SK287423B6 - Farmaceuticky účinné uridínové estery, ich použitie, spôsob ich prípravy a farmaceutický prostriedok - Google Patents

Farmaceuticky účinné uridínové estery, ich použitie, spôsob ich prípravy a farmaceutický prostriedok Download PDF

Info

Publication number: SK287423B6
Authority: SK; Slovakia
Prior art keywords: alkyl chain; acid; branched; dihydroxy; dioxo
Prior art date: 2001-04-30

Application number

SK1341-2003A

Other languages

English (en)

Slovak (sk)

Other versions

SK13412003A3 (sk

Inventor

Rudy Susilo

Original Assignee

Trommsdorff Gmbh & Co. Kg Arzneimittel

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2001-04-30

Filing date

2002-04-29

Publication date

2010-09-07

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27440125&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SK287423(B6) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

2002-04-29 Application filed by Trommsdorff Gmbh & Co. Kg Arzneimittel filed Critical Trommsdorff Gmbh & Co. Kg Arzneimittel

2004-05-04 Publication of SK13412003A3 publication Critical patent/SK13412003A3/sk

2010-09-07 Publication of SK287423B6 publication Critical patent/SK287423B6/sk

Links

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238000000034 method Methods 0.000 title claims abstract description 26
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-1 uridine ester Chemical group 0.000 claims abstract description 160
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Classifications

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- A61P9/00—Drugs for disorders of the cardiovascular system
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- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
- C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
- C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
- C07H19/06—Pyrimidine radicals

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SK1341-2003A 2001-04-30 2002-04-29 Farmaceuticky účinné uridínové estery, ich použitie, spôsob ich prípravy a farmaceutický prostriedok SK287423B6 (sk)

Applications Claiming Priority (5)

Application Number	Priority Date	Filing Date	Title
EP01110608		2001-04-30
US28809001P	2001-05-03	2001-05-03
EP01124879		2001-10-18
US33042901P	2001-10-22	2001-10-22
PCT/EP2002/004725 WO2002088159A1 (en)	2001-04-30	2002-04-29	Pharmaceutically active uridine esters

Publications (2)

Publication Number	Publication Date
SK13412003A3 SK13412003A3 (sk)	2004-05-04
SK287423B6 true SK287423B6 (sk)	2010-09-07

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Application Number	Title	Priority Date	Filing Date
SK1341-2003A SK287423B6 (sk)	2001-04-30	2002-04-29	Farmaceuticky účinné uridínové estery, ich použitie, spôsob ich prípravy a farmaceutický prostriedok

Country Status (25)

Country	Link
EP (2)	EP1390378B1 (de)
KR (1)	KR100660754B1 (de)
CN (1)	CN1505636A (de)
AT (1)	ATE433989T1 (de)
AU (2)	AU2002308068B2 (de)
BG (1)	BG108299A (de)
BR (1)	BR0209320A (de)
CA (2)	CA2445861A1 (de)
CZ (1)	CZ20032957A3 (de)
DE (1)	DE60232653D1 (de)
DK (1)	DK1390378T3 (de)
EE (1)	EE05434B1 (de)
ES (1)	ES2327397T3 (de)
HR (1)	HRP20030879A2 (de)
HU (1)	HUP0400732A3 (de)
IL (1)	IL158006A0 (de)
IS (1)	IS6997A (de)
MX (1)	MXPA03009737A (de)
NO (2)	NO326964B1 (de)
NZ (2)	NZ546060A (de)
PL (1)	PL209031B1 (de)
PT (1)	PT1390378E (de)
SK (1)	SK287423B6 (de)
UA (1)	UA74250C2 (de)
WO (1)	WO2002088159A1 (de)

