ZA837850B - New cephalosporins and a process for their preparation - Google Patents

New cephalosporins and a process for their preparation

Info

Publication number: ZA837850B
Authority: ZA; South Africa
Prior art keywords: preparation; new cephalosporins; alkyl; cephalosporins; new
Prior art date: 1982-10-23

Application number

ZA837850A

Other languages

English (en)

Inventor

Guenther Kinast

Michael Boberg

Karl Georg Metzger

Hans Joachim Zeiler

Original Assignee

Bayer Ag

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1982-10-23

Filing date

1983-10-21

Publication date

1984-06-27

1983-10-21 Application filed by Bayer Ag filed Critical Bayer Ag

1984-06-27 Publication of ZA837850B publication Critical patent/ZA837850B/xx

Links

229930186147 Cephalosporin Natural products 0.000 title abstract 2
229940124587 cephalosporin Drugs 0.000 title abstract 2
150000001780 cephalosporins Chemical class 0.000 title abstract 2
125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 2
125000004178 (C1-C4) alkyl group Chemical group 0.000 abstract 1
125000004169 (C1-C6) alkyl group Chemical group 0.000 abstract 1
WKBOTKDWSSQWDR-UHFFFAOYSA-N Bromine atom Chemical compound [Br] WKBOTKDWSSQWDR-UHFFFAOYSA-N 0.000 abstract 1
ZAMOUSCENKQFHK-UHFFFAOYSA-N Chlorine atom Chemical compound [Cl] ZAMOUSCENKQFHK-UHFFFAOYSA-N 0.000 abstract 1
GDTBXPJZTBHREO-UHFFFAOYSA-N bromine Substances BrBr GDTBXPJZTBHREO-UHFFFAOYSA-N 0.000 abstract 1
229910052794 bromium Inorganic materials 0.000 abstract 1
125000003917 carbamoyl group Chemical group [H]N([H])C(*)=O 0.000 abstract 1
229910052801 chlorine Inorganic materials 0.000 abstract 1
239000000460 chlorine Substances 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C07D501/14—Compounds having a nitrogen atom directly attached in position 7
- C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
- C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
- C07D501/24—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3
- C07D501/38—Methylene radicals, substituted by nitrogen atoms; Lactams thereof with the 2-carboxyl group; Methylene radicals substituted by nitrogen-containing hetero rings attached by the ring nitrogen atom; Quaternary compounds thereof
- C07D501/46—Methylene radicals, substituted by nitrogen atoms; Lactams thereof with the 2-carboxyl group; Methylene radicals substituted by nitrogen-containing hetero rings attached by the ring nitrogen atom; Quaternary compounds thereof with the 7-amino radical acylated by carboxylic acids containing hetero rings
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Life Sciences & Earth Sciences (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Communicable Diseases (AREA)
Pharmacology & Pharmacy (AREA)
Oncology (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Cephalosporin Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Saccharide Compounds (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

ZA837850A 1982-10-23 1983-10-21 New cephalosporins and a process for their preparation ZA837850B (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
DE19823239365 DE3239365A1 (de)	1982-10-23	1982-10-23	Neue cephalosporine und verfahren zu ihrer herstellung

Publications (1)

Publication Number	Publication Date
ZA837850B true ZA837850B (en)	1984-06-27

Family

ID=6176491

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
ZA837850A ZA837850B (en)	1982-10-23	1983-10-21	New cephalosporins and a process for their preparation

Country Status (19)

