UA77441C2 - 4,5-dihydro-1h-pyrazole derivatives as potent cb1 receptor antagonists, methods for their preparation (variants), intermediate, pharmaceutical composition and method for its preparation - Google Patents

4,5-dihydro-1h-pyrazole derivatives as potent cb1 receptor antagonists, methods for their preparation (variants), intermediate, pharmaceutical composition and method for its preparation Download PDF

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Publication number: UA77441C2
Authority: UA; Ukraine
Prior art keywords: group; formula; phenyl; dihydro; compound
Prior art date: 2001-09-21

Application number

UA20040402981A

Other languages

English (en)

Ukrainian (uk)

Inventor

Cornelis G Kruse

Arnoldus H J Herremans

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2001-09-21

Filing date

2002-09-17

Publication date

2006-12-15

2002-09-17 Application filed filed Critical

2006-12-15 Publication of UA77441C2 publication Critical patent/UA77441C2/uk

Links

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UA20040402981A 2001-09-21 2002-09-17 4,5-dihydro-1h-pyrazole derivatives as potent cb1 receptor antagonists, methods for their preparation (variants), intermediate, pharmaceutical composition and method for its preparation UA77441C2 (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
EP01203849		2001-09-21
PCT/EP2002/010435 WO2003026648A1 (en)	2001-09-21	2002-09-17	4,5-dihydro-1h-pyrazole derivatives having potent cb1-antagonistic activity

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UA77441C2 true UA77441C2 (en)	2006-12-15

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US (2)	US6974810B2 (pl)
EP (1)	EP1429762A1 (pl)
JP (1)	JP4313672B2 (pl)
KR (1)	KR100950430B1 (pl)
CN (2)	CN101195604A (pl)
AR (1)	AR036598A1 (pl)
AU (1)	AU2002333853B2 (pl)
BR (1)	BR0208253A (pl)
CA (1)	CA2442245C (pl)
HR (1)	HRP20030913A2 (pl)
HU (1)	HUP0402113A3 (pl)
IL (2)	IL157704A0 (pl)
MX (1)	MXPA03009439A (pl)
NO (1)	NO20041170L (pl)
NZ (1)	NZ528280A (pl)
PL (1)	PL367814A1 (pl)
RU (1)	RU2286988C2 (pl)
UA (1)	UA77441C2 (pl)
WO (1)	WO2003026648A1 (pl)
ZA (1)	ZA200307218B (pl)

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ZA200307218B (en)	2005-03-16
CA2442245C (en)	2010-03-30
NZ528280A (en)	2005-11-25
WO2003026648A1 (en)	2003-04-03
RU2286988C2 (ru)	2006-11-10
US20040106800A1 (en)	2004-06-03
CN101195604A (zh)	2008-06-11
US7608718B2 (en)	2009-10-27
EP1429762A1 (en)	2004-06-23
PL367814A1 (pl)	2005-03-07
HUP0402113A2 (hu)	2005-01-28
IL157704A0 (en)	2004-03-28
US20070259884A1 (en)	2007-11-08
CA2442245A1 (en)	2003-04-03
AU2002333853B2 (en)	2006-07-13
RU2003130268A (ru)	2005-01-27
HRP20030913A2 (en)	2004-06-30
JP2005503428A (ja)	2005-02-03
JP4313672B2 (ja)	2009-08-12
KR20040035845A (ko)	2004-04-29
AR036598A1 (es)	2004-09-22
KR100950430B1 (ko)	2010-04-02
HUP0402113A3 (en)	2012-05-29
IL157704A (en)	2008-07-08
NO20041170L (no)	2004-06-21
BR0208253A (pt)	2004-04-13
US6974810B2 (en)	2005-12-13
MXPA03009439A (es)	2004-02-12
CN1529595A (zh)	2004-09-15

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