DK0629189T3 - Fremstilling af mellemprodukter i syntesen af quinolinantbiotika - Google Patents

Fremstilling af mellemprodukter i syntesen af quinolinantbiotika

Info

Publication number: DK0629189T3
Authority: DK; Denmark
Prior art keywords: intermediates; quinolinant; biotics; synthesis; preparation
Prior art date: 1992-03-02

Application number

DK93902893.2T

Other languages

Danish (da)

English (en)

Inventor

Tamim F Braish

Original Assignee

Pfizer

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1992-03-02

Filing date

1993-01-07

Publication date

1997-12-08

1993-01-07 Application filed by Pfizer filed Critical Pfizer

1997-12-08 Application granted granted Critical

1997-12-08 Publication of DK0629189T3 publication Critical patent/DK0629189T3/da

Links

239000000543 intermediate Substances 0.000 title abstract 2
238000003786 synthesis reaction Methods 0.000 title abstract 2
230000015572 biosynthetic process Effects 0.000 title 1
238000002360 preparation method Methods 0.000 title 1
150000001875 compounds Chemical class 0.000 abstract 2
239000000126 substance Substances 0.000 abstract 2
230000000844 anti-bacterial effect Effects 0.000 abstract 1
LOAUVZALPPNFOQ-UHFFFAOYSA-N quinaldic acid Chemical class C1=CC=CC2=NC(C(=O)O)=CC=C21 LOAUVZALPPNFOQ-UHFFFAOYSA-N 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/52—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring condensed with a ring other than six-membered

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Plural Heterocyclic Compounds (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Indole Compounds (AREA)
Preparation Of Compounds By Using Micro-Organisms (AREA)

DK93902893.2T 1992-03-02 1993-01-07 Fremstilling af mellemprodukter i syntesen af quinolinantbiotika DK0629189T3 (da)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US07/844,367 US5256791A (en)	1992-03-02	1992-03-02	Preparation of intermediates in the synthesis of quinoline antibiotics

Publications (1)

Publication Number	Publication Date
DK0629189T3 true DK0629189T3 (da)	1997-12-08

Family

ID=25292537

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK93902893.2T DK0629189T3 (da)	1992-03-02	1993-01-07	Fremstilling af mellemprodukter i syntesen af quinolinantbiotika

Country Status (22)

Country	Link
US (2)	US5256791A (de)
EP (1)	EP0629189B1 (de)
JP (1)	JP2564247B2 (de)
KR (2)	KR950700251A (de)
CN (1)	CN1037100C (de)
AT (1)	ATE156480T1 (de)
AU (1)	AU667872B2 (de)
CA (1)	CA2131160C (de)
DE (1)	DE69312913T2 (de)
DK (1)	DK0629189T3 (de)
ES (1)	ES2105217T3 (de)
FI (1)	FI106022B (de)
GR (1)	GR3024789T3 (de)
HU (1)	HU215837B (de)
IL (1)	IL104818A (de)
MX (1)	MX9301138A (de)
MY (1)	MY107723A (de)
NO (1)	NO300681B1 (de)
NZ (1)	NZ246768A (de)
TW (1)	TW211002B (de)
WO (1)	WO1993018001A1 (de)
ZA (1)	ZA931428B (de)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
CZ286896B6 (en)	1994-01-18	2000-07-12	Pfizer	Process for preparing pharmaceutically acceptable salts of naphthyridone carboxylic acid and intermediates for this preparation
US5475116A (en) *	1994-04-29	1995-12-12	Pfizer Inc.	Aza bicyclo[3,1,0]hexane intermediates useful in the synthesis of quinolones
US5929240A (en) *	1994-12-12	1999-07-27	Pfizer Inc.	Process and intermediates for preparing naphthyridonecarboxylic acid salts
JPH0912547A (ja) *	1995-06-23	1997-01-14	Chisso Corp	ニューキノロン系化合物中間体の製造方法
GB9524466D0 (en) *	1995-11-30	1996-01-31	Pfizer Ltd	Process
US6057455A (en) *	1996-07-09	2000-05-02	Pfizer, Inc.	Preparation of intermediates useful in the synthesis of quinoline antibiotics
JPH1087617A (ja) *	1996-07-09	1998-04-07	Pfizer Inc	キノリン系抗生物質の合成に有用な中間体の製法
GB9614422D0 (en) *	1996-07-09	1996-09-04	Pfizer Ltd	Novel process
HN1998000106A (es)	1997-08-01	1999-01-08	Pfizer Prod Inc	Composiciones parenterales de alatroflaxacino
DE19733439A1 (de) *	1997-08-02	1999-02-04	Bayer Ag	Neue 6-endo-Amino-3-azabicyclo(3.1.0)hexande, Verfahren zu deren Herstellung und deren Verwendung zur Herstellung von Chinolon- und Naphthyridincarbonsäure-Derviaten mit verbesserten Eigenschaften
US6184380B1 (en) *	1999-01-25	2001-02-06	Pfizer Inc.	Process for preparing naphthyridones and intermediates
US7019142B2 (en)	1998-01-16	2006-03-28	Pfizer Inc.	Process for preparing naphthyridones and intermediates
PA8464701A1 (es) *	1998-01-16	2000-09-29	Pfizer Prod Inc	Procedimiento e intermedios para preparar naftiridonas
WO2008010061A2 (en) *	2006-07-17	2008-01-24	Glenmark Pharmaceuticals S.A.	3-azabicyclo [3.1.0] hexane vanilloid receptor ligands, pharmaceutical compositions containing them, and processes for their preparation
CA3142351A1 (en)	2019-05-31	2020-12-03	Ikena Oncology, Inc.	Tead inhibitors and uses thereof
CA3141826A1 (en)	2019-05-31	2020-12-03	Ikena Oncology, Inc.	Tead inhibitors and uses thereof
WO2023151188A1 (zh) *	2022-02-08	2023-08-17	上海皓元医药股份有限公司	一种抗病毒药物中间体的绿色合成方法

