ATE291019T1 - Heterocyclo-alkylsulfonylpyrazolderivate zur verwendung als anti-imflammatorische oder analgetische verbindungen - Google Patents

Heterocyclo-alkylsulfonylpyrazolderivate zur verwendung als anti-imflammatorische oder analgetische verbindungen

Info

Publication number: ATE291019T1
Authority: AT; Austria
Prior art keywords: alkylsulfonylpyrazole; imflammatory; heterocyclo; derivatives; analgesic compounds
Prior art date: 1999-12-03

Application number

AT00974741T

Other languages

English (en)

Inventor

Hengmiao Cheng

Jin Li

Kristin M Lundy

Martha Lou Minich

Subas Man Sakya

Chikara Uchida

Original Assignee

Pfizer Prod Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1999-12-03

Filing date

2000-11-24

Publication date

2005-04-15

2000-11-24 Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc

2005-04-15 Application granted granted Critical

2005-04-15 Publication of ATE291019T1 publication Critical patent/ATE291019T1/de

Links

230000000202 analgesic effect Effects 0.000 title 1
150000001875 compounds Chemical class 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
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- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings

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Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Veterinary Medicine (AREA)
Life Sciences & Earth Sciences (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
Animal Behavior & Ethology (AREA)
Pharmacology & Pharmacy (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Biomedical Technology (AREA)
Diabetes (AREA)
Immunology (AREA)
Physical Education & Sports Medicine (AREA)
Rheumatology (AREA)
Pain & Pain Management (AREA)
Hematology (AREA)
Cardiology (AREA)
Endocrinology (AREA)
Pulmonology (AREA)
Orthopedic Medicine & Surgery (AREA)
Reproductive Health (AREA)
Oncology (AREA)
Heart & Thoracic Surgery (AREA)
Psychiatry (AREA)
Dermatology (AREA)
Pregnancy & Childbirth (AREA)
Urology & Nephrology (AREA)
Communicable Diseases (AREA)
Hospice & Palliative Care (AREA)
Psychology (AREA)
Gynecology & Obstetrics (AREA)
Obesity (AREA)

AT00974741T 1999-12-03 2000-11-24 Heterocyclo-alkylsulfonylpyrazolderivate zur verwendung als anti-imflammatorische oder analgetische verbindungen ATE291019T1 (de)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US16870199P	1999-12-03	1999-12-03
PCT/IB2000/001748 WO2001040216A1 (en)	1999-12-03	2000-11-24	Heterocyclo-alkylsulfonyl pyrazole derivatives as anti-inflammatory/analgesic agents

Publications (1)

Publication Number	Publication Date
ATE291019T1 true ATE291019T1 (de)	2005-04-15

Family

ID=22612589

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT00974741T ATE291019T1 (de)	1999-12-03	2000-11-24	Heterocyclo-alkylsulfonylpyrazolderivate zur verwendung als anti-imflammatorische oder analgetische verbindungen

Country Status (34)

Country	Link
US (2)	US6531492B1 (de)
EP (1)	EP1233959B1 (de)
JP (1)	JP2003517475A (de)
KR (1)	KR20020058074A (de)
CN (1)	CN1423646A (de)
AP (1)	AP2002002532A0 (de)
AR (1)	AR026711A1 (de)
AT (1)	ATE291019T1 (de)
AU (1)	AU783359B2 (de)
BG (1)	BG106694A (de)
BR (1)	BR0016031A (de)
CA (1)	CA2392931A1 (de)
CO (1)	CO5261496A1 (de)
DE (1)	DE60018792T2 (de)
DZ (1)	DZ3246A1 (de)
EA (1)	EA200200520A1 (de)
ES (1)	ES2238324T3 (de)
GT (1)	GT200000204A (de)
HK (1)	HK1052701A1 (de)
HU (1)	HUP0300157A3 (de)
IL (1)	IL149581A0 (de)
IS (1)	IS6376A (de)
MA (1)	MA26848A1 (de)
MX (1)	MXPA02005539A (de)
NO (1)	NO20022624L (de)
OA (1)	OA12100A (de)
PA (1)	PA8508201A1 (de)
PE (1)	PE20010962A1 (de)
PL (1)	PL356669A1 (de)
SK (1)	SK7412002A3 (de)
TN (1)	TNSN00235A1 (de)
WO (1)	WO2001040216A1 (de)
YU (1)	YU35102A (de)
ZA (1)	ZA200204285B (de)

