ATE142205T1 - Substituierte piperidimylmethyl-ester von 3- indolcarbonsäure - Google Patents

Substituierte piperidimylmethyl-ester von 3- indolcarbonsäure

Info

Publication number: ATE142205T1
Authority: AT; Austria
Prior art keywords: piperidimylmethyl; indolecarboxic; esters; substituted; acid
Prior art date: 1991-02-25

Application number

AT92102900T

Other languages

English (en)

Inventor

Alexander William Oxford

John William Frank Whitehead

John Knight

Original Assignee

Glaxo Group Ltd

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1991-02-25

Filing date

1992-02-21

Publication date

1996-09-15

1992-02-21 Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd

1996-09-15 Application granted granted Critical

1996-09-15 Publication of ATE142205T1 publication Critical patent/ATE142205T1/de

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Bioinformatics & Cheminformatics (AREA)
Pharmacology & Pharmacy (AREA)
Engineering & Computer Science (AREA)
Animal Behavior & Ethology (AREA)
Chemical Kinetics & Catalysis (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Hospice & Palliative Care (AREA)
Otolaryngology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Hydrogenated Pyridines (AREA)
Indole Compounds (AREA)

AT92102900T 1991-02-25 1992-02-21 Substituierte piperidimylmethyl-ester von 3- indolcarbonsäure ATE142205T1 (de)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
GB919103862A GB9103862D0 (en)	1991-02-25	1991-02-25	Chemical compounds
APAP/P/1992/000417A AP295A (en)	1991-02-25	1992-08-17	3-Piperidinylmethylcarboxylate substituted indoles.
CN92110050A CN1083059A (zh)	1991-02-25	1992-08-24	3-哌啶甲基羧酸酯取代的吲哚

Publications (1)

Publication Number	Publication Date
ATE142205T1 true ATE142205T1 (de)	1996-09-15

Family

ID=36790873

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT92102900T ATE142205T1 (de)	1991-02-25	1992-02-21	Substituierte piperidimylmethyl-ester von 3- indolcarbonsäure

Country Status (18)

Country	Link
EP (1)	EP0501322B1 (de)
JP (1)	JPH06505238A (de)
CN (1)	CN1083059A (de)
AP (1)	AP295A (de)
AT (1)	ATE142205T1 (de)
AU (1)	AU645402B2 (de)
CA (1)	CA2105179A1 (de)
DE (1)	DE69213276T2 (de)
ES (1)	ES2091963T3 (de)
FI (1)	FI933697L (de)
GB (1)	GB9103862D0 (de)
HU (1)	HUT65486A (de)
IE (1)	IE920567A1 (de)
IL (1)	IL101042A (de)
MX (1)	MX9200762A (de)
NO (1)	NO933015D0 (de)
NZ (1)	NZ241704A (de)
WO (1)	WO1992014727A1 (de)

