UA108250C2 - Парентеральна фармацевтична композиція, її застосування та способи лікування або попередження віл-інфекції у людини - Google Patents

Парентеральна фармацевтична композиція, її застосування та способи лікування або попередження віл-інфекції у людини

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Publication number
UA108250C2
UA108250C2 UAA201303057A UAA201303057A UA108250C2 UA 108250 C2 UA108250 C2 UA 108250C2 UA A201303057 A UAA201303057 A UA A201303057A UA A201303057 A UAA201303057 A UA A201303057A UA 108250 C2 UA108250 C2 UA 108250C2
Authority
UA
Ukraine
Prior art keywords
prevention
hiv
treatment
methods
human
Prior art date
Application number
UAA201303057A
Other languages
English (en)
Ukrainian (uk)
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of UA108250C2 publication Critical patent/UA108250C2/ru

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Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/4985Pyrazines or piperazines ortho- or peri-condensed with heterocyclic ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/18Antivirals for RNA viruses for HIV

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Virology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • AIDS & HIV (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
UAA201303057A 2010-09-16 2011-09-15 Парентеральна фармацевтична композиція, її застосування та способи лікування або попередження віл-інфекції у людини UA108250C2 (uk)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US38354110P 2010-09-16 2010-09-16
PCT/US2011/051713 WO2012037320A2 (en) 2010-09-16 2011-09-15 Pharmaceutical compositions

Publications (1)

Publication Number Publication Date
UA108250C2 true UA108250C2 (uk) 2015-04-10

Family

ID=45832235

Family Applications (1)

Application Number Title Priority Date Filing Date
UAA201303057A UA108250C2 (uk) 2010-09-16 2011-09-15 Парентеральна фармацевтична композиція, її застосування та способи лікування або попередження віл-інфекції у людини

Country Status (28)

Country Link
US (7) US20130171214A1 (ru)
EP (1) EP2616076B1 (ru)
JP (1) JP6231385B2 (ru)
KR (1) KR101938662B1 (ru)
CN (1) CN103547266B (ru)
AU (1) AU2011302030B2 (ru)
BR (1) BR112013005907B1 (ru)
CA (1) CA2810524C (ru)
CL (1) CL2013000715A1 (ru)
CY (1) CY1118279T1 (ru)
DK (1) DK2616076T3 (ru)
EA (1) EA024924B1 (ru)
ES (1) ES2594557T3 (ru)
HR (1) HRP20161280T1 (ru)
HU (1) HUE031336T2 (ru)
IL (1) IL225028A (ru)
LT (1) LT2616076T (ru)
ME (1) ME02520B (ru)
MX (1) MX346193B (ru)
PL (1) PL2616076T3 (ru)
PT (1) PT2616076T (ru)
RS (1) RS55222B1 (ru)
SI (1) SI2616076T1 (ru)
SM (1) SMT201600350B (ru)
TW (1) TWI577377B (ru)
UA (1) UA108250C2 (ru)
WO (1) WO2012037320A2 (ru)
ZA (1) ZA201301766B (ru)

