ATE155456T1 - Verfahren zur herstellung und optischen auflösung von 2-phenyl-3-aminopiperidine - Google Patents

Verfahren zur herstellung und optischen auflösung von 2-phenyl-3-aminopiperidine

Info

Publication number
ATE155456T1
ATE155456T1 AT94910014T AT94910014T ATE155456T1 AT E155456 T1 ATE155456 T1 AT E155456T1 AT 94910014 T AT94910014 T AT 94910014T AT 94910014 T AT94910014 T AT 94910014T AT E155456 T1 ATE155456 T1 AT E155456T1
Authority
AT
Austria
Prior art keywords
phenyl
aminopiperidine
production
optical resolution
benzylaminopiperidines
Prior art date
Application number
AT94910014T
Other languages
English (en)
Inventor
William M Snyder
Harry A Watson Jr
Glenn E Wilcox
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Application granted granted Critical
Publication of ATE155456T1 publication Critical patent/ATE155456T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/56—Nitrogen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Hydrogenated Pyridines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
AT94910014T 1993-05-28 1994-04-06 Verfahren zur herstellung und optischen auflösung von 2-phenyl-3-aminopiperidine ATE155456T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US6847193A 1993-05-28 1993-05-28

Publications (1)

Publication Number Publication Date
ATE155456T1 true ATE155456T1 (de) 1997-08-15

Family

ID=22082784

Family Applications (1)

Application Number Title Priority Date Filing Date
AT94910014T ATE155456T1 (de) 1993-05-28 1994-04-06 Verfahren zur herstellung und optischen auflösung von 2-phenyl-3-aminopiperidine

Country Status (11)

Country Link
US (1) US6436961B1 (de)
EP (1) EP0700384B1 (de)
JP (1) JPH08507297A (de)
AT (1) ATE155456T1 (de)
CA (1) CA2162400A1 (de)
DE (1) DE69404306T2 (de)
DK (1) DK0700384T3 (de)
ES (1) ES2105664T3 (de)
FI (1) FI955708L (de)
GR (1) GR3024592T3 (de)
WO (1) WO1994027966A1 (de)

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WO2007075630A1 (en) * 2005-12-22 2007-07-05 Dow Global Technologies Inc. Method for producing 3-aminopiperidine diastereomer
DE102005063192A1 (de) 2005-12-30 2007-07-05 Basf Ag Racematspaltung von 2,6-trans-Dimethyl-morpholin
EP2121613A2 (de) * 2007-01-31 2009-11-25 Vertex Pharmaceuticals, Inc. 2-aminopyridinderivate als kinaseinhibitoren
MX2011000839A (es) 2008-07-23 2011-04-05 Vertex Pharma Inhibidores de pirazolpiridina cinasa.
AU2009274023A1 (en) 2008-07-23 2010-01-28 Vertex Pharmaceuticals Incorporated Tri-cyclic pyrazolopyridine kinase inhibitors
US8569337B2 (en) 2008-07-23 2013-10-29 Vertex Pharmaceuticals Incorporated Tri-cyclic pyrazolopyridine kinase inhibitors
WO2010017350A1 (en) * 2008-08-06 2010-02-11 Vertex Pharmaceuticals Incorporated Aminopyridine kinase inhibitors
MX2011011653A (es) 2009-05-06 2012-01-20 Vertex Pharma Pirazolopiridinas.
MX2012008643A (es) 2010-01-27 2013-02-26 Vertex Pharma Inhibidores de cinasas de pirazolopiridinas.
MX2012008641A (es) 2010-01-27 2012-11-23 Vertex Pharma Inhibidores de cinasas de pirazolopirazinas.
CA2787315A1 (en) 2010-01-27 2011-08-04 Vertex Pharmaceuticals Incorporated Pyrazolopyridine kinase inhibitors
WO2020019247A1 (en) 2018-07-26 2020-01-30 Xw Laboratories, Inc. Compounds as neurokinin-1 receptor antagonists and uses thereof

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Also Published As

Publication number Publication date
JPH08507297A (ja) 1996-08-06
FI955708A0 (fi) 1995-11-27
DE69404306T2 (de) 1997-10-30
FI955708A7 (fi) 1995-11-27
GR3024592T3 (en) 1997-12-31
DK0700384T3 (da) 1997-12-08
WO1994027966A1 (en) 1994-12-08
EP0700384A1 (de) 1996-03-13
CA2162400A1 (en) 1994-12-08
ES2105664T3 (es) 1997-10-16
FI955708L (fi) 1995-11-27
EP0700384B1 (de) 1997-07-16
DE69404306D1 (de) 1997-08-21
US6436961B1 (en) 2002-08-20

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Legal Events

Date Code Title Description
UEP Publication of translation of european patent specification
REN Ceased due to non-payment of the annual fee