AP2014007372A0 - Indazoles - Google Patents

Indazoles

Info

Publication number: AP2014007372A0
Authority: AP; ARIPO
Prior art keywords: indazoles
Prior art date: 2011-07-27

Application number

AP2014007372A

Other languages

English (en)

Inventor

Jotham Wadsworth Coe

Christoph Martin Dehnhardt

Peter Jones

Original Assignee

Pfizer Ltd

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2011-07-27

Filing date

2012-07-11

Publication date

2014-01-31

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=46826868&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AP2014007372(A0) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

2012-07-11 Application filed by Pfizer Ltd filed Critical Pfizer Ltd

2014-01-31 Publication of AP2014007372A0 publication Critical patent/AP2014007372A0/xx

Links

150000002473 indoazoles Chemical class 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A61P1/06—Anti-spasmodics, e.g. drugs for colics, esophagic dyskinesia
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- A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A61P11/06—Antiasthmatics
- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Public Health (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Chemical Kinetics & Catalysis (AREA)
Pharmacology & Pharmacy (AREA)
Veterinary Medicine (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Physical Education & Sports Medicine (AREA)
Immunology (AREA)
Pulmonology (AREA)
Neurology (AREA)
Rheumatology (AREA)
Diabetes (AREA)
Cardiology (AREA)
Biomedical Technology (AREA)
Orthopedic Medicine & Surgery (AREA)
Ophthalmology & Optometry (AREA)
Dermatology (AREA)
Neurosurgery (AREA)
Heart & Thoracic Surgery (AREA)
Endocrinology (AREA)
Pain & Pain Management (AREA)
Hematology (AREA)
Communicable Diseases (AREA)
Oncology (AREA)
Toxicology (AREA)
Urology & Nephrology (AREA)
Reproductive Health (AREA)
Obesity (AREA)
Hospice & Palliative Care (AREA)
Otolaryngology (AREA)
Child & Adolescent Psychology (AREA)

AP2014007372A 2011-07-27 2012-07-11 Indazoles AP2014007372A0 (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US201161512144P	2011-07-27	2011-07-27
PCT/IB2012/053546 WO2013014567A1 (en)	2011-07-27	2012-07-11	Indazoles

Publications (1)

Publication Number	Publication Date
AP2014007372A0 true AP2014007372A0 (en)	2014-01-31

Family

ID=46826868

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AP2014007372A AP2014007372A0 (en)	2011-07-27	2012-07-11	Indazoles

Country Status (30)

Country	Link
US (2)	US8575336B2 (xx)
EP (1)	EP2736907B1 (xx)
JP (1)	JP5579351B1 (xx)
KR (1)	KR20140026627A (xx)
CN (1)	CN103717599B (xx)
AP (1)	AP2014007372A0 (xx)
AR (1)	AR087348A1 (xx)
AU (1)	AU2012288491A1 (xx)
BR (1)	BR112014001801A2 (xx)
CA (1)	CA2841882A1 (xx)
CL (1)	CL2014000122A1 (xx)
CO (1)	CO6862160A2 (xx)
CR (1)	CR20140042A (xx)
CU (1)	CU20140009A7 (xx)
DO (1)	DOP2014000016A (xx)
EA (1)	EA201490357A1 (xx)
EC (1)	ECSP14013222A (xx)
GT (1)	GT201400016A (xx)
IL (1)	IL230662A0 (xx)
MA (1)	MA35285B1 (xx)
MD (1)	MD20140002A2 (xx)
MX (1)	MX2014001004A (xx)
NI (1)	NI201400005A (xx)
PE (1)	PE20141059A1 (xx)
PH (1)	PH12014500199A1 (xx)
TN (1)	TN2014000033A1 (xx)
TW (1)	TWI462922B (xx)
UA (1)	UA108442C2 (xx)
UY (1)	UY34220A (xx)
WO (1)	WO2013014567A1 (xx)

