ZA200305659B - Sulfamidothienopyrimidines and the use of the same as phosphodiesterase V inhibitors. - Google Patents

Sulfamidothienopyrimidines and the use of the same as phosphodiesterase V inhibitors. Download PDF

Info

Publication number: ZA200305659B
Authority: ZA; South Africa
Prior art keywords: formula; treatment; diseases; compound; substance
Prior art date: 2000-12-23

Application number

ZA200305659A

Other languages

English (en)

Inventor

Hans-Michael Eggenweiler

Pierre Schelling

Maria Christadler

Harry Schwartz

Norbert Beier

Original Assignee

Merck Patent Gmbh

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-12-23

Filing date

2003-07-22

Publication date

2004-08-27

2003-07-22 Application filed by Merck Patent Gmbh filed Critical Merck Patent Gmbh

2004-08-27 Publication of ZA200305659B publication Critical patent/ZA200305659B/en

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Classifications

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Urology & Nephrology (AREA)
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Reproductive Health (AREA)
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Ophthalmology & Optometry (AREA)
Vascular Medicine (AREA)
Rheumatology (AREA)
Hospice & Palliative Care (AREA)
Immunology (AREA)
Gynecology & Obstetrics (AREA)
Gastroenterology & Hepatology (AREA)
Physical Education & Sports Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

ZA200305659A 2000-12-23 2003-07-22 Sulfamidothienopyrimidines and the use of the same as phosphodiesterase V inhibitors. ZA200305659B (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
DE10064994A DE10064994A1 (de)	2000-12-23	2000-12-23	Sulfamidothienopyrimidine

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ZA200305659B true ZA200305659B (en)	2004-08-27

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ZA200305659A ZA200305659B (en)	2000-12-23	2003-07-22	Sulfamidothienopyrimidines and the use of the same as phosphodiesterase V inhibitors.

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US (1)	US7019013B2 (cs)
EP (1)	EP1353927B1 (cs)
JP (1)	JP4550361B2 (cs)
KR (1)	KR20030062438A (cs)
CN (1)	CN1483035A (cs)
AR (1)	AR035524A1 (cs)
AT (1)	ATE302781T1 (cs)
BR (1)	BR0115996A (cs)
CA (1)	CA2432582C (cs)
CZ (1)	CZ20031815A3 (cs)
DE (2)	DE10064994A1 (cs)
ES (1)	ES2247007T3 (cs)
HU (1)	HUP0302515A3 (cs)
MX (1)	MXPA03005714A (cs)
PL (1)	PL361733A1 (cs)
RU (1)	RU2003122189A (cs)
SK (1)	SK8432003A3 (cs)
WO (1)	WO2002051848A2 (cs)
ZA (1)	ZA200305659B (cs)

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CN101100472A (zh) *	2001-04-30	2008-01-09	美国拜尔公司	4-氨基-5,6-取代的噻吩并[2,3-d]嘧啶化合物及其应用
CN101163706A (zh) *	2005-04-21	2008-04-16	贝林格尔·英格海姆国际有限公司	用于治疗炎性疾病的二氢噻吩并嘧啶
EP1847543A1 (de)	2006-04-19	2007-10-24	Boehringer Ingelheim Pharma GmbH & Co. KG	Dihydrothienopyrimidine zur Behandlung von entzündlichen Erkrankungen
US8080549B2 (en) *	2007-01-12	2011-12-20	Concert Pharmaceuticals, Inc.	Endothelin receptor antagonists
US8071596B2 (en)	2007-01-12	2011-12-06	Concert Pharmaceuticals, Inc.	Endothelin receptor antagonists
JP2010516731A (ja)	2007-01-24	2010-05-20	グラクソグループリミテッド	２−メトキシ−５−（５−トリフルオロメチル−テトラゾール−１−イル）−ベンジル］−（２ｓ−フェニル−ピペリジン−３ｓ−イル）−アミンを含む医薬組成物
CN104069112A (zh) *	2007-10-19	2014-10-01	贝林格尔.英格海姆国际有限公司	取代的哌啶子基-二氢噻吩并嘧啶
CA2702524A1 (en)	2007-10-19	2009-04-23	Boehringer Ingelheim International Gmbh	Heterocycle-substituted piperazino-dihydrothienopyrimidines
CA2702518A1 (en)	2007-10-19	2009-04-23	Boehringer Ingelheim International Gmbh	New piperazino-dihydrothienopyrimidine derivatives
EP2595993B1 (en)	2010-07-23	2018-04-18	President and Fellows of Harvard College	Tricyclic proteasome activity enhancing compounds
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2000
- 2000-12-23 DE DE10064994A patent/DE10064994A1/de not_active Withdrawn
2001
- 2001-12-03 JP JP2002552942A patent/JP4550361B2/ja not_active Expired - Fee Related
- 2001-12-03 WO PCT/EP2001/014102 patent/WO2002051848A2/de not_active Ceased
- 2001-12-03 CA CA2432582A patent/CA2432582C/en not_active Expired - Fee Related
- 2001-12-03 CZ CZ20031815A patent/CZ20031815A3/cs unknown
- 2001-12-03 US US10/451,183 patent/US7019013B2/en not_active Expired - Fee Related
- 2001-12-03 RU RU2003122189/04A patent/RU2003122189A/ru not_active Application Discontinuation
- 2001-12-03 BR BR0115996-8A patent/BR0115996A/pt not_active Application Discontinuation
- 2001-12-03 PL PL01361733A patent/PL361733A1/xx unknown
- 2001-12-03 EP EP01271992A patent/EP1353927B1/de not_active Expired - Lifetime
- 2001-12-03 SK SK843-2003A patent/SK8432003A3/sk unknown
- 2001-12-03 KR KR10-2003-7008265A patent/KR20030062438A/ko not_active Withdrawn
- 2001-12-03 MX MXPA03005714A patent/MXPA03005714A/es not_active Application Discontinuation
- 2001-12-03 ES ES01271992T patent/ES2247007T3/es not_active Expired - Lifetime
- 2001-12-03 DE DE50107230T patent/DE50107230D1/de not_active Expired - Lifetime
- 2001-12-03 AT AT01271992T patent/ATE302781T1/de not_active IP Right Cessation
- 2001-12-03 HU HU0302515A patent/HUP0302515A3/hu unknown
- 2001-12-03 CN CNA018212190A patent/CN1483035A/zh active Pending
- 2001-12-19 AR ARP010105889A patent/AR035524A1/es not_active Application Discontinuation
2003
- 2003-07-22 ZA ZA200305659A patent/ZA200305659B/en unknown

