ATE181073T1 - Verfahren zur herstellung eines indazol-3- carbonamid derivates - Google Patents
Verfahren zur herstellung eines indazol-3- carbonamid derivatesInfo
- Publication number
- ATE181073T1 ATE181073T1 AT95912187T AT95912187T ATE181073T1 AT E181073 T1 ATE181073 T1 AT E181073T1 AT 95912187 T AT95912187 T AT 95912187T AT 95912187 T AT95912187 T AT 95912187T AT E181073 T1 ATE181073 T1 AT E181073T1
- Authority
- AT
- Austria
- Prior art keywords
- indazole
- producing
- carbonamide
- derivative
- pharmaceutically acceptable
- Prior art date
Links
- 238000004519 manufacturing process Methods 0.000 title abstract 2
- MFWNKCLOYSRHCJ-BTTYYORXSA-N granisetron Chemical compound C1=CC=C2C(C(=O)N[C@H]3C[C@H]4CCC[C@@H](C3)N4C)=NN(C)C2=C1 MFWNKCLOYSRHCJ-BTTYYORXSA-N 0.000 abstract 2
- 150000003839 salts Chemical class 0.000 abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 1
- 229960003727 granisetron Drugs 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 125000000467 secondary amino group Chemical group [H]N([*:1])[*:2] 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D451/00—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
- C07D451/14—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing 9-azabicyclo [3.3.1] nonane ring systems, e.g. granatane, 2-aza-adamantane; Cyclic acetals thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/18—Drugs for disorders of the alimentary tract or the digestive system for pancreatic disorders, e.g. pancreatic enzymes
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Otolaryngology (AREA)
- Hospice & Palliative Care (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Catalysts (AREA)
- Saccharide Compounds (AREA)
- Transition And Organic Metals Composition Catalysts For Addition Polymerization (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB9404055A GB9404055D0 (en) | 1994-03-03 | 1994-03-03 | Novel process |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE181073T1 true ATE181073T1 (de) | 1999-06-15 |
Family
ID=10751194
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT95912187T ATE181073T1 (de) | 1994-03-03 | 1995-02-28 | Verfahren zur herstellung eines indazol-3- carbonamid derivates |
Country Status (9)
| Country | Link |
|---|---|
| EP (1) | EP0748321B1 (de) |
| JP (1) | JP4034339B2 (de) |
| AT (1) | ATE181073T1 (de) |
| DE (1) | DE69510186D1 (de) |
| ES (1) | ES2132650T3 (de) |
| GB (1) | GB9404055D0 (de) |
| GR (1) | GR3031121T3 (de) |
| MX (1) | MX9603818A (de) |
| WO (1) | WO1995023799A1 (de) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB9502583D0 (en) * | 1995-02-10 | 1995-03-29 | Smithkline Beecham Plc | Novel process |
| GB9504078D0 (en) * | 1995-03-01 | 1995-04-19 | Smithkline Beecham Plc | Novel process |
| GB9504060D0 (en) * | 1995-03-01 | 1995-04-19 | Smithkline Beecham Plc | Novel process |
| GB9506119D0 (en) * | 1995-03-25 | 1995-05-10 | Smithkline Beecham Plc | Chemical process |
| GB9602862D0 (en) * | 1996-02-13 | 1996-04-10 | Smithkline Beecham Plc | Novel process |
| ES2197001B1 (es) * | 2002-03-26 | 2004-11-16 | Laboratorios Vita, S.A. | Procedimiento de obtencion de un compuesto farmaceuticamente activo. |
| WO2007088557A1 (en) * | 2006-02-01 | 2007-08-09 | Natco Pharma Limited | Process for highly pure crystalline granisetron base |
| US8193217B2 (en) * | 2008-08-19 | 2012-06-05 | Scinopharm Taiwan Ltd. | Polymorphic form of granisetron hydrochloride and methods of making the same |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IL59004A0 (en) * | 1978-12-30 | 1980-03-31 | Beecham Group Ltd | Substituted benzamides their preparation and pharmaceutical compositions containing them |
| DE3650772T2 (de) * | 1985-04-27 | 2003-04-03 | F. Hoffmann-La Roche Ag, Basel | Derivate von Indazole-3-carboxamide und -3-carboxylsäure |
-
1994
- 1994-03-03 GB GB9404055A patent/GB9404055D0/en active Pending
-
1995
- 1995-02-28 MX MX9603818A patent/MX9603818A/es unknown
- 1995-02-28 AT AT95912187T patent/ATE181073T1/de active
- 1995-02-28 EP EP95912187A patent/EP0748321B1/de not_active Expired - Lifetime
- 1995-02-28 ES ES95912187T patent/ES2132650T3/es not_active Expired - Lifetime
- 1995-02-28 JP JP52270295A patent/JP4034339B2/ja not_active Expired - Lifetime
- 1995-02-28 WO PCT/EP1995/000764 patent/WO1995023799A1/en not_active Ceased
- 1995-02-28 DE DE69510186T patent/DE69510186D1/de not_active Expired - Lifetime
-
1999
- 1999-08-31 GR GR990402203T patent/GR3031121T3/el unknown
Also Published As
| Publication number | Publication date |
|---|---|
| MX9603818A (es) | 1997-03-29 |
| GR3031121T3 (en) | 1999-12-31 |
| EP0748321A1 (de) | 1996-12-18 |
| WO1995023799A1 (en) | 1995-09-08 |
| JP4034339B2 (ja) | 2008-01-16 |
| EP0748321B1 (de) | 1999-06-09 |
| DE69510186D1 (de) | 1999-07-15 |
| JPH09509673A (ja) | 1997-09-30 |
| GB9404055D0 (en) | 1994-04-20 |
| ES2132650T3 (es) | 1999-08-16 |
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