ATE111884T1 - Verfahren zur herstellung von eicosatetraynsäure. - Google Patents

Verfahren zur herstellung von eicosatetraynsäure.

Info

Publication number: ATE111884T1
Authority: AT; Austria
Prior art keywords: nitrogen; oxygen; heterocyclic ring; treatment; hydrogen atom
Prior art date: 1986-12-31

Application number

AT91101995T

Other languages

English (en)

Inventor

Braham Shroot

Christopher Hensby

Jean Maignan

Gerard Lang

Serge Restle

Michel Colin

Original Assignee

Cird Galderma

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1986-12-31

Filing date

1987-12-30

Publication date

1994-10-15

1987-12-30 Application filed by Cird Galderma filed Critical Cird Galderma

1994-10-15 Application granted granted Critical

1994-10-15 Publication of ATE111884T1 publication Critical patent/ATE111884T1/de

Links

239000002253 acid Substances 0.000 title 1
IJGRMHOSHXDMSA-UHFFFAOYSA-N Atomic nitrogen Chemical compound N#N IJGRMHOSHXDMSA-UHFFFAOYSA-N 0.000 abstract 4
229910052757 nitrogen Inorganic materials 0.000 abstract 3
NINIDFKCEFEMDL-UHFFFAOYSA-N Sulfur Chemical compound [S] NINIDFKCEFEMDL-UHFFFAOYSA-N 0.000 abstract 2
125000003277 amino group Chemical group 0.000 abstract 2
QVGXLLKOCUKJST-UHFFFAOYSA-N atomic oxygen Chemical compound [O] QVGXLLKOCUKJST-UHFFFAOYSA-N 0.000 abstract 2
150000001875 compounds Chemical class 0.000 abstract 2
125000005842 heteroatom Chemical group 0.000 abstract 2
125000000623 heterocyclic group Chemical group 0.000 abstract 2
125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 2
229910052760 oxygen Inorganic materials 0.000 abstract 2
239000001301 oxygen Substances 0.000 abstract 2
238000011282 treatment Methods 0.000 abstract 2
201000004624 Dermatitis Diseases 0.000 abstract 1
239000005864 Sulphur Substances 0.000 abstract 1
125000000217 alkyl group Chemical group 0.000 abstract 1
208000026935 allergic disease Diseases 0.000 abstract 1
125000002887 hydroxy group Chemical group [H]O* 0.000 abstract 1
125000002768 hydroxyalkyl group Chemical group 0.000 abstract 1
208000027866 inflammatory disease Diseases 0.000 abstract 1
150000007522 mineralic acids Chemical class 0.000 abstract 1
125000004433 nitrogen atom Chemical group N* 0.000 abstract 1
150000007524 organic acids Chemical class 0.000 abstract 1
235000005985 organic acids Nutrition 0.000 abstract 1
238000011321 prophylaxis Methods 0.000 abstract 1
150000003839 salts Chemical class 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
- C07D295/18—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carboxylic acids, or sulfur or nitrogen analogues thereof
- C07D295/182—Radicals derived from carboxylic acids
- C07D295/185—Radicals derived from carboxylic acids from aliphatic carboxylic acids
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C21/00—Acyclic unsaturated compounds containing halogen atoms
- C07C21/22—Acyclic unsaturated compounds containing halogen atoms containing carbon-to-carbon triple bonds
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C231/00—Preparation of carboxylic acid amides
- C07C231/02—Preparation of carboxylic acid amides from carboxylic acids or from esters, anhydrides, or halides thereof by reaction with ammonia or amines
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C233/00—Carboxylic acid amides
- C07C233/01—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms
- C07C233/16—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by singly-bound oxygen atoms
- C07C233/17—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by singly-bound oxygen atoms with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom
- C07C233/20—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by singly-bound oxygen atoms with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom having the carbon atom of the carboxamide group bound to a carbon atom of an acyclic unsaturated carbon skeleton
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C51/00—Preparation of carboxylic acids or their salts, halides or anhydrides
- C07C51/347—Preparation of carboxylic acids or their salts, halides or anhydrides by reactions not involving formation of carboxyl groups
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C51/00—Preparation of carboxylic acids or their salts, halides or anhydrides
- C07C51/347—Preparation of carboxylic acids or their salts, halides or anhydrides by reactions not involving formation of carboxyl groups
- C07C51/353—Preparation of carboxylic acids or their salts, halides or anhydrides by reactions not involving formation of carboxyl groups by isomerisation; by change of size of the carbon skeleton
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C57/00—Unsaturated compounds having carboxyl groups bound to acyclic carbon atoms
- C07C57/18—Unsaturated compounds having carboxyl groups bound to acyclic carbon atoms with only carbon-to-carbon triple bonds as unsaturation

