ATE156480T1 - Verfahren zur herstellung von zwischenprodukten für die synthese von chinolin-antibiotika - Google Patents

Verfahren zur herstellung von zwischenprodukten für die synthese von chinolin-antibiotika

Info

Publication number: ATE156480T1
Authority: AT; Austria
Prior art keywords: synthesis; intermediate products; producing intermediate; quinoline antibiotics; quinoline
Prior art date: 1992-03-02

Application number

AT93902893T

Other languages

English (en)

Inventor

Tamim F Braish

Original Assignee

Pfizer

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1992-03-02

Filing date

1993-01-07

Publication date

1997-08-15

1993-01-07 Application filed by Pfizer filed Critical Pfizer

1997-08-15 Application granted granted Critical

1997-08-15 Publication of ATE156480T1 publication Critical patent/ATE156480T1/de

Links

238000003786 synthesis reaction Methods 0.000 title abstract 2
SMWDFEZZVXVKRB-UHFFFAOYSA-N Quinoline Chemical compound N1=CC=CC2=CC=CC=C21 SMWDFEZZVXVKRB-UHFFFAOYSA-N 0.000 title 2
239000003242 anti bacterial agent Substances 0.000 title 1
229940088710 antibiotic agent Drugs 0.000 title 1
230000015572 biosynthetic process Effects 0.000 title 1
239000013067 intermediate product Substances 0.000 title 1
238000004519 manufacturing process Methods 0.000 title 1
150000001875 compounds Chemical class 0.000 abstract 2
239000000126 substance Substances 0.000 abstract 2
230000000844 anti-bacterial effect Effects 0.000 abstract 1
239000000543 intermediate Substances 0.000 abstract 1
LOAUVZALPPNFOQ-UHFFFAOYSA-N quinaldic acid Chemical class C1=CC=CC2=NC(C(=O)O)=CC=C21 LOAUVZALPPNFOQ-UHFFFAOYSA-N 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/52—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring condensed with a ring other than six-membered

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Plural Heterocyclic Compounds (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Preparation Of Compounds By Using Micro-Organisms (AREA)
Indole Compounds (AREA)

AT93902893T 1992-03-02 1993-01-07 Verfahren zur herstellung von zwischenprodukten für die synthese von chinolin-antibiotika ATE156480T1 (de)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US07/844,367 US5256791A (en)	1992-03-02	1992-03-02	Preparation of intermediates in the synthesis of quinoline antibiotics

Publications (1)

Publication Number	Publication Date
ATE156480T1 true ATE156480T1 (de)	1997-08-15

Family

ID=25292537

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT93902893T ATE156480T1 (de)	1992-03-02	1993-01-07	Verfahren zur herstellung von zwischenprodukten für die synthese von chinolin-antibiotika

Country Status (22)

Country	Link
US (2)	US5256791A (de)
EP (1)	EP0629189B1 (de)
JP (1)	JP2564247B2 (de)
KR (2)	KR950700251A (de)
CN (1)	CN1037100C (de)
AT (1)	ATE156480T1 (de)
AU (1)	AU667872B2 (de)
CA (1)	CA2131160C (de)
DE (1)	DE69312913T2 (de)
DK (1)	DK0629189T3 (de)
ES (1)	ES2105217T3 (de)
FI (1)	FI106022B (de)
GR (1)	GR3024789T3 (de)
HU (1)	HU215837B (de)
IL (1)	IL104818A (de)
MX (1)	MX9301138A (de)
MY (1)	MY107723A (de)
NO (1)	NO300681B1 (de)
NZ (1)	NZ246768A (de)
TW (1)	TW211002B (de)
WO (1)	WO1993018001A1 (de)
ZA (1)	ZA931428B (de)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
CZ286896B6 (en)	1994-01-18	2000-07-12	Pfizer	Process for preparing pharmaceutically acceptable salts of naphthyridone carboxylic acid and intermediates for this preparation
US5475116A (en) *	1994-04-29	1995-12-12	Pfizer Inc.	Aza bicyclo[3,1,0]hexane intermediates useful in the synthesis of quinolones
US5929240A (en) *	1994-12-12	1999-07-27	Pfizer Inc.	Process and intermediates for preparing naphthyridonecarboxylic acid salts
JPH0912547A (ja) *	1995-06-23	1997-01-14	Chisso Corp	ニューキノロン系化合物中間体の製造方法
GB9524466D0 (en) *	1995-11-30	1996-01-31	Pfizer Ltd	Process
US6057455A (en) *	1996-07-09	2000-05-02	Pfizer, Inc.	Preparation of intermediates useful in the synthesis of quinoline antibiotics
GB9614422D0 (en) *	1996-07-09	1996-09-04	Pfizer Ltd	Novel process
JPH1087617A (ja) *	1996-07-09	1998-04-07	Pfizer Inc	キノリン系抗生物質の合成に有用な中間体の製法
HN1998000106A (es)	1997-08-01	1999-01-08	Pfizer Prod Inc	Composiciones parenterales de alatroflaxacino
DE19733439A1 (de) *	1997-08-02	1999-02-04	Bayer Ag	Neue 6-endo-Amino-3-azabicyclo(3.1.0)hexande, Verfahren zu deren Herstellung und deren Verwendung zur Herstellung von Chinolon- und Naphthyridincarbonsäure-Derviaten mit verbesserten Eigenschaften
US7019142B2 (en)	1998-01-16	2006-03-28	Pfizer Inc.	Process for preparing naphthyridones and intermediates
US6184380B1 (en) *	1999-01-25	2001-02-06	Pfizer Inc.	Process for preparing naphthyridones and intermediates
PA8464701A1 (es) *	1998-01-16	2000-09-29	Pfizer Prod Inc	Procedimiento e intermedios para preparar naftiridonas
WO2008010061A2 (en) *	2006-07-17	2008-01-24	Glenmark Pharmaceuticals S.A.	3-azabicyclo [3.1.0] hexane vanilloid receptor ligands, pharmaceutical compositions containing them, and processes for their preparation
WO2020243423A1 (en)	2019-05-31	2020-12-03	Ikena Oncology, Inc.	Tead inhibitors and uses thereof
KR20220030222A (ko)	2019-05-31	2022-03-10	이케나 온콜로지, 인코포레이티드	Tead 억제제 및 이의 용도
WO2023151188A1 (zh) *	2022-02-08	2023-08-17	上海皓元医药股份有限公司	一种抗病毒药物中间体的绿色合成方法

