TR200202109T2 - 5-[{6-(2-Flüorobenzil)oksi-2-naftil}metil]-2,4-tiyazolidin dion kristalleri - Google Patents
5-[{6-(2-Flüorobenzil)oksi-2-naftil}metil]-2,4-tiyazolidin dion kristalleriInfo
- Publication number
- TR200202109T2 TR200202109T2 TR2002/02109T TR200202109T TR200202109T2 TR 200202109 T2 TR200202109 T2 TR 200202109T2 TR 2002/02109 T TR2002/02109 T TR 2002/02109T TR 200202109 T TR200202109 T TR 200202109T TR 200202109 T2 TR200202109 T2 TR 200202109T2
- Authority
- TR
- Turkey
- Prior art keywords
- fluorobenzyl
- oxy
- naphthyl
- methyl
- crystals
- Prior art date
Links
- 239000013078 crystal Substances 0.000 title abstract 2
- PKWDZWYVIHVNKS-UHFFFAOYSA-N netoglitazone Chemical compound FC1=CC=CC=C1COC1=CC=C(C=C(CC2C(NC(=O)S2)=O)C=C2)C2=C1 PKWDZWYVIHVNKS-UHFFFAOYSA-N 0.000 title abstract 2
- 208000031226 Hyperlipidaemia Diseases 0.000 abstract 1
- 201000001431 Hyperuricemia Diseases 0.000 abstract 1
- 206010033645 Pancreatitis Diseases 0.000 abstract 1
- 239000004480 active ingredient Substances 0.000 abstract 1
- 206010012601 diabetes mellitus Diseases 0.000 abstract 1
- 201000010099 disease Diseases 0.000 abstract 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
- 208000032839 leukemia Diseases 0.000 abstract 1
- 230000001225 therapeutic effect Effects 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/34—Oxygen atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/18—Drugs for disorders of the alimentary tract or the digestive system for pancreatic disorders, e.g. pancreatic enzymes
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/06—Antigout agents, e.g. antihyperuricemic or uricosuric agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Rheumatology (AREA)
- Oncology (AREA)
- Physical Education & Sports Medicine (AREA)
- Pain & Pain Management (AREA)
- Emergency Medicine (AREA)
- Endocrinology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Cosmetics (AREA)
- Photoreceptors In Electrophotography (AREA)
Abstract
Mevcut bulus, 5-[{6-(2-Flüorobenzil)oksi-2-naftil}metil]-2,4-tiyazolidin dion' un kararli ve yeni C tipi kristallerine iliskin olup, bunlar asagidaki hastaliklarin tedavisine yönelik terapötik aktif bilesen olarak kullanilmaya uygundur: diyabet ve komplikasyonlari, hiperlipidemi ve komplikasyonlari, hiperürisemi, lösemi ve pankreatit.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP33054698 | 1998-11-20 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| TR200202109T2 true TR200202109T2 (tr) | 2002-11-21 |
Family
ID=18233859
Family Applications (4)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| TR2002/02110T TR200202110T2 (tr) | 1998-11-20 | 1999-11-19 | "5-[{6-(2-Flüore benzil) oksi-2-naftil}metil]-2,4-tiyazolidin dion kristalleri" |
| TR2001/01901T TR200101901T2 (tr) | 1998-11-20 | 1999-11-19 | 5-[{6-(2-Flüorobenzil)oksi-2-naftil}metil]-2,4-Tiyazolidin dion kristalleri |
| TR2002/02103T TR200202103T2 (tr) | 1998-11-20 | 1999-11-19 | ''5-[{6-(2-Flüorobenzil)oksi-2-naftil}metil]-2,4-tiyazolidin dion kristalleri'' |
| TR2002/02109T TR200202109T2 (tr) | 1998-11-20 | 1999-11-19 | 5-[{6-(2-Flüorobenzil)oksi-2-naftil}metil]-2,4-tiyazolidin dion kristalleri |
Family Applications Before (3)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| TR2002/02110T TR200202110T2 (tr) | 1998-11-20 | 1999-11-19 | "5-[{6-(2-Flüore benzil) oksi-2-naftil}metil]-2,4-tiyazolidin dion kristalleri" |
| TR2001/01901T TR200101901T2 (tr) | 1998-11-20 | 1999-11-19 | 5-[{6-(2-Flüorobenzil)oksi-2-naftil}metil]-2,4-Tiyazolidin dion kristalleri |
| TR2002/02103T TR200202103T2 (tr) | 1998-11-20 | 1999-11-19 | ''5-[{6-(2-Flüorobenzil)oksi-2-naftil}metil]-2,4-tiyazolidin dion kristalleri'' |
Country Status (23)
| Country | Link |
|---|---|
| US (3) | US6541493B1 (tr) |
| EP (1) | EP1131310B1 (tr) |
| JP (1) | JP3784001B2 (tr) |
| KR (1) | KR100652326B1 (tr) |
| CN (1) | CN1326449A (tr) |
| AT (1) | ATE315552T1 (tr) |
