ZA923538B - Amino acid azetidinyl substituted pyridone derivatives,their preparation and their application as medications - Google Patents

Amino acid azetidinyl substituted pyridone derivatives,their preparation and their application as medications

Info

Publication number
ZA923538B
ZA923538B ZA923538A ZA923538A ZA923538B ZA 923538 B ZA923538 B ZA 923538B ZA 923538 A ZA923538 A ZA 923538A ZA 923538 A ZA923538 A ZA 923538A ZA 923538 B ZA923538 B ZA 923538B
Authority
ZA
South Africa
Prior art keywords
medications
preparation
amino acid
application
pyridone derivatives
Prior art date
Application number
ZA923538A
Other languages
English (en)
Inventor
Jordi Corbera-Arjona
Corbera-Arjona Jordi
Jordi Frigola Constansa
Frigola Constansa Jordi
Juan Pares Corominas
Pares Corominas Juan
Original Assignee
Esteve Labor Dr
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Esteve Labor Dr filed Critical Esteve Labor Dr
Publication of ZA923538B publication Critical patent/ZA923538B/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/48—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • C07D215/54—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3
    • C07D215/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3 with oxygen atoms in position 4
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D205/04—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pyridine Compounds (AREA)
  • Peptides Or Proteins (AREA)
ZA923538A 1991-05-16 1992-05-15 Amino acid azetidinyl substituted pyridone derivatives,their preparation and their application as medications ZA923538B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9105937A FR2676445B1 (fr) 1991-05-16 1991-05-16 Derives de pyridone amino acide azetidinyl substitues, leur preparation et leur application en tant que medicaments.

Publications (1)

Publication Number Publication Date
ZA923538B true ZA923538B (en) 1993-01-27

Family

ID=9412841

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA923538A ZA923538B (en) 1991-05-16 1992-05-15 Amino acid azetidinyl substituted pyridone derivatives,their preparation and their application as medications

Country Status (20)

Country Link
EP (1) EP0514268A1 (cs)
JP (1) JPH05132479A (cs)
KR (1) KR920021528A (cs)
CN (1) CN1066656A (cs)
AU (1) AU660311B2 (cs)
CA (1) CA2068853A1 (cs)
CZ (1) CZ147992A3 (cs)
ES (1) ES2039192B1 (cs)
FI (1) FI922225A7 (cs)
FR (1) FR2676445B1 (cs)
HU (1) HUT61304A (cs)
IL (1) IL101886A0 (cs)
IS (1) IS3862A (cs)
MA (1) MA22526A1 (cs)
MX (1) MX9202273A (cs)
NO (1) NO921908L (cs)
NZ (1) NZ242733A (cs)
OA (1) OA09794A (cs)
PL (1) PL294561A1 (cs)
ZA (1) ZA923538B (cs)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE69732635T2 (de) 1996-07-12 2005-12-29 Daiichi Pharmaceutical Co., Ltd. Cis-substituierte aminocyclopropanderivate
KR100613690B1 (ko) * 2004-07-30 2006-08-21 한국화학연구원 4-퀴놀린온 유도체 및 이를 포함하는 농원예용 살균제조성물
KR100613688B1 (ko) * 2004-08-30 2006-08-21 한국화학연구원 2-아미노-4-퀴놀린온 유도체 및 이를 포함하는 농원예용살균제 조성물
WO2006068768A2 (en) 2004-11-24 2006-06-29 Hanna Skubatch Methods and compositions for treating conditions
US7557088B2 (en) 2006-03-28 2009-07-07 Neopro Labs, Llc Methods and compositions for treating conditions
US8217141B2 (en) 2007-05-17 2012-07-10 Neopro Labs, Llc Crystalline and amorphous forms of peptide
CN101898990B (zh) * 2009-06-01 2012-12-19 中国科学院化学研究所 微生物体系催化合成手性氮杂环丁烷酰胺和羧酸类化合物的方法
CA3213636A1 (en) 2021-03-18 2022-09-22 Seagen Inc. Selective drug release from internalized conjugates of biologically active compounds

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5746986A (en) * 1980-09-02 1982-03-17 Dai Ichi Seiyaku Co Ltd Pyrido(1,2,3-de)(1,4)benzoxazine derivative
IE55898B1 (en) * 1982-09-09 1991-02-14 Warner Lambert Co Antibacterial agents
DE3306771A1 (de) * 1983-02-25 1984-08-30 Bayer Ag, 5090 Leverkusen Chinoloncarbonsaeuren, verfahren zu ihrer herstellung sowie diese enthaltende antibakterielle mittel
CA1267413A (en) * 1984-04-26 1990-04-03 Abbott Laboratories Quino-benoxazine antibacterial compounds
US4617308A (en) * 1985-01-25 1986-10-14 Warner-Lambert Company 7-substituted amino-1-aryl-6,8-difluoro-1,4-dihydro-4-oxo-3-quinolinecarboxylic acids and derivatives thereof as antibacterial agents
US4851418A (en) * 1987-08-21 1989-07-25 Warner-Lambert Company Naphthyridine antibacterial agents containing an α-amino acid in the side chain of the 7-substituent
FR2634483B2 (fr) * 1987-12-29 1994-03-04 Esteve Labor Dr Derives des acides 7-(1-azetidinyl)-1,4-dihydro-4-oxoquinoleine-3-carboxyliques, leur preparation et leur application en tant que medicaments
IE76284B1 (en) * 1988-09-22 1997-10-08 Abbott Lab Amino acid quinoline and naphthyridine derivatives
AU5123690A (en) * 1989-03-13 1990-09-13 Bristol-Myers Squibb Company 5-substituted-1,4-dihydro-4-oxo-nephthyridine-3-carboxylate antibacterial agents
NO177302C (no) * 1989-03-16 1995-08-23 Esteve Labor Dr Analogifremgangsmåte til fremstilling av terapeutisk aktive substituerte azetidinylkinolon(naftyridon)karboksylsyrederivater
FR2645862B1 (fr) * 1989-04-18 1991-07-12 Esteve Labor Dr Derives d'isothiazolo-pyrydone azetidinyl substitues, leur preparation et leur application en tant que medicaments
FR2649100B1 (fr) * 1989-06-29 1994-03-04 Laboratorios Dr Esteve Sa Nouvelles azetidines, leur preparation et leur application comme intermediaires pour la preparation de composes avec activite antimicrobienne

Also Published As

Publication number Publication date
NO921908D0 (no) 1992-05-14
PL294561A1 (en) 1993-05-04
FI922225A0 (fi) 1992-05-15
HU9201621D0 (en) 1992-08-28
NZ242733A (en) 1994-06-27
EP0514268A1 (fr) 1992-11-19
JPH05132479A (ja) 1993-05-28
CZ147992A3 (en) 1993-09-15
MA22526A1 (fr) 1992-12-31
FR2676445A1 (fr) 1992-11-20
ES2039192B1 (es) 1994-04-01
IS3862A (is) 1992-11-17
CN1066656A (zh) 1992-12-02
FR2676445B1 (fr) 1995-02-03
AU660311B2 (en) 1995-06-22
IL101886A0 (en) 1992-12-30
CA2068853A1 (fr) 1992-11-17
KR920021528A (ko) 1992-12-18
OA09794A (fr) 1994-04-15
MX9202273A (es) 1993-05-01
FI922225A7 (fi) 1992-11-17
NO921908L (no) 1992-11-17
HUT61304A (en) 1992-12-28
AU1624992A (en) 1992-11-19
ES2039192A1 (es) 1993-09-01

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