ATE278654T1 - Verfahren zur herstellung eines 5- phthalancarbonitrils, zwischenprodukt dafür und verfahren zur herstellung des zwischenproduktes - Google Patents

Verfahren zur herstellung eines 5- phthalancarbonitrils, zwischenprodukt dafür und verfahren zur herstellung des zwischenproduktes

Info

Publication number: ATE278654T1
Authority: AT; Austria
Prior art keywords: producing; intermediate product; phthalane; carbonitrile; compound
Prior art date: 1999-11-01

Application number

AT00118562T

Other languages

English (en)

Inventor

Tetsuya Ikemoto

Masami Igi

Original Assignee

Sumika Fine Chemicals Co Ltd

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1999-11-01

Filing date

2000-08-26

Publication date

2004-10-15

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=18020462&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ATE278654(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

2000-08-26 Application filed by Sumika Fine Chemicals Co Ltd filed Critical Sumika Fine Chemicals Co Ltd

2004-10-15 Application granted granted Critical

2004-10-15 Publication of ATE278654T1 publication Critical patent/ATE278654T1/de

Links

238000004519 manufacturing process Methods 0.000 title abstract 4
239000013067 intermediate product Substances 0.000 title 2
LELOWRISYMNNSU-UHFFFAOYSA-N Hydrocyanic acid Natural products N#C LELOWRISYMNNSU-UHFFFAOYSA-N 0.000 title 1
-1 5-phthalancarbonitrile compound Chemical class 0.000 abstract 2
238000000034 method Methods 0.000 abstract 2
FYSNRJHAOHDILO-UHFFFAOYSA-N thionyl chloride Chemical compound ClS(Cl)=O FYSNRJHAOHDILO-UHFFFAOYSA-N 0.000 abstract 2
ZCYVEMRRCGMTRW-UHFFFAOYSA-N 7553-56-2 Chemical group [I] ZCYVEMRRCGMTRW-UHFFFAOYSA-N 0.000 abstract 1
WKBOTKDWSSQWDR-UHFFFAOYSA-N Bromine atom Chemical group [Br] WKBOTKDWSSQWDR-UHFFFAOYSA-N 0.000 abstract 1
XFXPMWWXUTWYJX-UHFFFAOYSA-N Cyanide Chemical compound N#[C-] XFXPMWWXUTWYJX-UHFFFAOYSA-N 0.000 abstract 1
239000003153 chemical reaction reagent Substances 0.000 abstract 1
229910052801 chlorine Inorganic materials 0.000 abstract 1
125000001309 chloro group Chemical group Cl* 0.000 abstract 1
150000001875 compounds Chemical class 0.000 abstract 1
230000007613 environmental effect Effects 0.000 abstract 1
229910001385 heavy metal Inorganic materials 0.000 abstract 1
229910052740 iodine Chemical group 0.000 abstract 1
229910052751 metal Inorganic materials 0.000 abstract 1
239000002184 metal Substances 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D307/78—Benzo [b] furans; Hydrogenated benzo [b] furans
- C07D307/79—Benzo [b] furans; Hydrogenated benzo [b] furans with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C29/00—Preparation of compounds having hydroxy or O-metal groups bound to a carbon atom not belonging to a six-membered aromatic ring
- C07C29/09—Preparation of compounds having hydroxy or O-metal groups bound to a carbon atom not belonging to a six-membered aromatic ring by hydrolysis
- C07C29/095—Preparation of compounds having hydroxy or O-metal groups bound to a carbon atom not belonging to a six-membered aromatic ring by hydrolysis of esters of organic acids
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C33/00—Unsaturated compounds having hydroxy or O-metal groups bound to acyclic carbon atoms
- C07C33/40—Halogenated unsaturated alcohols
- C07C33/46—Halogenated unsaturated alcohols containing only six-membered aromatic rings as cyclic parts
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C43/00—Ethers; Compounds having groups, groups or groups
- C07C43/30—Compounds having groups
- C07C43/313—Compounds having groups containing halogen
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C69/00—Esters of carboxylic acids; Esters of carbonic or haloformic acids
- C07C69/62—Halogen-containing esters
- C07C69/63—Halogen-containing esters of saturated acids
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D307/87—Benzo [c] furans; Hydrogenated benzo [c] furans
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2601/00—Systems containing only non-condensed rings
- C07C2601/12—Systems containing only non-condensed rings with a six-membered ring
- C07C2601/16—Systems containing only non-condensed rings with a six-membered ring the ring being unsaturated