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MX2010000224A (es)	2007-06-26	2010-05-03	Nutricia Nv	Mejoramiento de la memoria en individuos con mini-examen de estado mental de 24-26.
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MX2010000424A (es)	2007-07-09	2010-08-10	Easter Virginia Medical School	Derivados de nucleosidos sustituidos con propiedades antivirales y antimicrobianas.
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CN101951923B (zh)	2007-12-20	2013-10-30	N.V.努特里奇亚	含核苷酸/核苷的液态产品
US8257722B2 (en)	2008-09-15	2012-09-04	Cv Ingenuity Corp.	Local delivery of water-soluble or water-insoluble therapeutic agents to the surface of body lumens
US9198968B2 (en)	2008-09-15	2015-12-01	The Spectranetics Corporation	Local delivery of water-soluble or water-insoluble therapeutic agents to the surface of body lumens
US8114429B2 (en)	2008-09-15	2012-02-14	Cv Ingenuity Corp.	Local delivery of water-soluble or water-insoluble therapeutic agents to the surface of body lumens
WO2012091542A1 (en)	2010-12-28	2012-07-05	N.V. Nutricia	Combination of components for the prevention and treatment of frailty
US9956385B2 (en)	2012-06-28	2018-05-01	The Spectranetics Corporation	Post-processing of a medical device to control morphology and mechanical properties
CA2928190C (en) *	2013-10-23	2023-09-19	Chemgenes Corporation	Dithiolane functionalized nucleoside amidites and supports for stronger immobilization of bio-molecules on solid surfaces
WO2015084158A1 (en)	2013-12-06	2015-06-11	N.V. Nutricia	A pyrimidine derivative and a fatty acid source for use in the treatment of constipation
WO2016053085A1 (en)	2014-09-30	2016-04-07	N.V. Nutricia	Composition comprising a uridine source and butyrate producing fibres for preventing gastrointestinal disorders
DK3236972T3 (en)	2014-12-26	2021-10-04	Univ Emory	Antivirale N4-hydroxycytidin-derivativer
DE202015105351U1 (de)	2015-10-09	2016-01-07	Apotheke am Schlossplatz Inh. Mario Ganster e.K.	Diätetische Zusammensetzung
WO2017069613A1 (en)	2015-10-23	2017-04-27	N.V. Nutricia	Method for improving recognition and/or working memory in hyperphenylalanimenia and phenylketonuria patients
WO2017069611A1 (en)	2015-10-23	2017-04-27	N.V. Nutricia	Nutritional product for decreasing phenylalanine levels in pku patients
WO2017155387A1 (en)	2016-03-08	2017-09-14	N.V. Nutricia	Method for supporting memory function and/or cognitive function
WO2017155386A1 (en) *	2016-03-08	2017-09-14	N.V. Nutricia	Method for treating brain atrophy
JP6804790B1 (ja)	2017-12-07	2020-12-23	エモリーユニバーシティー	Ｎ４−ヒドロキシシチジンおよび誘導体ならびにそれらに関連する抗ウイルス用途
TW202317144A (zh)	2021-06-14	2023-05-01	美商維納拓爾斯製藥公司	口服生物可利用的核苷類似物
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2002
- 2002-04-29 PT PT02766645T patent/PT1390378E/pt unknown
- 2002-04-29 PL PL363178A patent/PL209031B1/pl not_active IP Right Cessation
- 2002-04-29 IL IL15800602A patent/IL158006A0/xx unknown
- 2002-04-29 AT AT02766645T patent/ATE433989T1/de active
- 2002-04-29 NZ NZ546060A patent/NZ546060A/en not_active IP Right Cessation
- 2002-04-29 CN CNA028091604A patent/CN1505636A/zh active Pending
- 2002-04-29 KR KR1020037014215A patent/KR100660754B1/ko not_active Expired - Fee Related
- 2002-04-29 HU HU0400732A patent/HUP0400732A3/hu unknown
- 2002-04-29 BR BR0209320-0A patent/BR0209320A/pt not_active IP Right Cessation
- 2002-04-29 HR HR20030879A patent/HRP20030879A2/xx not_active Application Discontinuation
- 2002-04-29 ES ES02766645T patent/ES2327397T3/es not_active Expired - Lifetime
- 2002-04-29 DE DE60232653T patent/DE60232653D1/de not_active Expired - Lifetime
- 2002-04-29 NZ NZ528634A patent/NZ528634A/en not_active IP Right Cessation
- 2002-04-29 CA CA002445861A patent/CA2445861A1/en not_active Abandoned
- 2002-04-29 EP EP02766645A patent/EP1390378B1/de not_active Revoked
- 2002-04-29 CA CA002594883A patent/CA2594883A1/en not_active Abandoned
- 2002-04-29 SK SK1341-2003A patent/SK287423B6/sk not_active IP Right Cessation
- 2002-04-29 MX MXPA03009737A patent/MXPA03009737A/es active IP Right Grant
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- 2002-04-29 AU AU2002308068A patent/AU2002308068B2/en not_active Ceased
- 2002-04-29 UA UA2003109720A patent/UA74250C2/uk unknown
2003
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2006
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Also Published As

