TR200000135T2 - Tiazolidinedion ve sülfonilüre ile diabet tedavisi. - Google Patents
Tiazolidinedion ve sülfonilüre ile diabet tedavisi.Info
- Publication number
- TR200000135T2 TR200000135T2 TR2000/00135T TR200000135T TR200000135T2 TR 200000135 T2 TR200000135 T2 TR 200000135T2 TR 2000/00135 T TR2000/00135 T TR 2000/00135T TR 200000135 T TR200000135 T TR 200000135T TR 200000135 T2 TR200000135 T2 TR 200000135T2
- Authority
- TR
- Turkey
- Prior art keywords
- thiazolidinedione
- sulfonylurea
- diabetes treatment
- mammal
- mellitus
- Prior art date
Links
- 206010012601 diabetes mellitus Diseases 0.000 title abstract 2
- ZOBPZXTWZATXDG-UHFFFAOYSA-N 1,3-thiazolidine-2,4-dione Chemical compound O=C1CSC(=O)N1 ZOBPZXTWZATXDG-UHFFFAOYSA-N 0.000 title 1
- 229940100389 Sulfonylurea Drugs 0.000 title 1
- 229940123464 Thiazolidinedione Drugs 0.000 title 1
- YROXIXLRRCOBKF-UHFFFAOYSA-N sulfonylurea Chemical class OC(=N)N=S(=O)=O YROXIXLRRCOBKF-UHFFFAOYSA-N 0.000 title 1
- 241000124008 Mammalia Species 0.000 abstract 2
- 229940122199 Insulin secretagogue Drugs 0.000 abstract 1
- 229940122355 Insulin sensitizer Drugs 0.000 abstract 1
- 231100000252 nontoxic Toxicity 0.000 abstract 1
- 230000003000 nontoxic effect Effects 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/64—Sulfonylureas, e.g. glibenclamide, tolbutamide, chlorpropamide
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/48—Drugs for disorders of the endocrine system of the pancreatic hormones
- A61P5/50—Drugs for disorders of the endocrine system of the pancreatic hormones for increasing or potentiating the activity of insulin
Landscapes
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Diabetes (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Obesity (AREA)
- Hematology (AREA)
- Endocrinology (AREA)
- Epidemiology (AREA)
- Emergency Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
Etkili, toksik olmayan ve eczacilik teknolojisi bakimindan kabul edilebilir tutarda bir ensülin yönünden duyarli duruma getiricinin, maksimum altinda miktarda bir insülin salgilattiricisinin, bunlara gereksinmesi bulunan bir memeliye verilmesini içeren diabetas mellitus' un memelide diabetes mellitus ile iliskili durumlarin tedavi edilmeleri için yöntem ile bu gibi yöntemin kullanilmasina yarar bilesim.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB9715306A GB9715306D0 (en) | 1997-07-18 | 1997-07-18 | Novel method of treatment |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| TR200000135T2 true TR200000135T2 (tr) | 2000-05-22 |
Family
ID=10816177
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| TR2000/00135T TR200000135T2 (tr) | 1997-07-18 | 1998-07-16 | Tiazolidinedion ve sülfonilüre ile diabet tedavisi. |
Country Status (40)
| Country | Link |
|---|---|
| EP (1) | EP0998291B2 (tr) |
| JP (2) | JP2001510158A (tr) |
| KR (1) | KR100680667B1 (tr) |
| CN (1) | CN1264302A (tr) |
| AP (1) | AP1318A (tr) |
| AR (2) | AR016768A1 (tr) |
| AT (1) | ATE366577T1 (tr) |
| AU (1) | AU743269B2 (tr) |
| BG (1) | BG64892B1 (tr) |
| BR (1) | BR9810904A (tr) |
| CA (1) | CA2297115C (tr) |
| CO (1) | CO4940422A1 (tr) |
| CY (1) | CY1107745T1 (tr) |
| CZ (1) | CZ302668B6 (tr) |
| DE (1) | DE69838066T3 (tr) |
| DK (1) | DK0998291T4 (tr) |
| DZ (1) | DZ2564A1 (tr) |
| EA (1) | EA003303B1 (tr) |
| ES (1) | ES2290989T5 (tr) |
| GB (1) | GB9715306D0 (tr) |
| HU (1) | HU229119B1 (tr) |
| ID (1) | ID24198A (tr) |
| IL (1) | IL134045A0 (tr) |
| IN (1) | IN189035B (tr) |
| MA (1) | MA26522A1 (tr) |
| MY (1) | MY138246A (tr) |
| NO (1) | NO326356B1 (tr) |
