ATE100107T1 - Heterozyklische verbindungen und ihre herstellung und verwendung. - Google Patents

Heterozyklische verbindungen und ihre herstellung und verwendung.

Info

Publication number: ATE100107T1
Authority: AT; Austria
Prior art keywords: heterocyclic compounds; chem; alkyl; production; compounds
Prior art date: 1987-10-06

Application number

AT88309153T

Other languages

English (en)

Inventor

Frank Waetjen

Holger Claus Hansen

Original Assignee

Novo Nordisk As

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1987-10-06

Filing date

1988-10-03

Publication date

1994-01-15

1988-10-03 Application filed by Novo Nordisk As filed Critical Novo Nordisk As

1994-01-15 Application granted granted Critical

1994-01-15 Publication of ATE100107T1 publication Critical patent/ATE100107T1/de

Links

150000002391 heterocyclic compounds Chemical class 0.000 title abstract 2
125000004169 (C1-C6) alkyl group Chemical group 0.000 abstract 3
125000006272 (C3-C7) cycloalkyl group Chemical group 0.000 abstract 1
241000124008 Mammalia Species 0.000 abstract 1
229940125681 anticonvulsant agent Drugs 0.000 abstract 1
239000001961 anticonvulsive agent Substances 0.000 abstract 1
239000002249 anxiolytic agent Substances 0.000 abstract 1
230000000949 anxiolytic effect Effects 0.000 abstract 1
229940005530 anxiolytics Drugs 0.000 abstract 1
125000003118 aryl group Chemical group 0.000 abstract 1
210000004556 brain Anatomy 0.000 abstract 1
230000003920 cognitive function Effects 0.000 abstract 1
150000001875 compounds Chemical class 0.000 abstract 1
229910052739 hydrogen Inorganic materials 0.000 abstract 1
239000001257 hydrogen Substances 0.000 abstract 1
125000004435 hydrogen atom Chemical class [H]* 0.000 abstract 1
239000003326 hypnotic agent Substances 0.000 abstract 1
230000000147 hypnotic effect Effects 0.000 abstract 1
238000002360 preparation method Methods 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
- C07D495/14—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives

Landscapes

Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
Organic Chemistry (AREA)
Veterinary Medicine (AREA)
Medicinal Chemistry (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Animal Behavior & Ethology (AREA)
Life Sciences & Earth Sciences (AREA)
Pharmacology & Pharmacy (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Engineering & Computer Science (AREA)
Biomedical Technology (AREA)
Chemical Kinetics & Catalysis (AREA)
Bioinformatics & Cheminformatics (AREA)
Neurosurgery (AREA)
Neurology (AREA)
Anesthesiology (AREA)
Pain & Pain Management (AREA)
Epidemiology (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Preparation Of Compounds By Using Micro-Organisms (AREA)
Plural Heterocyclic Compounds (AREA)
Agricultural Chemicals And Associated Chemicals (AREA)

AT88309153T 1987-10-06 1988-10-03 Heterozyklische verbindungen und ihre herstellung und verwendung. ATE100107T1 (de)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
DK522187A DK522187D0 (da)	1987-10-06	1987-10-06	Imidozothienopyrimidiner, deres fremstilling og anvendelse
EP88309153A EP0311321B1 (de)	1987-10-06	1988-10-03	Heterozyklische Verbindungen und ihre Herstellung und Verwendung

Publications (1)

Publication Number	Publication Date
ATE100107T1 true ATE100107T1 (de)	1994-01-15

Family

ID=8140567

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT88309153T ATE100107T1 (de)	1987-10-06	1988-10-03	Heterozyklische verbindungen und ihre herstellung und verwendung.

Country Status (18)

Country	Link
US (1)	US4866065A (de)
EP (1)	EP0311321B1 (de)
JP (1)	JP2662426B2 (de)
KR (1)	KR0130978B1 (de)
AT (1)	ATE100107T1 (de)
AU (1)	AU611718B2 (de)
CA (1)	CA1323365C (de)
DE (1)	DE3887064T2 (de)
DK (1)	DK522187D0 (de)
ES (1)	ES2061675T3 (de)
FI (1)	FI91759C (de)
IE (1)	IE64931B1 (de)
IL (1)	IL87780A (de)
NO (1)	NO168646C (de)
NZ (1)	NZ226461A (de)
PH (1)	PH25297A (de)
PT (1)	PT88673B (de)
ZA (1)	ZA887313B (de)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5185446A (en) *	1990-09-04	1993-02-09	Neurogen Corporation	Certain cycloalkyl imidazopyrimidines; a new class of gaba brainreceptor ligands
FR2872165B1 (fr) *	2004-06-24	2006-09-22	Sod Conseils Rech Applic	Nouveaux derives de pyrimido-benzimidazole
US20070208040A1 (en) *	2006-03-02	2007-09-06	Elfatih Elzein	A2a adenosine receptor antagonists

