AR010643A1 - Compuestos de 2-imidazolinilaminoindazol, composicion farmaceutica que lo contiene y uso de dicho compuesto para la fabricacion de un medicamento. - Google Patents

Compuestos de 2-imidazolinilaminoindazol, composicion farmaceutica que lo contiene y uso de dicho compuesto para la fabricacion de un medicamento.

Info

Publication number: AR010643A1
Authority: AR; Argentina
Prior art keywords: hydrogen; compounds; compound; unsubstituted; manufacture
Prior art date: 1996-11-25

Application number

ARP970105524A

Other languages

English (en)

Spanish (es)

Original Assignee

Procter & Gamble

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1996-11-25

Filing date

1997-11-25

Publication date

2000-06-28

1997-11-25 Application filed by Procter & Gamble filed Critical Procter & Gamble

2000-06-28 Publication of AR010643A1 publication Critical patent/AR010643A1/es

Links

150000001875 compounds Chemical class 0.000 title abstract 5
238000004519 manufacturing process Methods 0.000 title abstract 2
239000008194 pharmaceutical composition Substances 0.000 title abstract 2
229940126601 medicinal product Drugs 0.000 title 1
229910052739 hydrogen Inorganic materials 0.000 abstract 4
239000001257 hydrogen Substances 0.000 abstract 4
125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 3
125000006559 (C1-C3) alkylamino group Chemical group 0.000 abstract 2
125000000217 alkyl group Chemical group 0.000 abstract 2
102000030484 alpha-2 Adrenergic Receptor Human genes 0.000 abstract 2
108020004101 alpha-2 Adrenergic Receptor Proteins 0.000 abstract 2
-1 amino, hydroxy, mercapto Chemical class 0.000 abstract 2
208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 2
208000035475 disorder Diseases 0.000 abstract 2
125000004455 (C1-C3) alkylthio group Chemical group 0.000 abstract 1
125000006698 (C1-C3) dialkylamino group Chemical group 0.000 abstract 1
125000006274 (C1-C3)alkoxy group Chemical group 0.000 abstract 1
BAXOFTOLAUCFNW-UHFFFAOYSA-N 1H-indazole Chemical compound C1=CC=C2C=NNC2=C1 BAXOFTOLAUCFNW-UHFFFAOYSA-N 0.000 abstract 1
HBAQYPYDRFILMT-UHFFFAOYSA-N 8-[3-(1-cyclopropylpyrazol-4-yl)-1H-pyrazolo[4,3-d]pyrimidin-5-yl]-3-methyl-3,8-diazabicyclo[3.2.1]octan-2-one Chemical class C1(CC1)N1N=CC(=C1)C1=NNC2=C1N=C(N=C2)N1C2C(N(CC1CC2)C)=O HBAQYPYDRFILMT-UHFFFAOYSA-N 0.000 abstract 1
125000003342 alkenyl group Chemical group 0.000 abstract 1
125000004414 alkyl thio group Chemical group 0.000 abstract 1
150000001408 amides Chemical class 0.000 abstract 1
125000004093 cyano group Chemical group *C#N 0.000 abstract 1
239000003814 drug Substances 0.000 abstract 1
150000002148 esters Chemical class 0.000 abstract 1
229910052736 halogen Inorganic materials 0.000 abstract 1
125000001475 halogen functional group Chemical group 0.000 abstract 1
150000002367 halogens Chemical class 0.000 abstract 1
150000002431 hydrogen Chemical group 0.000 abstract 1
RGVBAADKKPKGQR-UHFFFAOYSA-N n-(4,5-dihydroimidazol-1-yl)-1h-indazol-3-amine Chemical class C1=NCCN1NC1=NNC2=CC=CC=C12 RGVBAADKKPKGQR-UHFFFAOYSA-N 0.000 abstract 1
230000003287 optical effect Effects 0.000 abstract 1
150000003839 salts Chemical class 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/475—Quinolines; Isoquinolines having an indole ring, e.g. yohimbine, reserpine, strychnine, vinblastine
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/16—Otologicals
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
Medicinal Chemistry (AREA)
Animal Behavior & Ethology (AREA)
Life Sciences & Earth Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Bioinformatics & Cheminformatics (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Engineering & Computer Science (AREA)
General Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Biomedical Technology (AREA)
Heart & Thoracic Surgery (AREA)
Ophthalmology & Optometry (AREA)
Cardiology (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Pulmonology (AREA)
Epidemiology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Epoxy Resins (AREA)

ARP970105524A 1996-11-25 1997-11-25 Compuestos de 2-imidazolinilaminoindazol, composicion farmaceutica que lo contiene y uso de dicho compuesto para la fabricacion de un medicamento. AR010643A1 (es)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US3174096P	1996-11-25	1996-11-25

Publications (1)

Publication Number	Publication Date
AR010643A1 true AR010643A1 (es)	2000-06-28

Family

ID=21861136

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
ARP970105524A AR010643A1 (es)	1996-11-25	1997-11-25	Compuestos de 2-imidazolinilaminoindazol, composicion farmaceutica que lo contiene y uso de dicho compuesto para la fabricacion de un medicamento.