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Engineering & Computer Science (AREA)
Oil, Petroleum & Natural Gas (AREA)
Life Sciences & Earth Sciences (AREA)
Veterinary Medicine (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Bioinformatics & Cheminformatics (AREA)
Pain & Pain Management (AREA)
Immunology (AREA)
Rheumatology (AREA)
Dermatology (AREA)
Pulmonology (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Cosmetics (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Measuring Or Testing Involving Enzymes Or Micro-Organisms (AREA)

AT91101995T 1986-12-31 1987-12-30 Verfahren zur herstellung von eicosatetraynsäure. ATE111884T1 (de)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
FR8618419A FR2609026B1 (fr)	1986-12-31	1986-12-31	Amides de l'acide eicosatetraynoique et leur application en pharmacie et en cosmetique

Publications (1)

Publication Number	Publication Date
ATE111884T1 true ATE111884T1 (de)	1994-10-15

Family

ID=9342478

Family Applications (2)

Application Number	Title	Priority Date	Filing Date
AT87119357T ATE86973T1 (de)	1986-12-31	1987-12-30	Eicosattraynsaeureamide, ihre verwendung in der arzneimittelkunde und kosmetika, ihre herstellung und verfahren zur herstellung von eicosattraynsaeure.
AT91101995T ATE111884T1 (de)	1986-12-31	1987-12-30	Verfahren zur herstellung von eicosatetraynsäure.

Family Applications Before (1)

Application Number	Title	Priority Date	Filing Date
AT87119357T ATE86973T1 (de)	1986-12-31	1987-12-30	Eicosattraynsaeureamide, ihre verwendung in der arzneimittelkunde und kosmetika, ihre herstellung und verfahren zur herstellung von eicosattraynsaeure.

Country Status (15)

Country	Link
US (1)	US4916136A (de)
EP (2)	EP0433267B1 (de)
JP (1)	JP2554683B2 (de)
AT (2)	ATE86973T1 (de)
AU (2)	AU606111B2 (de)
CA (2)	CA1299182C (de)
DE (2)	DE3750587T2 (de)
DK (1)	DK688587A (de)
FI (1)	FI875749A7 (de)
FR (1)	FR2609026B1 (de)
IE (1)	IE873551L (de)
NO (1)	NO875447L (de)
NZ (1)	NZ223070A (de)
PT (1)	PT86475B (de)
ZA (1)	ZA879726B (de)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
NZ216751A (en) *	1985-07-05	1990-01-29	Cird	Eicosatriynoic acid esters and amides,pharmaceutical compositions and process for preparing eicosatriynoic acid
FR2609026B1 (fr) *	1986-12-31	1989-03-31	Cird	Amides de l'acide eicosatetraynoique et leur application en pharmacie et en cosmetique
US5429394A (en) *	1993-11-15	1995-07-04	Dana Corporation	Quick connect cartridge assembly with plug
US7191000B2 (en) *	2001-07-31	2007-03-13	Cardiac Pacemakers, Inc.	Cardiac rhythm management system for edema
MX2008009215A (es) *	2006-01-17	2008-12-10	Barrier Therapeutics Inc	Tratamiento de trastornos inflamatorios con compuestos de triazol.