Families Citing this family (29)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JO3387B1 (ar) 2011-12-16 2019-03-13 Glaxosmithkline Llc مشتقات بيتولين
KR20150093819A (ko) 2012-12-14 2015-08-18 글락소스미스클라인 엘엘씨 약제 조성물
US9808428B2 (en) 2014-01-14 2017-11-07 Board Of Regents Of The University Of Nebraska Compositions and methods for the delivery of therapeutics
US20170165271A1 (en) * 2014-02-24 2017-06-15 The Board Of Regents Of The University Of Nebraska Compositions and Methods for the Delivery of Therapeutics
US10092523B2 (en) 2014-09-26 2018-10-09 Glaxosmithkline Intellectual Property (No. 2) Limited Long acting pharmaceutical compositions
WO2016057866A1 (en) 2014-10-09 2016-04-14 Board Of Regents Of The University Of Nebraska Compositions and methods for the delivery of therapeutics
TN2017000232A1 (en) * 2014-12-20 2018-10-19 Troikaa Pharmaceuticals Ltd Injectable formulations of paracetamol
EP4299133A3 (en) * 2016-06-23 2024-03-13 VIIV Healthcare Company Compositions and methods for the delivery of therapeutics
US11077050B2 (en) 2017-03-24 2021-08-03 Merck Sharp & Dohme Corp. Formulation for parenteral administration
SI3943070T1 (sl) 2017-07-14 2024-03-29 Janssen Pharmaceutica Nv, Dolgo delujoče formulacije bedakilina
WO2019016679A1 (en) * 2017-07-18 2019-01-24 Viiv Healthcare Company Combination drug therapy
EP3737359A4 (en) 2018-01-12 2021-11-03 Board of Regents of the University of Nebraska ANTIVIRAL MEDICINES AND FORMULATIONS OF THEM
CA3132832A1 (en) 2018-04-09 2019-10-17 Howard E. Gendelman Antiviral prodrugs and formulations thereof
ES2970251T3 (es) * 2018-10-22 2024-05-27 Univ Nebraska Profármacos antivirales y nanoformulaciones de los mismos
WO2020112931A1 (en) 2018-11-29 2020-06-04 Board Of Regents Of The University Of Nebraska Antiviral prodrugs and nanoformulations thereof
CN109646440B (zh) * 2019-01-11 2021-04-20 山东省农业科学院奶牛研究中心 Cabotegravir在制备抗牛传染性鼻气管炎药物中的应用
WO2020197991A1 (en) 2019-03-22 2020-10-01 Gilead Sciences, Inc. Bridged tricyclic carbamoylpyridone compounds and their pharmaceutical use
UY38982A (es) * 2019-12-09 2021-06-30 Viiv Healthcare Co Composiciones farmacéuticas
IL295677B1 (en) 2020-02-24 2026-04-01 Gilead Sciences Inc Tetracyclic compounds for the treatment of HIV infection
JP2023532981A (ja) * 2020-07-09 2023-08-01 ヤンセン ファーマシューティカ エヌ.ベー. 長時間作用型配合物
MX2023000439A (es) * 2020-07-09 2023-02-09 Janssen Pharmaceutica Nv Formulaciones a largo plazo.
WO2022051198A1 (en) * 2020-09-01 2022-03-10 Viiv Healthcare Company Combination of cabotegravir and levonorgestrel
CA3192145A1 (en) 2020-09-30 2022-04-07 Gilead Sciences, Inc. Bridged tricyclic carbamoylpyridone compounds and uses thereof
WO2022079739A1 (en) 2020-10-14 2022-04-21 Cipla Limited Fixed dose compositions of cabotegravir and rilpivirine
FI4196479T3 (fi) 2021-01-19 2024-01-17 Gilead Sciences Inc Substituoituja pyridotriatsiiniyhdisteitä ja niiden käyttöjä
TWI856796B (zh) 2022-04-06 2024-09-21 美商基利科學股份有限公司 橋聯三環胺甲醯基吡啶酮化合物及其用途
CN115844838B (zh) * 2022-12-01 2023-10-24 浙江萃泽医药科技有限公司 一种可注射的药物组合物
TW202602442A (zh) 2024-03-01 2026-01-16 英商Viiv醫療保健英國(No 3)有限公司 給藥方案
CN120424092B (zh) * 2025-07-02 2025-09-12 中国人民解放军军事科学院军事医学研究院 布尼亚病毒抑制剂及其制备方法和用途

