SK284013B6 - Farmaceutická kompozícia, spôsob jej prípravy a použitie - Google Patents

Farmaceutická kompozícia, spôsob jej prípravy a použitie Download PDF

Info

Publication number: SK284013B6
Authority: SK; Slovakia
Prior art keywords: composition; agent; mixture; hydroxyrisperidone; water
Prior art date: 1996-05-20

Application number

SK620-98A

Other languages

English (en)

Slovak (sk)

Other versions

SK62098A3 (en

Inventor

Marc Karel Jozef Fran�Ois

Roger Carolus Augusta Embrechts

Herman Karel Borghijs

Johan Monbaliu

Original Assignee

Janssen Pharmaceutica N. V.

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1996-05-20

Filing date

1997-05-12

Publication date

2004-08-03

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=8224016&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SK284013(B6) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

1997-05-12 Application filed by Janssen Pharmaceutica N. V. filed Critical Janssen Pharmaceutica N. V.

2000-04-10 Publication of SK62098A3 publication Critical patent/SK62098A3/sk

2004-08-03 Publication of SK284013B6 publication Critical patent/SK284013B6/sk

Links

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WVDDGKGOMKODPV-UHFFFAOYSA-N Benzyl alcohol Chemical group OCC1=CC=CC=C1 WVDDGKGOMKODPV-UHFFFAOYSA-N 0.000 claims description 21
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RAPZEAPATHNIPO-UHFFFAOYSA-N risperidone Chemical compound FC1=CC=C2C(C3CCN(CC3)CCC=3C(=O)N4CCCCC4=NC=3C)=NOC2=C1 RAPZEAPATHNIPO-UHFFFAOYSA-N 0.000 description 26
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PMXMIIMHBWHSKN-UHFFFAOYSA-N 3-{2-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]ethyl}-9-hydroxy-2-methyl-6,7,8,9-tetrahydropyrido[1,2-a]pyrimidin-4-one Chemical compound FC1=CC=C2C(C3CCN(CC3)CCC=3C(=O)N4CCCC(O)C4=NC=3C)=NOC2=C1 PMXMIIMHBWHSKN-UHFFFAOYSA-N 0.000 description 18
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Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/517—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with carbocyclic ring systems, e.g. quinazoline, perimidine
- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
- A—HUMAN NECESSITIES
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- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A61P25/24—Antidepressants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/02—Inorganic compounds
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
- A61K47/10—Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/26—Carbohydrates, e.g. sugar alcohols, amino sugars, nucleic acids, mono-, di- or oligo-saccharides; Derivatives thereof, e.g. polysorbates, sorbitan fatty acid esters or glycyrrhizin
- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
- A61K47/36—Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
- A61K47/38—Cellulose; Derivatives thereof

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Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Neurology (AREA)
Biomedical Technology (AREA)
Neurosurgery (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Organic Chemistry (AREA)
Epidemiology (AREA)
Psychiatry (AREA)
Dermatology (AREA)
Hospice & Palliative Care (AREA)
Pain & Pain Management (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Medicinal Preparation (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Agricultural Chemicals And Associated Chemicals (AREA)

SK620-98A 1996-05-20 1997-05-12 Farmaceutická kompozícia, spôsob jej prípravy a použitie SK284013B6 (sk)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
EP96201429		1996-05-20
PCT/EP1997/002504 WO1997044039A1 (fr)	1996-05-20	1997-05-12	Suspensions aqueuses d'esters d'acides gras de 9-hydroxyrisperidone

Publications (2)

Publication Number	Publication Date
SK62098A3 SK62098A3 (en)	2000-04-10
SK284013B6 true SK284013B6 (sk)	2004-08-03

Family

ID=8224016

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
SK620-98A SK284013B6 (sk)	1996-05-20	1997-05-12	Farmaceutická kompozícia, spôsob jej prípravy a použitie

Country Status (37)

