TW200716560A - Novel cannabinoid receptor ligands, pharmaceutical compositions containing them, and process for their preparation - Google Patents

Novel cannabinoid receptor ligands, pharmaceutical compositions containing them, and process for their preparation

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Publication number
TW200716560A
TW200716560A TW095119616A TW95119616A TW200716560A TW 200716560 A TW200716560 A TW 200716560A TW 095119616 A TW095119616 A TW 095119616A TW 95119616 A TW95119616 A TW 95119616A TW 200716560 A TW200716560 A TW 200716560A
Authority
TW
Taiwan
Prior art keywords
preparation
cannabinoid receptor
pharmaceutical compositions
compositions containing
receptor ligands
Prior art date
Application number
TW095119616A
Other languages
English (en)
Inventor
Meyyappan Muthuppalaniappan
Gopalan Balasubramanian
Srinivas Gullapalli
Neelima Khairatkar Joshi
Shridhar Narayanan
Original Assignee
Glenmark Pharmaceuticals Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glenmark Pharmaceuticals Sa filed Critical Glenmark Pharmaceuticals Sa
Publication of TW200716560A publication Critical patent/TW200716560A/zh

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/54Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
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  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
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  • Bioinformatics & Cheminformatics (AREA)
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  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Diabetes (AREA)
  • Immunology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Addiction (AREA)
  • Psychiatry (AREA)
  • Rheumatology (AREA)
  • Hematology (AREA)
  • Pain & Pain Management (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Endocrinology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Obesity (AREA)
  • Dermatology (AREA)
  • Reproductive Health (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Urology & Nephrology (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Virology (AREA)
  • Cardiology (AREA)
  • Pulmonology (AREA)
  • Hospice & Palliative Care (AREA)
TW095119616A 2005-06-02 2006-06-02 Novel cannabinoid receptor ligands, pharmaceutical compositions containing them, and process for their preparation TW200716560A (en)

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
IN659MU2005 2005-06-02
US69643305P 2005-07-01 2005-07-01
IN1370MU2005 2005-10-31
IN344MU2006 2006-03-09
US74407106P 2006-03-31 2006-03-31
IN689MU2006 2006-05-03

Publications (1)

Publication Number Publication Date
TW200716560A true TW200716560A (en) 2007-05-01

Family

ID=37056437

Family Applications (1)

Application Number Title Priority Date Filing Date
TW095119616A TW200716560A (en) 2005-06-02 2006-06-02 Novel cannabinoid receptor ligands, pharmaceutical compositions containing them, and process for their preparation

Country Status (11)

Country Link
US (1) US8420689B2 (zh)
EP (1) EP1902034B1 (zh)
JP (1) JP2008545739A (zh)
AR (1) AR055199A1 (zh)
AU (1) AU2006253842A1 (zh)
CA (1) CA2613678A1 (zh)
MY (1) MY142409A (zh)
PE (1) PE20070431A1 (zh)
PL (1) PL1902034T3 (zh)
TW (1) TW200716560A (zh)
WO (1) WO2006129178A1 (zh)

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US7923465B2 (en) 2005-06-02 2011-04-12 Glenmark Pharmaceuticals S.A. Cannabinoid receptor ligands, pharmaceutical compositions containing them, and process for their preparation
WO2008053341A2 (en) * 2006-11-03 2008-05-08 Glenmark Pharmaceuticals S.A. Bridged bicyclic indazoles as cannabinoid receptor ligands
WO2008093194A1 (en) * 2007-01-29 2008-08-07 Glenmark Pharmaceuticals, S.A. Cannabinoid receptor modulators for treating non-immediate type allergic diseases
KR101787116B1 (ko) 2009-01-28 2017-10-18 케러 테라퓨틱스, 인코포레이티드 바이시클릭 피라졸로-헤테로사이클
US7741350B1 (en) 2009-01-28 2010-06-22 Cara Therapeutics, Inc. Bicyclic pyrazolo-heterocycles
CA2770866C (en) * 2009-08-28 2017-10-10 Arena Pharmaceuticals, Inc. Cannabinoid receptor modulators
WO2012090179A2 (en) 2010-12-30 2012-07-05 Lupin Limited Isoquinoline derivatives as cannabinoid receptor modulators
WO2012090177A2 (en) 2010-12-30 2012-07-05 Lupin Limited Cannabinoid receptor modulators
CN103492369B (zh) * 2011-02-25 2019-03-29 艾尼纳制药公司 大麻素受体调节剂
US9597340B2 (en) 2011-02-25 2017-03-21 Arena Pharmaceuticals, Inc. Cannabinoid receptor modulators
US9458136B2 (en) 2011-02-25 2016-10-04 Arena Pharmaceuticals, Inc. Crystalline forms and processes for the preparation of cannabinoid receptor modulators
WO2013005168A2 (en) 2011-07-05 2013-01-10 Lupin Limited Cannabinoid receptor modulators
CN106063787A (zh) 2012-02-03 2016-11-02 泰华制药工业有限公司 拉喹莫德用于治疗一线抗TNFα疗法失败的克罗恩氏病患者的用途
TW201410243A (zh) * 2012-08-13 2014-03-16 Teva Pharma 用於治療大麻素受體型1(cb1)媒介之疾病之拉喹莫德(laquinimod)
JP2015535287A (ja) 2012-11-07 2015-12-10 テバ ファーマシューティカル インダストリーズ リミティド ラキニモドのアミン塩
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