ATE204281T1 - Rapamycinamidinocarbamate und diese enthaltende pharmazeutische zubereitungen - Google Patents

Rapamycinamidinocarbamate und diese enthaltende pharmazeutische zubereitungen

Info

Publication number
ATE204281T1
ATE204281T1 AT95922295T AT95922295T ATE204281T1 AT E204281 T1 ATE204281 T1 AT E204281T1 AT 95922295 T AT95922295 T AT 95922295T AT 95922295 T AT95922295 T AT 95922295T AT E204281 T1 ATE204281 T1 AT E204281T1
Authority
AT
Austria
Prior art keywords
hydrogen
rapamycinamidinocarbamates
alkynyl
alkenyl
alkyl
Prior art date
Application number
AT95922295T
Other languages
English (en)
Inventor
Jerauld Stanley Skotnicki
Yvette Latko Palmer
Original Assignee
American Home Prod
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by American Home Prod filed Critical American Home Prod
Application granted granted Critical
Publication of ATE204281T1 publication Critical patent/ATE204281T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
    • C07D498/18—Bridged systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Immunology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Transplantation (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
AT95922295T 1994-06-14 1995-06-09 Rapamycinamidinocarbamate und diese enthaltende pharmazeutische zubereitungen ATE204281T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US08/259,763 US5463048A (en) 1994-06-14 1994-06-14 Rapamycin amidino carbamates
PCT/US1995/007412 WO1995034565A1 (en) 1994-06-14 1995-06-09 Rapamycin amidino carbamates and pharmaceutical compositions containing them

Publications (1)

Publication Number Publication Date
ATE204281T1 true ATE204281T1 (de) 2001-09-15

Family

ID=22986267

Family Applications (1)

Application Number Title Priority Date Filing Date
AT95922295T ATE204281T1 (de) 1994-06-14 1995-06-09 Rapamycinamidinocarbamate und diese enthaltende pharmazeutische zubereitungen

Country Status (12)

Country Link
US (5) US5463048A (de)
EP (1) EP0765329B1 (de)
JP (1) JPH10501268A (de)
AT (1) ATE204281T1 (de)
AU (1) AU2703295A (de)
CA (1) CA2192972A1 (de)
DE (1) DE69522225T2 (de)
DK (1) DK0765329T3 (de)
ES (1) ES2159641T3 (de)
GR (1) GR3036940T3 (de)
PT (1) PT765329E (de)
WO (1) WO1995034565A1 (de)

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Also Published As

Publication number Publication date
WO1995034565A1 (en) 1995-12-21
JPH10501268A (ja) 1998-02-03
EP0765329B1 (de) 2001-08-16
DE69522225D1 (de) 2001-09-20
DE69522225T2 (de) 2002-03-21
US5463048A (en) 1995-10-31
US5541191A (en) 1996-07-30
PT765329E (pt) 2001-12-28
DK0765329T3 (da) 2001-10-08
CA2192972A1 (en) 1995-12-21
EP0765329A1 (de) 1997-04-02
US5541192A (en) 1996-07-30
US5637590A (en) 1997-06-10
US5508286A (en) 1996-04-16
GR3036940T3 (en) 2002-01-31
ES2159641T3 (es) 2001-10-16
AU2703295A (en) 1996-01-05
HK1011030A1 (en) 1999-07-02

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