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4183857A (en) *	1978-07-06	1980-01-15	Shell Oil Company	3-Benzyl-3-azabicyclo(3.1.0)hexane-2,4-dione
EP0010799B1 (de) *	1978-10-27	1982-05-19	Shell Internationale Researchmaatschappij B.V.	Verfahren zur Herstellung von 3-Azabicyclo(3.1.0)hexanderivaten und ihre Modifikationen
JPH0676400B2 (ja) *	1987-08-25	1994-09-28	大日本製薬株式会社	新規ピリドンカルボン酸誘導体、そのエステルおよびその塩
US5196548A (en) *	1989-05-11	1993-03-23	Pfizer Inc.	Preparation of diazabicyclic Intermediates
IE66202B1 (en) *	1989-08-16	1995-12-13	Pfizer	Azabicyclo quinolone carboxylic acids
US5200527A (en) *	1991-04-08	1993-04-06	Lonza Ltd.	Process for the production of 2-azabicyclo [2.2.1] hept-5-en-3-one

1992
- 1992-03-02 US US07/844,367 patent/US5256791A/en not_active Expired - Fee Related
1993
- 1993-01-07 DE DE69312913T patent/DE69312913T2/de not_active Expired - Fee Related
- 1993-01-07 NZ NZ246768A patent/NZ246768A/en unknown
- 1993-01-07 KR KR1019940703051A patent/KR950700251A/ko active Granted
- 1993-01-07 EP EP93902893A patent/EP0629189B1/de not_active Expired - Lifetime
- 1993-01-07 AU AU34300/93A patent/AU667872B2/en not_active Ceased
- 1993-01-07 KR KR1019940703051A patent/KR0135626B1/ko not_active Expired - Fee Related
- 1993-01-07 AT AT93902893T patent/ATE156480T1/de active
- 1993-01-07 JP JP5515648A patent/JP2564247B2/ja not_active Expired - Lifetime
- 1993-01-07 WO PCT/US1993/000008 patent/WO1993018001A1/en not_active Ceased
- 1993-01-07 ES ES93902893T patent/ES2105217T3/es not_active Expired - Lifetime
- 1993-01-07 HU HU9402530A patent/HU215837B/hu not_active IP Right Cessation
- 1993-01-07 CA CA002131160A patent/CA2131160C/en not_active Expired - Fee Related
- 1993-01-07 DK DK93902893.2T patent/DK0629189T3/da active
- 1993-01-11 TW TW082100123A patent/TW211002B/zh active
- 1993-02-22 IL IL104818A patent/IL104818A/xx not_active IP Right Cessation
- 1993-03-01 CN CN93102103A patent/CN1037100C/zh not_active Expired - Fee Related
- 1993-03-01 MX MX9301138A patent/MX9301138A/es not_active IP Right Cessation
- 1993-03-01 MY MYPI93000368A patent/MY107723A/en unknown
- 1993-03-01 ZA ZA931428A patent/ZA931428B/xx unknown
- 1993-08-04 US US08/101,879 patent/US5298629A/en not_active Expired - Fee Related
1994
- 1994-09-01 FI FI944013A patent/FI106022B/fi active
- 1994-09-01 NO NO943243A patent/NO300681B1/no not_active IP Right Cessation
1997
- 1997-09-17 GR GR970402413T patent/GR3024789T3/el unknown

Also Published As

Publication number	Publication date
MX9301138A (es)	1994-01-31
ES2105217T3 (es)	1997-10-16
EP0629189A1 (de)	1994-12-21
IL104818A (en)	1997-09-30
CA2131160C (en)	1997-11-18
HU9402530D0 (en)	1994-11-28
WO1993018001A1 (en)	1993-09-16
JP2564247B2 (ja)	1996-12-18
EP0629189B1 (de)	1997-08-06
AU667872B2 (en)	1996-04-18
NO943243L (no)	1994-09-01
HU215837B (en)	2001-03-28
CN1076440A (zh)	1993-09-22
KR0135626B1 (ko)	1998-04-23
AU3430093A (en)	1993-10-05
CA2131160A1 (en)	1993-09-16
DK0629189T3 (da)	1997-12-08
US5256791A (en)	1993-10-26
NO300681B1 (no)	1997-07-07
TW211002B (en)	1993-08-11
NZ246768A (en)	1995-09-26
ZA931428B (en)	1994-09-01
IL104818A0 (en)	1993-06-10
CN1037100C (zh)	1998-01-21
FI944013A0 (fi)	1994-09-01
HUT70497A (en)	1995-10-30
KR950700251A (ko)	1995-01-16
DE69312913T2 (de)	1997-11-20
MY107723A (en)	1996-05-30
DE69312913D1 (de)	1997-09-11
GR3024789T3 (en)	1998-01-30
JPH07500349A (ja)	1995-01-12
NO943243D0 (no)	1994-09-01
US5298629A (en)	1994-03-29
FI944013L (fi)	1994-09-01
FI106022B (fi)	2000-11-15

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