|
DE60020079T2
(de)
*
|
1999-01-15 |
2006-01-19 |
Altana Pharma Ag |
Phenanthridin-N-oxide mit PDE-IV-hemmender Wirkung
|
|
ES2241571T3
(es)
*
|
1999-01-15 |
2005-11-01 |
Altana Pharma Ag |
N-oxidos de fenantrinida con actividad inhividora de pde-iv.
|
|
CZ302882B6
(cs)
|
1999-08-21 |
2012-01-04 |
Nycomed Gmbh |
Farmaceutický prostredek
|
|
US6953774B2
(en)
|
2000-08-11 |
2005-10-11 |
Applied Research Systems Ars Holding N.V. |
Methods of inducing ovulation
|
|
US7250518B2
(en)
|
2001-01-31 |
2007-07-31 |
Pfizer Inc. |
Nicotinamide acids, amides, and their mimetics active as inhibitors of PDE4 isozymes
|
|
PL364135A1
(en)
|
2001-01-31 |
2004-12-13 |
Pfizer Products Inc. |
Nicotinamide biaryl derivatives useful as inhibitors of pde4 isozymes
|
|
BR0116850A
(pt)
|
2001-01-31 |
2004-02-25 |
Pfizer Prod Inc |
Derivados de amida de ácido tiazolil-, oxazolil-, pirrolil- e imidazolil- úteis como inibidores de isoenzimas de pde4
|
|
CN1527830A
(zh)
|
2001-01-31 |
2004-09-08 |
�Ʒ� |
用作pde4同工酶的抑制剂的醚衍生物
|
|
EP1389467B1
(de)
*
|
2001-05-23 |
2013-07-03 |
Mitsubishi Tanabe Pharma Corporation |
Therapeutische Zusammensetzungen für die regenerative Behandlung von Knorpelerkrankungen
|
|
BR0213660A
(pt)
*
|
2001-10-16 |
2004-08-24 |
Memory Pharm Corp |
Composto, composição farmacêutica e método para tratar pacientes
|
|
MY130622A
(en)
|
2001-11-05 |
2007-07-31 |
Novartis Ag |
Naphthyridine derivatives, their preparation and their use as phosphodiesterase isoenzyme 4 (pde4) inhibitors
|
|
DK1908463T3
(da)
|
2001-12-14 |
2011-11-28 |
Merck Serono Sa |
Fremgangsmåder til at inducere ægløsning ved anvendelse af en ikke polypeptid-CAMP-niveaumodulator
|
|
RU2356893C2
(ru)
|
2002-11-19 |
2009-05-27 |
Мемори Фармасьютиклз Корпорейшн |
Ингибиторы фосфодиэстеразы 4
|
|
GB0229281D0
(en)
*
|
2002-12-16 |
2003-01-22 |
Novartis Ag |
Organic compounds
|
|
US7153824B2
(en)
|
2003-04-01 |
2006-12-26 |
Applied Research Systems Ars Holding N.V. |
Inhibitors of phosphodiesterases in infertility
|
|
KR20060039392A
(ko)
*
|
2003-04-16 |
2006-05-08 |
메모리 파마슈티칼스 코포레이션 |
포스포디에스테라제 4 억제제
|
|
BRPI0409888A
(pt)
*
|
2003-04-18 |
2006-05-23 |
Memory Pharm Corp |
derivados de pirazol como inibidores de fosfodiesterase 4, composto, composição farmacêutica, método para efetuar a inibição da enzima pde4, incrementar a cognição e/ou tratar a psicose em um paciente, método para o tratamento de um paciente que tem uma doença que envolve nìveis de camp diminuìdos, método para o tratamento de um paciente que sofre de uma doença alérgica ou inflamatória e método para o tratamento de um paciente que sofre de neurodegeneração resultante de uma doença ou de um ferimento
|
|
TW200519106A
(en)
|
2003-05-02 |
2005-06-16 |
Novartis Ag |
Organic compounds
|
|
MY141255A
(en)
|
2003-12-11 |
2010-03-31 |
Memory Pharm Corp |
Phosphodiesterase 4 inhibitors, including n-substituted diarylamine analogs
|
|
GB0401334D0
(en)
|
2004-01-21 |
2004-02-25 |
Novartis Ag |
Organic compounds
|
|
US20090042951A1
(en)
*
|
2004-02-20 |
2009-02-12 |
Robert Danziger |
Blood Pressure Reduction in Salt-Sensitive Hypertension
|
|
GB0411056D0
(en)
|
2004-05-18 |
2004-06-23 |
Novartis Ag |
Organic compounds
|
|
JP2008503591A
(ja)
*
|
2004-06-22 |
2008-02-07 |
ライジェル ファーマシューティカルズ, インコーポレイテッド |
ユビキチンリガーゼ阻害剤
|
|
AU2005284826A1
(en)
*
|
2004-09-14 |
2006-03-23 |
Novartis Ag |
Process for the preparation of 6, 8-substituted `1, 7 naphthpyridin derivatives by reacting the 8-halo-`1, 7 naphthpyridin-derivate with an organic boronic acid derivatives and intermediates of this process
|
|
JP2008516964A
(ja)
*
|
2004-10-15 |
2008-05-22 |
メモリー ファーマシューティカルス コーポレーション |
ホスホジエステラーゼ4阻害剤としてのピラゾール誘導体
|
|
US7585882B2
(en)
*
|
2004-10-20 |
2009-09-08 |
Memory Pharmaceuticals Corporation |
Phosphodiesterase 4 inhibitors
|
|
GT200500281A
(es)
|
2004-10-22 |
2006-04-24 |
Novartis Ag |
Compuestos organicos.