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE2411274A1 (de) *	1974-03-06	1975-09-18	Schering Ag	Neue 2-nitrothieno eckige klammer auf 2,3-d eckige klammer zu pyrimidinon-derivate und verfahren zu ihrer herstellung
CA1142924A (en) *	1980-06-27	1983-03-15	Hoffmann-La Roche Limited	Pyrimidine derivatives
GB8432073D0 (en) *	1984-12-19	1985-01-30	Roussel Lab Ltd	Chemical compounds
AU587802B2 (en) *	1985-03-08	1989-08-31	Ferrosan A/S	Novel oxadiazolyl imidazobenzodiazepine derivatives and methods of preparing such compounds
US4622320A (en) *	1985-05-17	1986-11-11	As Ferrosan	Oxadiazolylimidazobenzodiazepine, compositions, and method
US4771051A (en) *	1985-05-17	1988-09-13	A/S Ferrosan	3-substituted-4,5-dihydro-5-oxo imidazoquinazolines, their preparation, and their use in treating benzodiazepin receptor-related ailments
DE3686723T2 (de) *	1985-10-17	1993-04-01	Novonordisk As	Oxadiazolylacetonitrile, ihre herstellung und anwendung.

1987
- 1987-10-06 DK DK522187A patent/DK522187D0/da not_active Application Discontinuation
1988
- 1988-09-15 IE IE279488A patent/IE64931B1/en not_active IP Right Cessation
- 1988-09-16 IL IL87780A patent/IL87780A/xx not_active IP Right Cessation
- 1988-09-29 ZA ZA887313A patent/ZA887313B/xx unknown
- 1988-10-03 EP EP88309153A patent/EP0311321B1/de not_active Expired - Lifetime
- 1988-10-03 DE DE88309153T patent/DE3887064T2/de not_active Expired - Fee Related
- 1988-10-03 AU AU23341/88A patent/AU611718B2/en not_active Ceased
- 1988-10-03 AT AT88309153T patent/ATE100107T1/de not_active IP Right Cessation
- 1988-10-03 ES ES88309153T patent/ES2061675T3/es not_active Expired - Lifetime
- 1988-10-04 NZ NZ226461A patent/NZ226461A/xx unknown
- 1988-10-04 KR KR1019880012905A patent/KR0130978B1/ko not_active Expired - Fee Related
- 1988-10-04 PT PT88673A patent/PT88673B/pt not_active IP Right Cessation
- 1988-10-05 CA CA000579431A patent/CA1323365C/en not_active Expired - Fee Related
- 1988-10-05 NO NO884431A patent/NO168646C/no unknown
- 1988-10-06 FI FI884595A patent/FI91759C/fi not_active IP Right Cessation
- 1988-10-06 US US07/254,421 patent/US4866065A/en not_active Expired - Fee Related
- 1988-10-06 PH PH8837645A patent/PH25297A/en unknown
- 1988-10-06 JP JP63251001A patent/JP2662426B2/ja not_active Expired - Lifetime

Also Published As

Publication number	Publication date
AU2334188A (en)	1989-04-06
DE3887064D1 (de)	1994-02-24
FI884595A7 (fi)	1989-04-07
EP0311321A3 (en)	1990-08-01
NZ226461A (en)	1990-05-28
FI884595A0 (fi)	1988-10-06
NO168646C (no)	1992-03-18
ZA887313B (en)	1989-06-28
KR890006653A (ko)	1989-06-15
NO884431L (no)	1989-04-07
IE882794L (en)	1989-04-06
FI91759C (fi)	1994-08-10
IL87780A (en)	1992-02-16
JP2662426B2 (ja)	1997-10-15
KR0130978B1 (ko)	1998-04-16
NO168646B (no)	1991-12-09
EP0311321A2 (de)	1989-04-12
NO884431D0 (no)	1988-10-05
FI91759B (fi)	1994-04-29
JPH01121291A (ja)	1989-05-12
EP0311321B1 (de)	1994-01-12
ES2061675T3 (es)	1994-12-16
PT88673B (pt)	1992-12-31
CA1323365C (en)	1993-10-19
IE64931B1 (en)	1995-09-20
DE3887064T2 (de)	1994-05-05
US4866065A (en)	1989-09-12
PH25297A (en)	1991-04-30
AU611718B2 (en)	1991-06-20
DK522187D0 (da)	1987-10-06

Legal Events

Date	Code	Title	Description
1994-09-15	UEP	Publication of translation of european patent specification
1999-07-15	REN	Ceased due to non-payment of the annual fee

Publication	Publication Date	Title
DE69329018D1 (de)	2000-08-17	Heterocyclische verbindungen, deren herstellung und verwendung
ATE109147T1 (de)	1994-08-15	Imidazochinoxalinverbindungen und ihre herstellung und verwendung.
DE3883033D1 (de)	1993-09-16	Heterocyclische verbindungen und ihre herstellung und anwendung.
ATE111100T1 (de)	1994-09-15	Imidazochinoxalinverbindungen und ihre herstellung und verwendung.
DE3766401D1 (de)	1991-01-10	Benzodiazepinderivate und ihre herstellung und verwendung.
ATE44381T1 (de)	1989-07-15	Heterocyclische verbindungen und ihre herstellung und verwendung.
DE3887064D1 (de)	1994-02-24	Heterozyklische Verbindungen und ihre Herstellung und Verwendung.
NO180635C (no)	1997-05-21	Analogifremgangsmåte for fremstilling av en terapeutisk aktiv tetracyklisk imidazolinforbindelse
ATE142209T1 (de)	1996-09-15	Heterocyclische verbindungen, herstellung und verwendung