ATE102206T1 - 6-(substituiertes methylen)peneme. - Google Patents
6-(substituiertes methylen)peneme.Info
- Publication number
- ATE102206T1 ATE102206T1 AT88311786T AT88311786T ATE102206T1 AT E102206 T1 ATE102206 T1 AT E102206T1 AT 88311786 T AT88311786 T AT 88311786T AT 88311786 T AT88311786 T AT 88311786T AT E102206 T1 ATE102206 T1 AT E102206T1
- Authority
- AT
- Austria
- Prior art keywords
- penems
- substituted methylene
- vivo hydrolysable
- denotes
- compounds
- Prior art date
Links
- 125000001570 methylene group Chemical class [H]C([H])([*:1])[*:2] 0.000 title 1
- 150000002961 penems Chemical class 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 2
- 238000001727 in vivo Methods 0.000 abstract 2
- 108090000204 Dipeptidase 1 Proteins 0.000 abstract 1
- 125000002252 acyl group Chemical group 0.000 abstract 1
- 230000000844 anti-bacterial effect Effects 0.000 abstract 1
- 102000006635 beta-lactamase Human genes 0.000 abstract 1
- 150000002148 esters Chemical class 0.000 abstract 1
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 1
- 230000002401 inhibitory effect Effects 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C07D499/88—Compounds with a double bond between positions 2 and 3 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Oncology (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Communicable Diseases (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Steroid Compounds (AREA)
- Photoreceptors In Electrophotography (AREA)
- Cephalosporin Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pens And Brushes (AREA)
- Medicines Containing Material From Animals Or Micro-Organisms (AREA)
- Peptides Or Proteins (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Mechanical Treatment Of Semiconductor (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB878729613A GB8729613D0 (en) | 1987-12-18 | 1987-12-18 | Novel compounds |
| EP88311786A EP0321186B1 (de) | 1987-12-18 | 1988-12-13 | 6-(Substituiertes Methylen)peneme |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE102206T1 true ATE102206T1 (de) | 1994-03-15 |
Family
ID=10628729
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT88311786T ATE102206T1 (de) | 1987-12-18 | 1988-12-13 | 6-(substituiertes methylen)peneme. |
Country Status (13)
| Country | Link |
|---|---|
| US (1) | US4923856A (de) |
| EP (1) | EP0321186B1 (de) |
| JP (1) | JPH02287A (de) |
| KR (1) | KR890009938A (de) |
| AT (1) | ATE102206T1 (de) |
| AU (1) | AU621846B2 (de) |
| CA (1) | CA1302402C (de) |
| DE (1) | DE3888127T2 (de) |
| DK (1) | DK702488A (de) |
| GB (1) | GB8729613D0 (de) |
| NZ (1) | NZ227355A (de) |
| PT (1) | PT89236B (de) |
| ZA (1) | ZA889397B (de) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4945466A (en) * | 1989-02-22 | 1990-07-31 | Borland Walter G | Resonant switching converter |
| AR039476A1 (es) * | 2002-05-01 | 2005-02-23 | Wyeth Corp | Proceso para preparar derivados de 6-alquiliden penem |
| AR039475A1 (es) | 2002-05-01 | 2005-02-23 | Wyeth Corp | 6-alquiliden-penems triciclicos como inhibidores de beta-lactamasa |
| AR039774A1 (es) | 2002-05-01 | 2005-03-02 | Wyeth Corp | 6-alquiliden-penems biciclicos como inhibidores de beta-lactamasas |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FI82471C (fi) * | 1984-01-26 | 1991-03-11 | Beecham Group Plc | Foerfarande foer framstaellning av farmakologiskt aktiva 6-metylenpenemderivater. |
| US4826833A (en) * | 1984-01-30 | 1989-05-02 | Pfizer Inc. | 6-(Substituted)methylene-penicillanic and 6-(substituted)hydroxymethylpenicillanic acids and derivatives thereof |
| GB8518422D0 (en) * | 1985-07-22 | 1985-08-29 | Beecham Group Plc | Compounds |
| GB8711391D0 (en) * | 1987-05-14 | 1987-06-17 | Beecham Group Plc | Process |
-
1987