Families Citing this family (24)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US20020128172A1 (en)	1991-12-21	2002-09-12	Smithkline Beecham Plc	Use of 5-HT4 modulators for the manufacture of a medicament for the treatment of the bladder diseases
DE69226961T2 (de) *	1991-12-21	1999-04-29	Smithkline Beecham P.L.C., Brentford, Middlesex	Verwendung von 5-ht4 - antagonisten zur herstellung eines arzneimittels zur behandlung von harninkontinenz
WO1993018036A1 (en) *	1992-03-12	1993-09-16	Smithkline Beecham Plc	Condensed indole derivatives as 5ht4-receptor antagonists
US5852014A (en) *	1992-03-12	1998-12-22	Smithkline Beecham P.L.C.	Condensed indole derivatives as 5HT4 -receptor antagonists
JPH07507290A (ja) *	1992-05-23	1995-08-10	スミスクライン・ビーチャム・パブリック・リミテッド・カンパニー	不安症の治療のための医薬
JPH07508276A (ja) *	1992-06-27	1995-09-14	スミスクライン・ビーチャム・パブリック・リミテッド・カンパニー	５−ｈｔ↓４受容体アンタゴニスト含有医薬品
MX9305947A (es) *	1992-09-29	1994-06-30	Smithkline Beecham Plc	Compuestos antagonistas del receptor 5-ht4, procedimiento para su preparacion y composiciones farmaceuticas que las contienen.
GB9221468D0 (en) *	1992-10-13	1992-11-25	Smithkline Beecham Plc	Pharmaceuticals
MX9306311A (es) *	1992-10-13	1994-04-29	Smithkline Beecham Plc	Compuestos antagonistas del receptor de 5-ht4, procedimiento para su preparacion y composiciones farmaceuticas que los contienen
WO1994008965A1 (en) *	1992-10-16	1994-04-28	Smithkline Beecham Plc	N-alkylpiperidinyl-4-methyl carboxylic esters/amides of condensed ring systems as 5-ht4 receptor antagonists
EP0667867A1 (de) *	1992-11-05	1995-08-23	Smithkline Beecham Plc	Piperidinderivate als 5-ht4 rezeptor antagonisten
GB9301660D0 (en) *	1993-01-28	1993-03-17	Smithkline Beecham Plc	Pharmaceuticals
GB9310582D0 (en) *	1993-05-22	1993-07-07	Smithkline Beecham Plc	Pharmaceuticals
GB9312348D0 (en) *	1993-06-16	1993-07-28	Smithkline Beecham Plc	Pharmaceuticals
IT1275903B1 (it) *	1995-03-14	1997-10-24	Boehringer Ingelheim Italia	Esteri e ammidi della 1,4-piperidina disostituita
GB9702194D0 (en)	1997-02-04	1997-03-26	Lilly Co Eli	Sulphonide derivatives
IT1291569B1 (it) *	1997-04-15	1999-01-11	Angelini Ricerche Spa	Indazolammidi come agenti serotoninergici
GB9725933D0 (en) *	1997-12-05	1998-02-04	Smithkline Beecham Plc	Pharmaceuticals
CA2418904A1 (en) *	2000-08-07	2002-02-14	Laboratoire Glaxosmithkline S.A.S.	Use of 5ht4 receptor antagonists in the manufacture of a medicament for the prophylaxis or treatment of atrial fibrillation
CN1293072C (zh) *	2001-04-20	2007-01-03	惠氏公司	作为5－羟色胺－6配体的杂环基氧基－、－硫代－和－氨基吲哚衍生物
CN1293073C (zh) *	2001-04-20	2007-01-03	惠氏公司	作为5－羟色胺－6配体的杂环基烷氧基－、－烷硫基－和－烷基氨基吲哚衍生物
GB0211230D0 (en)	2002-05-16	2002-06-26	Medinnova Sf	Treatment of heart failure
US8114894B2 (en) *	2008-12-03	2012-02-14	Nanotherapeutics, Inc.	Bicyclic compounds and methods of making and using same
JP2025500920A (ja) *	2021-12-23	2025-01-15	香港時代新能源科技有限公司	Ａ／ｍ／ｘ結晶材料、太陽光発電デバイス及びその製造方法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
JPS60123485A (ja) *	1983-12-08	1985-07-02	Yoshitomi Pharmaceut Ind Ltd	インド−ル−３−カルボキサミド誘導体
FR2557110B1 (fr) *	1983-12-23	1989-11-24	Sandoz Sa	Nouveaux derives d'amines cycliques, leur preparation et leur utilisation comme medicaments
GB8527052D0 (en) *	1985-11-02	1985-12-04	Beecham Group Plc	Compounds
DK623586A (da) *	1985-12-27	1987-06-28	Eisai Co Ltd	Piperidinderivater eller salte deraf og farmaceutiske kompositioner indeholdende forbindelserne
CA2030051C (en) *	1989-11-17	2001-08-07	Haruhiko Kikuchi	Indole derivatives

1991
- 1991-02-25 GB GB919103862A patent/GB9103862D0/en active Pending
1992
- 1992-02-21 WO PCT/EP1992/000371 patent/WO1992014727A1/en not_active Ceased
- 1992-02-21 FI FI933697A patent/FI933697L/fi not_active Application Discontinuation
- 1992-02-21 JP JP4504653A patent/JPH06505238A/ja active Pending
- 1992-02-21 HU HU9302414A patent/HUT65486A/hu unknown
- 1992-02-21 CA CA002105179A patent/CA2105179A1/en not_active Abandoned
- 1992-02-21 AU AU12094/92A patent/AU645402B2/en not_active Ceased
- 1992-02-21 DE DE69213276T patent/DE69213276T2/de not_active Expired - Fee Related
- 1992-02-21 ES ES92102900T patent/ES2091963T3/es not_active Expired - Lifetime
- 1992-02-21 AT AT92102900T patent/ATE142205T1/de not_active IP Right Cessation
- 1992-02-21 EP EP92102900A patent/EP0501322B1/de not_active Expired - Lifetime
- 1992-02-24 NZ NZ241704A patent/NZ241704A/xx unknown
- 1992-02-24 IL IL10104292A patent/IL101042A/en not_active IP Right Cessation
- 1992-02-24 IE IE056792A patent/IE920567A1/en unknown
- 1992-02-24 MX MX9200762A patent/MX9200762A/es unknown
- 1992-08-17 AP APAP/P/1992/000417A patent/AP295A/en active
- 1992-08-24 CN CN92110050A patent/CN1083059A/zh active Pending
1993
- 1993-08-24 NO NO933015A patent/NO933015D0/no unknown

