UA99132C2 - Производные дикарбоновых кислот как агонисты рецепторов s1p1 - Google Patents

Производные дикарбоновых кислот как агонисты рецепторов s1p1

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Publication number
UA99132C2
UA99132C2 UAA200912896A UAA200912896A UA99132C2 UA 99132 C2 UA99132 C2 UA 99132C2 UA A200912896 A UAA200912896 A UA A200912896A UA A200912896 A UAA200912896 A UA A200912896A UA 99132 C2 UA99132 C2 UA 99132C2
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Ukraine
Prior art keywords
dicarboxylic acid
acid derivatives
receptor agonists
compounds
conditions
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UAA200912896A
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English (en)
Ukrainian (uk)
Inventor
Марк Капе
Никола Левуан
Изабелла Берреби-Бертран
Филипп Робер
Жан-Шарль Шварц
Жан-Мари Леконт
Джайрадж Дилипбхаи Арадхье
Мутхукумаран Натараджан Пиллаи
Бхавеш Моханбхаи Панчал
Джигнеш Кантилал Дживани
Бисваджит Саманта
Ранджан Кумар Пал
Раджаманнар Тхеннати
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Биопроже
Сан Фарма Эдванст Рисёч Компани Лтд
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Publication of UA99132C2 publication Critical patent/UA99132C2/ru

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    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings

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  • Health & Medical Sciences (AREA)
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Abstract

Представленное изобретение касается новых соединений формулы (I), обладающих агонистической активность относительно рецепторов сфингозин-1-фосфата (S1P), способов их получения и их применения в качестве иммунодепрессантов.Изобретение касается также фармацевтических композиций, которые содержат упомянутые соединения, и применения таких композиций для лечения и профилактики заболеваний и состояний, опосредствованных иммунной системой, или воспалительных заболеваний и состояний.
UAA200912896A 2007-06-15 2008-06-16 Производные дикарбоновых кислот как агонисты рецепторов s1p1 UA99132C2 (ru)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP07290748A EP2014653A1 (en) 2007-06-15 2007-06-15 Novel dicarboxylic acid derivatives as S1P1 receptor agonists

Publications (1)

Publication Number Publication Date
UA99132C2 true UA99132C2 (ru) 2012-07-25

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Country Status (17)

Country Link
US (1) US8809539B2 (ru)
EP (2) EP2014653A1 (ru)
JP (1) JP5346016B2 (ru)
KR (1) KR20100040853A (ru)
CN (1) CN101784535A (ru)
BR (1) BRPI0811712A2 (ru)
CA (1) CA2693126A1 (ru)
CO (1) CO6251262A2 (ru)
EA (1) EA018826B1 (ru)
IL (1) IL202741A0 (ru)
MA (1) MA31447B1 (ru)
MX (1) MX2009013733A (ru)
NZ (1) NZ581933A (ru)
TN (1) TN2009000524A1 (ru)
UA (1) UA99132C2 (ru)
WO (1) WO2008152149A1 (ru)
ZA (1) ZA200908851B (ru)

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KR20190116416A (ko) 2017-02-16 2019-10-14 아레나 파마슈티칼스, 인크. 원발 담즙성 담관염을 치료하기 위한 화합물 및 방법
CN107827837B (zh) * 2017-11-21 2021-09-24 苏州朗科生物技术股份有限公司 鞘氨醇-1-磷酸受体调节剂化合物及其制备方法与应用
KR20200116953A (ko) * 2018-02-02 2020-10-13 고쿠리츠 다이가쿠 호진 교토 다이가쿠 안내 혈관 신생 및/또는 안내 혈관 투과성 항진을 수반하는 안과 질환의 예방 또는 치료를 위한 의약
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CO6251262A2 (es) 2011-02-21
BRPI0811712A2 (pt) 2014-11-04
EA201000024A1 (ru) 2010-06-30
ZA200908851B (en) 2010-07-28
EP2014653A1 (en) 2009-01-14
EP2170850B1 (en) 2014-09-24
IL202741A0 (en) 2010-06-30
TN2009000524A1 (en) 2011-03-31
KR20100040853A (ko) 2010-04-21
CA2693126A1 (en) 2008-12-18
EA018826B1 (ru) 2013-11-29
EP2170850A1 (en) 2010-04-07
CN101784535A (zh) 2010-07-21
MX2009013733A (es) 2010-04-22
WO2008152149A1 (en) 2008-12-18
MA31447B1 (fr) 2010-06-01
JP5346016B2 (ja) 2013-11-20
JP2010529977A (ja) 2010-09-02
NZ581933A (en) 2012-01-12
US20100249187A1 (en) 2010-09-30
US8809539B2 (en) 2014-08-19
AU2008263817A1 (en) 2008-12-18

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