Country Status (20)

Country	Link
EP (1)	EP0944620A1 (id)
JP (1)	JP2001506599A (id)
KR (1)	KR20000069104A (id)
CN (1)	CN1244864A (id)
AR (1)	AR010643A1 (id)
AU (1)	AU5433998A (id)
BR (1)	BR9713535A (id)
CA (1)	CA2272644A1 (id)
CO (1)	CO4910166A1 (id)
CZ (1)	CZ183999A3 (id)
HU (1)	HUP9904660A3 (id)
ID (1)	ID22676A (id)
IL (1)	IL130067A0 (id)
NO (1)	NO992502L (id)
NZ (1)	NZ335882A (id)
PE (1)	PE47099A1 (id)
SK (1)	SK69699A3 (id)
TR (1)	TR199901542T2 (id)
WO (1)	WO1998023609A1 (id)
ZA (1)	ZA9710576B (id)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB9908175D0 (en) *	1999-04-09	1999-06-02	Lilly Co Eli	Method of treating neurological disorders
US6433186B1 (en)	2000-08-16	2002-08-13	Astrazeneca Ab	Amidino derivatives and their use as thormbin inhibitors
EP2226315A4 (en)	2007-12-28	2012-01-25	Carna Biosciences Inc	2-aminoquinazoline DERIVATIVE
WO2010074753A1 (en)	2008-12-23	2010-07-01	Map Pharmaceuticals, Inc.	Inhalation devices and related methods for administration of sedative hypnotic compounds
CN112538074A (zh) *	2020-12-24	2021-03-23	艾希尔（深圳）药物研发有限公司	一种溴莫尼定脱溴杂质的制备方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
CH641782A5 (en) *	1978-12-07	1984-03-15	Siegfried Ag	1H- and 2H-indazole derivatives
US4526898A (en) *	1980-09-05	1985-07-02	Siegfried Aktiengesselschaft	Antihypertensive 4-(2-imidazolin-2-yl-amino)-2-methyl-indazole
US5478858A (en) *	1993-12-17	1995-12-26	The Procter & Gamble Company	5-(2-imidazolinylamino) benzimidazole compounds useful as alpha-2 adrenoceptor agonists
SG44628A1 (en) *	1993-12-17	1997-12-19	Procter & Gamble	6-(2-imidazolinylamino) Quinoxaline compounds useful as alpha-2 adrenoceptor agonists

1997
- 1997-11-21 ID IDW990412A patent/ID22676A/id unknown
- 1997-11-21 CZ CZ991839A patent/CZ183999A3/cs unknown
- 1997-11-21 BR BR9713535A patent/BR9713535A/pt unknown
- 1997-11-21 CA CA002272644A patent/CA2272644A1/en not_active Abandoned
- 1997-11-21 CN CN97181453A patent/CN1244864A/zh active Pending
- 1997-11-21 TR TR1999/01542T patent/TR199901542T2/xx unknown
- 1997-11-21 NZ NZ335882A patent/NZ335882A/xx unknown
- 1997-11-21 JP JP52468698A patent/JP2001506599A/ja active Pending
- 1997-11-21 WO PCT/US1997/020551 patent/WO1998023609A1/en not_active Ceased
- 1997-11-21 HU HU9904660A patent/HUP9904660A3/hu unknown
- 1997-11-21 KR KR1019997004569A patent/KR20000069104A/ko not_active Ceased
- 1997-11-21 EP EP97948238A patent/EP0944620A1/en not_active Withdrawn
- 1997-11-21 AU AU54339/98A patent/AU5433998A/en not_active Abandoned
- 1997-11-21 IL IL13006797A patent/IL130067A0/xx unknown
- 1997-11-24 CO CO97068615A patent/CO4910166A1/es unknown
- 1997-11-25 PE PE1997001067A patent/PE47099A1/es not_active Application Discontinuation
- 1997-11-25 ZA ZA9710576A patent/ZA9710576B/xx unknown
- 1997-11-25 AR ARP970105524A patent/AR010643A1/es unknown
1999
- 1999-05-25 NO NO992502A patent/NO992502L/no not_active Application Discontinuation
- 1999-05-25 SK SK696-99A patent/SK69699A3/sk unknown

Also Published As

Publication number	Publication date
IL130067A0 (en)	2000-02-29
WO1998023609A1 (en)	1998-06-04
SK69699A3 (en)	2000-06-12
CZ183999A3 (cs)	1999-11-17
CA2272644A1 (en)	1998-06-04
HUP9904660A3 (en)	2002-02-28
CO4910166A1 (es)	2000-04-24
BR9713535A (pt)	2000-03-21
CN1244864A (zh)	2000-02-16
NZ335882A (en)	2000-12-22
ID22676A (id)	1999-12-09
PE47099A1 (es)	1999-06-12
NO992502L (no)	1999-07-26
ZA9710576B (en)	1998-09-16
TR199901542T2 (xx)	2000-01-21
NO992502D0 (no)	1999-05-25
HUP9904660A2 (hu)	2000-06-28
JP2001506599A (ja)	2001-05-22
KR20000069104A (ko)	2000-11-25
EP0944620A1 (en)	1999-09-29
AU5433998A (en)	1998-06-22

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