AP2806A - 3H-imidazo[4,5-C] pyridine-6-carboxamides as anti-infammatory agents - Google Patents
3H-imidazo[4,5-C] pyridine-6-carboxamides as anti-infammatory agentsInfo
- Publication number
- AP2806A AP2806A AP2011005807A AP2011005807A AP2806A AP 2806 A AP2806 A AP 2806A AP 2011005807 A AP2011005807 A AP 2011005807A AP 2011005807 A AP2011005807 A AP 2011005807A AP 2806 A AP2806 A AP 2806A
- Authority
- AP
- ARIPO
- Prior art keywords
- carboxamides
- imidazo
- pyridine
- infammatory
- agents
- Prior art date
Links
- QIYBKHZLGLSNJX-UHFFFAOYSA-N 3h-imidazo[4,5-c]pyridine-6-carboxamide Chemical class C1=NC(C(=O)N)=CC2=C1N=CN2 QIYBKHZLGLSNJX-UHFFFAOYSA-N 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
- C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
- C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
- C07D235/24—Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- C07D235/30—Nitrogen atoms not forming part of a nitro radical
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Pain & Pain Management (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Rheumatology (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Pulmonology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Plural Heterocyclic Compounds (AREA)
- Macromolecular Compounds Obtained By Forming Nitrogen-Containing Linkages In General (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP09154414 | 2009-03-05 | ||
| EP09179618 | 2009-12-17 | ||
| PCT/EP2010/052799 WO2010100249A1 (en) | 2009-03-05 | 2010-03-05 | 3h-imidazo [4, 5 -c] pyridine- 6 -carboxamides as anti- inflammatory agents |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| AP2011005807A0 AP2011005807A0 (en) | 2011-08-31 |
| AP2806A true AP2806A (en) | 2013-11-30 |
Family
ID=42111729
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AP2011005807A AP2806A (en) | 2009-03-05 | 2010-03-05 | 3H-imidazo[4,5-C] pyridine-6-carboxamides as anti-infammatory agents |
Country Status (36)
| Country | Link |
|---|---|
| US (3) | US20100256188A1 (ar) |
| EP (1) | EP2403852B8 (ar) |
| JP (1) | JP5433708B2 (ar) |
| KR (1) | KR20110123764A (ar) |
| CN (1) | CN102341395B (ar) |
| AP (1) | AP2806A (ar) |
| AR (1) | AR075789A1 (ar) |
| AU (1) | AU2010220263B2 (ar) |
| BR (1) | BRPI1009118A2 (ar) |
| CA (1) | CA2753149A1 (ar) |
| CL (1) | CL2011002180A1 (ar) |
| CO (1) | CO6450668A2 (ar) |
| CY (1) | CY1115959T1 (ar) |
| DK (1) | DK2403852T3 (ar) |
| EA (1) | EA020282B1 (ar) |
| EC (1) | ECSP11011324A (ar) |
| ES (1) | ES2528730T3 (ar) |
| GE (1) | GEP20146034B (ar) |
| HR (1) | HRP20150096T1 (ar) |
| IL (1) | IL214033A0 (ar) |
| MA (1) | MA33239B1 (ar) |
| ME (1) | ME02117B (ar) |
| MX (1) | MX2011008948A (ar) |
| MY (1) | MY161092A (ar) |
| NZ (1) | NZ594589A (ar) |
| PE (1) | PE20120589A1 (ar) |
| PL (1) | PL2403852T3 (ar) |
| PT (1) | PT2403852E (ar) |
| RS (1) | RS53757B1 (ar) |
| SG (1) | SG174250A1 (ar) |
| SI (1) | SI2403852T1 (ar) |
| SM (1) | SMT201500053B (ar) |
| TN (1) | TN2011000446A1 (ar) |
| TW (1) | TWI466869B (ar) |
| UY (1) | UY32470A (ar) |
| WO (1) | WO2010100249A1 (ar) |
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| UY32470A (es) | 2009-03-05 | 2010-10-29 | Boehringer Ingelheim Int | Derivados de 2-{2-cloro-5-[(sustituido) metil]fenilamino} -1-metil]fenilamino}-1-metilbencimidazol-5-carboxamidas-n-(sustituidas) y sus sales fisiológicamente aceptables, composiciones conteniéndolos y aplicaciones |
| US8586604B2 (en) | 2010-08-20 | 2013-11-19 | Boehringer Ingelheim International Gmbh | Inhibitors of the microsomal prostaglandin E2 synthase-1 |
| US8759537B2 (en) * | 2010-08-20 | 2014-06-24 | Boehringer Ingelheim International Gmbh | 3H-imidazo [4, 5-C] pyridine-6-carboxamides as anti-inflammatory agents |
| TW201305178A (zh) | 2010-10-29 | 2013-02-01 | Glenmark Pharmaceuticals Sa | 作為ｍＰＧＥＳ－１抑制物的三環化合物 |
| US8466186B2 (en) * | 2010-12-10 | 2013-06-18 | Boehringer Ingelheim International Gmbh | Compounds |
| UY33779A (es) * | 2010-12-10 | 2012-07-31 | Boehringer Ingelheim Int | ?2-(fenilamino)-1H-bencimidazol-5-carboxamidas novedosas? |
| US8486968B2 (en) * | 2010-12-10 | 2013-07-16 | Boehringer Ingelheim International Gmbh | Compounds |