Family Cites Families (34)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR1215599A (fr) * 1958-06-27 1960-04-19 Rhone Poulenc Sa Nouveaux dérivés de l'iminodibenzyle substitués à l'azote par une chaîne pipérazinique et leur préparation
US5352459A (en) 1992-12-16 1994-10-04 Sterling Winthrop Inc. Use of purified surface modifiers to prevent particle aggregation during sterilization
US5484926A (en) 1993-10-07 1996-01-16 Agouron Pharmaceuticals, Inc. HIV protease inhibitors
AU723537B2 (en) 1995-06-07 2000-08-31 Trimeris Inc. The treatment of HIV and other viral infections using combinatorial therapy
US5834025A (en) * 1995-09-29 1998-11-10 Nanosystems L.L.C. Reduction of intravenously administered nanoparticulate-formulation-induced adverse physiological reactions
TW487572B (en) 1996-05-20 2002-05-21 Janssen Pharmaceutica Nv Aqueous suspensions of 9-hydroxyrisperidone fatty acid esters
US6045829A (en) 1997-02-13 2000-04-04 Elan Pharma International Limited Nanocrystalline formulations of human immunodeficiency virus (HIV) protease inhibitors using cellulosic surface stabilizers
US6066292A (en) * 1997-12-19 2000-05-23 Bayer Corporation Sterilization process for pharmaceutical suspensions
TW518218B (en) * 1999-05-27 2003-01-21 Merck Patent Gmbh Pharmaceutical compositions comprising 1-[4-(5-cyanoindol-3-yl)butyl]-4-(2-carbamoylbenzofuran-5-yl)piperazine or its physiologically acceptable salts for use in the treatment of sub-type anxiety disorders
JP5160005B2 (ja) * 2000-12-28 2013-03-13 武田薬品工業株式会社 徐放性製剤
US20050084490A1 (en) * 2002-07-09 2005-04-21 Point Therapeutics, Inc. Boroproline compound combination therapy
WO2004018312A1 (en) * 2002-08-21 2004-03-04 Pharmacia Corporation Injectable pharmaceutical suspension in a two-chamber vial
CA2523035C (en) 2003-05-22 2011-04-26 Elan Pharma International Ltd. Sterilization of dispersions of nanoparticulate active agents with gamma radiation
BRPI0507308A (pt) 2004-01-29 2007-06-26 Baxter Int nanossuspensões de agentes anti-retrovirais para entrega ao sistema nervoso central aumentada
US7985222B2 (en) 2004-04-21 2011-07-26 Medshape Solutions, Inc. Osteosynthetic implants and methods of use and manufacture
EP1879890A1 (en) 2005-04-25 2008-01-23 Janssen Pharmaceutica N.V. Preparation of aseptic 3-[2-[4-(6-fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl]ethyl]-6,7,8,9-tetrahydro-9-hydroxy-2-methyl-4h-pyridio[1,2-a]pyrimidin-4-one palmitate ester
US8129385B2 (en) * 2005-04-28 2012-03-06 Shionogi & Co., Ltd. Substituted 5-hydroxy-3,4,6,9,9a, 10-hexanhydro-2h-1-oxa04a,8a-diaza-anthracene-6,10-dioness
WO2007053189A2 (en) * 2005-06-01 2007-05-10 Northwestern University Compositions and methods for altering immune function
EP1904052A4 (en) 2005-06-17 2008-12-10 Hospira Australia Pty Ltd LIQUID PHARMACEUTICAL COMPOSITIONS OF DOCATEXEL
US20070001094A1 (en) 2005-06-29 2007-01-04 Micron Technology, Inc. Infrared filter for imagers
BRPI0707179A2 (pt) * 2006-01-20 2011-04-26 Tibotec Pharm Ltd tratamento de longo termo de infecção por hiv
US20070178051A1 (en) 2006-01-27 2007-08-02 Elan Pharma International, Ltd. Sterilized nanoparticulate glucocorticosteroid formulations
EP2040671B1 (en) 2006-06-23 2018-01-24 Janssen Sciences Ireland UC Aqueous suspensions of tmc278
SI2175857T1 (sl) * 2007-07-12 2014-01-31 Janssen R&D Ireland Kristalna oblika (E) 4-((4-((4-(2-cianoetenil)-2,6-dimetilfenil)amino) 2-pirimidinil)amino)benzonitrila
BRPI0821408A2 (pt) * 2007-12-19 2015-06-16 Janssen Pharmaceutica Nv Regime de dosagem associado a ésteres de paliperidona injetáveis de longa ação
TWI489994B (zh) 2008-03-17 2015-07-01 Baxter Healthcare Sa 供免疫球蛋白及玻尿酸酶之皮下投藥之用的組合及方法
US20090311237A1 (en) * 2008-04-14 2009-12-17 Frost Gregory I Combination therapy using a soluble hyaluronidase and a bisphosphonate
US8648119B2 (en) * 2008-05-23 2014-02-11 Otonomy, Inc. Controlled release immunomodulator compositions and methods for the treatment of otic disorders
EP2320909B8 (en) * 2008-07-25 2016-03-30 VIIV Healthcare Company Chemical compounds
WO2010011815A1 (en) * 2008-07-25 2010-01-28 Smithkline Beecham Corporation Chemical compounds
KR101682058B1 (ko) 2008-12-11 2016-12-02 비이브 헬쓰케어 컴퍼니 카르바모일피리돈 hiv 인테그라제 억제제를 위한 제조방법 및 중간체
CA2744019C (en) 2008-12-11 2017-03-14 Shionogi & Co., Ltd. Synthesis of carbamoylpyridone hiv integrase inhibitors and intermediates
WO2011017395A1 (en) 2009-08-04 2011-02-10 Glaxosmithkline Llc Chemical compounds
US20110152303A1 (en) 2009-12-18 2011-06-23 Glaxosmithkline Llc Chemical Compounds

