ATE271859T1 - Diphenyl ketoaldehyde-derivate mit wirkung gegen hiv - Google Patents

Diphenyl ketoaldehyde-derivate mit wirkung gegen hiv

Info

Publication number: ATE271859T1
Authority: AT; Austria
Prior art keywords: diphenyl; effect against; against hiv; xenaldial; group
Prior art date: 2000-03-24

Application number

AT01938038T

Other languages

English (en)

Inventor

Giulio Tarro

Original Assignee

Unihart Corp

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-03-24

Filing date

2001-03-23

Publication date

2004-08-15

2001-03-23 Application filed by Unihart Corp filed Critical Unihart Corp

2004-08-15 Application granted granted Critical

2004-08-15 Publication of ATE271859T1 publication Critical patent/ATE271859T1/de

Links

ZUOUZKKEUPVFJK-UHFFFAOYSA-N diphenyl Chemical compound C1=CC=CC=C1C1=CC=CC=C1 ZUOUZKKEUPVFJK-UHFFFAOYSA-N 0.000 title 2
235000010290 biphenyl Nutrition 0.000 title 1
239000004305 biphenyl Substances 0.000 title 1
ODRKIKHWTZCVCM-UHFFFAOYSA-N 2-[4-(4-oxaldehydoylphenyl)phenyl]-2-oxoacetaldehyde Chemical compound C1=CC(C(=O)C=O)=CC=C1C1=CC=C(C(=O)C=O)C=C1 ODRKIKHWTZCVCM-UHFFFAOYSA-N 0.000 abstract 2
PCESDWWIFVPSOX-UHFFFAOYSA-N 4-[[2-oxo-2-(4-phenylphenyl)ethylidene]amino]benzoic acid Chemical compound C1=CC(C(=O)O)=CC=C1N=CC(=O)C1=CC=C(C=2C=CC=CC=2)C=C1 PCESDWWIFVPSOX-UHFFFAOYSA-N 0.000 abstract 2
BPOMPTVRBWXZBY-UHFFFAOYSA-N 4-[[1-ethoxy-2-oxo-2-(4-phenylphenyl)ethyl]amino]benzoic acid Chemical compound C=1C=C(C=2C=CC=CC=2)C=CC=1C(=O)C(OCC)NC1=CC=C(C(O)=O)C=C1 BPOMPTVRBWXZBY-UHFFFAOYSA-N 0.000 abstract 1
208000030507 AIDS Diseases 0.000 abstract 1
102000004163 DNA-directed RNA polymerases Human genes 0.000 abstract 1
108090000626 DNA-directed RNA polymerases Proteins 0.000 abstract 1
208000031886 HIV Infections Diseases 0.000 abstract 1
239000002259 anti human immunodeficiency virus agent Substances 0.000 abstract 1
229940124411 anti-hiv antiviral agent Drugs 0.000 abstract 1
150000001875 compounds Chemical class 0.000 abstract 1
229940042399 direct acting antivirals protease inhibitors Drugs 0.000 abstract 1
239000003112 inhibitor Substances 0.000 abstract 1
229940124524 integrase inhibitor Drugs 0.000 abstract 1
239000002850 integrase inhibitor Substances 0.000 abstract 1
239000000137 peptide hydrolase inhibitor Substances 0.000 abstract 1
239000008194 pharmaceutical composition Substances 0.000 abstract 1
238000002360 preparation method Methods 0.000 abstract 1

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/12—Ketones
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/12—Ketones
- A61K31/121—Ketones acyclic
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
- A61K31/19—Carboxylic acids, e.g. valproic acid
- A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
- A61K31/196—Carboxylic acids, e.g. valproic acid having an amino group the amino group being directly attached to a ring, e.g. anthranilic acid, mefenamic acid, diclofenac, chlorambucil
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/18—Antivirals for RNA viruses for HIV

Landscapes

Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Medicinal Chemistry (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Animal Behavior & Ethology (AREA)
Pharmacology & Pharmacy (AREA)
Epidemiology (AREA)
Virology (AREA)
Communicable Diseases (AREA)
Tropical Medicine & Parasitology (AREA)
Organic Chemistry (AREA)
General Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Oncology (AREA)
Molecular Biology (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
AIDS & HIV (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

AT01938038T 2000-03-24 2001-03-23 Diphenyl ketoaldehyde-derivate mit wirkung gegen hiv ATE271859T1 (de)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
IT2000MI000629A IT1318424B1 (it)	2000-03-24	2000-03-24	Composti con attivita' anti-hiv.
PCT/EP2001/003343 WO2001070216A2 (en)	2000-03-24	2001-03-23	Diphenyl ketoaldehyde derivatives with anti-hiv activity

