TW200716560A - Novel cannabinoid receptor ligands, pharmaceutical compositions containing them, and process for their preparation - Google Patents
Novel cannabinoid receptor ligands, pharmaceutical compositions containing them, and process for their preparationInfo
- Publication number
- TW200716560A TW200716560A TW095119616A TW95119616A TW200716560A TW 200716560 A TW200716560 A TW 200716560A TW 095119616 A TW095119616 A TW 095119616A TW 95119616 A TW95119616 A TW 95119616A TW 200716560 A TW200716560 A TW 200716560A
- Authority
- TW
- Taiwan
- Prior art keywords
- preparation
- cannabinoid receptor
- pharmaceutical compositions
- compositions containing
- receptor ligands
- Prior art date
Links
- 102000018208 Cannabinoid Receptor Human genes 0.000 title abstract 2
- 108050007331 Cannabinoid receptor Proteins 0.000 title abstract 2
- 239000003446 ligand Substances 0.000 title 1
- 239000008194 pharmaceutical composition Substances 0.000 title 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 3
- 229930003827 cannabinoid Natural products 0.000 abstract 2
- 239000003557 cannabinoid Substances 0.000 abstract 2
- 208000035475 disorder Diseases 0.000 abstract 2
- 208000030814 Eating disease Diseases 0.000 abstract 1
- 208000019454 Feeding and Eating disease Diseases 0.000 abstract 1
- 208000008589 Obesity Diseases 0.000 abstract 1
- 239000003520 cannabinoid receptor affecting agent Substances 0.000 abstract 1
- 201000010099 disease Diseases 0.000 abstract 1
- 235000014632 disordered eating Nutrition 0.000 abstract 1
- 235000020824 obesity Nutrition 0.000 abstract 1
- 102000005962 receptors Human genes 0.000 abstract 1
- 108020003175 receptors Proteins 0.000 abstract 1
- 230000004580 weight loss Effects 0.000 abstract 1
- 208000016261 weight loss Diseases 0.000 abstract 1
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/54—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
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Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Diabetes (AREA)
- Immunology (AREA)
- Physical Education & Sports Medicine (AREA)
- Addiction (AREA)
- Psychiatry (AREA)
- Rheumatology (AREA)
- Hematology (AREA)
- Pain & Pain Management (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Endocrinology (AREA)
- Ophthalmology & Optometry (AREA)
- Obesity (AREA)
- Dermatology (AREA)
- Reproductive Health (AREA)
- Heart & Thoracic Surgery (AREA)
- Urology & Nephrology (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Virology (AREA)
- Cardiology (AREA)
- Pulmonology (AREA)
- Hospice & Palliative Care (AREA)
Applications Claiming Priority (6)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IN659MU2005 | 2005-06-02 | ||
| US69643305P | 2005-07-01 | 2005-07-01 | |
| IN1370MU2005 | 2005-10-31 | ||
| IN344MU2006 | 2006-03-09 | ||
| US74407106P | 2006-03-31 | 2006-03-31 | |
| IN689MU2006 | 2006-05-03 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| TW200716560A true TW200716560A (en) | 2007-05-01 |
Family
ID=37056437
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| TW095119616A TW200716560A (en) | 2005-06-02 | 2006-06-02 | Novel cannabinoid receptor ligands, pharmaceutical compositions containing them, and process for their preparation |
Country Status (11)
| Country | Link |
|---|---|
| US (1) | US8420689B2 (zh) |
| EP (1) | EP1902034B1 (zh) |
| JP (1) | JP2008545739A (zh) |
| AR (1) | AR055199A1 (zh) |
| AU (1) | AU2006253842A1 (zh) |
| CA (1) | CA2613678A1 (zh) |
| MY (1) | MY142409A (zh) |
| PE (1) | PE20070431A1 (zh) |
| PL (1) | PL1902034T3 (zh) |
| TW (1) | TW200716560A (zh) |
| WO (1) | WO2006129178A1 (zh) |
Families Citing this family (26)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7923465B2 (en) | 2005-06-02 | 2011-04-12 | Glenmark Pharmaceuticals S.A. | Cannabinoid receptor ligands, pharmaceutical compositions containing them, and process for their preparation |
| WO2008053341A2 (en) * | 2006-11-03 | 2008-05-08 | Glenmark Pharmaceuticals S.A. | Bridged bicyclic indazoles as cannabinoid receptor ligands |
| WO2008093194A1 (en) * | 2007-01-29 | 2008-08-07 | Glenmark Pharmaceuticals, S.A. | Cannabinoid receptor modulators for treating non-immediate type allergic diseases |
| KR101787116B1 (ko) | 2009-01-28 | 2017-10-18 | 케러 테라퓨틱스, 인코포레이티드 | 바이시클릭 피라졸로-헤테로사이클 |
| US7741350B1 (en) | 2009-01-28 | 2010-06-22 | Cara Therapeutics, Inc. | Bicyclic pyrazolo-heterocycles |
| CA2770866C (en) * | 2009-08-28 | 2017-10-10 | Arena Pharmaceuticals, Inc. | Cannabinoid receptor modulators |
| WO2012090179A2 (en) | 2010-12-30 | 2012-07-05 | Lupin Limited | Isoquinoline derivatives as cannabinoid receptor modulators |
| WO2012090177A2 (en) | 2010-12-30 | 2012-07-05 | Lupin Limited | Cannabinoid receptor modulators |
| CN103492369B (zh) * | 2011-02-25 | 2019-03-29 | 艾尼纳制药公司 | 大麻素受体调节剂 |
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2006
- 2006-06-01 CA CA002613678A patent/CA2613678A1/en not_active Abandoned
- 2006-06-01 WO PCT/IB2006/001437 patent/WO2006129178A1/en not_active Ceased
- 2006-06-01 PL PL06755930T patent/PL1902034T3/pl unknown
- 2006-06-01 EP EP06755930A patent/EP1902034B1/en active Active
- 2006-06-01 AU AU2006253842A patent/AU2006253842A1/en not_active Abandoned
- 2006-06-01 JP JP2008514222A patent/JP2008545739A/ja active Pending
- 2006-06-02 TW TW095119616A patent/TW200716560A/zh unknown
- 2006-06-02 PE PE2006000600A patent/PE20070431A1/es not_active Application Discontinuation
- 2006-06-02 MY MYPI20062558A patent/MY142409A/en unknown
- 2006-06-02 AR ARP060102327A patent/AR055199A1/es unknown
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2011
- 2011-01-14 US US13/006,560 patent/US8420689B2/en not_active Expired - Fee Related
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| AU2006253842A1 (en) | 2006-12-07 |
| EP1902034A1 (en) | 2008-03-26 |
| AR055199A1 (es) | 2007-08-08 |
| US20120142748A1 (en) | 2012-06-07 |
| PL1902034T3 (pl) | 2011-09-30 |
| WO2006129178A1 (en) | 2006-12-07 |
| EP1902034B1 (en) | 2011-03-30 |
| MY142409A (en) | 2010-11-30 |
| HK1118806A1 (zh) | 2009-02-20 |
| JP2008545739A (ja) | 2008-12-18 |
| PE20070431A1 (es) | 2007-06-27 |
| WO2006129178A8 (en) | 2007-01-11 |
| US8420689B2 (en) | 2013-04-16 |
| CA2613678A1 (en) | 2006-12-07 |
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