerol Chemical compound CCCCCCCC(=O)OCC(O)CO GHBFNMLVSPCDGN-UHFFFAOYSA-N 0.000 description 4
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LDVVMCZRFWMZSG-UHFFFAOYSA-N captan Chemical compound C1C=CCC2C(=O)N(SC(Cl)(Cl)Cl)C(=O)C21 LDVVMCZRFWMZSG-UHFFFAOYSA-N 0.000 description 3
GHVNFZFCNZKVNT-UHFFFAOYSA-M decanoate Chemical compound CCCCCCCCCC([O-])=O GHVNFZFCNZKVNT-UHFFFAOYSA-M 0.000 description 3
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GVJHHUAWPYXKBD-UHFFFAOYSA-N (±)-α-Tocopherol Chemical compound OC1=C(C)C(C)=C2OC(CCCC(C)CCCC(C)CCCC(C)C)(C)CCC2=C1C GVJHHUAWPYXKBD-UHFFFAOYSA-N 0.000 description 2
OIQOAYVCKAHSEJ-UHFFFAOYSA-N 2-[2,3-bis(2-hydroxyethoxy)propoxy]ethanol;hexadecanoic acid;octadecanoic acid Chemical compound OCCOCC(OCCO)COCCO.CCCCCCCCCCCCCCCC(O)=O.CCCCCCCCCCCCCCCCCC(O)=O OIQOAYVCKAHSEJ-UHFFFAOYSA-N 0.000 description 2
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125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 description 1
239000002480 mineral oil Substances 0.000 description 1
235000010446 mineral oil Nutrition 0.000 description 1
239000004941 mixed matrix membrane Substances 0.000 description 1
238000002156 mixing Methods 0.000 description 1
RZRNAYUHWVFMIP-UHFFFAOYSA-N monoelaidin Natural products CCCCCCCCC=CCCCCCCCC(=O)OCC(O)CO RZRNAYUHWVFMIP-UHFFFAOYSA-N 0.000 description 1
239000000178 monomer Substances 0.000 description 1
229940037959 monooctanoin Drugs 0.000 description 1
229940074096 monoolein Drugs 0.000 description 1
208000010125 myocardial infarction Diseases 0.000 description 1
230000008693 nausea Effects 0.000 description 1
FBUKVWPVBMHYJY-UHFFFAOYSA-N nonanoic acid Chemical compound CCCCCCCCC(O)=O FBUKVWPVBMHYJY-UHFFFAOYSA-N 0.000 description 1
235000020824 obesity Nutrition 0.000 description 1
239000003401 opiate antagonist Substances 0.000 description 1
229940126701 oral medication Drugs 0.000 description 1
235000011837 pasties Nutrition 0.000 description 1
JLFNLZLINWHATN-UHFFFAOYSA-N pentaethylene glycol Chemical compound OCCOCCOCCOCCOCCO JLFNLZLINWHATN-UHFFFAOYSA-N 0.000 description 1
NBIIXXVUZAFLBC-UHFFFAOYSA-K phosphate Chemical compound [O-]P([O-])([O-])=O NBIIXXVUZAFLBC-UHFFFAOYSA-K 0.000 description 1
239000010452 phosphate Substances 0.000 description 1
230000004962 physiological condition Effects 0.000 description 1
230000036470 plasma concentration Effects 0.000 description 1
208000028173 post-traumatic stress disease Diseases 0.000 description 1
239000002244 precipitate Substances 0.000 description 1
230000001376 precipitating effect Effects 0.000 description 1
230000008569 process Effects 0.000 description 1
238000011160 research Methods 0.000 description 1
230000004044 response Effects 0.000 description 1
238000004007 reversed phase HPLC Methods 0.000 description 1
239000012047 saturated solution Substances 0.000 description 1
229940124834 selective serotonin reuptake inhibitor Drugs 0.000 description 1
239000012896 selective serotonin reuptake inhibitor Substances 0.000 description 1
229940076279 serotonin Drugs 0.000 description 1
239000011734 sodium Substances 0.000 description 1
229910052708 sodium Inorganic materials 0.000 description 1
HPALAKNZSZLMCH-UHFFFAOYSA-M sodium;chloride;hydrate Chemical compound O.[Na+].[Cl-] HPALAKNZSZLMCH-UHFFFAOYSA-M 0.000 description 1
239000011877 solvent mixture Substances 0.000 description 1
230000002269 spontaneous effect Effects 0.000 description 1
239000012086 standard solution Substances 0.000 description 1
208000011117 substance-related disease Diseases 0.000 description 1
230000009747 swallowing Effects 0.000 description 1
230000009885 systemic effect Effects 0.000 description 1
YLQBMQCUIZJEEH-UHFFFAOYSA-N tetrahydrofuran Natural products C=1C=COC=1 YLQBMQCUIZJEEH-UHFFFAOYSA-N 0.000 description 1
238000002560 therapeutic procedure Methods 0.000 description 1
238000002627 tracheal intubation Methods 0.000 description 1
125000004044 trifluoroacetyl group Chemical group FC(C(=O)*)(F)F 0.000 description 1
238000011144 upstream manufacturing Methods 0.000 description 1
229940088594 vitamin Drugs 0.000 description 1
229930003231 vitamin Natural products 0.000 description 1
239000011782 vitamin Substances 0.000 description 1
235000013343 vitamin Nutrition 0.000 description 1
229940046009 vitamin E Drugs 0.000 description 1
235000019165 vitamin E Nutrition 0.000 description 1
239000011709 vitamin E Substances 0.000 description 1

