WO2009115267A3 - Diaminopyrimidine als pflanzenschutzmittel - Google Patents

Diaminopyrimidine als pflanzenschutzmittel Download PDF

Info

Publication number
WO2009115267A3
WO2009115267A3 PCT/EP2009/001902 EP2009001902W WO2009115267A3 WO 2009115267 A3 WO2009115267 A3 WO 2009115267A3 EP 2009001902 W EP2009001902 W EP 2009001902W WO 2009115267 A3 WO2009115267 A3 WO 2009115267A3
Authority
WO
WIPO (PCT)
Prior art keywords
diaminopyrimidines
plant protection
protection agents
formula
description
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
PCT/EP2009/001902
Other languages
English (en)
French (fr)
Other versions
WO2009115267A2 (de
Inventor
Jörg Nico GREUL
Oliver Gaertzen
Stefan Hillebrand
Amos Mattes
Ulrike Wachendorff-Neumann
Peter Dahmen
Arnd Voerste
Peter Schreier
Ulrich Görgens
Heinz Kehne
Christian Paulitz
Hiroyuki Hadano
Oliver Guth
Angela Becker
Olga Malsam
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Bayer CropScience AG
Original Assignee
Bayer CropScience AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer CropScience AG filed Critical Bayer CropScience AG
Priority to EA201001499A priority Critical patent/EA201001499A1/ru
Priority to EP09721756A priority patent/EP2268144A2/de
Priority to CN2009801181393A priority patent/CN102123591A/zh
Priority to MX2010009846A priority patent/MX2010009846A/es
Priority to US12/933,600 priority patent/US20110105472A1/en
Priority to JP2011500099A priority patent/JP2011519822A/ja
Publication of WO2009115267A2 publication Critical patent/WO2009115267A2/de
Anticipated expiration legal-status Critical
Publication of WO2009115267A3 publication Critical patent/WO2009115267A3/de
Ceased legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48—Two nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D411/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen and sulfur atoms as the only ring hetero atoms
    • C07D411/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen and sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D411/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen and sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Verwendung von Diaminopyrimidinen der Formel (I) in welcher R1 bis R11a,b,c und X1, X2 die in der Beschreibung angegebenen Bedeutungen haben, sowie agrochemisch wirksamen Salzen davon als Pflanzenschutzmittel. Diaminopyrimidine der Formeln (Ia), (Ib) und (Ic) in welcher R8a, R8b, R8c,, und R1, R2, R3, R4, R5, R6, R7, R8, R9, R10, R11a,b,c und X1, X2 die in der Beschreibung angegebenen Bedeutungen haben, sowie agrochemisch wirksame Salze davon und deren Verwendung zur Bekämpfung von tierischen Schädlingen und/oder pflanzenpathogenen Schadpilzen.
PCT/EP2009/001902 2008-03-20 2009-03-16 Diaminopyrimidine als pflanzenschutzmittel Ceased WO2009115267A2 (de)

Priority Applications (6)

Application Number Priority Date Filing Date Title
EA201001499A EA201001499A1 (ru) 2008-03-20 2009-03-16 Диаминопиримидины в качестве средств защиты растений
EP09721756A EP2268144A2 (de) 2008-03-20 2009-03-16 Diaminopyrimidine als pflanzenschutzmittel
CN2009801181393A CN102123591A (zh) 2008-03-20 2009-03-16 作为植物保护剂的二氨基嘧啶
MX2010009846A MX2010009846A (es) 2008-03-20 2009-03-16 Diaminopirimidinas como agentes fitosanitarios.
US12/933,600 US20110105472A1 (en) 2008-03-20 2009-03-16 Diaminopyrimidines as crop protection agents
JP2011500099A JP2011519822A (ja) 2008-03-20 2009-03-16 植物保護剤としてのジアミノピリミジン

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP08102819 2008-03-20
EP08102819.3 2008-03-20

Publications (2)

Publication Number Publication Date
WO2009115267A2 WO2009115267A2 (de) 2009-09-24
WO2009115267A3 true WO2009115267A3 (de) 2010-11-18

Family

ID=41091271

Family Applications (1)

Application Number Title Priority Date Filing Date
PCT/EP2009/001902 Ceased WO2009115267A2 (de) 2008-03-20 2009-03-16 Diaminopyrimidine als pflanzenschutzmittel

