FI955708L - Menetelmä 2-fenyyli-3-aminopiperidiinin valmistamiseksi ja erottamiseksi - Google Patents

Menetelmä 2-fenyyli-3-aminopiperidiinin valmistamiseksi ja erottamiseksi Download PDF

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Publication number
FI955708L
FI955708L FI955708A FI955708A FI955708L FI 955708 L FI955708 L FI 955708L FI 955708 A FI955708 A FI 955708A FI 955708 A FI955708 A FI 955708A FI 955708 L FI955708 L FI 955708L
Authority
FI
Finland
Prior art keywords
aminopiperidine
isolation
phenyl
preparation
Prior art date
Application number
FI955708A
Other languages
English (en)
Finnish (fi)
Swedish (sv)
Other versions
FI955708A7 (fi
FI955708A0 (fi
Inventor
William M Snyder
Jr Harry A Watson
Glenn E Wilcox
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of FI955708A7 publication Critical patent/FI955708A7/fi
Publication of FI955708A0 publication Critical patent/FI955708A0/fi
Publication of FI955708L publication Critical patent/FI955708L/fi

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/56—Nitrogen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Hydrogenated Pyridines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
FI955708A 1993-05-28 1994-04-06 Menetelmä 2-fenyyli-3-aminopiperidiinin valmistamiseksi ja erottamiseksi FI955708L (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US6847193A 1993-05-28 1993-05-28
PCT/IB1994/000059 WO1994027966A1 (en) 1993-05-28 1994-04-06 Process for preparing and resolving 2-phenyl-3-aminopiperidine

Publications (3)

Publication Number Publication Date
FI955708A7 FI955708A7 (fi) 1995-11-27
FI955708A0 FI955708A0 (fi) 1995-11-27
FI955708L true FI955708L (fi) 1995-11-27

Family

ID=22082784

Family Applications (1)

Application Number Title Priority Date Filing Date
FI955708A FI955708L (fi) 1993-05-28 1994-04-06 Menetelmä 2-fenyyli-3-aminopiperidiinin valmistamiseksi ja erottamiseksi

Country Status (11)

Country Link
US (1) US6436961B1 (de)
EP (1) EP0700384B1 (de)
JP (1) JPH08507297A (de)
AT (1) ATE155456T1 (de)
CA (1) CA2162400A1 (de)
DE (1) DE69404306T2 (de)
DK (1) DK0700384T3 (de)
ES (1) ES2105664T3 (de)
FI (1) FI955708L (de)
GR (1) GR3024592T3 (de)
WO (1) WO1994027966A1 (de)

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KR20050085673A (ko) 2002-12-18 2005-08-29 에프엠씨 코포레이션 N-(치환된 아릴메틸)-4-(이치환된 메틸)피페리딘 및피페라진
US6995270B2 (en) * 2003-03-17 2006-02-07 Pfizer Inc Hydrogenation process
WO2007075630A1 (en) * 2005-12-22 2007-07-05 Dow Global Technologies Inc. Method for producing 3-aminopiperidine diastereomer
DE102005063192A1 (de) * 2005-12-30 2007-07-05 Basf Ag Racematspaltung von 2,6-trans-Dimethyl-morpholin
EP2121613A2 (de) * 2007-01-31 2009-11-25 Vertex Pharmaceuticals, Inc. 2-aminopyridinderivate als kinaseinhibitoren
US8569337B2 (en) 2008-07-23 2013-10-29 Vertex Pharmaceuticals Incorporated Tri-cyclic pyrazolopyridine kinase inhibitors
NZ590784A (en) 2008-07-23 2012-12-21 Vertex Pharma Pyrazolopyridine kinase inhibitors
MX2011000837A (es) 2008-07-23 2011-04-05 Vertex Pharma Inhibidores de pirazolpiridina cinasa triciclica.
MX2011001319A (es) 2008-08-06 2011-04-05 Vertex Pharma Inhibidores de aminopiridina cinasa.
WO2010129668A1 (en) 2009-05-06 2010-11-11 Vertex Pharmaceuticals Incorporated Pyrazolopyridines
EP2582702A1 (de) 2010-01-27 2013-04-24 Vertex Pharmaceuticals Incorporated Pyrazolopyrimidinkinasehemmer
EP2528917B1 (de) 2010-01-27 2016-10-19 Vertex Pharmaceuticals Incorporated Zur behandlung von autoimmun-, entzündlichen oder (hyper)proliferativen erkrankungen geeignete pyrazolopyridine
AU2011209649A1 (en) 2010-01-27 2012-08-09 Vertex Pharmaceuticals Incorporated Pyrazolopyrazine kinase inhibitors
WO2020019247A1 (en) 2018-07-26 2020-01-30 Xw Laboratories, Inc. Compounds as neurokinin-1 receptor antagonists and uses thereof

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Also Published As

Publication number Publication date
US6436961B1 (en) 2002-08-20
CA2162400A1 (en) 1994-12-08
JPH08507297A (ja) 1996-08-06
DE69404306T2 (de) 1997-10-30
ES2105664T3 (es) 1997-10-16
DE69404306D1 (de) 1997-08-21
FI955708A7 (fi) 1995-11-27
EP0700384A1 (de) 1996-03-13
EP0700384B1 (de) 1997-07-16
GR3024592T3 (en) 1997-12-31
ATE155456T1 (de) 1997-08-15
WO1994027966A1 (en) 1994-12-08
DK0700384T3 (da) 1997-12-08
FI955708A0 (fi) 1995-11-27

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