UA77303C2 - Derivatives of thienopyridines substituted by benzocondensed heteroarylamide useful as therapeutic agents, pharmaceutical compositions and methods for their use - Google Patents

Derivatives of thienopyridines substituted by benzocondensed heteroarylamide useful as therapeutic agents, pharmaceutical compositions and methods for their use Download PDF

Info

Publication number: UA77303C2
Authority: UA; Ukraine
Prior art keywords: alkyl; compound; aryl; indole; carboxylic acid
Prior art date: 2002-06-14

Application number

UA20041210250A

Other languages

English (en)

Ukrainian (uk)

Original Assignee

Pfizer

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2002-06-14

Filing date

2003-04-06

Publication date

2006-11-15

2003-04-06 Application filed by Pfizer filed Critical Pfizer

2006-11-15 Publication of UA77303C2 publication Critical patent/UA77303C2/uk

Links

238000000034 method Methods 0.000 title claims abstract description 50
239000008194 pharmaceutical composition Substances 0.000 title claims abstract description 30
239000003814 drug Substances 0.000 title description 9
229940124597 therapeutic agent Drugs 0.000 title description 3
229940125670 thienopyridine Drugs 0.000 title description 2
239000002175 thienopyridine Substances 0.000 title description 2
150000001875 compounds Chemical class 0.000 claims abstract description 433
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-1 methylureido group Chemical group 0.000 claims description 80
125000000217 alkyl group Chemical group 0.000 claims description 64
125000000623 heterocyclic group Chemical group 0.000 claims description 61
125000003118 aryl group Chemical group 0.000 claims description 50
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Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
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Veterinary Medicine (AREA)
Medicinal Chemistry (AREA)
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Chemical Kinetics & Catalysis (AREA)
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Bioinformatics & Cheminformatics (AREA)
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Epidemiology (AREA)
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Heart & Thoracic Surgery (AREA)
Cardiology (AREA)
Urology & Nephrology (AREA)
Endocrinology (AREA)
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Biomedical Technology (AREA)
Neurology (AREA)
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Pain & Pain Management (AREA)
Gynecology & Obstetrics (AREA)
Pregnancy & Childbirth (AREA)
Hematology (AREA)
Pulmonology (AREA)
Emergency Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Plural Heterocyclic Compounds (AREA)

UA20041210250A 2002-06-14 2003-04-06 Derivatives of thienopyridines substituted by benzocondensed heteroarylamide useful as therapeutic agents, pharmaceutical compositions and methods for their use UA77303C2 (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US38911002P	2002-06-14	2002-06-14
PCT/IB2003/002393 WO2003106462A1 (en)	2002-06-14	2003-06-04	Benzofused heteroaryl amide derivatives of thienopyridines useful as therapeutic agents, pharmaceutical compositions including the same, and methods for their use

Publications (1)

Publication Number	Publication Date
UA77303C2 true UA77303C2 (en)	2006-11-15

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UA20041210250A UA77303C2 (en)	2002-06-14	2003-04-06	Derivatives of thienopyridines substituted by benzocondensed heteroarylamide useful as therapeutic agents, pharmaceutical compositions and methods for their use

Country Status (36)

Country	Link
US (3)	US6869962B2 (de)
EP (1)	EP1515975B1 (de)
JP (1)	JP2005534669A (de)
KR (2)	KR100714545B1 (de)
CN (1)	CN1671714A (de)
AP (1)	AP2004003184A0 (de)
AR (1)	AR039673A1 (de)
AT (1)	ATE373665T1 (de)
AU (1)	AU2003233134A1 (de)
BR (1)	BR0311806A (de)
CA (1)	CA2489466A1 (de)
CO (1)	CO5631447A2 (de)
DE (1)	DE60316440T2 (de)
EA (1)	EA008255B1 (de)
EC (1)	ECSP045483A (de)
ES (1)	ES2290460T3 (de)
GE (1)	GEP20074033B (de)
GT (1)	GT200300129A (de)
HN (1)	HN2003000182A (de)
HR (1)	HRP20041173A2 (de)
IL (1)	IL165591A0 (de)
IS (1)	IS7552A (de)
MA (1)	MA27596A1 (de)
MX (1)	MXPA04011637A (de)
NO (1)	NO20045103L (de)
NZ (1)	NZ537140A (de)
OA (1)	OA12865A (de)
PA (1)	PA8575401A1 (de)
PE (1)	PE20050123A1 (de)
PL (1)	PL374542A1 (de)
RS (1)	RS107504A (de)
TN (1)	TNSN04246A1 (de)
TW (1)	TW200404070A (de)
UA (1)	UA77303C2 (de)
WO (1)	WO2003106462A1 (de)
ZA (1)	ZA200409862B (de)

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US20040186126A1 (en)	2004-09-23
AR039673A1 (es)	2005-03-09
US7045528B2 (en)	2006-05-16
RS107504A (sr)	2006-10-27
CO5631447A2 (es)	2006-04-28
ECSP045483A (es)	2005-01-28
WO2003106462A1 (en)	2003-12-24
JP2005534669A (ja)	2005-11-17
DE60316440T2 (de)	2008-01-24
AP2004003184A0 (en)	2004-12-31
MA27596A1 (fr)	2005-11-01
TNSN04246A1 (fr)	2007-03-12
KR20060110011A (ko)	2006-10-23
US20040009965A1 (en)	2004-01-15
DE60316440D1 (de)	2007-10-31
EA008255B1 (ru)	2007-04-27
GEP20074033B (en)	2007-02-12
GT200300129A (es)	2004-03-17
EP1515975B1 (de)	2007-09-19
PA8575401A1 (es)	2004-05-07
EP1515975A1 (de)	2005-03-23
US20060079548A1 (en)	2006-04-13
NO20045103L (no)	2005-02-17
NZ537140A (en)	2006-10-27
US6869962B2 (en)	2005-03-22
ES2290460T3 (es)	2008-02-16
ATE373665T1 (de)	2007-10-15
CN1671714A (zh)	2005-09-21
CA2489466A1 (en)	2003-12-24
KR100714545B1 (ko)	2007-05-07
ZA200409862B (en)	2006-05-31
PE20050123A1 (es)	2005-03-22
TW200404070A (en)	2004-03-16
EA200500018A1 (ru)	2005-06-30
HN2003000182A (es)	2004-07-27
BR0311806A (pt)	2005-03-29
MXPA04011637A (es)	2005-03-07
KR20050008821A (ko)	2005-01-21
PL374542A1 (en)	2005-10-31
IL165591A0 (en)	2006-01-15
AU2003233134A1 (en)	2003-12-31
KR100671632B1 (ko)	2007-02-28
HRP20041173A2 (en)	2005-06-30
IS7552A (is)	2004-11-25
OA12865A (en)	2006-09-15

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