|
|
GB0424284D0
(en)
|
2004-11-02 |
2004-12-01 |
Novartis Ag |
Organic compounds
|
|
GB0426164D0
(en)
|
2004-11-29 |
2004-12-29 |
Novartis Ag |
Organic compounds
|
|
JP2006241111A
(ja)
*
|
2005-03-04 |
2006-09-14 |
Univ Nihon |
新規ベンゾフロキサン及びその合成法
|
|
GB0507577D0
(en)
|
2005-04-14 |
2005-05-18 |
Novartis Ag |
Organic compounds
|
|
GB0510390D0
(en)
|
2005-05-20 |
2005-06-29 |
Novartis Ag |
Organic compounds
|
|
JP2009506069A
(ja)
|
2005-08-26 |
2009-02-12 |
ブレインセルス,インコーポレイティド |
ムスカリン性受容体調節による神経発生
|
|
EP2258359A3
(de)
|
2005-08-26 |
2011-04-06 |
Braincells, Inc. |
Neurogenese durch Modulation des Muscarinrezeptors mit Sabcomelin
|
|
JP2009512711A
(ja)
|
2005-10-21 |
2009-03-26 |
ブレインセルス,インコーポレイティド |
Pde阻害による神経新生の調節
|
|
AU2006335042A1
(en)
*
|
2005-10-21 |
2007-07-19 |
Glaxo Group Limited |
Compounds
|
|
MY144906A
(en)
|
2005-10-21 |
2011-11-30 |
Novartis Ag |
Human antibodies against il13 and therapeutic uses
|
|
EP2314289A1
(de)
|
2005-10-31 |
2011-04-27 |
Braincells, Inc. |
Gaba-rezeptor-vermittelte modulation von neurogenese
|
|
GB0526244D0
(en)
|
2005-12-22 |
2006-02-01 |
Novartis Ag |
Organic compounds
|
|
ES2344523T3
(es)
|
2005-12-22 |
2010-08-30 |
Glaxo Group Limited |
Compuestos heterociclicos, su preparacion y su uso como agentes antibacterianos.