Country	Link
US (1)	US6077843A (fr)
EP (1)	EP0904081B1 (fr)
JP (1)	JP3274687B2 (fr)
KR (1)	KR100358373B1 (fr)
CN (1)	CN1093762C (fr)
AR (1)	AR007194A1 (fr)
AT (1)	ATE208619T1 (fr)
AU (1)	AU715572B2 (fr)
BG (1)	BG62684B1 (fr)
BR (1)	BR9706824B8 (fr)
CA (1)	CA2236691C (fr)
CY (2)	CY2270B1 (fr)
CZ (1)	CZ291284B6 (fr)
DE (2)	DE122011100027I1 (fr)
DK (1)	DK0904081T3 (fr)
EA (1)	EA000536B1 (fr)
EE (1)	EE03594B1 (fr)
ES (1)	ES2167745T3 (fr)
FR (1)	FR11C0035I2 (fr)
HR (1)	HRP970276B1 (fr)
HU (2)	HU224025B1 (fr)
ID (1)	ID16927A (fr)
IL (1)	IL124551A (fr)
LU (1)	LU91842I2 (fr)
MX (1)	MX9804816A (fr)
MY (1)	MY126302A (fr)
NO (2)	NO315931B1 (fr)
NZ (1)	NZ330369A (fr)
PL (1)	PL188309B1 (fr)
PT (1)	PT904081E (fr)
SI (1)	SI0904081T1 (fr)
SK (1)	SK284013B6 (fr)
TR (1)	TR199800923T2 (fr)
TW (1)	TW487572B (fr)
UA (1)	UA61898C2 (fr)
WO (1)	WO1997044039A1 (fr)
ZA (1)	ZA974331B (fr)

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KR101760953B1 (ko)	2008-09-04	2017-07-24	아밀린 파마슈티칼스, 엘엘씨.	비-수성 담체를 이용한 서방성 제형물
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1997
- 1997-05-01 TW TW086105768A patent/TW487572B/zh not_active IP Right Cessation
- 1997-05-12 EE EE9800136A patent/EE03594B1/xx active Protection Beyond IP Right Term
- 1997-05-12 NZ NZ330369A patent/NZ330369A/xx not_active IP Right Cessation
- 1997-05-12 BR BRPI9706824-1B8A patent/BR9706824B8/pt not_active IP Right Cessation
- 1997-05-12 PT PT97923912T patent/PT904081E/pt unknown
- 1997-05-12 HU HU9901319A patent/HU224025B1/hu active Protection Beyond IP Right Term
- 1997-05-12 EP EP97923912A patent/EP0904081B1/fr not_active Expired - Lifetime
- 1997-05-12 ES ES97923912T patent/ES2167745T3/es not_active Expired - Lifetime
- 1997-05-12 WO PCT/EP1997/002504 patent/WO1997044039A1/fr not_active Ceased
- 1997-05-12 TR TR1998/00923T patent/TR199800923T2/xx unknown
- 1997-05-12 AT AT97923912T patent/ATE208619T1/de active
- 1997-05-12 DE DE201112100027 patent/DE122011100027I1/de active Pending
- 1997-05-12 DK DK97923912T patent/DK0904081T3/da active
- 1997-05-12 SI SI9730272T patent/SI0904081T1/xx unknown
- 1997-05-12 AU AU29559/97A patent/AU715572B2/en not_active Expired
- 1997-05-12 PL PL97327995A patent/PL188309B1/pl unknown
- 1997-05-12 CN CN97191494A patent/CN1093762C/zh not_active Expired - Lifetime
- 1997-05-12 EA EA199800531A patent/EA000536B1/ru not_active IP Right Cessation
- 1997-05-12 KR KR10-1998-0703629A patent/KR100358373B1/ko not_active Expired - Lifetime
- 1997-05-12 JP JP54150097A patent/JP3274687B2/ja not_active Expired - Lifetime
- 1997-05-12 CA CA002236691A patent/CA2236691C/fr not_active Expired - Lifetime
- 1997-05-12 IL IL12455197A patent/IL124551A/xx not_active IP Right Cessation
- 1997-05-12 DE DE69708284T patent/DE69708284T2/de not_active Expired - Lifetime
- 1997-05-12 US US09/180,659 patent/US6077843A/en not_active Expired - Lifetime
- 1997-05-12 SK SK620-98A patent/SK284013B6/sk not_active IP Right Cessation
- 1997-05-12 CZ CZ19981401A patent/CZ291284B6/cs not_active IP Right Cessation
- 1997-05-19 MY MYPI97002172A patent/MY126302A/en unknown
- 1997-05-19 ZA ZA974331A patent/ZA974331B/xx unknown
- 1997-05-19 AR ARP970102112A patent/AR007194A1/es active IP Right Grant
- 1997-05-19 ID IDP971649A patent/ID16927A/id unknown
- 1997-05-20 HR HR970276A patent/HRP970276B1/xx not_active IP Right Cessation
- 1997-12-05 UA UA98052747A patent/UA61898C2/uk unknown
1998
- 1998-04-30 NO NO19981984A patent/NO315931B1/no not_active IP Right Cessation
- 1998-05-12 BG BG102443A patent/BG62684B1/bg unknown
- 1998-06-15 MX MX9804816A patent/MX9804816A/es unknown
2002
- 2002-04-25 CY CY0200021A patent/CY2270B1/xx unknown
2011
- 2011-07-20 LU LU91842C patent/LU91842I2/fr unknown
- 2011-08-18 CY CY2011011C patent/CY2011011I1/el unknown
- 2011-08-18 HU HUS1100013C patent/HUS1100013I1/hu unknown
- 2011-08-29 NO NO2011015C patent/NO2011015I2/no unknown
- 2011-09-02 FR FR11C0035C patent/FR11C0035I2/fr active Active

