AT257038B - Verfahren zur Herstellung von Aminoacylanalogen von Cephalosporin C - Google Patents

Verfahren zur Herstellung von Aminoacylanalogen von Cephalosporin C

Info

Publication number
AT257038B
AT257038B AT579463A AT579463A AT257038B AT 257038 B AT257038 B AT 257038B AT 579463 A AT579463 A AT 579463A AT 579463 A AT579463 A AT 579463A AT 257038 B AT257038 B AT 257038B
Authority
AT
Austria
Prior art keywords
aminoacyl
cephalosporin
analogs
preparation
aminoacyl analogs
Prior art date
Application number
AT579463A
Other languages
German (de)
English (en)
Original Assignee
Glaxo Lab Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Lab Ltd filed Critical Glaxo Lab Ltd
Application granted granted Critical
Publication of AT257038B publication Critical patent/AT257038B/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D501/00Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/207-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
    • C07D501/247-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3
    • C07D501/26Methylene radicals, substituted by oxygen atoms; Lactones thereof with the 2-carboxyl group
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • A61K31/542Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/545Compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins, cefaclor, or cephalexine
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D501/00Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/207-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
    • C07D501/247-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3
    • C07D501/26Methylene radicals, substituted by oxygen atoms; Lactones thereof with the 2-carboxyl group
    • C07D501/32Methylene radicals, substituted by oxygen atoms; Lactones thereof with the 2-carboxyl group with the 7-amino radical acylated by an araliphatic carboxylic acid, which is substituted on the aliphatic radical by hetero atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Cephalosporin Compounds (AREA)
AT579463A 1962-07-20 1963-07-19 Verfahren zur Herstellung von Aminoacylanalogen von Cephalosporin C AT257038B (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB2803962 1962-07-20

Publications (1)

Publication Number Publication Date
AT257038B true AT257038B (de) 1967-09-25

Family

ID=10269280

Family Applications (1)

Application Number Title Priority Date Filing Date
AT579463A AT257038B (de) 1962-07-20 1963-07-19 Verfahren zur Herstellung von Aminoacylanalogen von Cephalosporin C

Country Status (8)

Country Link
AT (1) AT257038B (fr)
CH (1) CH441323A (fr)
DE (1) DE1445822C3 (fr)
DK (1) DK118083B (fr)
ES (1) ES289733A1 (fr)
FR (1) FR3065M (fr)
NL (1) NL142164B (fr)
SE (1) SE334891B (fr)

Also Published As

Publication number Publication date
DE1445822C3 (de) 1973-12-13
NL142164B (nl) 1974-05-15
DE1445822B2 (de) 1973-05-24
CH441323A (de) 1967-08-15
SE334891B (fr) 1971-05-10
DE1445822A1 (de) 1969-04-17
FR3065M (fr) 1965-01-18
ES289733A1 (es) 1963-12-01
DK118083B (da) 1970-07-06

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