Country Status (12)

Country Link
US (1) US20110105472A1 (de)
EP (1) EP2268144A2 (de)
JP (1) JP2011519822A (de)
KR (1) KR20100134048A (de)
CN (1) CN102123591A (de)
AR (1) AR070982A1 (de)
CL (1) CL2009000600A1 (de)
CO (1) CO6280578A2 (de)
EA (1) EA201001499A1 (de)
MX (1) MX2010009846A (de)
TW (1) TW201000011A (de)
WO (1) WO2009115267A2 (de)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8796296B2 (en) * 2011-11-29 2014-08-05 Genentech, Inc. Aminopyrimidine derivatives as LRRK2 modulators

Families Citing this family (38)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RU2008152195A (ru) * 2006-06-15 2010-07-20 БЕРИНГЕР ИНГЕЛЬХАЙМ ИНТЕРНАЦИОНАЛЬ ГмбХ (DE) 2-анилино-4-(гетероциклил)аминопиримидины, как ингибиторы протеинкиназы с-альфа
US9273077B2 (en) 2008-05-21 2016-03-01 Ariad Pharmaceuticals, Inc. Phosphorus derivatives as kinase inhibitors
MX353308B (es) 2008-05-21 2018-01-08 Ariad Pharma Inc Derivados fosforosos como inhibidores de cinasa.
US8338439B2 (en) 2008-06-27 2012-12-25 Celgene Avilomics Research, Inc. 2,4-disubstituted pyrimidines useful as kinase inhibitors
NZ603525A (en) 2008-06-27 2015-02-27 Celgene Avilomics Res Inc Pyrimidine based compound and uses thereof
US11351168B1 (en) 2008-06-27 2022-06-07 Celgene Car Llc 2,4-disubstituted pyrimidines useful as kinase inhibitors
BRPI0918062A2 (pt) * 2008-09-03 2015-08-11 Bayer Cropscience Ag Tienilaminopirimidinas como fungicidas
KR20110049905A (ko) * 2008-09-03 2011-05-12 바이엘 크롭사이언스 아게 4-알킬-치환된 디아미노피리미딘
US9908884B2 (en) 2009-05-05 2018-03-06 Dana-Farber Cancer Institute, Inc. EGFR inhibitors and methods of treating disorders
ES2577829T3 (es) 2010-06-04 2016-07-19 F. Hoffmann-La Roche Ag Derivados de aminopirimidina como moduladores de la LRRK2
MX336875B (es) 2010-08-10 2016-02-04 Celgene Avilomics Res Inc Sal de besilato de un inhibidor de tirosina cinasa de bruton (btk).
WO2012061303A1 (en) 2010-11-01 2012-05-10 Avila Therapeutics, Inc. Heteroaryl compounds and uses thereof
EP2635284B1 (de) 2010-11-01 2019-12-18 Celgene CAR LLC Heterocyclische verbindungen und ihre verwendung
NO2638031T3 (de) 2010-11-10 2018-03-10
WO2012064706A1 (en) 2010-11-10 2012-05-18 Avila Therapeutics, Inc. Mutant-selective egfr inhibitors and uses thereof
EP2704572B1 (de) 2011-05-04 2015-12-30 Ariad Pharmaceuticals, Inc. Verfahren zur hemmung der zellproliferation bei efgr-vermitteltem krebs
US9364476B2 (en) 2011-10-28 2016-06-14 Celgene Avilomics Research, Inc. Methods of treating a Bruton's Tyrosine Kinase disease or disorder
CA2866852C (en) 2012-03-15 2020-12-29 Celgene Avilomics Research, Inc. Solid forms of an epidermal growth factor receptor kinase inhibitor
BR112014022790B1 (pt) 2012-03-15 2022-04-19 Celgene Car Llc Sais de um inibidor de quinase de receptor de fator do crescimento epidermal, composição farmacêutica e usos do mesmo
WO2013169401A1 (en) 2012-05-05 2013-11-14 Ariad Pharmaceuticals, Inc. Compounds for inhibiting cell proliferation in egfr-driven cancers
US9126950B2 (en) 2012-12-21 2015-09-08 Celgene Avilomics Research, Inc. Heteroaryl compounds and uses thereof
MX2015009952A (es) 2013-02-08 2015-10-05 Celgene Avilomics Res Inc Inhibidores de cinasas reguladas por señales extracelulares (erk) y sus usos.
US9611283B1 (en) 2013-04-10 2017-04-04 Ariad Pharmaceuticals, Inc. Methods for inhibiting cell proliferation in ALK-driven cancers
US9492471B2 (en) 2013-08-27 2016-11-15 Celgene Avilomics Research, Inc. Methods of treating a disease or disorder associated with Bruton'S Tyrosine Kinase
WO2015054662A1 (en) 2013-10-10 2015-04-16 Eastern Virginia Medical School 4-((2-hydroxy-3-methoxybenzyl)amino) benzenesulfonamide derivatives as 12-lipoxygenase inhibitors
US9415049B2 (en) 2013-12-20 2016-08-16 Celgene Avilomics Research, Inc. Heteroaryl compounds and uses thereof
US9556126B2 (en) 2013-12-20 2017-01-31 Signal Pharmaceuticals, Llc Substituted diaminopyrimidyl compounds, compositions thereof, and methods of treatment therewith
EP3144292B1 (de) * 2014-04-14 2020-08-26 Shanghai Haiyan Pharmaceutical Technology Co., Ltd 2,3,4,6-tetrasubstituierte benzol-1,5-diamin-derivate, herstellungsverfahren dafür und medizinische verwendung davon
EP3179858B1 (de) 2014-08-13 2019-05-15 Celgene Car Llc Formen und zusammensetzungen eines erk-inhibitors
EP3319968A1 (de) 2015-07-06 2018-05-16 Rodin Therapeutics, Inc. Heterobicyclische n-aminophenyl-amide als inhibitoren der histondeacetylase
WO2017007756A1 (en) 2015-07-06 2017-01-12 Rodin Therapeutics, Inc Hetero-halo inhibitors of histone deacetylase
HUE057849T2 (hu) 2017-01-11 2022-06-28 Alkermes Inc Hiszton deacetiláz biciklusos gátlói
LT3664802T (lt) 2017-08-07 2022-06-27 Alkermes, Inc. Bicikliniai histonų deacetilazės inhibitoriai
EP3717479B1 (de) * 2017-11-29 2023-07-05 Syngenta Participations AG Mikrobiozide thiazolderivate
CN108299416A (zh) * 2018-04-14 2018-07-20 张汝伟 一种乙酰乳酸合成酶抑制剂及其在除草剂中的应用
CN110759898B (zh) * 2018-07-26 2022-12-13 南开大学 Hyrtinadine类生物碱及其衍生物在防治植物病毒病菌病中的应用
WO2020193474A1 (de) 2019-03-27 2020-10-01 Bayer Aktiengesellschaft Substituierte 2-heteroarylaminobenzole sowie deren salze und ihre verwendung als herbizide wirkstoffe
CN111830158B (zh) * 2020-07-17 2022-04-01 大连美创药业有限公司 一种合成艾地骨化醇中间体的液相色谱检测方法