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB859897A (en) *	1958-07-05	1961-01-25	Roche Products Ltd	Novel unsaturated acids and esters thereof and a process for the manufacture and conversion of same
US4190669A (en) *	1976-03-08	1980-02-26	The Regents Of The University Of Michigan	Method for treating psoriasis
US4497827A (en) *	1982-08-30	1985-02-05	Syntex (U.S.A.) Inc.	Arachidonic acid analogues as anti-inflammatory and anti-allergic agents
US4619938A (en) *	1984-03-21	1986-10-28	Terumo Kabushiki Kaisha	Fatty acid derivatives of aminoalkyl nicotinic acid esters and platelet aggregation inhibitors
NZ216751A (en) *	1985-07-05	1990-01-29	Cird	Eicosatriynoic acid esters and amides,pharmaceutical compositions and process for preparing eicosatriynoic acid
FR2609026B1 (fr) *	1986-12-31	1989-03-31	Cird	Amides de l'acide eicosatetraynoique et leur application en pharmacie et en cosmetique

1986
- 1986-12-31 FR FR8618419A patent/FR2609026B1/fr not_active Expired
1987
- 1987-12-23 NZ NZ223070A patent/NZ223070A/xx unknown
- 1987-12-28 US US07/138,791 patent/US4916136A/en not_active Expired - Lifetime
- 1987-12-28 DK DK688587A patent/DK688587A/da not_active Application Discontinuation
- 1987-12-28 NO NO875447A patent/NO875447L/no unknown
- 1987-12-29 PT PT86475A patent/PT86475B/pt not_active IP Right Cessation
- 1987-12-29 ZA ZA879726A patent/ZA879726B/xx unknown
- 1987-12-29 FI FI875749A patent/FI875749A7/fi not_active Application Discontinuation
- 1987-12-29 JP JP62336805A patent/JP2554683B2/ja not_active Expired - Fee Related
- 1987-12-30 EP EP91101995A patent/EP0433267B1/de not_active Expired - Lifetime
- 1987-12-30 AT AT87119357T patent/ATE86973T1/de active
- 1987-12-30 EP EP87119357A patent/EP0279954B1/de not_active Expired - Lifetime
- 1987-12-30 DE DE3750587T patent/DE3750587T2/de not_active Expired - Fee Related
- 1987-12-30 IE IE873551A patent/IE873551L/xx unknown
- 1987-12-30 AT AT91101995T patent/ATE111884T1/de not_active IP Right Cessation
- 1987-12-30 AU AU83139/87A patent/AU606111B2/en not_active Ceased
- 1987-12-30 DE DE8787119357T patent/DE3784913T2/de not_active Expired - Fee Related
- 1987-12-31 CA CA000555730A patent/CA1299182C/fr not_active Expired - Lifetime
1990
- 1990-05-31 CA CA000615760A patent/CA1300642C/fr not_active Expired - Lifetime
- 1990-11-06 AU AU65818/90A patent/AU629422B2/en not_active Expired - Fee Related

