UA97536C2 - Proteasome inhibitors - Google Patents

Proteasome inhibitors

Info

Publication number
UA97536C2
UA97536C2 UAA201002409A UAA201002409A UA97536C2 UA 97536 C2 UA97536 C2 UA 97536C2 UA A201002409 A UAA201002409 A UA A201002409A UA A201002409 A UAA201002409 A UA A201002409A UA 97536 C2 UA97536 C2 UA 97536C2
Authority
UA
Ukraine
Prior art keywords
proteasome inhibitors
compositions
treatment
methods
various diseases
Prior art date
Application number
UAA201002409A
Other languages
English (en)
Russian (ru)
Inventor
Эдвард Дж. Олхава
Михаэла Д. Данка
Original Assignee
Милленниум Фармасьютикалз, Инк.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=38691782&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=UA97536(C2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Милленниум Фармасьютикалз, Инк. filed Critical Милленниум Фармасьютикалз, Инк.
Publication of UA97536C2 publication Critical patent/UA97536C2/ru

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
    • C07F5/02—Boron compounds
    • C07F5/025—Boronic and borinic acid compounds
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
    • C07F5/02—Boron compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/69—Boron compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P39/00—General protective or antinoxious agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Epidemiology (AREA)
  • Toxicology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Immunology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

У даному винаході запропоновані нові сполуки, придатні для застосування як інгібітори протеасом.У даному винаході також запропоновані фармацевтичні композиції, що містять сполуки згідно з даним винаходом, і застосування зазначених композицій для лікування різних захворювань.
UAA201002409A 2007-08-06 2007-08-06 Proteasome inhibitors UA97536C2 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
PCT/US2007/017440 WO2009020448A1 (en) 2007-08-06 2007-08-06 Proteasome inhibitors

Publications (1)

Publication Number Publication Date
UA97536C2 true UA97536C2 (en) 2012-02-27

Family

ID=38691782

Family Applications (1)

Application Number Title Priority Date Filing Date
UAA201002409A UA97536C2 (en) 2007-08-06 2007-08-06 Proteasome inhibitors

Country Status (32)

Country Link
EP (3) EP3210987A1 (uk)
JP (1) JP5261488B2 (uk)
KR (6) KR20160040735A (uk)
CN (1) CN101772507B (uk)
AU (1) AU2007357338B2 (uk)
BR (1) BRPI0721905B8 (uk)
CA (1) CA2695082C (uk)
CY (2) CY1113386T1 (uk)
DK (1) DK2178888T3 (uk)
EA (1) EA028622B1 (uk)
EC (1) ECSP10010015A (uk)
ES (1) ES2390606T3 (uk)
FR (1) FR17C1011I2 (uk)
GE (1) GEP20125599B (uk)
HR (1) HRP20120745T1 (uk)
HU (1) HUS1700018I1 (uk)
IL (4) IL203641A (uk)
LT (1) LTC2178888I2 (uk)
LU (1) LUC00013I2 (uk)
MY (1) MY161991A (uk)
NL (1) NL300871I2 (uk)
NZ (1) NZ582693A (uk)
PH (1) PH12014500053B1 (uk)
PL (1) PL2178888T3 (uk)
PT (1) PT2178888E (uk)
RS (1) RS52435B (uk)
SG (1) SG10201508712QA (uk)
SI (1) SI2178888T1 (uk)
TN (1) TN2010000060A1 (uk)
UA (1) UA97536C2 (uk)
WO (1) WO2009020448A1 (uk)
ZA (1) ZA201000348B (uk)

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Also Published As

Publication number Publication date
FR17C1011I2 (fr) 2018-04-27
HK1182924A1 (zh) 2013-12-13
EP2178888A1 (en) 2010-04-28
PL2178888T3 (pl) 2012-11-30
KR20150010802A (ko) 2015-01-28
CY2017016I2 (el) 2017-07-12
ECSP10010015A (es) 2010-04-30
DK2178888T3 (da) 2012-10-01
KR20100059811A (ko) 2010-06-04
JP2010535759A (ja) 2010-11-25
BRPI0721905B8 (pt) 2021-05-25
GEP20125599B (en) 2012-08-10
BRPI0721905A2 (pt) 2014-02-25
NZ582693A (en) 2012-01-12
CN101772507B (zh) 2012-12-12
KR20140042932A (ko) 2014-04-07
KR20170004031A (ko) 2017-01-10
TN2010000060A1 (en) 2011-09-26
LUC00013I2 (uk) 2017-06-19
AU2007357338B2 (en) 2014-03-20
JP5261488B2 (ja) 2013-08-14
IL242291A0 (en) 2015-11-30
EP3210987A1 (en) 2017-08-30
EA028622B1 (ru) 2017-12-29
CN101772507A (zh) 2010-07-07
HK1143595A1 (en) 2011-01-07
IL242290A0 (en) 2015-11-30
CY2017016I1 (el) 2017-07-12
CA2695082C (en) 2015-07-28
LTC2178888I2 (lt) 2018-03-12
SG10201508712QA (en) 2015-11-27
ES2390606T3 (es) 2012-11-14
PH12014500053A1 (en) 2015-03-30
EP2527347A1 (en) 2012-11-28
CA2695082A1 (en) 2009-02-12
LTPA2017010I1 (lt) 2017-05-10
IL203641A (en) 2015-11-30
HRP20120745T1 (hr) 2012-10-31
SI2178888T1 (sl) 2012-11-30
IL242292A0 (en) 2015-11-30
LUC00013I1 (uk) 2017-04-06
BRPI0721905B1 (pt) 2020-11-17
CY1113386T1 (el) 2016-06-22
NL300871I2 (nl) 2017-12-07
EP2178888B1 (en) 2012-07-04
HUS1700018I1 (hu) 2017-05-29
IL242291A (en) 2017-12-31
KR101474831B1 (ko) 2014-12-19
IL242292A (en) 2017-12-31
KR101831674B1 (ko) 2018-02-23
RS52435B (sr) 2013-02-28
ZA201000348B (en) 2011-03-30
AU2007357338A1 (en) 2009-02-12
WO2009020448A1 (en) 2009-02-12
EA201070247A1 (ru) 2010-06-30
KR20160040735A (ko) 2016-04-14
PH12014500053B1 (en) 2015-03-30
KR20140042933A (ko) 2014-04-07
PT2178888E (pt) 2012-10-04
MY161991A (en) 2017-05-31
IL242290A (en) 2017-12-31
FR17C1011I1 (uk) 2017-05-26

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