ZA200406548B - Process for the preparation of morpholine derivatives and intermediates therefor. - Google Patents
Process for the preparation of morpholine derivatives and intermediates therefor. Download PDFInfo
- Publication number
- ZA200406548B ZA200406548B ZA200406548A ZA200406548A ZA200406548B ZA 200406548 B ZA200406548 B ZA 200406548B ZA 200406548 A ZA200406548 A ZA 200406548A ZA 200406548 A ZA200406548 A ZA 200406548A ZA 200406548 B ZA200406548 B ZA 200406548B
- Authority
- ZA
- South Africa
- Prior art keywords
- formula
- alkyl
- compound
- aryl
- heteroaryl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/44—Iso-indoles; Hydrogenated iso-indoles
- C07D209/48—Iso-indoles; Hydrogenated iso-indoles with oxygen atoms in positions 1 and 3, e.g. phthalimide
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D265/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
- C07D265/28—1,4-Oxazines; Hydrogenated 1,4-oxazines
- C07D265/30—1,4-Oxazines; Hydrogenated 1,4-oxazines not condensed with other rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB0207450.8A GB0207450D0 (en) | 2002-03-28 | 2002-03-28 | Novel compounds |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ZA200406548B true ZA200406548B (en) | 2005-09-19 |
Family
ID=9933999
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ZA200406548A ZA200406548B (en) | 2002-03-28 | 2004-08-17 | Process for the preparation of morpholine derivatives and intermediates therefor. |
Country Status (20)
| Country | Link |
|---|---|
| EP (1) | EP1487809B1 (de) |
| JP (1) | JP2005532281A (de) |
| KR (1) | KR20050008664A (de) |
| CN (1) | CN1642928A (de) |
| AR (1) | AR039178A1 (de) |
| AT (1) | ATE383349T1 (de) |
| AU (1) | AU2003226760A1 (de) |
| BR (1) | BR0308720A (de) |
| CA (1) | CA2479819A1 (de) |
| DE (1) | DE60318559T2 (de) |
| ES (1) | ES2298539T3 (de) |
| GB (1) | GB0207450D0 (de) |
| IS (1) | IS7401A (de) |
| MX (1) | MXPA04009457A (de) |
| NO (1) | NO20044036L (de) |
| PL (1) | PL373972A1 (de) |
| RU (1) | RU2004125289A (de) |
| TW (1) | TW200401772A (de) |
| WO (1) | WO2003082835A1 (de) |
| ZA (1) | ZA200406548B (de) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP1992628A1 (de) | 2007-05-18 | 2008-11-19 | Glaxo Group Limited | Derivate und Analoge von N-Ethylquinolonen und N-Ethylazaquinolonen |
| US10702521B2 (en) | 2014-08-22 | 2020-07-07 | Glaxosmithkline Intellectual Property Development Limited | Methods for treating neisseria gonorrhoeae infection with substituted 1,2-dihydro-2A,5,8A-triazaacenaphthylene-3,8-diones |
| WO2019168874A1 (en) | 2018-02-27 | 2019-09-06 | The Research Foundation For The State University Of New York | Difluoromethoxylation and trifluoromethoxylation compositions and methods for synthesizing same |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE2447732A1 (de) * | 1974-10-07 | 1976-04-08 | Wuelfing J A Fa | Neue morpholinverbindungen, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel |
| KR20010014105A (ko) * | 1997-06-23 | 2001-02-26 | 가마쿠라 아키오 | 헬리코박터 감염에 기인한 질환의 예방 또는 치료제 |
| BR0114321A (pt) * | 2000-09-29 | 2003-07-01 | Glaxo Group Ltd | Composto, composição farmacêutica, uso de um composto, método de tratamento ou profilaxia de doenças inflamatórias, e, processo para preparar um composto |
-
2002
- 2002-03-28 GB GBGB0207450.8A patent/GB0207450D0/en not_active Ceased
-
2003
- 2003-03-26 TW TW092106783A patent/TW200401772A/zh unknown
- 2003-03-27 ES ES03745297T patent/ES2298539T3/es not_active Expired - Lifetime
- 2003-03-27 DE DE60318559T patent/DE60318559T2/de not_active Expired - Lifetime
- 2003-03-27 CN CNA038073862A patent/CN1642928A/zh active Pending
- 2003-03-27 PL PL03373972A patent/PL373972A1/xx not_active Application Discontinuation
- 2003-03-27 MX MXPA04009457A patent/MXPA04009457A/es not_active Application Discontinuation
- 2003-03-27 JP JP2003580303A patent/JP2005532281A/ja active Pending