Also Published As

Publication number	Publication date
EP1353927A2 (de)	2003-10-22
CA2432582A1 (en)	2002-07-04
MXPA03005714A (es)	2003-10-06
KR20030062438A (ko)	2003-07-25
JP4550361B2 (ja)	2010-09-22
AR035524A1 (es)	2004-06-02
CN1483035A (zh)	2004-03-17
WO2002051848A3 (de)	2002-10-24
CA2432582C (en)	2011-01-25
SK8432003A3 (en)	2003-10-07
DE10064994A1 (de)	2002-07-04
US7019013B2 (en)	2006-03-28
DE50107230D1 (de)	2005-09-29
HUP0302515A3 (en)	2005-06-28
CZ20031815A3 (cs)	2003-10-15
JP2004516329A (ja)	2004-06-03
WO2002051848A2 (de)	2002-07-04
US20040063943A1 (en)	2004-04-01
ATE302781T1 (de)	2005-09-15
RU2003122189A (ru)	2004-12-27
ES2247007T3 (es)	2006-03-01
EP1353927B1 (de)	2005-08-24
PL361733A1 (en)	2004-10-04
HUP0302515A2 (hu)	2003-11-28
BR0115996A (pt)	2004-01-06

Publication	Publication Date	Title
US20040063730A1 (en)	2004-04-01	Pharmacuetical formulation comprising puyrazolo[4,-3-d]pyrimidines and antithrombotics, calcium antagonists, or prostaglandins or prostaglandin derivatives
US20040034040A1 (en)	2004-02-19	Use of thienopyrimidines
CA2432582C (en)	2011-01-25	Sulfamidothienopyrimidines
AU742433B2 (en)	2002-01-03	Thienopyrimidines
AU2002362806B2 (en)	2008-09-18	Pyrimidine derivatives
US20040072846A1 (en)	2004-04-15	Pharmaceutical formulation containing thienopyrimidines and antithrombotics, calcium antagonists, prostaglandins or prostaglandin derivatives
JP2004525890A (ja)	2004-08-26	ピラゾロ［４，３−ｄ］ピリミジンおよびエンドセリンレセプターアンタゴニストまたはチエノピリミジンおよびエンドセリンレセプターアンタゴニストを含む医薬製剤
CA2429645A1 (en)	2002-05-30	Use of pyrazolo[4,3-d]pyrimidines
US20040058940A1 (en)	2004-03-25	Pharmaceutical formulation comprising thienopyrimidines and antithrombotics, calcium antagonists, prostaglandins or prostaglandin derivatives (2)
ZA200302513B (en)	2004-08-24	Thienopyrimidines.
ZA200306730B (en)	2004-09-01	Pharmaceutical formulation containing pyrazolo[4,3-d] pyrimidine and nitrates or thienopyrimidines and nitrates.
ZA200305548B (en)	2005-01-26	Pharmaceutical formulation containing thienopyrimidines and antithrombotics calcium antagonists prostaglandins or prostaglandin derivatives (2)
ZA200305542B (en)	2005-01-26	Pharmaceutical formulation containing pyrazole [4,3-d]pymidines and antithrombotic agents calcium antagonists prostaglandins or prostaglandin derivatives