Also Published As

Publication number Publication date
CN103547266A (zh) 2014-01-29
SI2616076T1 (sl) 2016-11-30
US20170027933A1 (en) 2017-02-02
US20250268893A1 (en) 2025-08-28
ZA201301766B (en) 2016-11-30
PL2616076T3 (pl) 2017-07-31
ME02520B (me) 2017-02-20
EP2616076B1 (en) 2016-07-13
CA2810524C (en) 2018-06-26
ES2594557T3 (es) 2016-12-21
MX2013003037A (es) 2013-09-02
CA2810524A1 (en) 2012-03-22
CY1118279T1 (el) 2017-06-28
EP2616076A2 (en) 2013-07-24
US20130171214A1 (en) 2013-07-04
EA201390233A1 (ru) 2014-03-31
HUE031336T2 (hu) 2017-07-28
BR112013005907B1 (pt) 2021-04-27
TWI577377B (zh) 2017-04-11
US11224597B2 (en) 2022-01-18
HRP20161280T1 (hr) 2016-11-18
EA024924B1 (ru) 2016-11-30
AU2011302030B2 (en) 2015-01-22
JP6231385B2 (ja) 2017-11-15
US20220096469A1 (en) 2022-03-31
US20240307387A1 (en) 2024-09-19
IL225028A (en) 2017-04-30
KR101938662B1 (ko) 2019-01-15
KR20130116254A (ko) 2013-10-23
AU2011302030A1 (en) 2013-04-04
MX346193B (es) 2017-03-10
CL2013000715A1 (es) 2013-07-05
DK2616076T3 (en) 2016-10-24
JP2014500849A (ja) 2014-01-16
RS55222B1 (sr) 2017-02-28
SMT201600350B (it) 2016-11-10
TW201223529A (en) 2012-06-16
WO2012037320A2 (en) 2012-03-22
US20250017923A1 (en) 2025-01-16
EP2616076A4 (en) 2015-01-21
CN103547266B (zh) 2016-04-06
US12138264B2 (en) 2024-11-12
LT2616076T (lt) 2016-10-10
BR112013005907A2 (pt) 2016-06-07
US20250017924A1 (en) 2025-01-16
PT2616076T (pt) 2016-09-30
WO2012037320A3 (en) 2014-03-27

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