UA89787C2 - Фторгликозидные производные пиразолов, лекарственное средство, которое содержит их, и их применение - Google Patents

Фторгликозидные производные пиразолов, лекарственное средство, которое содержит их, и их применение

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Publication number
UA89787C2
UA89787C2 UAA200700259A UAA200700259A UA89787C2 UA 89787 C2 UA89787 C2 UA 89787C2 UA A200700259 A UAA200700259 A UA A200700259A UA A200700259 A UAA200700259 A UA A200700259A UA 89787 C2 UA89787 C2 UA 89787C2
Authority
UA
Ukraine
Prior art keywords
pyrazoles
compounds
medicaments containing
fluoroglycoside derivatives
derivatives
Prior art date
Application number
UAA200700259A
Other languages
English (en)
Ukrainian (uk)
Inventor
Харм Бруммерхоп
Венделин Фрик
Хайнер Гломбик
Оливер ПЛЕТТЕНБУРГ
Мартин Биккель
Хуберт Хойер
Штефан Тайс
Original Assignee
Санофи-Авентис Дойчланд Гмбх
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Санофи-Авентис Дойчланд Гмбх filed Critical Санофи-Авентис Дойчланд Гмбх
Publication of UA89787C2 publication Critical patent/UA89787C2/ru

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/02—Heterocyclic radicals containing only nitrogen as ring hetero atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/12—Drugs for disorders of the urinary system of the kidneys
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/06—Antipsoriatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
    • A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/18—Antivirals for RNA viruses for HIV
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/12—Antidiuretics, e.g. drugs for diabetes insipidus
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Immunology (AREA)
  • Rheumatology (AREA)
  • Obesity (AREA)
  • Molecular Biology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Psychiatry (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Pulmonology (AREA)
  • Urology & Nephrology (AREA)
  • Virology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • AIDS & HIV (AREA)
  • Ophthalmology & Optometry (AREA)
  • Pain & Pain Management (AREA)

Abstract

Изобретение касается замещенных фторгликозидных производных пиразолов формулы (И), в которой остатки имеют указанные значения, а также их физиологически совместимых солей и способов их получения. Соединения используют, например, как антидиабетические средства.
UAA200700259A 2004-06-11 2005-06-03 Фторгликозидные производные пиразолов, лекарственное средство, которое содержит их, и их применение UA89787C2 (ru)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE102004028241A DE102004028241B4 (de) 2004-06-11 2004-06-11 Neue Fluorglykosidderivate von Pyrazolen, diese Verbindungen enthaltende Arzneimittel und Herstellung dieser Arzneimittel

Publications (1)

Publication Number Publication Date
UA89787C2 true UA89787C2 (ru) 2010-03-10

Family

ID=35355753

Family Applications (1)

Application Number Title Priority Date Filing Date
UAA200700259A UA89787C2 (ru) 2004-06-11 2005-06-03 Фторгликозидные производные пиразолов, лекарственное средство, которое содержит их, и их применение

Country Status (33)

Country Link
US (1) US7820804B2 (ru)
EP (1) EP1758914B1 (ru)
JP (1) JP4996464B2 (ru)
CN (1) CN100582116C (ru)
AR (1) AR049393A1 (ru)
AU (1) AU2005252329B2 (ru)
BR (1) BRPI0510770A (ru)
CA (1) CA2570042C (ru)
CR (1) CR8773A (ru)
CY (1) CY1107426T1 (ru)
DE (2) DE102004028241B4 (ru)
DK (1) DK1758914T3 (ru)
EC (1) ECSP067054A (ru)
ES (1) ES2296180T3 (ru)
HR (1) HRP20080023T3 (ru)
IL (1) IL179757A (ru)
MA (1) MA28653B1 (ru)
MX (1) MXPA06013513A (ru)
MY (1) MY143565A (ru)
NO (1) NO20070176L (ru)
NZ (1) NZ551948A (ru)
PE (1) PE20060297A1 (ru)
PL (1) PL1758914T3 (ru)
PT (1) PT1758914E (ru)
RS (1) RS50541B (ru)
RU (1) RU2370499C2 (ru)
SI (1) SI1758914T1 (ru)
TN (1) TNSN06409A1 (ru)
TW (1) TWI382030B (ru)
UA (1) UA89787C2 (ru)
UY (1) UY28955A1 (ru)
WO (1) WO2005121161A1 (ru)
ZA (1) ZA200608832B (ru)

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Also Published As

Publication number Publication date
PL1758914T3 (pl) 2008-04-30
CR8773A (es) 2008-02-28
AR049393A1 (es) 2006-07-26
CN100582116C (zh) 2010-01-20
RU2370499C2 (ru) 2009-10-20
DE502005002056D1 (de) 2008-01-03
MXPA06013513A (es) 2007-03-01
AU2005252329A1 (en) 2005-12-22
CY1107426T1 (el) 2012-12-19
MY143565A (en) 2011-05-31
PT1758914E (pt) 2008-01-31
RS50541B (sr) 2010-05-07
TNSN06409A1 (en) 2008-02-22
IL179757A0 (en) 2007-05-15
WO2005121161A1 (de) 2005-12-22
DE102004028241A1 (de) 2006-01-05
HRP20080023T3 (en) 2008-06-30
TWI382030B (zh) 2013-01-11
US7820804B2 (en) 2010-10-26
RU2007101154A (ru) 2008-07-20
PE20060297A1 (es) 2006-05-25
NO20070176L (no) 2007-03-09
US20070197623A1 (en) 2007-08-23
TW200610527A (en) 2006-04-01
CA2570042C (en) 2013-01-15
ZA200608832B (en) 2008-05-28
CN1964984A (zh) 2007-05-16
AU2005252329B2 (en) 2011-02-10
BRPI0510770A (pt) 2007-11-20
SI1758914T1 (sl) 2008-04-30
UY28955A1 (es) 2006-01-31
HK1100411A1 (zh) 2007-09-21
CA2570042A1 (en) 2005-12-22
DK1758914T3 (da) 2008-03-17
ECSP067054A (es) 2007-01-26
JP2008501745A (ja) 2008-01-24
MA28653B1 (fr) 2007-06-01
DE102004028241B4 (de) 2007-09-13
ES2296180T3 (es) 2008-04-16
IL179757A (en) 2010-12-30
JP4996464B2 (ja) 2012-08-08
EP1758914A1 (de) 2007-03-07
EP1758914B1 (de) 2007-11-21
NZ551948A (en) 2010-04-30

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