Also Published As

Publication number	Publication date
HUS1100013I1 (hu)	2017-03-28
FR11C0035I1 (fr)	2011-07-10
DE69708284T2 (de)	2002-07-25
HK1017852A1 (en)	1999-12-03
EE9800136A (et)	1998-10-15
PL327995A1 (en)	1999-01-04
JP2000513718A (ja)	2000-10-17
HU224025B1 (hu)	2005-05-30
NZ330369A (en)	2000-04-28
US6077843A (en)	2000-06-20
ZA974331B (en)	1998-11-19
KR100358373B1 (ko)	2003-02-11
EP0904081A1 (fr)	1999-03-31
NO2011015I1 (no)	2011-09-19
EA199800531A1 (ru)	1998-12-24
NO981984L (no)	1998-11-19
BR9706824B8 (pt)	2015-02-18
HUP9901319A3 (en)	1999-11-29
SI0904081T1 (en)	2002-04-30
NO2011015I2 (no)	2013-03-11
DE122011100027I1 (de)	2011-11-17
PL188309B1 (pl)	2005-01-31
CY2270B1 (en)	2003-07-04
HRP970276B1 (en)	2002-04-30
EP0904081B1 (fr)	2001-11-14
MY126302A (en)	2006-09-29
CN1206347A (zh)	1999-01-27
IL124551A (en)	2001-08-26
EE03594B1 (et)	2002-02-15
HUP9901319A2 (hu)	1999-08-30
LU91842I2 (fr)	2011-09-20
AR007194A1 (es)	1999-10-13
CA2236691A1 (fr)	1997-11-27
FR11C0035I2 (fr)	2013-08-16
NO981984D0 (no)	1998-04-30
KR19990067603A (ko)	1999-08-25
PT904081E (pt)	2002-04-29
DK0904081T3 (da)	2002-02-25
NO315931B1 (no)	2003-11-17
BG102443A (en)	1999-06-30
ES2167745T3 (es)	2002-05-16
HRP970276A2 (en)	1998-04-30
WO1997044039A1 (fr)	1997-11-27
CZ140198A3 (cs)	1999-04-14
CZ291284B6 (cs)	2003-01-15
TR199800923T2 (xx)	1999-09-21
ID16927A (id)	1997-11-20
SK62098A3 (en)	2000-04-10
CN1093762C (zh)	2002-11-06
BG62684B1 (bg)	2000-05-31
EA000536B1 (ru)	1999-10-28
DE69708284D1 (de)	2001-12-20
BR9706824A (pt)	1999-03-23
AU715572B2 (en)	2000-02-03
CA2236691C (fr)	2007-01-02
AU2955997A (en)	1997-12-09
MX9804816A (es)	1998-10-31
CY2011011I2 (el)	2016-12-14
ATE208619T1 (de)	2001-11-15
JP3274687B2 (ja)	2002-04-15
TW487572B (en)	2002-05-21
UA61898C2 (en)	2003-12-15
IL124551A0 (en)	1998-12-06
CY2011011I1 (el)	2016-12-14

Legal Events

Date

Code

Title

Description

2012-03-02

SPCF

Filing of an spc

Free format text: PRODUCT NAME: PALIPERIDON; REGISTRATION NO/DATE: EU/1/11/672/001 - EU/1/11/672/006 20110304

Spc suppl protection certif: 5007-2011

Filing date: 20110804

2015-08-04

SPCG

Grant of an spc