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Peptides Or Proteins (AREA)
Indole Compounds (AREA)

AT00118562T 1999-11-01 2000-08-26 Verfahren zur herstellung eines 5- phthalancarbonitrils, zwischenprodukt dafür und verfahren zur herstellung des zwischenproduktes ATE278654T1 (de)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
JP31170399		1999-11-01

Publications (1)

Publication Number	Publication Date
ATE278654T1 true ATE278654T1 (de)	2004-10-15

Family

ID=18020462

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT00118562T ATE278654T1 (de)	1999-11-01	2000-08-26	Verfahren zur herstellung eines 5- phthalancarbonitrils, zwischenprodukt dafür und verfahren zur herstellung des zwischenproduktes

Country Status (10)

Country	Link
US (7)	US6310222B1 (de)
EP (1)	EP1095926B1 (de)
AT (1)	ATE278654T1 (de)
AU (1)	AU781464B2 (de)
CA (1)	CA2317002A1 (de)
DE (1)	DE60014548T2 (de)
DK (1)	DK1095926T3 (de)
ES (1)	ES2228369T3 (de)
PT (1)	PT1095926E (de)
SI (1)	SI1095926T1 (de)

Families Citing this family (35)

* Cited by examiner, † Cited by third party
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DE69904853T2 (de)	1998-10-20	2003-09-04	Lundbeck As Valby H	Verfahren zur herstellung von citalopram
SI1140886T1 (en)	1998-12-23	2003-08-31	H. Lundbeck A/S	Method for the preparation of 5-cyanophthalide
AR022329A1 (es)	1999-01-29	2002-09-04	Lundbeck & Co As H	Metodo para la preparacion de 5-cianoftalida
TR200102957T2 (tr)	1999-04-14	2004-12-21	H. Lundbeck A/S	Sitalopram hazırlanması için metod.
ITMI991579A1 (it)	1999-06-25	2001-01-15	Lundbeck & Co As H	Metodo per la preparazione di citalopram
EP1228056B1 (de)	1999-10-25	2004-09-22	H. Lundbeck A/S	Verfahren zur herstellung von citalopram
HRP20020344B1 (hr)	1999-10-25	2010-10-31	H. Lundbeck A/S	Način priprave citaloprama
US6310222B1 (en) *	1999-11-01	2001-10-30	Sumika Fine Chemicals Co., Ltd.	Production method of 5-phthalancarbonitrile compound, intermediate therefor and production method of the intermediate
US20020055971A1 (en) *	1999-11-01	2002-05-09	Interdigital Technology Corporation	Method and system for a low-overhead mobility management protocol in the internet protocol layer
AR026063A1 (es)	1999-11-01	2002-12-26	Lundbeck & Co As H	Metodo para la preparacion de 5-carboxiftalida.
EP1246812B1 (de)	1999-12-28	2004-03-17	H. Lundbeck A/S	Verfahren zur herstellung von citalopram
SI1246813T1 (en)	1999-12-30	2004-08-31	H. Lundbeck A/S	Method for the preparation of citalopram
PL197821B1 (pl) *	2000-01-14	2008-04-30	Lundbeck & Co As H	Sposób wytwarzania 5-cyjanoftalidu