Country	Link
US (1)	US4489076A (da)
EP (1)	EP0107138B1 (da)
JP (1)	JPS5993086A (da)
KR (1)	KR840006487A (da)
AT (1)	ATE29498T1 (da)
AU (1)	AU556826B2 (da)
CA (1)	CA1208206A (da)
DE (2)	DE3239365A1 (da)
DK (1)	DK486183A (da)
ES (1)	ES526674A0 (da)
FI (1)	FI73689C (da)
GR (1)	GR79682B (da)
HU (1)	HU189763B (da)
IL (1)	IL70012A (da)
NO (1)	NO833644L (da)
NZ (1)	NZ206017A (da)
PH (3)	PH20918A (da)
PT (1)	PT77501B (da)
ZA (1)	ZA837850B (da)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE3300593A1 (de) *	1983-01-11	1984-07-12	Bayer Ag, 5090 Leverkusen	Neue cephalosporine und verfahren zu ihrer herstellung
DE3343208A1 (de) *	1983-11-30	1985-06-05	Bayer Ag, 5090 Leverkusen	Neue cephalosporine und verfahren zu ihrer herstellung
DE3418376A1 (de) *	1984-05-17	1985-11-21	Bayer Ag, 5090 Leverkusen	Zwischenprodukte sowie verfahren zur herstellung von zwischenprodukten fuer die synthese von cephalosporinen
DE3419012A1 (de) *	1984-05-22	1985-11-28	Bayer Ag, 5090 Leverkusen	Ss-lactamantibiotika, verfahren zu deren herstellung sowie ihre verwendung als arzneimittel oder wachstumsfoerderer in der tieraufzucht oder als antioxidantien
JP2501785B2 (ja) *	1984-07-09	1996-05-29	明治製菓株式会社	新規セフアロスポリン系化合物
AT397963B (de) *	1985-03-29	1994-08-25	Shionogi & Co	Verfahren zur herstellung von neuen 7 beta-(2-(2- amino-4-thiazolyl)-alkenoylamimo)-3-cephem-4- carbonsäureestern
AU580855B2 (en) *	1985-03-29	1989-02-02	Shionogi & Co., Ltd.	Alkeneamidocephalosporin esters
JP4554395B2 (ja)	2005-02-17	2010-09-29	浜松ホトニクス株式会社	光源装置
JP4589142B2 (ja)	2005-02-17	2010-12-01	浜松ホトニクス株式会社	光源装置

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
JPS4970990A (da) *	1973-09-29	1974-07-09
NZ176206A (en) *	1973-12-25	1978-03-06	Takeda Chemical Industries Ltd	Cephalosporins
DK154939C (da) *	1974-12-19	1989-06-12	Takeda Chemical Industries Ltd	Analogifremgangsmaade til fremstilling af thiazolylacetamido-cephemforbindelser eller farmaceutisk acceptable salte eller estere deraf
US4148997A (en) *	1977-11-07	1979-04-10	Yeda Research And Development Co., Ltd.	7-[Sulfomethyl)phenyl]acetamidocephalosporin derivatives
KR830000606B1 (ko) *	1978-05-26	1983-03-17	헤롤드 월터 마틴	세팔로스포린 항생제의 제조방법
IT1148888B (it) *	1980-07-15	1986-12-03	Schiena Ricerche Di	Composti antibiotici
DE3037997A1 (de) *	1980-10-08	1982-05-13	Bayer Ag	(beta) -lactamantibiotika, verfahren zu deren herstellung sowie sie enthaltende mittel
DE3145727A1 (de) *	1981-11-19	1983-05-26	Bayer Ag, 5090 Leverkusen	Zwischenprodukte, verfahren zu deren herstellung und verfahren zur herstellung von cephalosporinen

1982
- 1982-10-23 DE DE19823239365 patent/DE3239365A1/de not_active Withdrawn
1983
- 1983-10-06 NO NO833644A patent/NO833644L/no unknown
- 1983-10-11 DE DE8383110116T patent/DE3373476D1/de not_active Expired
- 1983-10-11 EP EP83110116A patent/EP0107138B1/de not_active Expired
- 1983-10-11 AT AT83110116T patent/ATE29498T1/de active
- 1983-10-13 PT PT77501A patent/PT77501B/pt unknown
- 1983-10-17 US US06/542,833 patent/US4489076A/en not_active Expired - Fee Related
- 1983-10-20 FI FI833846A patent/FI73689C/fi not_active IP Right Cessation
- 1983-10-20 NZ NZ206017A patent/NZ206017A/en unknown
- 1983-10-20 IL IL70012A patent/IL70012A/xx unknown
- 1983-10-21 AU AU20447/83A patent/AU556826B2/en not_active Ceased
- 1983-10-21 ZA ZA837850A patent/ZA837850B/xx unknown
- 1983-10-21 GR GR72763A patent/GR79682B/el unknown
- 1983-10-21 DK DK486183A patent/DK486183A/da not_active Application Discontinuation
- 1983-10-21 PH PH29734A patent/PH20918A/en unknown
- 1983-10-21 ES ES526674A patent/ES526674A0/es active Granted
- 1983-10-21 CA CA000439476A patent/CA1208206A/en not_active Expired
- 1983-10-21 HU HU833636A patent/HU189763B/hu not_active IP Right Cessation
- 1983-10-22 KR KR1019830005011A patent/KR840006487A/ko not_active Ceased
- 1983-10-22 JP JP58198180A patent/JPS5993086A/ja active Pending
1985
- 1985-07-15 PH PH32523A patent/PH20908A/en unknown
- 1985-07-15 PH PH32524A patent/PH20665A/en unknown