- 1987-12-18 GB GB878729613A patent/GB8729613D0/en active Pending
-
1988
- 1988-12-13 AT AT88311786T patent/ATE102206T1/de not_active IP Right Cessation
- 1988-12-13 EP EP88311786A patent/EP0321186B1/de not_active Expired - Lifetime
- 1988-12-13 DE DE3888127T patent/DE3888127T2/de not_active Expired - Fee Related
- 1988-12-15 ZA ZA889397A patent/ZA889397B/xx unknown
- 1988-12-16 NZ NZ227355A patent/NZ227355A/en unknown
- 1988-12-16 US US07/286,375 patent/US4923856A/en not_active Expired - Fee Related
- 1988-12-16 AU AU26931/88A patent/AU621846B2/en not_active Ceased
- 1988-12-16 CA CA000586210A patent/CA1302402C/en not_active Expired - Fee Related
- 1988-12-16 PT PT89236A patent/PT89236B/pt not_active IP Right Cessation
- 1988-12-16 DK DK702488A patent/DK702488A/da not_active Application Discontinuation
- 1988-12-17 KR KR1019880016903A patent/KR890009938A/ko not_active Withdrawn
- 1988-12-19 JP JP63320334A patent/JPH02287A/ja active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| EP0321186A1 (de) | 1989-06-21 |
| ZA889397B (en) | 1990-08-29 |
| PT89236A (pt) | 1989-12-29 |
| EP0321186B1 (de) | 1994-03-02 |
| DK702488D0 (da) | 1988-12-16 |
| CA1302402C (en) | 1992-06-02 |
| DE3888127D1 (de) | 1994-04-07 |
| JPH02287A (ja) | 1990-01-05 |
| US4923856A (en) | 1990-05-08 |
| AU621846B2 (en) | 1992-03-26 |
| PT89236B (pt) | 1993-07-30 |
| AU2693188A (en) | 1989-06-22 |
| GB8729613D0 (en) | 1988-02-03 |
| DK702488A (da) | 1989-06-19 |
| KR890009938A (ko) | 1989-08-05 |
| NZ227355A (en) | 1991-04-26 |
| DE3888127T2 (de) | 1994-07-07 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| WO2001007433A3 (en) | Quinoline derivatives and their use as antibacterial agents | |
| IL133409A0 (en) | Retroviral protease inhibiting compounds | |
| ATE110729T1 (de) | Cephalosporinverbindungen, verfahren zu ihrer herstellung und antibakterielle mittel. | |
| MY101970A (en) | Zwitterionic bicyclic compounds and their salts, solvates, hydrates and esters. | |
| FI911286A0 (fi) | Kemiska foereningar. | |
| LU83820A1 (fr) | Derives de la 2-oxoazetidine,leur preparation et leur utilisation | |
| IE782546L (en) | Amino-thiazolyl cephalosporins | |
| ATE97901T1 (de) | Cephalosporinderivate, verfahren zu ihrer herstellung sowie entsprechende pharmazeutische praeparate. | |
| ES2089136T3 (es) | Tratamiento de enfermedades inflamatorias con la ayuda de derivados 15-ceto-prostaglandinas. | |
| DK297385A (da) | Carbapenemer med externt alkyleret mono- eller bicyclisk heteroarylalkylthiosubstituent samt laegemiddel indeholdende saadanne forbindelser | |
| ATE102206T1 (de) | 6-(substituiertes methylen)peneme. | |
| DE3876712D1 (de) | Antianaerobe naphthyridinverbindungen. | |
| FI915245A0 (fi) | 7-acyl-3-(substitueradkarbamoyloxi) cefemfoereningar samt foerfarande foer framstaellning av dessa. | |
| ATE140460T1 (de) | Echinocandin-b-derivat | |
| NO911081L (no) | Fremgangsmaate for fremstilling av substituerte puriner, og deres anvendelse som antivirale midler. | |
| EP0487996B1 (de) | 3-substituierte Cephalosporine, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel | |
| FI880334A0 (fi) | 6- (substituerad)-(s)-hydroximetyl -penicillansyror och derivat daerav. | |
| FI880385A0 (fi) | Substituerade 3-fenyl-7h-tiazolo /3,2-b//1,2,4/-triazin-7-oner, foerfaranden foer deras framstaellning, dessa innehaollande laekemedel och deras anvaendning, samt naogra vid framstaellningen av naemnda foereningar bildade mellanprodukter. | |
| ES8503353A1 (es) | Un procedimiento para la preparacion de derivados del acido clavolanico. | |
| SU1573800A1 (ru) | Производные о-аминобензойной кислоты, обладающие фунгицидными свойствами |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| RER | Ceased as to paragraph 5 lit. 3 law introducing patent treaties |