|
|
GB0601951D0
(en)
|
2006-01-31 |
2006-03-15 |
Novartis Ag |
Organic compounds
|
|
US20100216734A1
(en)
|
2006-03-08 |
2010-08-26 |
Braincells, Inc. |
Modulation of neurogenesis by nootropic agents
|
|
PE20080361A1
(es)
|
2006-04-21 |
2008-06-03 |
Novartis Ag |
Compuestos derivados de purina como activadores del receptor de adenosina a2a
|
|
CA2651862A1
(en)
|
2006-05-09 |
2007-11-22 |
Braincells, Inc. |
5 ht receptor mediated neurogenesis
|
|
AU2007249399A1
(en)
|
2006-05-09 |
2007-11-22 |
Braincells, Inc. |
Neurogenesis by modulating angiotensin
|
|
WO2008030651A1
(en)
|
2006-09-08 |
2008-03-13 |
Braincells, Inc. |
Combinations containing a 4-acylaminopyridine derivative
|
|
US20100184806A1
(en)
|
2006-09-19 |
2010-07-22 |
Braincells, Inc. |
Modulation of neurogenesis by ppar agents
|
|
RU2009115954A
(ru)
|
2006-09-29 |
2010-11-10 |
Новартис АГ (CH) |
Пиразолопиримидины в качестве ингибиторов липидной киназы р13к
|
|
JP2010508315A
(ja)
|
2006-10-30 |
2010-03-18 |
ノバルティス アーゲー |
抗炎症剤としてのヘテロ環式化合物
|
|
DE602007011670D1
(de)
|
2007-01-10 |
2011-02-10 |
Irm Llc |
Verbindungen und zusammensetzungen als kanal-aktivierende proteasehemmer
|
|
US8318935B2
(en)
|
2007-05-07 |
2012-11-27 |
Novartis Ag |
Organic compounds 75074
|
|
EP2231280B1
(de)
|
2007-12-10 |
2016-08-10 |
Novartis AG |
Amiloride-ähnliche Pyrazine-carboxamide als ENaC Blocker
|
|
KR20100113557A
(ko)
|
2008-01-11 |
2010-10-21 |
노파르티스 아게 |
키나제 억제제로서의 피리미딘
|
|
US8268834B2
(en)
|
2008-03-19 |
2012-09-18 |
Novartis Ag |
Pyrazine derivatives that inhibit phosphatidylinositol 3-kinase enzyme
|
|
BRPI0915018A2
(pt)
|
2008-06-10 |
2015-10-27 |
Novartis Ag |
compostos orgânicos
|
|
HRP20121006T1
(hr)
|
2009-01-29 |
2013-01-31 |
Novartis Ag |
Supstituirani benzimidazoli za lijeäśenje astrocitoma
|
|
US20100216805A1
(en)
|
2009-02-25 |
2010-08-26 |
Braincells, Inc. |
Modulation of neurogenesis using d-cycloserine combinations
|
|
US8389526B2
(en)
|
2009-08-07 |
2013-03-05 |
Novartis Ag |
3-heteroarylmethyl-imidazo[1,2-b]pyridazin-6-yl derivatives
|
|
CA2770873A1
(en)
|
2009-08-12 |
2011-02-17 |
Novartis Ag |
Heterocyclic hydrazone compounds and their uses to treat cancer and inflammation
|
|
GEP201706639B
(en)
|
2009-08-17 |
2017-03-27 |
Intellikine Llc |
Heterocyclic compounds and uses thereof
|
|
CA2771432A1
(en)
|
2009-08-20 |
2011-02-24 |
Novartis Ag |
Heterocyclic oxime compounds
|
|
EP2813227A1
(de)
|
2009-10-22 |
2014-12-17 |
Vertex Pharmaceuticals Incorporated |
Zusammensetzungen für die Behandlung von Mukoviszidose und anderen chronischen Erkrankungen
|
|
US8247436B2
(en)
|
2010-03-19 |
2012-08-21 |
Novartis Ag |
Pyridine and pyrazine derivative for the treatment of CF
|
|
MA34373B1
(fr)
|
2010-07-14 |
2013-07-03 |
Novartis Ag |
Composés hétérocycliques agonistes du récepteur ip
|
|
UY33597A
(es)
|
2010-09-09 |
2012-04-30 |
Irm Llc |
Compuestos y composiciones como inhibidores de la trk
|
|
WO2012034095A1
(en)
|
2010-09-09 |
2012-03-15 |
Irm Llc |
Compounds and compositions as trk inhibitors
|
|
US8372845B2
(en)
|
2010-09-17 |
2013-02-12 |
Novartis Ag |
Pyrazine derivatives as enac blockers
|
|
JP2014505088A
(ja)
|
2011-02-10 |
2014-02-27 |
ノバルティス アーゲー |
C−METチロシンキナーゼ阻害剤としての[1,2,4]トリアゾロ[4,3−b]ピリダジン化合物
|
|
JP5808826B2
(ja)
|
2011-02-23 |
2015-11-10 |
インテリカイン, エルエルシー |