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/4841—Filling excipients; Inactive ingredients
- A61K9/4858—Organic compounds
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

Health & Medical Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Veterinary Medicine (AREA)
Chemical & Material Sciences (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
Animal Behavior & Ethology (AREA)
Life Sciences & Earth Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Engineering & Computer Science (AREA)
General Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Bioinformatics & Cheminformatics (AREA)
Organic Chemistry (AREA)
Epidemiology (AREA)
Neurosurgery (AREA)
Neurology (AREA)
Biomedical Technology (AREA)
Psychiatry (AREA)
Child & Adolescent Psychology (AREA)
Addiction (AREA)
Obesity (AREA)
Hematology (AREA)
Pain & Pain Management (AREA)
Endocrinology (AREA)
Reproductive Health (AREA)
Diabetes (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Medicinal Preparation (AREA)

SK1805-99A 1997-07-01 1998-06-16 Sertralínová dávkovacia forma SK282914B6 (sk)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US5140197P	1997-07-01	1997-07-01
PCT/IB1998/000936 WO1999001113A1 (en)	1997-07-01	1998-06-16	Gelatine encapsulated solution dosage forms of sertraline

Publications (2)

Publication Number	Publication Date
SK180599A3 SK180599A3 (en)	2001-01-18
SK282914B6 true SK282914B6 (sk)	2003-01-09

Family

ID=21971076

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
SK1805-99A SK282914B6 (sk)	1997-07-01	1998-06-16	Sertralínová dávkovacia forma

Country Status (40)

Country	Link
EP (1)	EP0980241B1 (de)
JP (1)	JP3585245B2 (de)
KR (1)	KR100371730B1 (de)
CN (1)	CN1261792A (de)
AP (1)	AP945A (de)
AR (1)	AR015916A1 (de)
AT (1)	ATE256457T1 (de)
AU (1)	AU724635B2 (de)
BG (1)	BG103917A (de)
BR (1)	BR9809712A (de)
CA (1)	CA2290973C (de)
CO (1)	CO4940405A1 (de)
DE (1)	DE69820608T2 (de)
DK (1)	DK0980241T3 (de)
DZ (1)	DZ2544A1 (de)
EA (1)	EA001905B1 (de)
ES (1)	ES2210760T3 (de)
GT (1)	GT199800090A (de)
HR (1)	HRP980378B1 (de)
HU (1)	HUP0002250A3 (de)
ID (1)	ID24673A (de)
IL (1)	IL133075A0 (de)
IS (1)	IS5266A (de)
MA (1)	MA24586A1 (de)
MY (1)	MY119728A (de)
NO (1)	NO996492L (de)
NZ (1)	NZ501252A (de)
OA (1)	OA11246A (de)
PA (1)	PA8454001A1 (de)
PE (1)	PE97299A1 (de)
PL (1)	PL337807A1 (de)
PT (1)	PT980241E (de)
SK (1)	SK282914B6 (de)
TN (1)	TNSN98123A1 (de)
TR (1)	TR199903282T2 (de)
TW (1)	TW382597B (de)
UA (1)	UA68350C2 (de)
UY (1)	UY25070A1 (de)
WO (1)	WO1999001113A1 (de)
ZA (1)	ZA985709B (de)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US6727283B2 (en)	1998-10-13	2004-04-27	Pfizer Inc.	Sertraline oral concentrate
WO2000021521A2 (en) *	1998-10-13	2000-04-20	Pfizer Products Inc.	Sertraline oral concentrate
PL211402B1 (pl)	1999-09-03	2012-05-31	Apbi Holdings	Zastosowanie dapoksetyny do leczenia lub zwalczania przedwczesnej ejakulacji
MXPA03001771A (es)	2000-08-30	2003-06-04	Pfizer Prod Inc	Formulaciones de liberacion sostenida para secretagogos de hormona del crecimiento.
EP1375659A1 (de) *	2002-06-18	2004-01-02	Laboratorio di Diagnostica Moleculare	Konzentratmischungen in löslichen Kapseln zur einfachen Zubereitung von chemischen oder biologischen Lösungen
EP1556000A1 (de) *	2002-10-31	2005-07-27	Alza Corporation	Pharmazeutische formulierung zur erhöhten bioverfügbarkeit hydrophober arzneistoffe
WO2016020936A2 (en) *	2014-07-21	2016-02-11	Patel Jayendrakumar Dasharathlal	A novel oral gastroretentive pharmaceutical dosage form
CN108014087A (zh) *	2017-12-27	2018-05-11	江苏联环药业股份有限公司	一种盐酸舍曲林胶囊的制备方法
GB2630572A (en)	2023-05-29	2024-12-04	Novumgen Ltd	An orally disintegrating tablet of sertraline and its process of preparation