| AR084174A1 (es) | 2010-12-21 | 2013-04-24 | Lilly Co Eli | Compuestos de imidazol-2-benzamida utiles para el tratamiento de osteoartritis y una composicion farmaceutica |
| AR086254A1 (es) | 2011-05-26 | 2013-11-27 | Lilly Co Eli | Derivados de imidazol utiles para el tratamiento de artritis |
| WO2013038308A1 (en) | 2011-09-15 | 2013-03-21 | Glenmark Pharmaceuticals S.A. | SUBSTITUTED BICYCLIC HETEROARYL COMPOUNDS AS mPGES-1 INHIBITORS |
| MY167575A (en) * | 2011-10-14 | 2018-09-20 | Ambit Biosciences Corp | Heterocyclic compounds and use thereof as modulators of type iii receptor tyrosine kinases |
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| US9006257B2 (en) | 2012-02-09 | 2015-04-14 | Glenmark Pharmaceuticals S.A. | Bicyclic compounds as mPGES-1 inhibitors |
| US9580398B2 (en) | 2012-04-02 | 2017-02-28 | The Trustees Of Columbia University In The City Of New York | Compounds, compositions, and methods for modulating ferroptosis and treating excitotoxic disorders |
| WO2013153535A1 (en) | 2012-04-13 | 2013-10-17 | Glenmark Pharmaceuticals S.A. | TRICYCLIC COMPOUNDS AS mPGES-1 INHIBITORS |
| CN103450329B (zh) * | 2012-05-29 | 2015-05-27 | 首都医科大学 | 3h-咪唑并吡啶-6-甲酰氨基酸苄酯、其合成、抗肿瘤活性和应用 |
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| WO2014167444A1 (en) | 2013-04-08 | 2014-10-16 | Glenmark Pharmaceuticals S.A. | SUBSTITUTED BICYCLIC COMPOUNDS AS mPGES-1 INHIBITORS |
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| WO2015059618A1 (en) | 2013-10-22 | 2015-04-30 | Glenmark Pharmaceuticals S.A. | SUBSTITUTED PYRIMIDINE COMPOUNDS AS mPGES-1 INHIBITORS |
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| EP3209660B1 (en) | 2014-10-23 | 2020-06-17 | Deutsches Krebsforschungszentrum Stiftung des öffentlichen Rechts | 1-cyclohexyl-2-phenylaminobenzimidazoles as midh1 inhibitors for the treatment of tumors |
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- 2010-03-04 AR ARP100100651A patent/AR075789A1/es unknown
- 2010-03-04 US US12/717,407 patent/US20100256188A1/en not_active Abandoned
- 2010-03-04 TW TW99106302A patent/TWI466869B/zh not_active IP Right Cessation
- 2010-03-05 SG SG2011063765A patent/SG174250A1/en unknown
- 2010-03-05 EA EA201101243A patent/EA020282B1/ru not_active IP Right Cessation
- 2010-03-05 RS RS20150066A patent/RS53757B1/sr unknown
- 2010-03-05 AP AP2011005807A patent/AP2806A/xx active
- 2010-03-05 NZ NZ594589A patent/NZ594589A/en not_active IP Right Cessation
- 2010-03-05 EP EP10706659.9A patent/EP2403852B8/en active Active
- 2010-03-05 GE GEAP201012405A patent/GEP20146034B/en unknown
- 2010-03-05 CN CN201080010352.5A patent/CN102341395B/zh not_active Expired - Fee Related
- 2010-03-05 CA CA2753149A patent/CA2753149A1/en not_active Abandoned
- 2010-03-05 HR HRP20150096AT patent/HRP20150096T1/hr unknown
- 2010-03-05 BR BRPI1009118A patent/BRPI1009118A2/pt not_active IP Right Cessation
- 2010-03-05 MA MA34131A patent/MA33239B1/ar unknown
- 2010-03-05 WO PCT/EP2010/052799 patent/WO2010100249A1/en not_active Ceased
- 2010-03-05 PL PL10706659T patent/PL2403852T3/pl unknown
- 2010-03-05 MY MYPI2011004122A patent/MY161092A/en unknown
- 2010-03-05 PE PE2011001560A patent/PE20120589A1/es not_active Application Discontinuation
- 2010-03-05 SI SI201030855T patent/SI2403852T1/sl unknown
- 2010-03-05 DK DK10706659.9T patent/DK2403852T3/en active
- 2010-03-05 AU AU2010220263A patent/AU2010220263B2/en not_active Ceased
- 2010-03-05 PT PT107066599T patent/PT2403852E/pt unknown
- 2010-03-05 MX MX2011008948A patent/MX2011008948A/es active IP Right Grant
- 2010-03-05 ME MEP-2015-11A patent/ME02117B/me unknown
- 2010-03-05 JP JP2011552460A patent/JP5433708B2/ja not_active Expired - Fee Related
- 2010-03-05 KR KR1020117020598A patent/KR20110123764A/ko not_active Ceased
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2011
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2012
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2013
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- 2015-01-27 CY CY20151100083T patent/CY1115959T1/el unknown
- 2015-03-09 SM SM201500053T patent/SMT201500053B/xx unknown
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