ATE277071T1 - Durch 11-beta-aryl-17,17-spirothiolan substituierte steroide - Google Patents

Durch 11-beta-aryl-17,17-spirothiolan substituierte steroide

Info

Publication number
ATE277071T1
ATE277071T1 AT00948741T AT00948741T ATE277071T1 AT E277071 T1 ATE277071 T1 AT E277071T1 AT 00948741 T AT00948741 T AT 00948741T AT 00948741 T AT00948741 T AT 00948741T AT E277071 T1 ATE277071 T1 AT E277071T1
Authority
AT
Austria
Prior art keywords
spirothiolane
beta
aryl
steroids substituted
substituted
Prior art date
Application number
AT00948741T
Other languages
English (en)
Inventor
Edgar C Cook
Rupa S Shetty
John A Kepler
David Y-W Lee
Original Assignee
Res Triangle Inst
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Res Triangle Inst filed Critical Res Triangle Inst
Application granted granted Critical
Publication of ATE277071T1 publication Critical patent/ATE277071T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J33/00—Normal steroids having a sulfur-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Endocrinology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Reproductive Health (AREA)
  • Diabetes (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pregnancy & Childbirth (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
AT00948741T 1999-07-21 2000-07-20 Durch 11-beta-aryl-17,17-spirothiolan substituierte steroide ATE277071T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US09/357,923 US6043235A (en) 1999-07-21 1999-07-21 11β-aryl-17, 17-spirothiolane-substituted steroids
PCT/US2000/019537 WO2001007462A1 (en) 1999-07-21 2000-07-20 11β-ARYL-17,17-SPIROTHIOLANE-SUBSTITUTED STEROIDS

Publications (1)

Publication Number Publication Date
ATE277071T1 true ATE277071T1 (de) 2004-10-15

Family

ID=23407590

Family Applications (1)

Application Number Title Priority Date Filing Date
AT00948741T ATE277071T1 (de) 1999-07-21 2000-07-20 Durch 11-beta-aryl-17,17-spirothiolan substituierte steroide

Country Status (14)

Country Link
US (1) US6043235A (de)
EP (1) EP1196428B1 (de)
JP (1) JP4768181B2 (de)
KR (1) KR100616025B1 (de)
AT (1) ATE277071T1 (de)
AU (1) AU774472B2 (de)
CA (1) CA2379995C (de)
DE (1) DE60014096T2 (de)
DK (1) DK1196428T3 (de)
ES (1) ES2228584T3 (de)
HK (1) HK1044542B (de)
NO (1) NO321524B1 (de)
PT (1) PT1196428E (de)
WO (1) WO2001007462A1 (de)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6262042B1 (en) * 1998-05-29 2001-07-17 Research Triangle Institute 17β-amino and hydroxylamino-11β-arylsteroids and their derivatives having agonist or antagonist hormonal properties
JP5649786B2 (ja) 2006-03-07 2015-01-07 ギータ シュロフ ヒト胚性幹細胞およびそれらの誘導体を含む組成物、使用方法、ならびに調製方法
KR200451979Y1 (ko) * 2008-04-11 2011-01-24 정종오 회전형 광고장치
DE102009034367A1 (de) * 2009-07-20 2011-01-27 Bayer Schering Pharma Aktiengesellschaft 17-Hydroxy-17-pentafluorethyl-estra-4,9(10)-dien-11-benzyliden-Derivate, Verfahren zu deren Herstellung und deren Verwendung zur Behandlung von Krankheiten
DE102009034526A1 (de) * 2009-07-21 2011-02-10 Bayer Schering Pharma Aktiengesellschaft 17-Hydroxy-17-pentafluorethyl-estra-4,9(10)-dien-11-ethinylphenyl-Derivate, Verfahren zu deren Herstellung und deren Verwendung zur Behandlung von Krankheiten

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2344286A1 (fr) * 1976-03-16 1977-10-14 Roussel Uclaf Nouveaux derives 17-spirosultines, les g-hydroxy acides correspondants, leur procede de preparation et leur application comme medicament
FR2374037A1 (fr) * 1976-10-27 1978-07-13 Roussel Uclaf Nouveaux derives steroides 17-spirosultines les g-hydroxy acides correspondants, leur procede de preparation et leur application comme medicament
ZA929315B (en) * 1991-12-20 1993-05-24 Akzo Nv 17-spirofuran-3'-ylidene steroids.
IL115659A (en) * 1994-10-27 2000-06-01 Akzo Nobel Nv Steroids with a 17-spiromethylene lactone or lactol group process for their preparation and pharmaceutical compositions containing them

Also Published As

Publication number Publication date
KR100616025B1 (ko) 2006-08-30
HK1044542B (en) 2005-02-25
PT1196428E (pt) 2005-02-28
JP2003531815A (ja) 2003-10-28
DK1196428T3 (da) 2005-01-24
WO2001007462A1 (en) 2001-02-01
KR20020092893A (ko) 2002-12-12
JP4768181B2 (ja) 2011-09-07
DE60014096T2 (de) 2005-10-06
NO20020260D0 (no) 2002-01-17
AU774472B2 (en) 2004-07-01
HK1044542A1 (en) 2002-10-25
NO321524B1 (no) 2006-05-15
AU6220000A (en) 2001-02-13
EP1196428A1 (de) 2002-04-17
DE60014096D1 (de) 2004-10-28
EP1196428A4 (de) 2002-10-16
ES2228584T3 (es) 2005-04-16
CA2379995C (en) 2008-10-14
NO20020260L (no) 2002-03-14
CA2379995A1 (en) 2001-02-01
US6043235A (en) 2000-03-28
EP1196428B1 (de) 2004-09-22

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