ATE231873T1 - Kondensierte pyridazinonverbindungen - Google Patents

Kondensierte pyridazinonverbindungen

Info

Publication number: ATE231873T1
Authority: AT; Austria
Prior art keywords: group; stands; formula; alkyl; hydrogen
Prior art date: 1998-11-09

Application number

AT99971809T

Other languages

English (en)

Inventor

Ferenc Andrasi

Agnes Angyal

Pal Berzsenyi

Sandor Boros

Laszlo Harsing

Katalin Horvath

Peter Matyus

Imre Moravcsik

Agnes Papp

Antal Simay

Erzsebet Szabo

Katalin Szabo

Istvan Tarnawa

Ildiko Varga

Original Assignee

Gyogyszerkutato Intezet

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1998-11-09

Filing date

1999-11-09

Publication date

2003-02-15

1999-11-09 Application filed by Gyogyszerkutato Intezet filed Critical Gyogyszerkutato Intezet

2003-02-15 Application granted granted Critical

2003-02-15 Publication of ATE231873T1 publication Critical patent/ATE231873T1/de

Links

AAILEWXSEQLMNI-UHFFFAOYSA-N 1h-pyridazin-6-one Chemical class OC1=CC=CN=N1 AAILEWXSEQLMNI-UHFFFAOYSA-N 0.000 title 1
125000004178 (C1-C4) alkyl group Chemical group 0.000 abstract 4
125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 4
NINIDFKCEFEMDL-UHFFFAOYSA-N Sulfur Chemical group [S] NINIDFKCEFEMDL-UHFFFAOYSA-N 0.000 abstract 2
QVGXLLKOCUKJST-UHFFFAOYSA-N atomic oxygen Chemical compound [O] QVGXLLKOCUKJST-UHFFFAOYSA-N 0.000 abstract 2
125000002915 carbonyl group Chemical group [*:2]C([*:1])=O 0.000 abstract 2
150000001875 compounds Chemical class 0.000 abstract 2
229910052739 hydrogen Inorganic materials 0.000 abstract 2
239000001257 hydrogen Substances 0.000 abstract 2
125000000325 methylidene group Chemical group [H]C([H])=* 0.000 abstract 2
229910052760 oxygen Inorganic materials 0.000 abstract 2
239000001301 oxygen Substances 0.000 abstract 2
125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 2
125000000229 (C1-C4)alkoxy group Chemical group 0.000 abstract 1
125000006656 (C2-C4) alkenyl group Chemical group 0.000 abstract 1
DJFWTWULJOZOGK-UHFFFAOYSA-N 3h-pyridazino[4,5-f][1,4]oxazepin-2-one Chemical compound O1C(=O)CN=CC2=CN=NC=C21 DJFWTWULJOZOGK-UHFFFAOYSA-N 0.000 abstract 1
UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 abstract 1
125000002252 acyl group Chemical group 0.000 abstract 1
DHZYXWMZLAKTQV-UHFFFAOYSA-N diazepin-3-one Chemical class O=C1C=CC=CN=N1 DHZYXWMZLAKTQV-UHFFFAOYSA-N 0.000 abstract 1
125000005843 halogen group Chemical group 0.000 abstract 1
230000006883 memory enhancing effect Effects 0.000 abstract 1
230000000324 neuroprotective effect Effects 0.000 abstract 1
125000000449 nitro group Chemical group [O-][N+](*)=O 0.000 abstract 1
150000003839 salts Chemical class 0.000 abstract 1
JKCJXAVMBWFTTC-UHFFFAOYSA-N thiazepine 1-oxide Chemical compound O=S1C=CC=CC=N1 JKCJXAVMBWFTTC-UHFFFAOYSA-N 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Health & Medical Sciences (AREA)
General Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Medicinal Chemistry (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Hospice & Palliative Care (AREA)
Psychiatry (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)