Publication number	Publication date
HRP20030879A2 (en)	2005-08-31
NZ546060A (en)	2006-11-30
KR100660754B1 (ko)	2006-12-26
DK1390378T3 (da)	2009-09-14
AU2006200874A1 (en)	2006-03-23
AU2002308068B2 (en)	2006-06-15
EP1390378B1 (de)	2009-06-17
HUP0400732A2 (hu)	2004-06-28
EP1666092A3 (de)	2006-11-29
CN1505636A (zh)	2004-06-16
MXPA03009737A (es)	2005-03-07
BG108299A (bg)	2004-09-30
CA2594883A1 (en)	2002-11-07
ES2327397T3 (es)	2009-10-29
CA2445861A1 (en)	2002-11-07
PL363178A1 (en)	2004-11-15
BR0209320A (pt)	2004-07-20
PL209031B1 (pl)	2011-07-29
PT1390378E (pt)	2009-07-23
IS6997A (is)	2003-10-21
NO326964B1 (no)	2009-03-23
ATE433989T1 (de)	2009-07-15
NO20034782L (no)	2003-12-12
IL158006A0 (en)	2004-03-28
EP1390378A1 (de)	2004-02-25
CZ20032957A3 (cs)	2004-02-18
DE60232653D1 (de)	2009-07-30
NO20082222L (no)	2003-12-12
UA74250C2 (uk)	2005-11-15
EE200300536A (et)	2004-02-16
NZ528634A (en)	2005-04-29
WO2002088159A1 (en)	2002-11-07
HUP0400732A3 (en)	2007-05-29
EE05434B1 (et)	2011-06-15
SK13412003A3 (sk)	2004-05-04
KR20040016859A (ko)	2004-02-25
NO20034782D0 (no)	2003-10-24
EP1666092A2 (de)	2006-06-07

Legal Events

Date	Code	Title	Description
2014-01-08	MM4A	Patent lapsed due to non-payment of maintenance fees	Effective date: 20130429

Publication	Publication Date	Title
SK287423B6 (sk)	2010-09-07	Farmaceuticky účinné uridínové estery, ich použitie, spôsob ich prípravy a farmaceutický prostriedok
US7417034B2 (en)	2008-08-26	Pharmaceutically active uridine esters
AU2002308068A1 (en)	2003-04-17	Pharmaceutically active uridine esters
EP1957086B1 (de)	2018-05-02	Nicotinoyl-ribosid-zusammensetzungen und anwendungsverfahren
MXPA06010075A (es)	2007-04-10	Compuestos terapeuticos.
IL153379A (en)	2007-02-11	2' - deoxy - 3' - d - valinyl - ?? - l - cytidine and similar compounds as prodrugs and pharmaceutical compositions containing them
WO2012158811A2 (en)	2012-11-22	Purine monophosphate prodrugs for treatment of viral infections
EP2935304A1 (de)	2015-10-28	4'-fluor-nukleoside zur behandlung von hcv
MX2008012185A (es)	2008-10-02	Compuestos de purina y metodos de uso de los mismos.
ZA200308420B (en)	2004-10-29	Pharmaceutically active uridine esters.
CN1227489A (zh)	1999-09-01	腺嘌呤核苷脱氨酶抑制剂
DE60020891T2 (de)	2005-12-08	Arylphosphatderivate von d4t
KR101425228B1 (ko)	2014-08-06	암의 치료를 위한 디옥솔란 유도체
HK1065318A (en)	2005-02-18	Pharmaceutically active uridine esters
HK1094149A (en)	2007-03-23	Pharmaceutically active uridine esters