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
ATE214276T1 (de) *	1994-09-19	2002-03-15	Du Pont Pharm Co	Zusammensetzungen von opioid antagonisten mit selektiven serotonin-aufnahme inhibitoren, zur behandlung von alkoholismus und alkohoabhängigkeit
EP0768083B1 (de) *	1995-07-17	2003-03-26	Pfizer Inc.	Sertralin zur Behandlung von Post-Myocard-Infarkt-Patienten

1998
- 1998-06-16 BR BR9809712-1A patent/BR9809712A/pt not_active Application Discontinuation
- 1998-06-16 ID IDW991697A patent/ID24673A/id unknown
- 1998-06-16 CA CA002290973A patent/CA2290973C/en not_active Expired - Fee Related
- 1998-06-16 AU AU75450/98A patent/AU724635B2/en not_active Ceased
- 1998-06-16 HU HU0002250A patent/HUP0002250A3/hu unknown
- 1998-06-16 SK SK1805-99A patent/SK282914B6/sk unknown
- 1998-06-16 DE DE69820608T patent/DE69820608T2/de not_active Expired - Fee Related
- 1998-06-16 TR TR1999/03282T patent/TR199903282T2/xx unknown
- 1998-06-16 EA EA199900963A patent/EA001905B1/ru not_active IP Right Cessation
- 1998-06-16 KR KR10-1999-7011596A patent/KR100371730B1/ko not_active Expired - Fee Related
- 1998-06-16 IL IL13307598A patent/IL133075A0/xx unknown
- 1998-06-16 NZ NZ501252A patent/NZ501252A/en unknown
- 1998-06-16 DK DK98923021T patent/DK0980241T3/da active
- 1998-06-16 PT PT98923021T patent/PT980241E/pt unknown
- 1998-06-16 ES ES98923021T patent/ES2210760T3/es not_active Expired - Lifetime
- 1998-06-16 JP JP50677699A patent/JP3585245B2/ja not_active Expired - Fee Related
- 1998-06-16 PL PL98337807A patent/PL337807A1/xx unknown
- 1998-06-16 UA UA99116393A patent/UA68350C2/uk unknown
- 1998-06-16 EP EP98923021A patent/EP0980241B1/de not_active Expired - Lifetime
- 1998-06-16 CN CN98806765A patent/CN1261792A/zh active Pending
- 1998-06-16 WO PCT/IB1998/000936 patent/WO1999001113A1/en not_active Ceased
- 1998-06-16 AT AT98923021T patent/ATE256457T1/de not_active IP Right Cessation
- 1998-06-19 PA PA19988454001A patent/PA8454001A1/es unknown
- 1998-06-25 AP APAP/P/1998/001279A patent/AP945A/en active
- 1998-06-25 TW TW087110254A patent/TW382597B/zh not_active IP Right Cessation
- 1998-06-26 PE PE1998000575A patent/PE97299A1/es not_active Application Discontinuation
- 1998-06-29 GT GT199800090A patent/GT199800090A/es unknown
- 1998-06-29 AR ARP980103145A patent/AR015916A1/es not_active Application Discontinuation
- 1998-06-29 MY MYPI98002949A patent/MY119728A/en unknown
- 1998-06-29 UY UY25070A patent/UY25070A1/es not_active IP Right Cessation
- 1998-06-30 DZ DZ980154A patent/DZ2544A1/xx active
- 1998-06-30 MA MA25145A patent/MA24586A1/fr unknown
- 1998-06-30 ZA ZA9805709A patent/ZA985709B/xx unknown
- 1998-06-30 TN TNTNSN98123A patent/TNSN98123A1/fr unknown
- 1998-07-01 CO CO98037136A patent/CO4940405A1/es unknown
- 1998-07-01 HR HR980378A patent/HRP980378B1/xx not_active IP Right Cessation
1999
- 1999-11-23 IS IS5266A patent/IS5266A/is unknown
- 1999-11-23 BG BG103917A patent/BG103917A/bg unknown
- 1999-12-23 OA OA9900306A patent/OA11246A/en unknown
- 1999-12-27 NO NO996492A patent/NO996492L/no not_active Application Discontinuation