複素環化合物およびその使用
|
|
KR20140014184A
(ko)
|
2011-02-25 |
2014-02-05 |
아이알엠 엘엘씨 |
Trk 억제제로서의 화합물 및 조성물
|
|
US8883819B2
(en)
|
2011-09-01 |
2014-11-11 |
Irm Llc |
Bicyclic heterocycle derivatives for the treatment of pulmonary arterial hypertension
|
|
AU2012310168B2
(en)
|
2011-09-15 |
2015-07-16 |
Novartis Ag |
6 - substituted 3 - (quinolin- 6 - ylthio) - [1,2,4] triazolo [4, 3 -a] pyradines as tyrosine kinase
|
|
WO2013038381A1
(en)
|
2011-09-16 |
2013-03-21 |
Novartis Ag |
Pyridine/pyrazine amide derivatives
|
|
ES2558457T3
(es)
|
2011-09-16 |
2016-02-04 |
Novartis Ag |
Compuestos heterocíclicos para el tratamiento de fibrosis quística
|
|
WO2013038378A1
(en)
|
2011-09-16 |
2013-03-21 |
Novartis Ag |
Pyridine amide derivatives
|
|
US9056867B2
(en)
|
2011-09-16 |
2015-06-16 |
Novartis Ag |
N-substituted heterocyclyl carboxamides
|
|
WO2013038373A1
(en)
|
2011-09-16 |
2013-03-21 |
Novartis Ag |
Pyridine amide derivatives
|
|
WO2013078440A2
(en)
|
2011-11-23 |
2013-05-30 |
Intellikine, Llc |
Enhanced treatment regimens using mtor inhibitors
|
|
WO2013106547A1
(en)
|
2012-01-10 |
2013-07-18 |
President And Fellows Of Harvard College |
Beta-cell replication promoting compounds and methods of their use
|
|
ES2565826T3
(es)
|
2012-01-13 |
2016-04-07 |
Novartis Ag |
Pirroles fusionados como agonistas del receptor IP para el tratamiento de hipertensión arterial pulmonar (PAH) y trastornos relacionados
|
|
US8809340B2
(en)
|
2012-03-19 |
2014-08-19 |
Novartis Ag |
Crystalline form
|
|
EP3964513A1
(de)
|
2012-04-03 |
2022-03-09 |
Novartis AG |
Kombinationsprodukte mit tyrosinkinaseinhibitoren und deren verwendung
|
|
JP5907006B2
(ja)
*
|
2012-09-04 |
2016-04-20 |
エヌ・イーケムキャット株式会社 |
ビフェニル化合物の合成方法
|
|
JP5907005B2
(ja)
*
|
2012-09-04 |
2016-04-20 |
エヌ・イーケムキャット株式会社 |
ビフェニル化合物の合成方法
|
|
US9604981B2
(en)
|
2013-02-13 |
2017-03-28 |
Novartis Ag |
IP receptor agonist heterocyclic compounds
|
|
US9073921B2
(en)
|
2013-03-01 |
2015-07-07 |
Novartis Ag |
Salt forms of bicyclic heterocyclic derivatives
|
|
WO2014151147A1
(en)
|
2013-03-15 |
2014-09-25 |
Intellikine, Llc |
Combination of kinase inhibitors and uses thereof
|
|
TW201605450A
(zh)
|
2013-12-03 |
2016-02-16 |
諾華公司 |
Mdm2抑制劑與BRAF抑制劑之組合及其用途
|
|
CN106458980A
(zh)
|
2014-04-24 |
2017-02-22 |
诺华股份有限公司 |
作为磷脂酰肌醇3‑激酶抑制剂的氨基吡啶衍生物
|
|
BR112016024533A8
(pt)
|
2014-04-24 |
2021-03-30 |
Novartis Ag |
derivados de amino pirazina como inibidores de fosfatidilinositol 3-cinase ou sal, seu uso, e composição e combinação farmacêuticas
|
|
KR20160141856A
(ko)
|
2014-04-24 |
2016-12-09 |
노파르티스 아게 |
포스파티딜이노시톨 3-키나제 억제제로서의 피라진 유도체
|
|
US9741941B2
(en)
|
2014-04-29 |
2017-08-22 |
Universal Display Corporation |
Organic electroluminescent materials and devices
|
|
WO2016011658A1
(en)
|
2014-07-25 |
2016-01-28 |
Novartis Ag |
Combination therapy
|
|
BR112017001695A2
(pt)
|
2014-07-31 |
2017-11-21 |
Novartis Ag |
terapia de combinação
|
|
KR20220019015A
(ko)
|
2019-06-10 |
2022-02-15 |
노파르티스 아게 |
Cf, copd, 및 기관지확장증 치료를 위한 피리딘 및 피라진 유도체
|
|
UY38860A
(es)
|
2019-08-28 |
2021-02-26 |
Novartis Ag |
Derivados de 1,3–fenil heteroarilo sustituidos, composiciones para su uso en el tratamiento de enfermedades y formas cristalinas
|
|
TW202140550A
(zh)
|
2020-01-29 |
2021-11-01 |
瑞士商諾華公司 |
使用抗tslp抗體治療炎性或阻塞性氣道疾病之方法
|