Families Citing this family (41)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US8575336B2 (en)	2011-07-27	2013-11-05	Pfizer Limited	Indazoles
KR20170002623A (ko) *	2014-05-14	2017-01-06	화이자 인코포레이티드	피라졸로피리딘 및 피라졸로피리미딘
JP2018507236A (ja)	2015-03-04	2018-03-15	エフ．ホフマン−ラロシュアーゲーＦ．Ｈｏｆｆｍａｎｎ−ＬａＲｏｃｈｅＡｋｔｉｅｎｇｅｓｅｌｌｓｃｈａｆｔ	トリアゾロピリジン化合物及びその使用法
LT3286181T (lt)	2015-04-22	2021-04-26	Rigel Pharmaceuticals, Inc.	Pirazolo junginiai ir junginių gamybos bei naudojimo būdas
WO2017077283A1 (en) *	2015-11-03	2017-05-11	Topivert Pharma Limited	4,5,6,7-tetrahydro-1h-imidazo[4,5-c]pyridine and 1,4,5,6,7,8-hexahydroimidazo[4,5-d]azepine derivatives as janus kinase inhibitors
DK3371185T3 (da)	2015-11-03	2020-11-30	Topivert Pharma Ltd	4,5,6,7-tetrahydro-1h-imidazo[4,5-c]pyridin og 1,4,5,6,7,8-hexahydroimidazo[4,5-d]azepinderivater som janus-kinase-inhibitorer
UA123633C2 (uk) *	2015-11-03	2021-05-05	Тереванс Байофарма Ар Енд Ді Айпі, Елелсі	Сполуки інгібітору jak-кінази для лікування респіраторного захворювання
TW201720828A (zh)	2015-11-23	2017-06-16	赫孚孟拉羅股份公司	治療性化合物及組合物以及其使用方法
WO2017096262A1 (en)	2015-12-04	2017-06-08	Jomoco, Corp.	Compositions and methods to mitigate or prevent an immune response to an immunogenic therapeutic molecule in non-human primates
JP6936236B2 (ja)	2016-02-18	2021-09-15	エフ．ホフマン−ラロシュアーゲーＦ．Ｈｏｆｆｍａｎｎ−ＬａＲｏｃｈｅＡｋｔｉｅｎｇｅｓｅｌｌｓｃｈａｆｔ	治療化合物、組成物及びその方法の使用
JP7034942B2 (ja)	2016-05-05	2022-03-14	エフ．ホフマン－ラロシュアーゲー	ピラゾール誘導体、その組成物及び治療的使用
MX394560B (es) *	2016-06-01	2025-03-24	Bayer Pharma AG	Uso de indazoles sustituidos para el tratamiento y la prevencion de enfermedades en animales.
CN109890817B (zh)	2016-09-06	2022-06-17	豪夫迈·罗氏有限公司	8-(氮杂环丁烷-1-基)-[1,2,4]三唑并[1,5-a]吡啶基化合物、其组合物和应用方法
CR20190310A (es)	2016-12-29	2019-08-21	Hoffmann La Roche	Compuestos de pirazolopirimidina y métodos de uso de los mismos
WO2018165392A1 (en) *	2017-03-09	2018-09-13	Theravance Biopharma R&D Ip, Llc	Jak inhibitors containing a 4-membered heterocyclic amide
JP2020510061A (ja)	2017-03-14	2020-04-02	エフ．ホフマン−ラロシュアーゲーＦ．Ｈｏｆｆｍａｎｎ−ＬａＲｏｃｈｅＡｋｔｉｅｎｇｅｓｅｌｌｓｃｈａｆｔ	ピラゾロクロロフェニル化合物、組成物及びその使用方法
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Also Published As

Publication number	Publication date
NI201400005A (es)	2014-04-23
IL230662A0 (en)	2014-03-31
MX2014001004A (es)	2014-05-13
JP5579351B1 (ja)	2014-08-27
US8895544B2 (en)	2014-11-25
KR20140026627A (ko)	2014-03-05
US20130029968A1 (en)	2013-01-31
CA2841882A1 (en)	2013-01-31
TWI462922B (zh)	2014-12-01
CU20140009A7 (es)	2014-03-26
UY34220A (es)	2013-02-28
PE20141059A1 (es)	2014-08-30
EA201490357A1 (ru)	2014-05-30
UA108442C2 (xx)	2015-04-27
MD20140002A2 (ro)	2014-06-30
EP2736907B1 (en)	2015-10-07
EP2736907A1 (en)	2014-06-04
AR087348A1 (es)	2014-03-19
ECSP14013222A (es)	2014-03-31
WO2013014567A1 (en)	2013-01-31
JP2014522865A (ja)	2014-09-08
CN103717599B (zh)	2015-11-25
CN103717599A (zh)	2014-04-09
CO6862160A2 (es)	2014-02-10
TN2014000033A1 (fr)	2015-07-01
DOP2014000016A (es)	2014-07-15
GT201400016A (es)	2015-02-19
TW201313712A (zh)	2013-04-01
CL2014000122A1 (es)	2014-08-18
AU2012288491A1 (en)	2014-01-30
US8575336B2 (en)	2013-11-05
MA35285B1 (fr)	2014-07-03
US20140024634A1 (en)	2014-01-23
BR112014001801A2 (pt)	2017-02-14
CR20140042A (es)	2014-03-19
PH12014500199A1 (en)	2014-03-03

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AP2014007372A0 (en)	2014-01-31	Indazoles
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EP2566328A4 (en)	2013-10-16	indazoles
AP2014007621A0 (en)	2014-05-31	2-Thiopyrimidinones
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GB201102519D0 (en)	2011-03-30	Mirrorcane
GB201102755D0 (en)	2011-03-30	Protectaridge
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GB201106115D0 (en)	2011-05-25	BanksAway
GB201107098D0 (en)	2011-06-08	Corcost-ZZ1000
GB201112214D0 (en)	2011-08-31	Wheelaway