| NZ (3) | NZ520652A (tr) |
| OA (1) | OA11632A (tr) |
| PE (1) | PE99799A1 (tr) |
| PL (2) | PL338127A1 (tr) |
| PT (1) | PT998291E (tr) |
| SI (1) | SI0998291T2 (tr) |
| SK (2) | SK288053B6 (tr) |
| TR (1) | TR200000135T2 (tr) |
| TW (1) | TW586926B (tr) |
| UA (1) | UA70302C2 (tr) |
| UY (1) | UY25103A1 (tr) |
| WO (1) | WO1999003476A1 (tr) |
| ZA (1) | ZA986365B (tr) |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7045519B2 (en) | 1998-06-19 | 2006-05-16 | Chiron Corporation | Inhibitors of glycogen synthase kinase 3 |
| EP1897547A1 (en) * | 1999-07-13 | 2008-03-12 | Medicure Inc. | Use of pyridoxal phosphate derivatives for the treatment of diabetes and related complications |
| EP1832291A3 (en) * | 1999-07-13 | 2009-11-04 | Medicure Inc. | use of pyridoxal phosphate for the treatment of diabetes and related complications |
| US6586438B2 (en) | 1999-11-03 | 2003-07-01 | Bristol-Myers Squibb Co. | Antidiabetic formulation and method |
| US20010036479A1 (en) | 2000-01-14 | 2001-11-01 | Gillian Cave | Glyburide composition |
| CA2725833A1 (en) | 2001-01-12 | 2002-07-18 | Sun Pharmaceutical Industries Limited | Spaced drug delivery system |
| GEP20084570B (en) | 2003-10-31 | 2008-12-25 | Takeda Pharmaceutical | Solid preparation comprising an insulin sensitizer, an insulin secretagogue and a polyoxyethylene sorbitan fatty acid ester |
| JP2008019169A (ja) * | 2004-10-25 | 2008-01-31 | Osaka Univ | 新規ppar調節剤およびそのスクリーニング方法 |
| AU2006328328B2 (en) | 2005-12-22 | 2012-08-30 | Takeda Pharmaceutical Company Limited | Solid preparation containing an insulin sensitizer |
Family Cites Families (19)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS5522636A (en) * | 1978-08-04 | 1980-02-18 | Takeda Chem Ind Ltd | Thiazoliding derivative |
| JPS5697277A (en) * | 1980-01-07 | 1981-08-05 | Takeda Chem Ind Ltd | Thiazolidine derivative |
| JPS6051189A (ja) * | 1983-08-30 | 1985-03-22 | Sankyo Co Ltd | チアゾリジン誘導体およびその製造法 |
| US4582839A (en) * | 1984-03-21 | 1986-04-15 | Takeda Chemical Industries, Ltd. | 2,4-thiazolidinediones |
| CN1003445B (zh) * | 1984-10-03 | 1989-03-01 | 武田药品工业株式会社 | 噻唑烷二酮衍生物,其制备方法和用途 |
| JPH06779B2 (ja) * | 1985-06-10 | 1994-01-05 | 武田薬品工業株式会社 | チアゾリジオン誘導体およびそれを含んでなる医薬組成物 |
| US4812570A (en) * | 1986-07-24 | 1989-03-14 | Takeda Chemical Industries, Ltd. | Method for producing thiazolidinedione derivatives |
| ATE186724T1 (de) * | 1987-09-04 | 1999-12-15 | Beecham Group Plc | Substituierte thiazolidindionderivate |
| US4791125A (en) * | 1987-12-02 | 1988-12-13 | Pfizer Inc. | Thiazolidinediones as hypoglycemic and anti-atherosclerosis agents |
| MX15171A (es) * | 1988-03-08 | 1993-05-01 | Pfizer | Derivados de tiazolidinodiona hipoglicemicos |
| WO1989008650A1 (en) * | 1988-03-08 | 1989-09-21 | Pfizer Inc. | Thiazolidinedione hypoglycemic agents |
| WO1991007107A1 (en) * | 1989-11-13 | 1991-05-30 | Pfizer Inc. | Oxazolidinedione hypoglycemic agents |
| JPH04210683A (ja) * | 1990-12-06 | 1992-07-31 | Terumo Corp | チアゾリジン−2,4−ジオン誘導体およびこれを含有する糖尿病合併症治療薬 |
| US5183823A (en) * | 1991-04-11 | 1993-02-02 | Takeda Chemical Industries, Ltd. | Pyridine n-oxide compounds which are useful as hypoglycemic and hypolipidemic agents |
| ES2089474T3 (es) * | 1991-08-16 | 1996-10-01 | Sandoz Ltd | Inhalador para la administracion de sustancias en polvo. |
| DE69219136T2 (de) * | 1991-08-26 | 1997-08-28 | Pharmacia & Upjohn Co., Kalamazoo, Mich. | Flüssiges nahrungsmittel, das 3-guanidinopropionsäure enthält |
| GB9218830D0 (en) * | 1992-09-05 | 1992-10-21 | Smithkline Beecham Plc | Novel compounds |