US6433196B1 (en) *	2000-02-17	2002-08-13	Sumika Fine Chemicals Co., Ltd.	Production method of citalopram, intermediate therefor and production method of the intermediate
IES20010143A2 (en) *	2000-02-24	2001-07-25	Lundbeck & Co As H	Method for the preparation of citalopram
FR2805812A1 (fr)	2000-02-24	2001-09-07	Lundbeck & Co As H	Procede de preparation du citalopram
NL1017417C1 (nl)	2000-03-03	2001-03-16	Lundbeck & Co As H	Werkwijze voor de bereiding van Citalopram.
GB0005477D0 (en)	2000-03-07	2000-04-26	Resolution Chemicals Limited	Process for the preparation of citalopram
BR0109364A (pt) *	2000-03-13	2002-12-24	Lundbeck & Co As H	Métodos para fabricação de citalopram através de alquilação escalonada de 5-substituìda 1- (4-fluorofenil) - 1,3- diidroisobenzofuranos e citalopram
PL360110A1 (en)	2000-03-13	2004-09-06	H.Lundbeck A/S	Method for the preparation of citalopram
NL1017500C1 (nl)	2000-03-13	2001-04-26	Lundbeck & Co As H	Werkwijze voor de bereiding van Citalopram.
JP2003527386A (ja)	2000-03-14	2003-09-16	ハー・ルンドベック・アクチエゼルスカベット	シタロプラムの製造方法
CH692148A5 (de) *	2000-03-16	2002-02-28	Lundbeck & Co As H	Verfahren zur Herstellung von Citalopram.
AR032455A1 (es)	2000-05-12	2003-11-12	Lundbeck & Co As H	Metodo para la preparacion de citalopram, un intermediario empleado en el metodo, un metodo para la preparacion del intermediario empleado en el metodo y composicion farmaceutica antidepresiva
CA2354877C (en)	2000-08-18	2006-05-02	H. Lundbeck A/S	Method for the preparation of citalopram
EA003581B1 (ru)	2000-12-22	2003-06-26	Х.Лундбекк А/С	Способ получения чистого циталопрама
AU2001100399B4 (en)	2000-12-28	2002-03-21	H Lundbeck As	Process for the preparation of pure citalopram
WO2004035526A1 (ja) *	2002-10-21	2004-04-29	Ihara Chemical Industry Co., Ltd.	芳香族ニトリル化合物の製造方法
US6812355B2 (en)	2002-10-22	2004-11-02	Sekhsaria Chemicals Limited	Process for the manufacture of citalopram hydrobromide from 5-bromophthalide
ITMI20030479A1 (it)	2003-03-13	2004-09-14	Adorkem Technology S P A	Procedimento per la preparazione di un ciano-isobenzofurano.
WO2004085416A1 (en) *	2003-03-24	2004-10-07	Hetero Drugs Limited	Novel crystalline forms of (s)-citalopram oxalate
JP2007503466A (ja) *	2003-05-16	2007-02-22	ワイス	アリール−カルボアルデヒドオキシム誘導体およびエストロゲン様物質としてのその使用
CA2546422A1 (en) *	2003-10-28	2005-05-12	Wockhardt Limited	Improved process for the manufacture of citalopram hydrobromide
US20060043024A1 (en) *	2004-08-31	2006-03-02	Eric Taylor	Multi-stage Carbon Block Filters
CN108794439B (zh) *	2017-05-02	2021-09-21	中国科学院大连化学物理研究所	一种苯酞的制备方法

