ATE339415T1 - Benzocarbazol und indenoindole derivate als östrogene agentien - Google Patents

Benzocarbazol und indenoindole derivate als östrogene agentien

Info

Publication number: ATE339415T1
Authority: AT; Austria
Prior art keywords: benzocarbazole; estrogenic agents; indenoindole derivatives; indenoindole; derivatives
Prior art date: 1998-05-12

Application number

AT99921833T

Other languages

English (en)

Inventor

Chris Paul Miller

Michael David Collini

Bach Dinh Tran

Original Assignee

Wyeth Corp

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1998-05-12

Filing date

1999-05-11

Publication date

2006-10-15

1999-05-11 Application filed by Wyeth Corp filed Critical Wyeth Corp

2006-10-15 Application granted granted Critical

2006-10-15 Publication of ATE339415T1 publication Critical patent/ATE339415T1/de

Links

239000000262 estrogen Substances 0.000 title abstract 3
MYKQKWIPLZEVOW-UHFFFAOYSA-N 11h-benzo[a]carbazole Chemical compound C1=CC2=CC=CC=C2C2=C1C1=CC=CC=C1N2 MYKQKWIPLZEVOW-UHFFFAOYSA-N 0.000 title abstract 2
RXXXUIOZOITBII-UHFFFAOYSA-N indeno[1,2-g]indole Chemical class C1=C2C=CC=CC2=C2C1=C1N=CC=C1C=C2 RXXXUIOZOITBII-UHFFFAOYSA-N 0.000 title abstract 2
150000001875 compounds Chemical class 0.000 abstract 1
229940011871 estrogen Drugs 0.000 abstract 1
239000008194 pharmaceutical composition Substances 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/56—Ring systems containing three or more rings
- C07D209/80—[b, c]- or [b, d]-condensed
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
- A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A61P5/30—Oestrogens
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/56—Ring systems containing three or more rings
- C07D209/80—[b, c]- or [b, d]-condensed
- C07D209/94—[b, c]- or [b, d]-condensed containing carbocyclic rings other than six-membered

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Physical Education & Sports Medicine (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Engineering & Computer Science (AREA)
Pharmacology & Pharmacy (AREA)
Bioinformatics & Cheminformatics (AREA)
Veterinary Medicine (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Orthopedic Medicine & Surgery (AREA)
Rheumatology (AREA)
Endocrinology (AREA)
Cardiology (AREA)
Heart & Thoracic Surgery (AREA)
Diabetes (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Indole Compounds (AREA)

AT99921833T 1998-05-12 1999-05-11 Benzocarbazol und indenoindole derivate als östrogene agentien ATE339415T1 (de)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US7671198A	1998-05-12	1998-05-12
US7640798A	1998-05-12	1998-05-12

Publications (1)

Publication Number	Publication Date
ATE339415T1 true ATE339415T1 (de)	2006-10-15

Family

ID=26758069

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT99921833T ATE339415T1 (de)	1998-05-12	1999-05-11	Benzocarbazol und indenoindole derivate als östrogene agentien

Country Status (8)

Country	Link
EP (1)	EP1082319B1 (de)
JP (1)	JP2002514641A (de)
CN (1)	CN1173973C (de)
AT (1)	ATE339415T1 (de)
AU (1)	AU3894399A (de)
CA (1)	CA2331631A1 (de)
DE (1)	DE69933212D1 (de)
WO (1)	WO1999058524A1 (de)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
AU2005300030B2 (en)	2004-09-20	2012-01-12	Janssen Pharmaceutica N.V.	Novel tetracyclic heteroatom containing derivatives useful as sex steroid hormone receptor modulators

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE3821148A1 (de) *	1988-06-23	1989-12-28	Erwin Von Dr Angerer	Aminoalkylindole, verfahren zu deren herstellung und diese enthaltende pharmazeutische praeparate
EP0639567A1 (de) *	1992-05-08	1995-02-22	Otsuka Pharmaceutical Factory, Inc.	Indol-derivate
DE4426625A1 (de) *	1994-07-27	1996-03-14	Schering Ag	2-Phenylindole, Verfahren zu deren Herstellung, diese enthaltende pharmazeutische Präparate sowie deren Verwendung zur Herstellung von Arzneimitteln
TW397821B (en) *	1996-04-19	2000-07-11	American Home Produits Corp	3-[4-(2-phenyl-indole-1-ylmethyl)-phenyl]-acrylamides and 2-phenyl-1-[4-(amino-1-yl-alk-1-ynyl)-benzyl]-1H-indol-5-ol as well as pharmaceutical compositions of estrogenic agents thereof
PT802183E (pt) *	1996-04-19	2002-03-28	American Home Prod	Agentes estrogenicos

1999
- 1999-05-11 AU AU38943/99A patent/AU3894399A/en not_active Abandoned
- 1999-05-11 CN CNB998084409A patent/CN1173973C/zh not_active Expired - Fee Related
- 1999-05-11 JP JP2000548328A patent/JP2002514641A/ja not_active Withdrawn
- 1999-05-11 CA CA002331631A patent/CA2331631A1/en not_active Abandoned
- 1999-05-11 DE DE69933212T patent/DE69933212D1/de not_active Expired - Lifetime
- 1999-05-11 AT AT99921833T patent/ATE339415T1/de not_active IP Right Cessation
- 1999-05-11 WO PCT/US1999/010216 patent/WO1999058524A1/en not_active Ceased
- 1999-05-11 EP EP99921833A patent/EP1082319B1/de not_active Expired - Lifetime

Also Published As

Publication number	Publication date
WO1999058524A1 (en)	1999-11-18
EP1082319B1 (de)	2006-09-13
EP1082319A1 (de)	2001-03-14
DE69933212D1 (de)	2006-10-26
AU3894399A (en)	1999-11-29
CN1173973C (zh)	2004-11-03
CN1308630A (zh)	2001-08-15
CA2331631A1 (en)	1999-11-18
JP2002514641A (ja)	2002-05-21

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Legal Events

Date	Code	Title	Description
2007-03-15	RER	Ceased as to paragraph 5 lit. 3 law introducing patent treaties