Publications (1)

Publication Number	Publication Date
ATE271859T1 true ATE271859T1 (de)	2004-08-15

Family

ID=11444629

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT01938038T ATE271859T1 (de)	2000-03-24	2001-03-23	Diphenyl ketoaldehyde-derivate mit wirkung gegen hiv

Country Status (16)

Country	Link
US (1)	US20040058999A1 (de)
EP (1)	EP1267858B1 (de)
JP (1)	JP2003527419A (de)
CN (1)	CN1193747C (de)
AT (1)	ATE271859T1 (de)
AU (1)	AU2001263803A1 (de)
BR (1)	BR0109345A (de)
CA (1)	CA2403707A1 (de)
DE (1)	DE60104530T2 (de)
ES (1)	ES2225550T3 (de)
IT (1)	IT1318424B1 (de)
MX (1)	MXPA02009173A (de)
NO (1)	NO20024522L (de)
RU (1)	RU2002125444A (de)
WO (1)	WO2001070216A2 (de)
ZA (1)	ZA200207586B (de)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
ITMI20020966A1 (it) *	2002-05-08	2003-11-10	Unihart Corp	Composti attivi contro i rhinovirus
UA87884C2 (uk) *	2004-12-03	2009-08-25	Мерк Энд Ко., Инк.	Безводна кристалічна калієва сіль інгібітора віл-інтегрази
CN104031117B (zh) *	2014-04-23	2017-07-11	南开大学	美国癌症数据库化合物在抗艾滋病毒1型蛋白酶活性上的新用途

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4724232A (en) *	1985-03-16	1988-02-09	Burroughs Wellcome Co.	Treatment of human viral infections
US5147652A (en) *	1990-07-03	1992-09-15	Cell Research Corporation	Autobiotics and their use in eliminating nonself cells in vivo

2000
- 2000-03-24 IT IT2000MI000629A patent/IT1318424B1/it active
2001
- 2001-03-23 CN CNB018069568A patent/CN1193747C/zh not_active Expired - Fee Related
- 2001-03-23 WO PCT/EP2001/003343 patent/WO2001070216A2/en not_active Ceased
- 2001-03-23 AU AU2001263803A patent/AU2001263803A1/en not_active Abandoned
- 2001-03-23 JP JP2001568414A patent/JP2003527419A/ja active Pending
- 2001-03-23 ES ES01938038T patent/ES2225550T3/es not_active Expired - Lifetime
- 2001-03-23 US US10/239,239 patent/US20040058999A1/en not_active Abandoned
- 2001-03-23 AT AT01938038T patent/ATE271859T1/de not_active IP Right Cessation
- 2001-03-23 CA CA002403707A patent/CA2403707A1/en not_active Abandoned
- 2001-03-23 DE DE60104530T patent/DE60104530T2/de not_active Expired - Fee Related
- 2001-03-23 BR BR0109345-2A patent/BR0109345A/pt not_active Application Discontinuation
- 2001-03-23 RU RU2002125444/15A patent/RU2002125444A/ru unknown
- 2001-03-23 MX MXPA02009173A patent/MXPA02009173A/es not_active Application Discontinuation
- 2001-03-23 EP EP01938038A patent/EP1267858B1/de not_active Expired - Lifetime
2002
- 2002-09-20 NO NO20024522A patent/NO20024522L/no not_active Application Discontinuation
- 2002-09-20 ZA ZA200207586A patent/ZA200207586B/xx unknown

Also Published As

Publication number	Publication date
WO2001070216A3 (en)	2001-12-27
ZA200207586B (en)	2003-09-22
US20040058999A1 (en)	2004-03-25
CN1193747C (zh)	2005-03-23
ITMI20000629A1 (it)	2001-09-24
EP1267858A2 (de)	2003-01-02
BR0109345A (pt)	2002-12-17
CN1419447A (zh)	2003-05-21
NO20024522L (no)	2002-11-25
JP2003527419A (ja)	2003-09-16
WO2001070216A2 (en)	2001-09-27
NO20024522D0 (no)	2002-09-20
CA2403707A1 (en)	2001-09-27
ITMI20000629A0 (it)	2000-03-24
EP1267858B1 (de)	2004-07-28
DE60104530T2 (de)	2005-09-01
ES2225550T3 (es)	2005-03-16
AU2001263803A1 (en)	2001-10-03
MXPA02009173A (es)	2003-03-12
DE60104530D1 (de)	2004-09-02
RU2002125444A (ru)	2004-03-20
IT1318424B1 (it)	2003-08-25

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Legal Events

Date	Code	Title	Description
2005-01-15	RER	Ceased as to paragraph 5 lit. 3 law introducing patent treaties