ATE287871T1 - Modulatoren von anregbaren aminosäurerezeptoren - Google Patents
Modulatoren von anregbaren aminosäurerezeptorenInfo
- Publication number
- ATE287871T1 ATE287871T1 AT00938702T AT00938702T ATE287871T1 AT E287871 T1 ATE287871 T1 AT E287871T1 AT 00938702 T AT00938702 T AT 00938702T AT 00938702 T AT00938702 T AT 00938702T AT E287871 T1 ATE287871 T1 AT E287871T1
- Authority
- AT
- Austria
- Prior art keywords
- stimulatable
- modulators
- amino acid
- acid receptors
- alkenyl
- Prior art date
Links
- 102000015404 Amino Acid Receptors Human genes 0.000 title 1
- 108010025177 Amino Acid Receptors Proteins 0.000 title 1
- 125000003903 2-propenyl group Chemical group [H]C([*])([H])C([H])=C([H])[H] 0.000 abstract 1
- 125000006374 C2-C10 alkenyl group Chemical group 0.000 abstract 1
- 102000016193 Metabotropic glutamate receptors Human genes 0.000 abstract 1
- 108010010914 Metabotropic glutamate receptors Proteins 0.000 abstract 1
- 125000000217 alkyl group Chemical group 0.000 abstract 1
- 125000000304 alkynyl group Chemical group 0.000 abstract 1
- 210000003169 central nervous system Anatomy 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 150000002148 esters Chemical class 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C229/00—Compounds containing amino and carboxyl groups bound to the same carbon skeleton
- C07C229/46—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino or carboxyl groups bound to carbon atoms of rings other than six-membered aromatic rings of the same carbon skeleton
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/07—Optical isomers
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2601/00—Systems containing only non-condensed rings
- C07C2601/02—Systems containing only non-condensed rings with a three-membered ring
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP99500089 | 1999-06-03 | ||
| PCT/EP2000/004896 WO2000075102A1 (en) | 1999-06-03 | 2000-05-26 | Excitatory amino acid receptor modulators |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE287871T1 true ATE287871T1 (de) | 2005-02-15 |
Family
ID=8242501
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT00938702T ATE287871T1 (de) | 1999-06-03 | 2000-05-26 | Modulatoren von anregbaren aminosäurerezeptoren |
Country Status (7)
| Country | Link |
|---|---|
| US (1) | US6504052B1 (de) |
| EP (1) | EP1189874B1 (de) |
| AT (1) | ATE287871T1 (de) |
| AU (1) | AU5398300A (de) |
| DE (1) | DE60017737T2 (de) |
| ES (1) | ES2235894T3 (de) |
| WO (1) | WO2000075102A1 (de) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7125871B2 (en) * | 2000-05-31 | 2006-10-24 | Eli Lilly And Company | Excitatory amino acid receptor modulators |
| US7081481B2 (en) * | 2000-05-31 | 2006-07-25 | Eli Lilly And Company | Excitatory amino acid receptor modulators |
| US9499586B2 (en) * | 2012-10-16 | 2016-11-22 | Hong Kong Baptist University | Anticancer and anti-obesity cyclic peptide agents |
| US9963485B2 (en) | 2012-10-16 | 2018-05-08 | Hong Kong Baptist University | Cycloheptapeptide agents for treatment of cancer and obesity diseases |
| WO2018068757A1 (en) * | 2016-10-14 | 2018-04-19 | Hong Kong Baptist University | Cycloheptapeptide agents for treatment of cancer and obesity diseases |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP3481975B2 (ja) | 1992-09-08 | 2003-12-22 | サントリー株式会社 | (2s,1’s,2’r)−2−(2−カルボキシ−3−置換オキシメチルシクロプロピル)グリシン及びその製造法 |
| JPH08301825A (ja) | 1995-03-07 | 1996-11-19 | Suntory Ltd | 3’−置換−(2−カルボキシシクロプロピル)グリシン |
| IT1276153B1 (it) | 1995-11-17 | 1997-10-27 | Roberto Pellicciari | Derivati di glicina ad attivita' antagonista dei recettori metabotropi del glutammato |
| EP0913389A4 (de) | 1996-06-28 | 2000-02-02 | Nippon Chemiphar Co | Cyclopropylglycinderivate und agonisten des l-glutamatrezeptors vom typ der metabolitenregulation |
| ES2131463B1 (es) * | 1997-04-08 | 2000-03-01 | Lilly Sa | Derivados de ciclopropilglicina con propiedades farmaceuticas. |
-
2000
- 2000-05-26 ES ES00938702T patent/ES2235894T3/es not_active Expired - Lifetime
- 2000-05-26 DE DE60017737T patent/DE60017737T2/de not_active Expired - Fee Related
- 2000-05-26 US US09/979,437 patent/US6504052B1/en not_active Expired - Fee Related
- 2000-05-26 AT AT00938702T patent/ATE287871T1/de not_active IP Right Cessation
- 2000-05-26 AU AU53983/00A patent/AU5398300A/en not_active Abandoned
- 2000-05-26 EP EP00938702A patent/EP1189874B1/de not_active Expired - Lifetime
- 2000-05-26 WO PCT/EP2000/004896 patent/WO2000075102A1/en not_active Ceased
Also Published As
| Publication number | Publication date |
|---|---|
| US6504052B1 (en) | 2003-01-07 |
| EP1189874B1 (de) | 2005-01-26 |
| ES2235894T3 (es) | 2005-07-16 |
| DE60017737T2 (de) | 2006-01-05 |
| WO2000075102A1 (en) | 2000-12-14 |
| EP1189874A1 (de) | 2002-03-27 |
| AU5398300A (en) | 2000-12-28 |
| DE60017737D1 (de) | 2005-03-03 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| RER | Ceased as to paragraph 5 lit. 3 law introducing patent treaties |