Also Published As

Publication number	Publication date
EA001905B1 (ru)	2001-10-22
KR100371730B1 (ko)	2003-02-07
NO996492L (no)	2000-02-29
WO1999001113A1 (en)	1999-01-14
PL337807A1 (en)	2000-09-11
IS5266A (is)	1999-11-23
EA199900963A1 (ru)	2000-08-28
BR9809712A (pt)	2000-07-11
NO996492D0 (no)	1999-12-27
KR20010013588A (ko)	2001-02-26
SK180599A3 (en)	2001-01-18
CA2290973C (en)	2003-06-17
ES2210760T3 (es)	2004-07-01
EP0980241A1 (de)	2000-02-23
PT980241E (pt)	2004-03-31
HRP980378A2 (en)	1999-04-30
TR199903282T2 (xx)	2000-08-21
JP2000512316A (ja)	2000-09-19
PA8454001A1 (es)	2000-05-24
EP0980241B1 (de)	2003-12-17
OA11246A (en)	2002-11-19
CO4940405A1 (es)	2000-07-24
CA2290973A1 (en)	1999-01-14
AP945A (en)	2001-02-28
AU724635B2 (en)	2000-09-28
TNSN98123A1 (fr)	2005-03-15
AP9801279A0 (en)	1998-06-30
NZ501252A (en)	2004-11-26
IL133075A0 (en)	2001-03-19
MA24586A1 (fr)	1998-12-31
ID24673A (id)	2000-07-27
TW382597B (en)	2000-02-21
ZA985709B (en)	2000-01-10
ATE256457T1 (de)	2004-01-15
DZ2544A1 (fr)	2003-02-08
DK0980241T3 (da)	2004-04-05
AU7545098A (en)	1999-01-25
DE69820608T2 (de)	2004-12-23
HUP0002250A2 (hu)	2000-12-28
DE69820608D1 (de)	2004-01-29
HRP980378B1 (en)	2001-12-31
MY119728A (en)	2005-07-29
PE97299A1 (es)	1999-10-13
UY25070A1 (es)	2000-12-29
UA68350C2 (en)	2004-08-16
JP3585245B2 (ja)	2004-11-04
GT199800090A (es)	1999-12-21
HUP0002250A3 (en)	2001-01-29
CN1261792A (zh)	2000-08-02
BG103917A (bg)	2000-07-31
AR015916A1 (es)	2001-05-30

Publication	Publication Date	Title
EP0553178B1 (de)	1995-05-24	Zweiphasige freigabezusammensetzungen für lipophile wirkstoffe
AU692255B2 (en)	1998-06-04	Self-emulsifiable formulation producing an oil-in-water emulsion
ES2326783T3 (es)	2009-10-20	Composiciones de n-benzoilestaurosporina espontaneamente dispersables.
US20220096461A1 (en)	2022-03-31	Liquid oral dosage formulations of methylnaltrexone
CA2290973C (en)	2003-06-17	Encapsulated solution dosage forms of sertraline
JPH0840936A (ja)	1996-02-13	経口投与薬物のための製剤
US20030133974A1 (en)	2003-07-17	Encapsulated solution dosage forms of sertraline
JP3277735B2 (ja)	2002-04-22	ナフトエ酸誘導体の吸収促進組成物
WO1992014443A1 (en)	1992-09-03	Microsphere-in-oil emulsion
CZ464299A3 (cs)	2000-04-12	Želatinové zapouzdření roztokové dávkovači formy sertralinu
MXPA99012099A (en)	2000-09-04	Gelatine encapsulated solution dosage forms of sertraline
WO2012066347A1 (en)	2012-05-24	Oil based formulations
HK1028882A (en)	2001-03-09	Gelatine encapsulated solution dosage forms of sertraline
WO2026015623A2 (en)	2026-01-15	Pharmaceutical formulations comprising dydrogesterone and methods of preparation thereof
JPWO2001005406A1 (ja)	2003-02-04	粘膜吸収グリチルリチン製剤
KR20100022626A (ko)	2010-03-03	나노입자 형성을 이용하는 리세드로네이트 경질캡슐