Also Published As

Publication number	Publication date
MX9200762A (es)	1992-08-01
IL101042A0 (en)	1992-11-15
IL101042A (en)	1996-06-18
GB9103862D0 (en)	1991-04-10
AP295A (en)	1993-12-29
ES2091963T3 (es)	1996-11-16
AU1209492A (en)	1992-09-15
FI933697A0 (fi)	1993-08-23
DE69213276D1 (de)	1996-10-10
AP9200417A0 (en)	1992-10-31
IE920567A1 (en)	1992-08-26
EP0501322B1 (de)	1996-09-04
NO933015L (no)	1993-08-24
CA2105179A1 (en)	1992-08-26
NO933015D0 (no)	1993-08-24
HUT65486A (en)	1994-06-28
EP0501322A1 (de)	1992-09-02
CN1083059A (zh)	1994-03-02
HU9302414D0 (en)	1993-11-29
FI933697A7 (fi)	1993-08-23
NZ241704A (en)	1993-11-25
JPH06505238A (ja)	1994-06-16
AU645402B2 (en)	1994-01-13
WO1992014727A1 (en)	1992-09-03
FI933697L (fi)	1993-08-23
DE69213276T2 (de)	1997-01-23

Legal Events

Date	Code	Title	Description
1997-04-15	UEP	Publication of translation of european patent specification
2000-11-15	REN	Ceased due to non-payment of the annual fee

Publication	Publication Date	Title
ATE142205T1 (de)	1996-09-15	Substituierte piperidimylmethyl-ester von 3- indolcarbonsäure
ATE113610T1 (de)	1994-11-15	Ester von alginsäure.
DK0383117T3 (da)	1994-07-25	Pyridylsubstituerede acrylsyreestere
MX9101139A (es)	1992-05-04	Esteres de acido carboxilico de rapamicina
FI904230A7 (fi)	1990-08-27	Akryylihappojohdannaisia
DE69320556D1 (de)	1998-10-01	Carbonylierung von Epoxyden
DE69426245D1 (de)	2000-12-14	Monoester der Harzsäure
DE69417496D1 (de)	1999-05-06	Sulfonierung von Fettsäureestern
NO172688C (no)	1993-08-25	Karbaminsyre-ester
DE69212968D1 (de)	1996-09-26	Herstellung von Ethylendiamintriessigsäure
DE69302098D1 (de)	1996-05-09	Zusammensetzungen von hexitan-fettsäureestern
DK0464381T3 (da)	1995-11-06	2-Methoximinocarboxylsyreestere
DE59207354D1 (de)	1996-11-21	Triazinyl-substituierte Acrylsäureester
DK0384211T3 (da)	1994-12-05	Substituerede acrylsyreestere
DE69207387D1 (de)	1996-02-15	Herstellung von Carbonsäureestern
ATE42751T1 (de)	1989-05-15	Carboxylsaeureesterderivate von deglucoteicoplanin.
FI881959L (fi)	1988-10-28	Karboksyylihappoestereiden pelkistys
DK637888D0 (da)	1988-11-15	Carboxylsyreestere
DE58902314D1 (de)	1992-10-29	Substituierte acrylsaeureester.
DE59205221D1 (de)	1996-03-14	1-Alkoxyhexatrien-2-carbonsäureester
FI946085L (fi)	1994-12-23	Uusia nikotiinihappoestereitä
FI933300L (fi)	1994-01-24	Foerfarande foer rengoering av klorvaetesyra i gasform
DE69229616D1 (de)	1999-08-26	Enzymatische Resolution von Alpha-tertiären-Karbonsäureestern
FI922125L (fi)	1992-12-22	Mikrobidogiskt foerfarande foer framstaellning av 5-hydroxipyrazinkarboxylsyra
DK670589A (da)	1990-06-30	Carboxylsyrederivater