ATE161253T1 - Derivate und analoge der 2-deoxy-2,3-didehydro-n- acetyl-neuraminsäure und ihre verwendung als antivirale agentien - Google Patents

Derivate und analoge der 2-deoxy-2,3-didehydro-n- acetyl-neuraminsäure und ihre verwendung als antivirale agentien

Info

Publication number
ATE161253T1
ATE161253T1 AT91908682T AT91908682T ATE161253T1 AT E161253 T1 ATE161253 T1 AT E161253T1 AT 91908682 T AT91908682 T AT 91908682T AT 91908682 T AT91908682 T AT 91908682T AT E161253 T1 ATE161253 T1 AT E161253T1
Authority
AT
Austria
Prior art keywords
didehydro
deoxy
analogues
derivatives
antiviral agents
Prior art date
Application number
AT91908682T
Other languages
English (en)
Inventor
Itzstein Laurence Mark Von
Wen-Yang Wu
Tho Van Phan
Basil Danylec
Betty Jin
Peter Malcolm Colman
Joseph Noozhumurry Varghese
Original Assignee
Biota Scient Management
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Biota Scient Management filed Critical Biota Scient Management
Application granted granted Critical
Publication of ATE161253T1 publication Critical patent/ATE161253T1/de

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D309/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings
    • C07D309/16—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D309/28—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D309/30—Oxygen atoms, e.g. delta-lactones
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D309/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings
    • C07D309/16—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D309/28—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Virology (AREA)
  • Veterinary Medicine (AREA)
  • Oncology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Pyrane Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Heterocyclic Compounds Containing Sulfur Atoms (AREA)
AT91908682T 1990-04-24 1991-04-24 Derivate und analoge der 2-deoxy-2,3-didehydro-n- acetyl-neuraminsäure und ihre verwendung als antivirale agentien ATE161253T1 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
AUPJ980090 1990-04-24
AUPK289690 1990-10-19
AUPK453791 1991-02-11

Publications (1)

Publication Number Publication Date
ATE161253T1 true ATE161253T1 (de) 1998-01-15

Family

ID=27157556

Family Applications (2)

Application Number Title Priority Date Filing Date
AT97100119T ATE406358T1 (de) 1990-04-24 1991-04-24 Derivate und analoge der 2-deoxy-2,3-didehydro-n- acetyl-neuraminsäure und ihre verwendung als antivirale agentien
AT91908682T ATE161253T1 (de) 1990-04-24 1991-04-24 Derivate und analoge der 2-deoxy-2,3-didehydro-n- acetyl-neuraminsäure und ihre verwendung als antivirale agentien

Family Applications Before (1)

Application Number Title Priority Date Filing Date
AT97100119T ATE406358T1 (de) 1990-04-24 1991-04-24 Derivate und analoge der 2-deoxy-2,3-didehydro-n- acetyl-neuraminsäure und ihre verwendung als antivirale agentien

Country Status (37)

Country Link
US (2) US5360817A (de)
EP (2) EP0526543B1 (de)
JP (1) JP2944750B2 (de)
KR (1) KR0169496B1 (de)
CN (3) CN1143853C (de)
AP (1) AP249A (de)
AT (2) ATE406358T1 (de)
AU (2) AU654815B2 (de)
BG (1) BG62092B1 (de)
CA (2) CA2081356C (de)
CY (1) CY2186B1 (de)
CZ (1) CZ288492B6 (de)
DE (3) DE69128469T2 (de)
DK (1) DK0526543T3 (de)
ES (2) ES2113881T3 (de)
FI (2) FI105478B (de)
GR (1) GR3026225T3 (de)
HK (1) HK1003834A1 (de)
HU (2) HU219355B (de)
IE (2) IE980526A1 (de)
IL (1) IL97936A (de)
LU (1) LU90468I2 (de)
MY (1) MY107843A (de)
NL (1) NL990030I2 (de)
NO (3) NO302751B1 (de)
NZ (1) NZ237936A (de)
OA (1) OA09679A (de)
PL (3) PL167630B1 (de)
PT (1) PT97460B (de)
RU (1) RU2119487C1 (de)
SG (1) SG43170A1 (de)
SI (1) SI9110745B (de)
SK (1) SK282950B6 (de)
UA (1) UA41252C2 (de)
WO (1) WO1991016320A1 (de)
YU (1) YU48741B (de)
ZA (1) ZA913086B (de)

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