Citations (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE4029650A1 (de) * 1990-09-19 1992-03-26 Hoechst Ag 2-anilino-pyrimidine, verfahren zu ihrer herstellung, sie enthaltene mittel und ihre verwendung als fungizide
WO2004056807A1 (en) * 2002-12-20 2004-07-08 Pfizer Products Inc. Pyrimidine derivatives for the treatment of abnormal cell growth
WO2005111022A1 (en) * 2004-05-14 2005-11-24 Pfizer Products Inc. Pyrimidines derivatives for the treatment of abnormal cell growth
WO2007132010A1 (de) * 2006-05-15 2007-11-22 Boehringer Ingelheim International Gmbh 2, 4 -diamino pyrimidine als inhibitoren von zellzykluskinasen

Patent Citations (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE4029650A1 (de) * 1990-09-19 1992-03-26 Hoechst Ag 2-anilino-pyrimidine, verfahren zu ihrer herstellung, sie enthaltene mittel und ihre verwendung als fungizide
WO2004056807A1 (en) * 2002-12-20 2004-07-08 Pfizer Products Inc. Pyrimidine derivatives for the treatment of abnormal cell growth
WO2005111022A1 (en) * 2004-05-14 2005-11-24 Pfizer Products Inc. Pyrimidines derivatives for the treatment of abnormal cell growth
WO2007132010A1 (de) * 2006-05-15 2007-11-22 Boehringer Ingelheim International Gmbh 2, 4 -diamino pyrimidine als inhibitoren von zellzykluskinasen

