UA81994C2 - 5,7-diaminopyrazolo [4,3-d] pyrimidines with pde-5 inhibiting activity - Google Patents

5,7-diaminopyrazolo [4,3-d] pyrimidines with pde-5 inhibiting activity Download PDF

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Publication number
UA81994C2
UA81994C2 UAA200605669A UAA200605669A UA81994C2 UA 81994 C2 UA81994 C2 UA 81994C2 UA A200605669 A UAA200605669 A UA A200605669A UA A200605669 A UAA200605669 A UA A200605669A UA 81994 C2 UA81994 C2 UA 81994C2
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preparation
formula
nmr
solution
compounds
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UAA200605669A
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Ukrainian (uk)
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Кевин Нил Декк
Девид Натан Абрахам Фокс
Ян Роджер Марш
Эндрю Ян Моррелл
Керол Энн Уинслоу
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Пфайзер Инк.
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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
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    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/14—Vasoprotectives; Antihaemorrhoidals; Drugs for varicose therapy; Capillary stabilisers
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
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    • Y02P20/582—Recycling of unreacted starting or intermediate materials

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Abstract

Это изобретение касается соединений формулы (І)(I).
UAA200605669A 2003-11-24 2004-12-11 5,7-diaminopyrazolo [4,3-d] pyrimidines with pde-5 inhibiting activity UA81994C2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0327319.0A GB0327319D0 (en) 2003-11-24 2003-11-24 Novel pharmaceuticals
PCT/IB2004/003747 WO2005049616A1 (en) 2003-11-24 2004-11-12 5,7-DIAMINOPYRAZOLO [4,3-d] PYRIMIDINES WITH PDE-5 INHIBITING ACTIVITY

Publications (1)

Publication Number Publication Date
UA81994C2 true UA81994C2 (en) 2008-02-25

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UAA200605669A UA81994C2 (en) 2003-11-24 2004-12-11 5,7-diaminopyrazolo [4,3-d] pyrimidines with pde-5 inhibiting activity

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EP (1) EP1689751B1 (ru)
JP (1) JP4056015B2 (ru)
KR (2) KR100848216B1 (ru)
CN (4) CN101362764B (ru)
AP (1) AP2227A (ru)
AR (1) AR046711A1 (ru)
AT (1) ATE485297T1 (ru)
AU (1) AU2004290643B2 (ru)
BR (1) BRPI0416869A (ru)
CA (1) CA2546987C (ru)
CR (1) CR8416A (ru)
CY (1) CY1110933T1 (ru)
DE (1) DE602004029705D1 (ru)
DK (1) DK1689751T3 (ru)
EA (1) EA011772B1 (ru)
EC (1) ECSP066580A (ru)
ES (1) ES2351622T3 (ru)
GB (1) GB0327319D0 (ru)
GE (1) GEP20084528B (ru)
HR (1) HRP20100651T1 (ru)
IL (1) IL175433A (ru)
IS (1) IS8406A (ru)
MA (1) MA28172A1 (ru)
ME (1) ME01216B (ru)
MX (1) MXPA06005914A (ru)
MY (1) MY140872A (ru)
NL (1) NL1027568C2 (ru)
NO (1) NO336526B1 (ru)
NZ (1) NZ548097A (ru)
OA (1) OA13289A (ru)
PA (1) PA8617701A1 (ru)
PE (1) PE20051061A1 (ru)
PL (1) PL1689751T3 (ru)
PT (1) PT1689751E (ru)
RS (1) RS51556B (ru)
SG (1) SG133614A1 (ru)
SI (1) SI1689751T1 (ru)
TN (1) TNSN06154A1 (ru)
TW (1) TWI265031B (ru)
UA (1) UA81994C2 (ru)
UY (1) UY28625A1 (ru)
WO (1) WO2005049616A1 (ru)
ZA (1) ZA200602899B (ru)

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