Also Published As

Publication number	Publication date
DK486183D0 (da)	1983-10-21
EP0107138A2 (de)	1984-05-02
FI73689B (fi)	1987-07-31
FI833846L (fi)	1984-04-24
NZ206017A (en)	1985-11-08
ES8406491A1 (es)	1984-07-01
IL70012A0 (en)	1984-01-31
HU189763B (en)	1986-07-28
AU556826B2 (en)	1986-11-20
PH20665A (en)	1987-03-23
AU2044783A (en)	1984-05-03
US4489076A (en)	1984-12-18
EP0107138B1 (de)	1987-09-09
EP0107138A3 (en)	1985-05-15
FI833846A0 (fi)	1983-10-20
HUT34210A (en)	1985-02-28
PT77501B (en)	1986-02-12
ATE29498T1 (de)	1987-09-15
DK486183A (da)	1984-04-24
GR79682B (da)	1984-10-31
ES526674A0 (es)	1984-07-01
FI73689C (fi)	1987-11-09
PH20908A (en)	1987-05-27
CA1208206A (en)	1986-07-22
DE3239365A1 (de)	1984-04-26
IL70012A (en)	1987-09-16
PH20918A (en)	1987-05-28
NO833644L (no)	1984-04-24
JPS5993086A (ja)	1984-05-29
PT77501A (en)	1983-11-01
DE3373476D1 (en)	1987-10-15
KR840006487A (ko)	1984-11-30

Publication	Publication Date	Title
AU539519B2 (en)	1984-10-04	7(2-(2-aminothiazol-4-yl)-2(2-carboxyprop-2-oxyimino) acteamido)-3-(1-pyridiniumethyl)ceph 3-em-4-carboxylate
ZA857274B (en)	1986-05-28	Diarylacetylenes,their preparation and their use
AU556826B2 (en)	1986-11-20	And a process for their preparation
GR3005624T3 (da)	1993-06-07
ZA801787B (en)	1981-03-25	7-(2-(amino-4-thiazolyl)-2-((1-carboxy-1,1-dialkyl)-alkoxyimino)acetamido)cephem sulfoxides
ES2001338A6 (es)	1988-05-16	Un procedimiento para la preparacion de un solvato cristalino con dimetilformamida del acido 7-(d)-2-amino-2-(4-hidroxifenil) acetamido -3-(z)-1-propenil cef -3-em-4-carboxilico.
AU572916B2 (en)	1988-05-19	Cephalosporin derivatives
IL52699A (en)	1980-09-16	7-(2-(substituted benzoyl amino)acetamido)cephalosporins
AU553493B2 (en)	1986-07-17	3,7alpha-diazacyclohepta(j,k)fluoriene derivatives
PT83712A (de)	1986-12-01	Cephalosporinderivate und verfahren zu ihrer herstellung
AU2231783A (en)	1984-06-21	Substitution of acylamino beta-lactam at the carbon atom carrying the acylamino group
GB2068959B (en)	1984-02-22	7-(2-amino-4-thiazolyl) acetamido cephalosporins
IE790065L (en)	1979-07-17	Penicillins, cephalosporins and related intermediates
YU72283A (en)	1985-12-31	Process for the manufcture of n-(2-pyrridyl)-2-alkyl-4-hydroxy-2h-1,2-benzothiazine-3-carboxamide-1,1-dioxide
YU42883B (en)	1988-12-31	Process for the manufacture of n-(2-pyridil)-2-methyl-4-hydroxy-2h-1,2-benzothiazine-3-carboxamide-1,1-dioxide