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8796296B2 (en) * 2011-11-29 2014-08-05 Genentech, Inc. Aminopyrimidine derivatives as LRRK2 modulators

Also Published As

Publication number Publication date
CO6280578A2 (es) 2011-05-20
CL2009000600A1 (es) 2010-05-07
US20110105472A1 (en) 2011-05-05
CN102123591A (zh) 2011-07-13
EP2268144A2 (de) 2011-01-05
TW201000011A (en) 2010-01-01
MX2010009846A (es) 2010-10-05
JP2011519822A (ja) 2011-07-14
EA201001499A1 (ru) 2011-04-29
KR20100134048A (ko) 2010-12-22
WO2009115267A2 (de) 2009-09-24
AR070982A1 (es) 2010-05-19

Similar Documents

Publication Publication Date Title
WO2009115267A3 (de) Diaminopyrimidine als pflanzenschutzmittel
WO2009132785A8 (de) Thiazol-4-carbonsäureester und thioester als pflanzenschutzmittel
WO2010069502A8 (de) Tetrazolsubstituierte anthranilsäureamide als pestizide
WO2009027820A3 (en) Substituted-quinoxaline-type-piperidine compounds and the uses thereof
WO2010025863A3 (de) 4-alkyl-substituierte diaminopyrimidine
WO2007093529A3 (de) Heteroaroylsubstituierte alanine
UA96314C2 (ru) Замещенные 1-(3-пиридинил)пиразол-4-илуксусные кислоты и их применение в качестве гербицидов и регуляторов роста растений
WO2009115557A3 (en) Fungicide hydroximoyl-tetrazole derivatives
WO2012082580A3 (en) Fungicidal azocyclic amides
WO2009098223A3 (en) Plant health composition
TW200734314A (en) Piperazine compounds having herbicidal action
MX2011009732A (es) Combinaciones de principios activos sinergicas.
MX2009007345A (es) Compuestos con (fenil sustituido), con restos de propenal, sus derivados, actividad biologica y uso del mismo.
MX2011013706A (es) Derivados de tiazoliliperidina como fungicidas.
ZA200809714B (en) Synergistic active ingredient combinations
WO2011039444A3 (fr) Composition, utilisation et procédé de conservation
WO2009048752A3 (en) Insecticidal substituted azinyl derivatives
WO2014102592A3 (en) Oxime/substituted quinoxaline-type piperidine compounds and uses thereof
WO2010083955A3 (de) Verwendung von enaminocarbonylverbindungen zur bekämpfung von durch insekten übertragenen virosen
WO2008087182A3 (de) Fungizide mischungen aus 1-methylpyrazol-4-ylcarbonsäureaniliden und azolopyrimidinylaminen
WO2014020405A8 (en) Cyclic urea- or lactam-substituted quinoxaline-type piperidine compounds and the uses thereof
TW200833248A (en) Bisoximes as fungicides
UA83314C2 (ru) 2-(пиридин-2-ил)пиримидиновые соединения и их применение для борьбы с вредными грибами
EP2135622A3 (de) Zusammensetzungen zur Bereitstellung eines schmerzlindernden Effekts auf der Haut
TW200800993A (en) Organic compounds

Legal Events

Date Code Title Description
WWE Wipo information: entry into national phase

Ref document number: 200980118139.3

Country of ref document: CN

WWE Wipo information: entry into national phase

Ref document number: 2009721756

Country of ref document: EP

WWE Wipo information: entry into national phase

Ref document number: MX/A/2010/009846

Country of ref document: MX

WWE Wipo information: entry into national phase

Ref document number: 10111169

Country of ref document: CO

WWE Wipo information: entry into national phase

Ref document number: 2011500099

Country of ref document: JP

NENP Non-entry into the national phase

Ref country code: DE

WWE Wipo information: entry into national phase

Ref document number: 201001499

Country of ref document: EA

ENP Entry into the national phase

Ref document number: 20107023278

Country of ref document: KR

Kind code of ref document: A

WWE Wipo information: entry into national phase

Ref document number: 7365/DELNP/2010

Country of ref document: IN

WWE Wipo information: entry into national phase

Ref document number: 12933600

Country of ref document: US