Also Published As

Publication number	Publication date
AU606111B2 (en)	1991-01-31
EP0279954A3 (en)	1988-10-26
EP0279954B1 (de)	1993-03-17
US4916136A (en)	1990-04-10
FR2609026B1 (fr)	1989-03-31
DK688587D0 (da)	1987-12-28
ATE86973T1 (de)	1993-04-15
EP0279954A2 (de)	1988-08-31
NZ223070A (en)	1990-07-26
NO875447L (no)	1988-07-01
JPS63253059A (ja)	1988-10-20
EP0433267B1 (de)	1994-09-21
FI875749A0 (fi)	1987-12-29
ZA879726B (en)	1989-08-30
NO875447D0 (no)	1987-12-28
CA1299182C (fr)	1992-04-21
AU8313987A (en)	1988-07-07
JP2554683B2 (ja)	1996-11-13
PT86475A (fr)	1988-01-01
CA1300642C (fr)	1992-05-12
PT86475B (pt)	1990-11-20
FI875749A7 (fi)	1988-07-01
DE3750587T2 (de)	1995-01-26
AU629422B2 (en)	1992-10-01
EP0433267A3 (en)	1991-10-23
DE3784913T2 (de)	1993-06-24
DE3784913D1 (de)	1993-04-22
FR2609026A1 (fr)	1988-07-01
AU6581890A (en)	1991-02-28
EP0433267A2 (de)	1991-06-19
DE3750587D1 (de)	1994-10-27
DK688587A (da)	1988-07-01
IE873551L (en)	1988-06-30

Legal Events

Date	Code	Title	Description
1995-03-15	RER	Ceased as to paragraph 5 lit. 3 law introducing patent treaties

Publication	Publication Date	Title
ATE21699T1 (de)	1986-09-15	Verfahren zur herstellung von 2-penemverbindungen.
ATE89822T1 (de)	1993-06-15	Durch benzhydryl n-substituierte heterocyclische derivate, ihre herstellung und ihre verwendung.
BR8601978A (pt)	1987-01-06	Processo de estabilizar uma pelicula polimera ou artigo moldado contra a acao da luz,umidade e oxigenio,combinacao estabilizadora sinergistica para um polimero e composicao estavel leve
ES387553A1 (es)	1974-01-16	Procedimiento para la preparacion de 4-morfolino-tieno (3,-2-d)-pirimidinas.
ES8200868A1 (es)	1981-11-16	Un procedimiento para la preparacion de un derivado de aze- tidina
ES505116A0 (es)	1983-01-01	Un procedimiento para la preparacion del acido 9-halo-7-oxo-2,3-dihidro-7m-pirido-1,2,3-de-1,4 benzoxazin 6-carboxilico.
DE3750587D1 (de)	1994-10-27	Verfahren zur Herstellung von Eicosatetraynsäure.
PT86526A (pt)	1989-09-14	Processo para a preparacao de mono-hidrato de cefadroxil cristalino e de composicoes farmaceuticas que o contem
PT73841B (en)	1983-11-07	Process for preparing novel guanidine derivatives
ES8106713A1 (es)	1981-09-01	Procedimiento para la preparacion de n-aril-n-acil-3-amino- oxazolidin-2-onas
SE8005686L (sv)	1981-02-14	Nya halogenvinkamonderivat jemte sett for deras framstellning
MA19842A1 (fr)	1984-04-01	Procede de preparation de derives de peneme antibacteriens .
PT76861A (fr)	1983-07-01	Procede de preparation de nouveaux derives d'oxazinobenzothiazine-6,6-dioxide et de compositions pharmaceutiques les contenant
ES8604388A1 (es)	1985-08-01	Metodo de producir compuestos 1(2h)-isoquinolonicos y analogos
ES8207530A1 (es)	1982-10-01	Un procedimiento para la produccion de nuevos derivados del tetrahidroimidazo (2,1-b)tiazol
SE7910430L (sv)	1980-06-20	Cyklododekanderivat jemte sett for deras framstellning
FI841058A0 (fi)	1984-03-15	Tillvaextregulatorer foer vaexter
ES8104198A1 (es)	1981-04-01	Un procedimiento para la preparacion de un derivado de mo- noamida del acido tereftalico
BR8401229A (pt)	1984-10-23	Processo para a preparacao de um ester de acido fosfonico,composicao inseticida,acaricida ou nematicida,processo para combater parasitas e processo para preparar uma tal composicao
DK157869C (da)	1990-08-06	Analogifremgangsmaade til fremstilling af azatetracycliske carbonitriler eller syreadditionssalte deraf
ES550292A1 (es)	1989-04-16	Procedimiento para la preparacion de derivados de piperazina