| AU (1) | AU1185100A (tr) |
| BR (1) | BR9916795A (tr) |
| CA (1) | CA2351727C (tr) |
| CZ (1) | CZ20011763A3 (tr) |
| DE (1) | DE69929476T2 (tr) |
| ES (1) | ES2257104T3 (tr) |
| HU (1) | HUP0104139A3 (tr) |
| ID (1) | ID30064A (tr) |
| IL (1) | IL143177A0 (tr) |
| NO (1) | NO20012444L (tr) |
| NZ (1) | NZ512429A (tr) |
| PL (1) | PL348502A1 (tr) |
| PT (1) | PT1131310E (tr) |
| TR (4) | TR200202110T2 (tr) |
| TW (2) | TWI272944B (tr) |
| WO (1) | WO2000031055A1 (tr) |
| ZA (1) | ZA200104081B (tr) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TR200202110T2 (tr) * | 1998-11-20 | 2002-10-21 | Mitsubishi Chemical Corporation | "5-[{6-(2-Flüore benzil) oksi-2-naftil}metil]-2,4-tiyazolidin dion kristalleri" |
| BR0015702A (pt) * | 1999-11-19 | 2002-07-16 | Johnson & Johnson | Formas de estado sólido de 5-[[6-[(2-fluorofenil)metoxi]-2naftalenil] metil] 2,4-tiazolidinediona |
| JP4590159B2 (ja) * | 2001-04-04 | 2010-12-01 | オーソ−マクニール・フアーマシユーチカル・インコーポレーテツド | グルコース再吸収阻害剤およびpparモジュレーターを含んで成る併用療法 |
| WO2007049050A2 (en) * | 2005-10-27 | 2007-05-03 | Heptahelix Ab | Modulators of gpr40 for the treatment of diabetes |
| AU2009211072B2 (en) | 2008-02-04 | 2014-01-23 | Pfizer Limited | Polymorphic form of a [1, 2, 4] triazolo [4, 3-A] pyridine derivative for treating inflammatory diseases |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5594016A (en) * | 1992-12-28 | 1997-01-14 | Mitsubishi Chemical Corporation | Naphthalene derivatives |
| JP2845743B2 (ja) * | 1992-12-28 | 1999-01-13 | 三菱化学株式会社 | 新規なナフタレン誘導体 |
| JP4023697B2 (ja) | 1996-11-14 | 2007-12-19 | 三菱化学株式会社 | ナフタレン誘導体の製造方法 |
| TR200202110T2 (tr) * | 1998-11-20 | 2002-10-21 | Mitsubishi Chemical Corporation | "5-[{6-(2-Flüore benzil) oksi-2-naftil}metil]-2,4-tiyazolidin dion kristalleri" |
-
1999
- 1999-11-19 TR TR2002/02110T patent/TR200202110T2/tr unknown
- 1999-11-19 AU AU11851/00A patent/AU1185100A/en not_active Abandoned
- 1999-11-19 JP JP2000583883A patent/JP3784001B2/ja not_active Expired - Fee Related
- 1999-11-19 BR BR9916795-6A patent/BR9916795A/pt not_active IP Right Cessation
- 1999-11-19 US US09/856,295 patent/US6541493B1/en not_active Expired - Fee Related
- 1999-11-19 KR KR1020017006299A patent/KR100652326B1/ko not_active Expired - Fee Related
- 1999-11-19 ES ES99972628T patent/ES2257104T3/es not_active Expired - Lifetime
- 1999-11-19 CZ CZ20011763A patent/CZ20011763A3/cs unknown
- 1999-11-19 ID IDW00200101331A patent/ID30064A/id unknown
- 1999-11-19 CN CN99813380A patent/CN1326449A/zh active Pending
- 1999-11-19 TR TR2001/01901T patent/TR200101901T2/tr unknown
- 1999-11-19 TR TR2002/02103T patent/TR200202103T2/tr unknown
- 1999-11-19 NZ NZ512429A patent/NZ512429A/en unknown
- 1999-11-19 EP EP99972628A patent/EP1131310B1/en not_active Expired - Lifetime
- 1999-11-19 WO PCT/JP1999/006492 patent/WO2000031055A1/en not_active Ceased
- 1999-11-19 HU HU0104139A patent/HUP0104139A3/hu unknown
- 1999-11-19 TR TR2002/02109T patent/TR200202109T2/tr unknown
- 1999-11-19 IL IL14317799A patent/IL143177A0/xx unknown
- 1999-11-19 CA CA002351727A patent/CA2351727C/en not_active Expired - Fee Related
- 1999-11-19 AT AT99972628T patent/ATE315552T1/de not_active IP Right Cessation
- 1999-11-19 PL PL99348502A patent/PL348502A1/xx unknown
- 1999-11-19 DE DE69929476T patent/DE69929476T2/de not_active Expired - Fee Related
- 1999-11-19 PT PT99972628T patent/PT1131310E/pt unknown
- 1999-11-20 TW TW094136910A patent/TWI272944B/zh not_active IP Right Cessation
- 1999-11-20 TW TW088120305A patent/TWI250156B/zh not_active IP Right Cessation
-
2001
- 2001-05-18 NO NO20012444A patent/NO20012444L/no not_active Application Discontinuation
- 2001-05-18 ZA ZA200104081A patent/ZA200104081B/en unknown
-
2003
- 2003-01-31 US US10/355,160 patent/US20030158241A1/en not_active Abandoned
-
2006
- 2006-02-21 US US11/357,208 patent/US20060149075A1/en not_active Abandoned
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