| TW438587B (en) * | 1995-06-20 | 2001-06-07 | Takeda Chemical Industries Ltd | A pharmaceutical composition for prophylaxis and treatment of diabetes |
| US5859037A (en) * | 1997-02-19 | 1999-01-12 | Warner-Lambert Company | Sulfonylurea-glitazone combinations for diabetes |
-
1997
- 1997-07-18 GB GB9715306A patent/GB9715306D0/en active Pending
-
1998
- 1998-07-15 DZ DZ980174A patent/DZ2564A1/xx active
- 1998-07-16 AU AU84487/98A patent/AU743269B2/en not_active Expired
- 1998-07-16 AP APAP/P/2000/001734A patent/AP1318A/en active
- 1998-07-16 SK SK89-2005A patent/SK288053B6/sk not_active IP Right Cessation
- 1998-07-16 PL PL98338127A patent/PL338127A1/xx not_active Application Discontinuation
- 1998-07-16 MA MA25173A patent/MA26522A1/fr unknown
- 1998-07-16 NZ NZ520652A patent/NZ520652A/en not_active IP Right Cessation
- 1998-07-16 ES ES98935126T patent/ES2290989T5/es not_active Expired - Lifetime
- 1998-07-16 DE DE69838066T patent/DE69838066T3/de not_active Expired - Lifetime
- 1998-07-16 CN CN98807221A patent/CN1264302A/zh active Pending
- 1998-07-16 UA UA2000010215A patent/UA70302C2/uk unknown
- 1998-07-16 SK SK60-2000A patent/SK287823B6/sk not_active IP Right Cessation
- 1998-07-16 NZ NZ515555A patent/NZ515555A/xx not_active IP Right Cessation
- 1998-07-16 AT AT98935126T patent/ATE366577T1/de active
- 1998-07-16 JP JP2000502775A patent/JP2001510158A/ja not_active Withdrawn
- 1998-07-16 SI SI9830892T patent/SI0998291T2/sl unknown
- 1998-07-16 HU HU0003634A patent/HU229119B1/hu unknown
- 1998-07-16 PL PL375989A patent/PL199125B1/pl unknown
- 1998-07-16 EP EP98935126A patent/EP0998291B2/en not_active Expired - Lifetime
- 1998-07-16 PT PT98935126T patent/PT998291E/pt unknown
- 1998-07-16 WO PCT/GB1998/002109 patent/WO1999003476A1/en not_active Ceased
- 1998-07-16 IL IL13404598A patent/IL134045A0/xx unknown
- 1998-07-16 ID IDW20000074A patent/ID24198A/id unknown
- 1998-07-16 CA CA2297115A patent/CA2297115C/en not_active Expired - Lifetime
- 1998-07-16 EA EA200000141A patent/EA003303B1/ru not_active IP Right Cessation
- 1998-07-16 BR BR9810904-9A patent/BR9810904A/pt not_active Application Discontinuation
- 1998-07-16 TR TR2000/00135T patent/TR200000135T2/tr unknown
- 1998-07-16 NZ NZ501256A patent/NZ501256A/xx not_active IP Right Cessation
- 1998-07-16 DK DK98935126.7T patent/DK0998291T4/da active
- 1998-07-16 OA OA1200000014A patent/OA11632A/en unknown
- 1998-07-16 CZ CZ20000173A patent/CZ302668B6/cs not_active IP Right Cessation
- 1998-07-16 PE PE1998000631A patent/PE99799A1/es not_active Application Discontinuation
- 1998-07-16 KR KR1020007000513A patent/KR100680667B1/ko not_active Expired - Lifetime
- 1998-07-17 CO CO98040748A patent/CO4940422A1/es unknown
- 1998-07-17 UY UY25103A patent/UY25103A1/es not_active IP Right Cessation
- 1998-07-17 MY MYPI98003290A patent/MY138246A/en unknown
- 1998-07-17 TW TW087111768A patent/TW586926B/zh not_active IP Right Cessation
- 1998-07-17 ZA ZA9806365A patent/ZA986365B/xx unknown
- 1998-07-17 AR ARP980103516A patent/AR016768A1/es not_active Application Discontinuation
- 1998-07-20 IN IN2089DE1998 patent/IN189035B/en unknown
-
1999
- 1999-06-18 AR ARP990102953A patent/AR019331A2/es unknown
-
2000
- 2000-01-17 NO NO20000229A patent/NO326356B1/no not_active IP Right Cessation
- 2000-02-08 BG BG104139A patent/BG64892B1/bg unknown
-
2005
- 2005-04-21 JP JP2005123586A patent/JP2005247865A/ja active Pending
-
2007
- 2007-09-27 CY CY20071101241T patent/CY1107745T1/el unknown
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