ZA200203295B - Sodium-hydrogen exchanger type 1 inhibitor crystals. - Google Patents

Sodium-hydrogen exchanger type 1 inhibitor crystals.

Info

Publication number
ZA200203295B
ZA200203295B ZA200203295A ZA200203295A ZA200203295B ZA 200203295 B ZA200203295 B ZA 200203295B ZA 200203295 A ZA200203295 A ZA 200203295A ZA 200203295 A ZA200203295 A ZA 200203295A ZA 200203295 B ZA200203295 B ZA 200203295B
Authority
ZA
South Africa
Prior art keywords
sodium
exchanger type
hydrogen exchanger
inhibitor crystals
crystals
Prior art date
Application number
ZA200203295A
Other languages
English (en)
Inventor
Lyle Robinson Brostrom
Terrence Joseph Connolly
Zheng Jane Li
Susan Lee Orrill
Bharat Kiritkumar Shah
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of ZA200203295B publication Critical patent/ZA200203295B/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/08Drugs for disorders of the urinary system of the prostate
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00Drugs for disorders of the muscular or neuromuscular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P39/00General protective or antinoxious agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P41/00Drugs used in surgical methods, e.g. surgery adjuvants for preventing adhesion or for vitreum substitution
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Diabetes (AREA)
  • Urology & Nephrology (AREA)
  • Emergency Medicine (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Endocrinology (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Toxicology (AREA)
  • Vascular Medicine (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pulmonology (AREA)
  • Neurology (AREA)
  • Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Treatment Of Water By Ion Exchange (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
ZA200203295A 1999-10-29 2002-04-25 Sodium-hydrogen exchanger type 1 inhibitor crystals. ZA200203295B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US16237499P 1999-10-29 1999-10-29

Publications (1)

Publication Number Publication Date
ZA200203295B true ZA200203295B (en) 2003-06-25

Family

ID=22585355

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA200203295A ZA200203295B (en) 1999-10-29 2002-04-25 Sodium-hydrogen exchanger type 1 inhibitor crystals.

Country Status (44)

Country Link
EP (1) EP1224179B1 (fr)
JP (1) JP2003512455A (fr)
KR (1) KR100464526B1 (fr)
CN (2) CN1205205C (fr)
AP (1) AP2002002493A0 (fr)
AR (1) AR029402A1 (fr)
AT (1) ATE271047T1 (fr)
AU (1) AU778573B2 (fr)
BG (1) BG106729A (fr)
BR (1) BR0015275A (fr)
CA (1) CA2389020A1 (fr)
CO (1) CO5271714A1 (fr)
CZ (1) CZ20021332A3 (fr)
DE (1) DE60012208T2 (fr)
DK (1) DK1224179T3 (fr)
DZ (1) DZ3463A1 (fr)
EA (1) EA004937B1 (fr)
EE (1) EE200200227A (fr)
ES (1) ES2222923T3 (fr)
GE (1) GEP20043222B (fr)
GT (1) GT200000180A (fr)
HK (1) HK1048472B (fr)
HR (1) HRP20020366B1 (fr)
HU (1) HUP0204009A3 (fr)
IL (1) IL148581A0 (fr)
IS (1) IS6302A (fr)
MA (1) MA26840A1 (fr)
MX (1) MXPA02004358A (fr)
NO (1) NO20021821L (fr)
NZ (1) NZ517738A (fr)
OA (1) OA12080A (fr)
PA (1) PA8505501A1 (fr)
PE (1) PE20010764A1 (fr)
PL (1) PL354869A1 (fr)
PT (1) PT1224179E (fr)
SI (1) SI1224179T1 (fr)
SK (1) SK5312002A3 (fr)
SV (1) SV2002000209A (fr)
TN (1) TNSN00210A1 (fr)
TR (1) TR200201167T2 (fr)
UA (1) UA72002C2 (fr)
WO (1) WO2001030759A2 (fr)
YU (1) YU31502A (fr)
ZA (1) ZA200203295B (fr)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6441176B1 (en) 1999-10-29 2002-08-27 Pfizer Inc. Method for preparing sodium-hydrogen exchanger type 1 inhibitor
CN1479737A (zh) * 2001-01-31 2004-03-03 �Ʒ� 钠-质子交换蛋白1型抑制剂的乙醇盐
BR0307195A (pt) * 2002-01-30 2004-11-03 Pfizer Prod Inc Composições farmacêuticas de mesilato de zoniporide e processos para melhorar a solubilidade do zoniporide
MXPA04008646A (es) * 2002-05-02 2004-12-06 Pfizer Prod Inc Tratamiento para la diabetes y complicaciones diabeticas con inhibidores del nhe-1.

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PT1056729E (pt) * 1998-02-27 2005-04-29 Pfizer Prod Inc Derivados de n-[ciclo di- ou tri-aza di-insaturado de cinco membros substituido) carbonil] guanidina para o tratamento de isquemia

Also Published As

Publication number Publication date
DE60012208D1 (de) 2004-08-19
CA2389020A1 (fr) 2001-05-03
HRP20020366B1 (en) 2005-04-30
AP2002002493A0 (en) 2002-06-30
NO20021821D0 (no) 2002-04-18
DZ3463A1 (fr) 2001-05-03
BR0015275A (pt) 2002-07-16
PL354869A1 (en) 2004-03-08
HK1048472B (zh) 2005-09-16
NZ517738A (en) 2005-06-24
ES2222923T3 (es) 2005-02-16
IL148581A0 (en) 2002-09-12
BG106729A (bg) 2002-12-29
IS6302A (is) 2002-03-15
OA12080A (en) 2003-08-25
CZ20021332A3 (cs) 2002-10-16
HUP0204009A2 (hu) 2003-03-28
CN1384829A (zh) 2002-12-11
KR20020040918A (ko) 2002-05-30
EA004937B1 (ru) 2004-10-28
EP1224179B1 (fr) 2004-07-14
TNSN00210A1 (fr) 2005-11-10
GT200000180A (es) 2002-04-11
EP1224179A2 (fr) 2002-07-24
HUP0204009A3 (en) 2004-07-28
CO5271714A1 (es) 2003-04-30
HK1048472A1 (en) 2003-04-04
SV2002000209A (es) 2002-07-16
YU31502A (sh) 2004-12-31
PE20010764A1 (es) 2001-07-23
AU7441500A (en) 2001-05-08
GEP20043222B (en) 2004-04-26
ATE271047T1 (de) 2004-07-15
DK1224179T3 (da) 2004-10-25
NO20021821L (no) 2002-04-18
AU778573B2 (en) 2004-12-09
JP2003512455A (ja) 2003-04-02
EA200200416A1 (ru) 2002-10-31
CN1636991A (zh) 2005-07-13
UA72002C2 (en) 2005-01-17
CN1205205C (zh) 2005-06-08
KR100464526B1 (ko) 2005-01-03
AR029402A1 (es) 2003-06-25
MA26840A1 (fr) 2004-12-20
DE60012208T2 (de) 2005-07-21
SK5312002A3 (en) 2003-01-09
EE200200227A (et) 2003-06-16
PA8505501A1 (es) 2003-09-05
HRP20020366A2 (en) 2004-02-29
WO2001030759A2 (fr) 2001-05-03
WO2001030759A3 (fr) 2001-09-13
MXPA02004358A (es) 2002-11-07
SI1224179T1 (en) 2004-10-31
TR200201167T2 (tr) 2002-08-21
PT1224179E (pt) 2004-10-29

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