AT99971809T 1998-11-09 1999-11-09 Kondensierte pyridazinonverbindungen ATE231873T1 (de)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
HU9802585A HUP9802585A3 (en)	1998-11-09	1998-11-09	Pyridazinooxazepine, -thiazepine, -diazepine and thiazine derivatives and pharmaceutical compositions containing them
PCT/HU1999/000077 WO2000027851A1 (en)	1998-11-09	1999-11-09	Novel type condensed pyridazinone compounds

Publications (1)

Publication Number	Publication Date
ATE231873T1 true ATE231873T1 (de)	2003-02-15

Family

ID=89997316

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT99971809T ATE231873T1 (de)	1998-11-09	1999-11-09	Kondensierte pyridazinonverbindungen

Country Status (12)

Country	Link
EP (1)	EP1129097B1 (de)
JP (1)	JP2002529470A (de)
KR (1)	KR100636515B1 (de)
AT (1)	ATE231873T1 (de)
AU (1)	AU762526B2 (de)
CA (1)	CA2350560C (de)
DE (1)	DE69905191T2 (de)
DK (1)	DK1129097T3 (de)
ES (1)	ES2192104T3 (de)
HU (1)	HUP9802585A3 (de)
PT (1)	PT1129097E (de)
WO (1)	WO2000027851A1 (de)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB0405034D0 (en) *	2004-03-05	2004-04-07	Novartis Ag	Organic compounds
BRPI0916540B8 (pt)	2008-07-23	2021-05-25	Us Health	inibidores do canal de ânion de superficíe de plasmódio como agentes antimaláricos
WO2012142125A2 (en)	2011-04-12	2012-10-18	The United States Of America, As Represented By The Secretary, Department Of Health And Human Services	Plasmodial surface anion channel inhibitors for the treatment or prevention of malaria

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB9411955D0 (en) *	1994-06-15	1994-08-03	Merck Sharp & Dohme	Therapeutic agents

1998
- 1998-11-09 HU HU9802585A patent/HUP9802585A3/hu unknown
1999
- 1999-11-09 KR KR1020017005304A patent/KR100636515B1/ko not_active Expired - Fee Related
- 1999-11-09 EP EP99971809A patent/EP1129097B1/de not_active Expired - Lifetime
- 1999-11-09 JP JP2000581029A patent/JP2002529470A/ja active Pending
- 1999-11-09 CA CA002350560A patent/CA2350560C/en not_active Expired - Fee Related
- 1999-11-09 DE DE69905191T patent/DE69905191T2/de not_active Expired - Fee Related
- 1999-11-09 DK DK99971809T patent/DK1129097T3/da active
- 1999-11-09 AT AT99971809T patent/ATE231873T1/de not_active IP Right Cessation
- 1999-11-09 PT PT99971809T patent/PT1129097E/pt unknown
- 1999-11-09 AU AU14016/00A patent/AU762526B2/en not_active Ceased
- 1999-11-09 ES ES99971809T patent/ES2192104T3/es not_active Expired - Lifetime
- 1999-11-09 WO PCT/HU1999/000077 patent/WO2000027851A1/en not_active Ceased

Also Published As

Publication number	Publication date
AU762526B2 (en)	2003-06-26
DE69905191D1 (de)	2003-03-06
AU1401600A (en)	2000-05-29
CA2350560C (en)	2006-10-31
WO2000027851A1 (en)	2000-05-18
PT1129097E (pt)	2003-06-30
JP2002529470A (ja)	2002-09-10
KR100636515B1 (ko)	2006-10-18
EP1129097A1 (de)	2001-09-05
KR20010092424A (ko)	2001-10-24
DE69905191T2 (de)	2003-10-16
HUP9802585A3 (en)	2000-09-28
DK1129097T3 (da)	2003-06-02
HUP9802585A2 (hu)	2000-08-28
CA2350560A1 (en)	2000-05-18
HU9802585D0 (en)	1999-01-28
EP1129097B1 (de)	2003-01-29
ES2192104T3 (es)	2003-09-16

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Legal Events

Date

Code

Title

Description

2003-08-15

UEP

Publication of translation of european patent specification

Ref document number: 1129097

Country of ref document: EP

2004-07-15

EEFA

Change of the company name

2008-08-15

REN

Ceased due to non-payment of the annual fee