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US134895A (en) *		1873-01-14		Improvement in folding-cribs
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US3835167A (en)	1972-12-18	1974-09-10	Syntex Inc	Anthrone carboxylic acids and derivatives
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ES8700647A1 (es)	1984-10-11	1986-11-16	Raychem Corp	Procedimiento para la preparacion de un compuesto carbonilo aromatico
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JPH04210687A (ja) *	1990-03-30	1992-07-31	Mitsubishi Rayon Co Ltd	ヒドロイソクマリン誘導体
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UA62985C2 (en) *	1997-11-10	2004-01-15	Lunnbeck As H	A method for the preparation of citalopram
FR2785284B1 (fr) *	1998-11-02	2000-12-01	Galderma Res & Dev	Analogues de la vitamine d
TR200102957T2 (tr)	1999-04-14	2004-12-21	H. Lundbeck A/S	Sitalopram hazırlanması için metod.
US6310222B1 (en)	1999-11-01	2001-10-30	Sumika Fine Chemicals Co., Ltd.	Production method of 5-phthalancarbonitrile compound, intermediate therefor and production method of the intermediate
US6433196B1 (en)	2000-02-17	2002-08-13	Sumika Fine Chemicals Co., Ltd.	Production method of citalopram, intermediate therefor and production method of the intermediate
IES20010143A2 (en)	2000-02-24	2001-07-25	Lundbeck & Co As H	Method for the preparation of citalopram
FR2805812A1 (fr)	2000-02-24	2001-09-07	Lundbeck & Co As H	Procede de preparation du citalopram
CH692148A5 (de)	2000-03-16	2002-02-28	Lundbeck & Co As H	Verfahren zur Herstellung von Citalopram.
AR032455A1 (es)	2000-05-12	2003-11-12	Lundbeck & Co As H	Metodo para la preparacion de citalopram, un intermediario empleado en el metodo, un metodo para la preparacion del intermediario empleado en el metodo y composicion farmaceutica antidepresiva
US20030109577A1 (en)	2000-10-27	2003-06-12	Ken Liljegren	Pharmaceutical composition containing citalopram

2000
- 2000-08-25 US US09/648,048 patent/US6310222B1/en not_active Expired - Fee Related
- 2000-08-26 SI SI200030563T patent/SI1095926T1/xx unknown
- 2000-08-26 DE DE60014548T patent/DE60014548T2/de not_active Expired - Fee Related
- 2000-08-26 AT AT00118562T patent/ATE278654T1/de not_active IP Right Cessation
- 2000-08-26 PT PT00118562T patent/PT1095926E/pt unknown
- 2000-08-26 DK DK00118562T patent/DK1095926T3/da active
- 2000-08-26 EP EP00118562A patent/EP1095926B1/de not_active Expired - Lifetime
- 2000-08-26 ES ES00118562T patent/ES2228369T3/es not_active Expired - Lifetime
- 2000-08-29 CA CA002317002A patent/CA2317002A1/en not_active Abandoned
- 2000-08-30 AU AU55008/00A patent/AU781464B2/en not_active Ceased
2001
- 2001-07-20 US US09/909,596 patent/US6395910B2/en not_active Expired - Fee Related
- 2001-11-30 US US09/997,992 patent/US6433195B1/en not_active Expired - Fee Related
2002
- 2002-06-21 US US10/176,721 patent/US20020151728A1/en not_active Abandoned
2003
- 2003-08-28 US US10/650,876 patent/US6930211B2/en not_active Expired - Fee Related
- 2003-08-28 US US10/650,875 patent/US20050080278A1/en not_active Abandoned
2006
- 2006-03-21 US US11/386,018 patent/US20060167285A1/en not_active Abandoned

Also Published As

Publication number	Publication date
SI1095926T1 (en)	2005-04-30
EP1095926A3 (de)	2003-05-07
US20020045770A1 (en)	2002-04-18
US6930211B2 (en)	2005-08-16
EP1095926A2 (de)	2001-05-02
US6433195B1 (en)	2002-08-13
PT1095926E (pt)	2004-12-31
US6395910B2 (en)	2002-05-28
AU781464B2 (en)	2005-05-26
US6310222B1 (en)	2001-10-30
EP1095926B1 (de)	2004-10-06
CA2317002A1 (en)	2001-05-01
US20040044232A1 (en)	2004-03-04
DE60014548D1 (de)	2004-11-11
DK1095926T3 (da)	2004-12-20
AU5500800A (en)	2001-05-03
US20060167285A1 (en)	2006-07-27
ES2228369T3 (es)	2005-04-16
US20050080278A1 (en)	2005-04-14
US20010056194A1 (en)	2001-12-27
US20020151728A1 (en)	2002-10-17
DE60014548T2 (de)	2006-03-09

Legal Events

Date

Code

Title

Description

2006-07-15

UEP

Publication of translation of european patent specification

Ref document number: 1095926

Country of ref document: EP

2008-05-15

REN

Ceased due to non-payment of the annual fee

Publication	Publication Date	Title
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