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4183857A (en) *	1978-07-06	1980-01-15	Shell Oil Company	3-Benzyl-3-azabicyclo(3.1.0)hexane-2,4-dione
DE2962910D1 (en) *	1978-10-27	1982-07-08	Shell Int Research	A process for the preparation of 3-azabicyclo(3.1.0)hexane derivatives and modifications thereof
JPH0676400B2 (ja) *	1987-08-25	1994-09-28	大日本製薬株式会社	新規ピリドンカルボン酸誘導体、そのエステルおよびその塩
US5196548A (en) *	1989-05-11	1993-03-23	Pfizer Inc.	Preparation of diazabicyclic Intermediates
WO1991002526A1 (en) *	1989-08-16	1991-03-07	Pfizer Inc.	Azabicyclo quinolone carboxylic acids
US5200527A (en) *	1991-04-08	1993-04-06	Lonza Ltd.	Process for the production of 2-azabicyclo [2.2.1] hept-5-en-3-one

1992
- 1992-03-02 US US07/844,367 patent/US5256791A/en not_active Expired - Fee Related
1993
- 1993-01-07 KR KR1019940703051A patent/KR950700251A/ko active Granted
- 1993-01-07 JP JP5515648A patent/JP2564247B2/ja not_active Expired - Lifetime
- 1993-01-07 NZ NZ246768A patent/NZ246768A/en unknown
- 1993-01-07 EP EP93902893A patent/EP0629189B1/de not_active Expired - Lifetime
- 1993-01-07 KR KR1019940703051A patent/KR0135626B1/ko not_active Expired - Fee Related
- 1993-01-07 AT AT93902893T patent/ATE156480T1/de active
- 1993-01-07 DK DK93902893.2T patent/DK0629189T3/da active
- 1993-01-07 DE DE69312913T patent/DE69312913T2/de not_active Expired - Fee Related
- 1993-01-07 ES ES93902893T patent/ES2105217T3/es not_active Expired - Lifetime
- 1993-01-07 WO PCT/US1993/000008 patent/WO1993018001A1/en not_active Ceased
- 1993-01-07 AU AU34300/93A patent/AU667872B2/en not_active Ceased
- 1993-01-07 CA CA002131160A patent/CA2131160C/en not_active Expired - Fee Related
- 1993-01-07 HU HU9402530A patent/HU215837B/hu not_active IP Right Cessation
- 1993-01-11 TW TW082100123A patent/TW211002B/zh active
- 1993-02-22 IL IL104818A patent/IL104818A/xx not_active IP Right Cessation
- 1993-03-01 ZA ZA931428A patent/ZA931428B/xx unknown
- 1993-03-01 CN CN93102103A patent/CN1037100C/zh not_active Expired - Fee Related
- 1993-03-01 MX MX9301138A patent/MX9301138A/es not_active IP Right Cessation
- 1993-03-01 MY MYPI93000368A patent/MY107723A/en unknown
- 1993-08-04 US US08/101,879 patent/US5298629A/en not_active Expired - Fee Related
1994
- 1994-09-01 NO NO943243A patent/NO300681B1/no not_active IP Right Cessation
- 1994-09-01 FI FI944013A patent/FI106022B/fi active
1997
- 1997-09-17 GR GR970402413T patent/GR3024789T3/el unknown

Also Published As

Publication number	Publication date
EP0629189B1 (de)	1997-08-06
US5298629A (en)	1994-03-29
NO943243D0 (no)	1994-09-01
JP2564247B2 (ja)	1996-12-18
IL104818A0 (en)	1993-06-10
NO300681B1 (no)	1997-07-07
TW211002B (en)	1993-08-11
MY107723A (en)	1996-05-30
HU9402530D0 (en)	1994-11-28
MX9301138A (es)	1994-01-31
DE69312913D1 (de)	1997-09-11
KR950700251A (ko)	1995-01-16
IL104818A (en)	1997-09-30
EP0629189A1 (de)	1994-12-21
ATE156480T1 (de)	1997-08-15
JPH07500349A (ja)	1995-01-12
HU215837B (en)	2001-03-28
AU3430093A (en)	1993-10-05
WO1993018001A1 (en)	1993-09-16
FI106022B (fi)	2000-11-15
ZA931428B (en)	1994-09-01
GR3024789T3 (en)	1998-01-30
CA2131160A1 (en)	1993-09-16
DE69312913T2 (de)	1997-11-20
KR0135626B1 (ko)	1998-04-23
AU667872B2 (en)	1996-04-18
NZ246768A (en)	1995-09-26
ES2105217T3 (es)	1997-10-16
CN1076440A (zh)	1993-09-22
HUT70497A (en)	1995-10-30
US5256791A (en)	1993-10-26
CA2131160C (en)	1997-11-18
CN1037100C (zh)	1998-01-21
NO943243L (no)	1994-09-01
FI944013L (fi)	1994-09-01
FI944013A0 (fi)	1994-09-01

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