ZA961994B - Piperidine derivatives process for the preparation thereof and application thereof in therapeutics - Google Patents
Piperidine derivatives process for the preparation thereof and application thereof in therapeuticsInfo
- Publication number
- ZA961994B ZA961994B ZA961994A ZA961994A ZA961994B ZA 961994 B ZA961994 B ZA 961994B ZA 961994 A ZA961994 A ZA 961994A ZA 961994 A ZA961994 A ZA 961994A ZA 961994 B ZA961994 B ZA 961994B
- Authority
- ZA
- South Africa
- Prior art keywords
- therapeutics
- preparation
- application
- piperidine derivatives
- derivatives process
- Prior art date
Links
- 239000003814 drug Substances 0.000 title 1
- 150000003053 piperidines Chemical class 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/06—Peri-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Psychiatry (AREA)
- Heart & Thoracic Surgery (AREA)
- Hospice & Palliative Care (AREA)
- Cardiology (AREA)
- Pain & Pain Management (AREA)
- Pulmonology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Hydrogenated Pyridines (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR9502863A FR2731708B1 (en) | 1995-03-13 | 1995-03-13 | PIPERIDINE DERIVATIVES, THEIR PREPARATION PROCESS AND THEIR THERAPEUTIC APPLICATION |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ZA961994B true ZA961994B (en) | 1996-09-03 |
Family
ID=9476960
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ZA961994A ZA961994B (en) | 1995-03-13 | 1996-03-12 | Piperidine derivatives process for the preparation thereof and application thereof in therapeutics |
Country Status (15)
| Country | Link |
|---|---|
| EP (1) | EP0732334A1 (en) |
| JP (1) | JPH08269058A (en) |
| KR (1) | KR960034205A (en) |
| CN (1) | CN1140174A (en) |
| AU (1) | AU4800896A (en) |
| CA (1) | CA2171579A1 (en) |
| CZ (1) | CZ75496A3 (en) |
| FR (1) | FR2731708B1 (en) |
| HU (1) | HUP9600624A2 (en) |
| IL (1) | IL117455A0 (en) |
| NO (1) | NO961000L (en) |
| NZ (1) | NZ286164A (en) |
| PL (1) | PL313204A1 (en) |
| SK (1) | SK34196A3 (en) |
| ZA (1) | ZA961994B (en) |
Families Citing this family (18)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR19990045728A (en) * | 1995-09-18 | 1999-06-25 | 그레이엄 브레레톤, 레슬리 에드워즈 | 5-HT3 receptor antagonist for dyskinesia |
| TW527186B (en) | 1996-03-19 | 2003-04-11 | Janssen Pharmaceutica Nv | Fused imidazole derivatives as multidrug resistance modulators |
| FR2801589A1 (en) * | 1999-11-25 | 2001-06-01 | Sanofi Synthelabo | 2-Aryl quinoline derivatives useful for the treatment of urinary incontinence. venous ulcers, migraine or gastro-intestinal disorders |
| EP1309594B1 (en) * | 2000-08-08 | 2004-12-15 | Sanofi-Aventis | Benzimidazole derivatives, preparation and therapeutic use thereof |
| FR2816619B1 (en) * | 2000-11-15 | 2003-01-31 | Sanofi Synthelabo | BENZIMIDAZOLE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION |
| FR2816941B1 (en) * | 2000-11-23 | 2003-01-31 | Sanofi Synthelabo | BENZIMIDAZOLE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION |
| FR2816942B1 (en) | 2000-11-23 | 2003-05-09 | Sanofi Synthelabo | BENZIMIDAZOLE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION |
| MX366703B (en) * | 2013-03-15 | 2019-07-22 | Incyte Holdings Corp | Tricyclic heterocycles as bet protein inhibitors. |
| AR096837A1 (en) * | 2013-07-08 | 2016-02-03 | Incyte Corp | TRICYCLIC HETEROCICLES AS BET PROTEIN INHIBITORS |
