UA66801C2 - Триазоло[4,5-d]піримідинові сполуки, спосіб їх одержання (варіанти), фармацевтична композиція на їх основі та спосіб лікування порушень агрегації тромбоцитів - Google Patents

Триазоло[4,5-d]піримідинові сполуки, спосіб їх одержання (варіанти), фармацевтична композиція на їх основі та спосіб лікування порушень агрегації тромбоцитів

Info

Publication number
UA66801C2
UA66801C2 UA2000020981A UA00020981A UA66801C2 UA 66801 C2 UA66801 C2 UA 66801C2 UA 2000020981 A UA2000020981 A UA 2000020981A UA 00020981 A UA00020981 A UA 00020981A UA 66801 C2 UA66801 C2 UA 66801C2
Authority
UA
Ukraine
Prior art keywords
novel compounds
medicaments
processes
formula
preparation
Prior art date
Application number
UA2000020981A
Other languages
English (en)
Russian (ru)
Inventor
Сімон Гайл
Ентоні Інголл
Брайан Спрінгторп
Пол Уілліс
Original Assignee
Астра Фармасьютікалз Лтд.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=26663042&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=UA66801(C2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from SE9702775A external-priority patent/SE9702775D0/xx
Priority claimed from SE9702773A external-priority patent/SE9702773D0/xx
Application filed by Астра Фармасьютікалз Лтд. filed Critical Астра Фармасьютікалз Лтд.
Publication of UA66801C2 publication Critical patent/UA66801C2/uk

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/04—Drugs for disorders of the respiratory system for throat disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/14—Vasoprotectives; Antihaemorrhoidals; Drugs for varicose therapy; Capillary stabilisers

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pulmonology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Vascular Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Otolaryngology (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)

Abstract

Винахід стосується нових триазоло[4,5-d]піримідинових сполук формули (І), їх застосування як лікарських засобів, композицій, що їх містять, та способів їх одержання.
UA2000020981A 1997-07-22 1998-07-15 Триазоло[4,5-d]піримідинові сполуки, спосіб їх одержання (варіанти), фармацевтична композиція на їх основі та спосіб лікування порушень агрегації тромбоцитів UA66801C2 (uk)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
SE9702775A SE9702775D0 (sv) 1997-07-22 1997-07-22 Novel compounds
SE9702773A SE9702773D0 (sv) 1997-07-22 1997-07-22 Novel compounds
PCT/SE1998/001393 WO1999005143A1 (en) 1997-07-22 1998-07-15 Novel compounds

Publications (1)

Publication Number Publication Date
UA66801C2 true UA66801C2 (uk) 2004-06-15

Family

ID=26663042

Family Applications (1)

Application Number Title Priority Date Filing Date
UA2000020981A UA66801C2 (uk) 1997-07-22 1998-07-15 Триазоло[4,5-d]піримідинові сполуки, спосіб їх одержання (варіанти), фармацевтична композиція на їх основі та спосіб лікування порушень агрегації тромбоцитів

Country Status (30)

Country Link
EP (1) EP0996621B1 (uk)
JP (1) JP4187406B2 (uk)
KR (2) KR20050084540A (uk)
CN (1) CN1154650C (uk)
AR (2) AR017014A1 (uk)
AT (1) ATE251161T1 (uk)
AU (1) AU745381B2 (uk)
BR (1) BR9810802B1 (uk)
CA (1) CA2296665C (uk)
CZ (1) CZ302629B6 (uk)
DE (1) DE69818668T2 (uk)
DK (1) DK0996621T3 (uk)
EE (1) EE04193B1 (uk)
EG (1) EG24412A (uk)
ES (1) ES2207846T3 (uk)
HU (1) HU230074B1 (uk)
IL (2) IL133959A0 (uk)
IS (1) IS2236B (uk)
MY (1) MY123196A (uk)
NO (1) NO315854B1 (uk)
NZ (1) NZ502381A (uk)
PL (1) PL200325B1 (uk)
PT (1) PT996621E (uk)
RU (1) RU2225407C2 (uk)
SA (1) SA98190487B1 (uk)
SK (1) SK284199B6 (uk)
TR (1) TR200000197T2 (uk)
TW (1) TW530058B (uk)
UA (1) UA66801C2 (uk)
WO (1) WO1999005143A1 (uk)

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SE9904128D0 (sv) * 1999-11-15 1999-11-15 Astra Pharma Prod Novel compounds
SE9904129D0 (sv) * 1999-11-15 1999-11-15 Astra Pharma Prod Novel compounds
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SE0004099D0 (sv) * 2000-11-09 2000-11-09 Astrazeneca Ab Novel compounds
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WO2023213198A1 (zh) * 2022-05-04 2023-11-09 华东师范大学 芳香稠环化合物作为trek-1激活剂的用途、包含其的药物组合物、镇痛剂
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CN115710275B (zh) * 2022-11-21 2024-02-02 河南中医药大学 一种嘧啶-tcp类化合物、制备方法和医药用途

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Also Published As

Publication number Publication date
KR20050084540A (ko) 2005-08-26
EP0996621A1 (en) 2000-05-03
KR20010022083A (ko) 2001-03-15
CN1270590A (zh) 2000-10-18
HK1026421A1 (en) 2000-12-15
NO20000312D0 (no) 2000-01-21
JP2001510842A (ja) 2001-08-07
NO20000312L (no) 2000-03-21
SA98190487B1 (ar) 2006-08-20
PL200325B1 (pl) 2008-12-31
EE200000044A (et) 2000-10-16
CN1154650C (zh) 2004-06-23
RU2225407C2 (ru) 2004-03-10
CA2296665C (en) 2008-06-10
TW530058B (en) 2003-05-01
SK284199B6 (sk) 2004-10-05
IL133959A0 (en) 2001-04-30
HUP0004333A3 (en) 2001-11-28
AU8370698A (en) 1999-02-16
SK188199A3 (en) 2000-10-09
MY123196A (en) 2006-05-31
ATE251161T1 (de) 2003-10-15
NO315854B1 (no) 2003-11-03
TR200000197T2 (tr) 2000-06-21
AR077553A2 (es) 2011-09-07
BR9810802A (pt) 2000-09-12
PL338516A1 (en) 2000-11-06
AU745381B2 (en) 2002-03-21
BR9810802B1 (pt) 2010-10-19
KR100535837B1 (ko) 2006-01-12
DE69818668D1 (de) 2003-11-06
EP0996621B1 (en) 2003-10-01
IL133959A (en) 2007-10-31
IS2236B (is) 2007-05-15
EG24412A (en) 2009-05-25
ES2207846T3 (es) 2004-06-01
JP4187406B2 (ja) 2008-11-26
CA2296665A1 (en) 1999-02-04
HU230074B1 (hu) 2015-06-29
HUP0004333A2 (hu) 2001-04-28
DK0996621T3 (da) 2004-02-02
EE04193B1 (et) 2003-12-15
WO1999005143A1 (en) 1999-02-04
PT996621E (pt) 2004-02-27
DE69818668T2 (de) 2004-08-12
IS5354A (is) 2000-01-20
AR017014A1 (es) 2001-08-22
CZ302629B6 (cs) 2011-08-10
CZ2000233A3 (cs) 2000-07-12
NZ502381A (en) 2001-12-21

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