ZA85696B - Pyrimido(2,1-b)benzothiazoles - Google Patents

Pyrimido(2,1-b)benzothiazoles

Info

Publication number: ZA85696B
Authority: ZA; South Africa
Prior art keywords: group; branched; straight; hydrogen atom; alkyl
Prior art date: 1984-02-13

Application number

ZA85696A

Other languages

English (en)

Inventor

David Alun Rowlands

Julian Marian Charles Golec

Original Assignee

Roussel Uclaf

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1984-02-13

Filing date

1985-01-29

Publication date

1986-03-26

1985-01-29 Application filed by Roussel Uclaf filed Critical Roussel Uclaf

1986-03-26 Publication of ZA85696B publication Critical patent/ZA85696B/xx

Links

RWVLSUFUYXWYKA-UHFFFAOYSA-N 4h-pyrimido[2,1-b][1,3]benzothiazole Chemical class C1=CC=C2N3CC=CN=C3SC2=C1 RWVLSUFUYXWYKA-UHFFFAOYSA-N 0.000 title 1
125000004169 (C1-C6) alkyl group Chemical group 0.000 abstract 3
125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 3
125000004191 (C1-C6) alkoxy group Chemical group 0.000 abstract 2
125000005913 (C3-C6) cycloalkyl group Chemical group 0.000 abstract 2
125000004453 alkoxycarbonyl group Chemical group 0.000 abstract 1
125000000217 alkyl group Chemical group 0.000 abstract 1
239000000043 antiallergic agent Substances 0.000 abstract 1
125000003710 aryl alkyl group Chemical group 0.000 abstract 1
125000003118 aryl group Chemical group 0.000 abstract 1
229910052799 carbon Inorganic materials 0.000 abstract 1
125000004432 carbon atom Chemical group C* 0.000 abstract 1
150000001875 compounds Chemical class 0.000 abstract 1
125000005843 halogen group Chemical group 0.000 abstract 1
125000001072 heteroaryl group Chemical group 0.000 abstract 1
125000002887 hydroxy group Chemical group [H]O* 0.000 abstract 1
125000004573 morpholin-4-yl group Chemical group N1(CCOCC1)* 0.000 abstract 1
125000000449 nitro group Chemical group [O-][N+](*)=O 0.000 abstract 1
229910052757 nitrogen Inorganic materials 0.000 abstract 1
125000004433 nitrogen atom Chemical group N* 0.000 abstract 1
125000000587 piperidin-1-yl group Chemical group [H]C1([H])N(*)C([H])([H])C([H])([H])C([H])([H])C1([H])[H] 0.000 abstract 1
150000003839 salts Chemical class 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
- C07D277/62—Benzothiazoles
- C07D277/68—Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- C07D277/82—Nitrogen atoms

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Bioinformatics & Cheminformatics (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Engineering & Computer Science (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Pulmonology (AREA)
Public Health (AREA)
Immunology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Agricultural Chemicals And Associated Chemicals (AREA)
Luminescent Compositions (AREA)
Transition And Organic Metals Composition Catalysts For Addition Polymerization (AREA)
Saccharide Compounds (AREA)
Compositions Of Macromolecular Compounds (AREA)
Thiazole And Isothizaole Compounds (AREA)
Macromolecular Compounds Obtained By Forming Nitrogen-Containing Linkages In General (AREA)
Indole Compounds (AREA)
Polymerisation Methods In General (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)

ZA85696A 1984-02-13 1985-01-29 Pyrimido(2,1-b)benzothiazoles ZA85696B (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
GB848403739A GB8403739D0 (en)	1984-02-13	1984-02-13	Chemical compounds

Publications (1)

Publication Number	Publication Date
ZA85696B true ZA85696B (en)	1986-03-26

Family

ID=10556508

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
ZA85696A ZA85696B (en)	1984-02-13	1985-01-29	Pyrimido(2,1-b)benzothiazoles

Country Status (16)

Country	Link
EP (1)	EP0153230B1 (da)
JP (1)	JPS60184086A (da)
KR (1)	KR850005847A (da)
AT (1)	ATE44745T1 (da)
AU (1)	AU574131B2 (da)
CA (1)	CA1257259A (da)
DE (1)	DE3571621D1 (da)
DK (1)	DK63385A (da)
ES (2)	ES8702421A1 (da)
FI (1)	FI79323C (da)
GB (2)	GB8403739D0 (da)
GR (1)	GR850369B (da)
HU (1)	HU192318B (da)
NZ (1)	NZ211104A (da)
PT (1)	PT79955B (da)
ZA (1)	ZA85696B (da)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4762840A (en) *	1984-02-13	1988-08-09	Roussel Uclaf	Pyrimido[2,1-b]benzothiazoles having antiallergic activity
GB8519261D0 (en) *	1985-07-31	1985-09-04	Roussel Lab Ltd	Chemical compounds
AP2013006706A0 (en)	2010-07-02	2013-02-28	Gilead Sciences Inc	Napht-2-ylacetic acid derivatives to treat AIDS
SG186821A1 (en)	2010-07-02	2013-02-28	Gilead Sciences Inc	2 -quinolinyl- acetic acid derivatives as hiv antiviral compounds
SG194512A1 (en) *	2011-04-21	2013-12-30	Gilead Sciences Inc	Benzothiazole compounds and their pharmaceutical use
US9376392B2 (en)	2012-01-04	2016-06-28	Gilead Sciences, Inc.	2-(tert-butoxy)-2-(7-methylquinolin-6-yl) acetic acid derivatives for treating AIDS
WO2013103738A1 (en)	2012-01-04	2013-07-11	Gilead Sciences, Inc.	Napthalene acetic acid derivatives against hiv infection
CN105121418A (zh)	2012-04-20	2015-12-02	吉利德科学公司	苯并噻唑-6-基乙酸衍生物及其治疗hiv感染的用途