| US9399640B2 (en) | 2013-11-26 | 2016-07-26 | Incyte Corporation | Substituted pyrrolo[2,3-c]pyridines and pyrazolo[3,4-c]pyridines as BET protein inhibitors |
| WO2015081189A1 (en) | 2013-11-26 | 2015-06-04 | Incyte Corporation | Bicyclic heterocycles as bet protein inhibitors |
| WO2015095492A1 (en) | 2013-12-19 | 2015-06-25 | Incyte Corporation | Tricyclic heterocycles as bet protein inhibitors |
| EA034972B1 (en) | 2014-04-23 | 2020-04-13 | Инсайт Корпорейшн | 1H-PYRROLO[2,3-c]PYRIDIN-7(6H)-ONES AS INHIBITORS OF BET PROTEINS |
| US9527864B2 (en) | 2014-09-15 | 2016-12-27 | Incyte Corporation | Tricyclic heterocycles as BET protein inhibitors |
| TW201722966A (en) | 2015-10-29 | 2017-07-01 | 英塞特公司 | Amorphous solid form of a BET protein inhibitor |
| KR102643344B1 (en) | 2016-06-20 | 2024-03-07 | 인사이트 코포레이션 | Crystalline solid forms of a bet inhibitor |
| JP2021530442A (en) * | 2018-06-28 | 2021-11-11 | ジエンス ヘンルイ メデイシンカンパニー リミテッドJiangsu Hengrui Medicine Co., Ltd. | Condensed tricyclic heterocyclic compounds and their therapeutic use |
| US11833155B2 (en) | 2020-06-03 | 2023-12-05 | Incyte Corporation | Combination therapy for treatment of myeloproliferative neoplasms |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2674855B1 (en) * | 1991-04-03 | 1994-01-14 | Synthelabo | PIPERIDINE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION. |
| FR2696176B1 (en) * | 1992-09-28 | 1994-11-10 | Synthelabo | Piperidine derivatives, their preparation and their therapeutic application. |
| FR2710915B1 (en) * | 1993-10-04 | 1995-11-24 | Synthelabo | Piperidine derivatives, their preparation and their therapeutic use. |
-
1995
- 1995-03-13 FR FR9502863A patent/FR2731708B1/en not_active Expired - Fee Related
-
1996
- 1996-03-04 EP EP96400452A patent/EP0732334A1/en not_active Withdrawn
- 1996-03-12 JP JP8054560A patent/JPH08269058A/en active Pending
- 1996-03-12 SK SK341-96A patent/SK34196A3/en unknown
- 1996-03-12 NO NO961000A patent/NO961000L/en unknown
- 1996-03-12 KR KR1019960006462A patent/KR960034205A/en not_active Withdrawn
- 1996-03-12 AU AU48008/96A patent/AU4800896A/en not_active Abandoned
- 1996-03-12 PL PL96313204A patent/PL313204A1/en unknown
- 1996-03-12 IL IL11745596A patent/IL117455A0/en unknown
- 1996-03-12 NZ NZ286164A patent/NZ286164A/en unknown
- 1996-03-12 HU HU9600624A patent/HUP9600624A2/en unknown
- 1996-03-12 CN CN96107315A patent/CN1140174A/en active Pending
- 1996-03-12 CA CA002171579A patent/CA2171579A1/en not_active Abandoned
- 1996-03-12 CZ CZ96754A patent/CZ75496A3/en unknown
- 1996-03-12 ZA ZA961994A patent/ZA961994B/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| NZ286164A (en) | 1996-11-26 |
| HUP9600624A2 (en) | 1997-01-28 |
| PL313204A1 (en) | 1996-09-16 |
| NO961000D0 (en) | 1996-03-12 |
| FR2731708A1 (en) | 1996-09-20 |
| HU9600624D0 (en) | 1996-05-28 |
| KR960034205A (en) | 1996-10-22 |
| AU4800896A (en) | 1996-09-26 |
| CA2171579A1 (en) | 1996-09-14 |
| EP0732334A1 (en) | 1996-09-18 |
| NO961000L (en) | 1996-09-16 |
| JPH08269058A (en) | 1996-10-15 |
| CZ75496A3 (en) | 1996-10-16 |
| IL117455A0 (en) | 1996-07-23 |
| CN1140174A (en) | 1997-01-15 |
| SK34196A3 (en) | 1996-10-02 |
| FR2731708B1 (en) | 1997-04-30 |
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