- 2003-03-27 KR KR10-2004-7015446A patent/KR20050008664A/ko not_active Withdrawn
- 2003-03-27 EP EP03745297A patent/EP1487809B1/de not_active Expired - Lifetime
- 2003-03-27 AU AU2003226760A patent/AU2003226760A1/en not_active Abandoned
- 2003-03-27 AR ARP030101091A patent/AR039178A1/es unknown
- 2003-03-27 CA CA002479819A patent/CA2479819A1/en not_active Abandoned
- 2003-03-27 BR BR0308720-4A patent/BR0308720A/pt not_active Application Discontinuation
- 2003-03-27 WO PCT/EP2003/003343 patent/WO2003082835A1/en not_active Ceased
- 2003-03-27 RU RU2004125289/04A patent/RU2004125289A/ru not_active Application Discontinuation
- 2003-03-27 AT AT03745297T patent/ATE383349T1/de not_active IP Right Cessation
-
2004
- 2004-08-12 IS IS7401A patent/IS7401A/is unknown
- 2004-08-17 ZA ZA200406548A patent/ZA200406548B/en unknown
- 2004-09-24 NO NO20044036A patent/NO20044036L/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| RU2004125289A (ru) | 2005-06-27 |
| DE60318559D1 (de) | 2008-02-21 |
| EP1487809B1 (de) | 2008-01-09 |
| BR0308720A (pt) | 2005-01-04 |
| PL373972A1 (en) | 2005-09-19 |
| CA2479819A1 (en) | 2003-10-09 |
| JP2005532281A (ja) | 2005-10-27 |
| DE60318559T2 (de) | 2009-01-08 |
| EP1487809A1 (de) | 2004-12-22 |
| IS7401A (is) | 2004-08-12 |
| GB0207450D0 (en) | 2002-05-08 |
| TW200401772A (en) | 2004-02-01 |
| NO20044036L (no) | 2004-09-29 |
| AU2003226760A1 (en) | 2003-10-13 |
| ES2298539T3 (es) | 2008-05-16 |
| ATE383349T1 (de) | 2008-01-15 |
| WO2003082835A1 (en) | 2003-10-09 |
| MXPA04009457A (es) | 2005-01-25 |
| KR20050008664A (ko) | 2005-01-21 |
| CN1642928A (zh) | 2005-07-20 |
| AR039178A1 (es) | 2005-02-09 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| JP6777398B2 (ja) | 薬剤を調製するための方法と中間体 | |
| CA2530159C (en) | N-pyrrolidin-3-yl-amide derivatives as serotonin and noradrenaline re-uptake inhibitors | |
| FR2921657A1 (fr) | Derives de nicotinamide, leur preparation et leur application en therapeutique | |
| JP2020524158A (ja) | Ｓｓａｏ阻害剤 | |
| MXPA04002653A (es) | Metodo para preparar compuestos de pirimidinona y sales farmaceuticamente aceptables del mismo. | |
| CN118047774A (zh) | 一种制备非奈利酮及其中间体的方法 | |
| US7915427B2 (en) | Process for producing aminoacetyl pyrrolidine carbonitrile derivative and intermediate for production thereof | |
| ZA200406548B (en) | Process for the preparation of morpholine derivatives and intermediates therefor. | |
| Huang et al. | A facile approach to trans-4, 5-pyrrolidine lactam and application in the synthesis of nemonapride and streptopyrrolidine | |
| JP2022528690A (ja) | （３ｒ，４ｒ）－１－ベンジル－ｎ，４－ジメチルピペリジン－３－アミンまたはその塩の製造方法、およびそれを使用したトファシチニブの製造方法 | |
| Nagamine et al. | A New Chiral Synthesis of a Bicyclic Enedlone Containing a Seven-Membered Ring Mediated by a Combination of Chiral Amine and Bronsted Acid | |
| AU2006277710A1 (en) | Preparation of diazapentalene derivatives via epoxydation of dihydropyrroles | |
| FR2943675A1 (fr) | Composes anticancereux, leur preparation et leur application en therapeutique | |
| Chai et al. | Urazole synthesis. Part 2: facilitating N4 substitution | |
| Chen et al. | Synthesis, Characterization and Suppression of Impurities during Optimization of Dabigatran Etexilate | |
| EP2058300A1 (de) | Bernsteinsäurediesterderivat, verfahren zu dessen herstellung und verwendung des derivats bei der herstellung einer pharmazeutischen zubereitung | |
| Xu et al. | Impact of atropisomerism on a non-steroidal glucocorticoid receptor agonist | |
| OA13178A (en) | N-pyrrolidin-3-yl-amide derivatives as serotonin and noradrenaline re-uptake inhibitors. | |
| Zhang et al. | A facile and efficient synthesis of d3‐labelled Reyataz™ | |
| FR2943670A1 (fr) | Derives anticancereux,leur preparation et leur application en therapeutique | |
| KR20220011669A (ko) | Btk 억제제 제조를 위한 방법 및 중간체 | |
| WO2010092286A1 (fr) | Derives de n-[(2-aza-bicyclo[2.1.1]hex-1-yl]-aryl-methyl]-benzamide, leur preparation et leur application en therapeutique |