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3919201A (en) *	1970-09-30	1975-11-11	Lilly Industries Ltd	2-({62 -Aminoacryloyl)iminobenzothiazolines
DE2810863A1 (de) *	1978-03-13	1979-09-27	Boehringer Mannheim Gmbh	1-oxo-1h-pyrimido eckige klammer auf 6,1-b eckige klammer zu benzthiazol-derivate und verfahren zu ihrer herstellung
GB8519261D0 (en) *	1985-07-31	1985-09-04	Roussel Lab Ltd	Chemical compounds

1984
- 1984-02-13 GB GB848403739A patent/GB8403739D0/en active Pending
1985
- 1985-01-13 KR KR1019850000879A patent/KR850005847A/ko not_active Ceased
- 1985-01-29 ZA ZA85696A patent/ZA85696B/xx unknown
- 1985-02-11 DE DE8585400219T patent/DE3571621D1/de not_active Expired
- 1985-02-11 AT AT85400219T patent/ATE44745T1/de not_active IP Right Cessation
- 1985-02-11 EP EP85400219A patent/EP0153230B1/fr not_active Expired
- 1985-02-12 GR GR850369A patent/GR850369B/el unknown
- 1985-02-12 GB GB08503541A patent/GB2154583B/en not_active Expired
- 1985-02-12 NZ NZ211104A patent/NZ211104A/en unknown
- 1985-02-12 HU HU85529A patent/HU192318B/hu not_active IP Right Cessation
- 1985-02-12 DK DK63385A patent/DK63385A/da not_active Application Discontinuation
- 1985-02-12 ES ES540332A patent/ES8702421A1/es not_active Expired
- 1985-02-12 CA CA000474113A patent/CA1257259A/en not_active Expired
- 1985-02-12 PT PT79955A patent/PT79955B/pt not_active IP Right Cessation
- 1985-02-12 JP JP60023706A patent/JPS60184086A/ja active Pending
- 1985-02-12 FI FI850582A patent/FI79323C/fi not_active IP Right Cessation
- 1985-02-13 AU AU38672/85A patent/AU574131B2/en not_active Ceased
1986
- 1986-04-01 ES ES553574A patent/ES8800243A1/es not_active Expired

Also Published As

Publication number	Publication date
GB8403739D0 (en)	1984-03-14
FI79323C (fi)	1989-12-11
ES8702421A1 (es)	1986-12-16
HUT38649A (en)	1986-06-30
PT79955A (en)	1985-03-01
FI850582L (fi)	1985-08-14
ES553574A0 (es)	1987-10-16
AU574131B2 (en)	1988-06-30
EP0153230A2 (fr)	1985-08-28
ES540332A0 (es)	1986-12-16
NZ211104A (en)	1987-08-31
ATE44745T1 (de)	1989-08-15
ES8800243A1 (es)	1987-10-16
AU3867285A (en)	1985-08-22
DK63385D0 (da)	1985-02-12
HU192318B (en)	1987-05-28
GR850369B (da)	1985-06-14
JPS60184086A (ja)	1985-09-19
GB2154583A (en)	1985-09-11
GB2154583B (en)	1987-10-28
PT79955B (en)	1987-02-02
GB8503541D0 (en)	1985-03-13
EP0153230B1 (fr)	1989-07-19
DE3571621D1 (en)	1989-08-24
CA1257259A (en)	1989-07-11
EP0153230A3 (en)	1986-10-01
FI850582A0 (fi)	1985-02-12
DK63385A (da)	1985-08-14
KR850005847A (ko)	1985-09-26
FI79323B (fi)	1989-08-31

Publication	Publication Date	Title
DE3588100D1 (de)	1996-05-23	Carbamidsäureester-Derivate, Mittel und Herstellungsverfahren
DE69426157D1 (de)	2000-11-23	1,4-di(phenylalkyl)piperazinderivate
AU5228190A (en)	1990-10-04	Novel quinolone derivatives, preparation processes thereof, and antibacterial agents containing the same
AU574131B2 (en)	1988-06-30	Pyrimido (2,1-b)benzothiazoles
TW290539B (da)	1996-11-11
AU582621B2 (en)	1989-04-06	Imidazole derivatives, their preparation and their use as fungicides
EP0214292A4 (en)	1988-05-03	STABILIZATION COMPOSITION FOR POLYURETHANE.
AU561008B2 (en)	1987-04-30	N,n,-disubstituted alkenamides and phenylalkenamides and heterocyclic starting compounds
PT83099A (en)	1986-08-01	Process for the preparation of new pyrimide <2,1-b> benzothiazoles with anti-allergical properties
DE69113901D1 (de)	1995-11-23	Pyrazolo(1,5-a)pyridine, deren Herstellung und Verwendung.
GB2167750A (en)	1986-06-04	Isothiuronium salts