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US20040248945A1 (en) *	1999-04-23	2004-12-09	Smithkline Beecham P.L.C.	Thiazolidinedione derivative and its use as antidiabetic
DE60018792T2 (de) *	1999-12-03	2006-01-26	Pfizer Products Inc., Groton	Heterocyclo-alkylsulfonylpyrazolderivate zur verwendung als anti-imflammatorische oder analgetische verbindungen
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EP1419770A4 (de) *	2001-08-24	2005-08-03	Shionogi & Co	Mittel zur beschleunigung der expression von apo ai
YU67702A (sh) *	2001-09-28	2004-12-31	Pfizer Products Inc.	Postupak za dobijanje alkansulfonil piridina
GT200200183A (es) *	2001-09-28	2003-05-23		Procedimiento para preparar derivados de heterocicloalquilsulfonil pirazol
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RU2332412C2 (ru)	2003-02-07	2008-08-27	Дайити Фармасьютикал Ко., Лтд.	Производные пиразола
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2000
- 2000-11-24 DE DE60018792T patent/DE60018792T2/de not_active Expired - Fee Related
- 2000-11-24 CN CN00818329A patent/CN1423646A/zh active Pending
- 2000-11-24 ES ES00974741T patent/ES2238324T3/es not_active Expired - Lifetime
- 2000-11-24 DZ DZ003246A patent/DZ3246A1/fr active
- 2000-11-24 HU HU0300157A patent/HUP0300157A3/hu unknown
- 2000-11-24 KR KR1020027007082A patent/KR20020058074A/ko not_active Ceased
- 2000-11-24 IL IL14958100A patent/IL149581A0/xx unknown
- 2000-11-24 EP EP00974741A patent/EP1233959B1/de not_active Expired - Lifetime
- 2000-11-24 AU AU12953/01A patent/AU783359B2/en not_active Ceased
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- 2000-11-24 AT AT00974741T patent/ATE291019T1/de not_active IP Right Cessation
- 2000-11-24 YU YU35102A patent/YU35102A/sh unknown
- 2000-11-24 PL PL00356669A patent/PL356669A1/xx not_active Application Discontinuation
- 2000-11-24 HK HK03104988.3A patent/HK1052701A1/zh unknown
- 2000-11-24 JP JP2001541900A patent/JP2003517475A/ja active Pending
- 2000-11-24 WO PCT/IB2000/001748 patent/WO2001040216A1/en not_active Ceased
- 2000-11-24 SK SK741-2002A patent/SK7412002A3/sk unknown
- 2000-11-24 MX MXPA02005539A patent/MXPA02005539A/es unknown
- 2000-11-24 BR BR0016031-8A patent/BR0016031A/pt not_active IP Right Cessation
- 2000-11-24 EA EA200200520A patent/EA200200520A1/ru unknown
- 2000-11-24 AP APAP/P/2002/002532A patent/AP2002002532A0/en unknown
- 2000-11-24 CA CA002392931A patent/CA2392931A1/en not_active Abandoned
- 2000-11-28 US US09/724,446 patent/US6531492B1/en not_active Expired - Fee Related
- 2000-12-01 PE PE2000001289A patent/PE20010962A1/es not_active Application Discontinuation
- 2000-12-01 TN TNTNSN00235A patent/TNSN00235A1/fr unknown
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- 2000-12-04 AR ARP000106402A patent/AR026711A1/es unknown
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2002
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- 2002-05-13 BG BG106694A patent/BG106694A/xx unknown
- 2002-05-29 ZA ZA200204285A patent/ZA200204285B/en unknown
- 2002-05-31 MA MA26662A patent/MA26848A1/fr unknown
- 2002-06-03 NO NO20022624A patent/NO20022624L/no unknown
2003
- 2003-01-14 US US10/342,666 patent/US20030236258A1/en not_active Abandoned

Also Published As

Publication number	Publication date
BG106694A (en)	2003-03-31
SK7412002A3 (en)	2003-08-05
CA2392931A1 (en)	2001-06-07
JP2003517475A (ja)	2003-05-27
BR0016031A (pt)	2002-07-23
PE20010962A1 (es)	2001-09-22
EP1233959A1 (de)	2002-08-28
NO20022624L (no)	2002-07-30
AU1295301A (en)	2001-06-12
DZ3246A1 (fr)	2001-06-07
WO2001040216A1 (en)	2001-06-07
AU783359B2 (en)	2005-10-20
ES2238324T3 (es)	2005-09-01
US20030236258A1 (en)	2003-12-25
KR20020058074A (ko)	2002-07-12
EA200200520A1 (ru)	2002-10-31
NO20022624D0 (no)	2002-06-03
OA12100A (en)	2006-05-04
US6531492B1 (en)	2003-03-11
YU35102A (sh)	2005-03-15
HUP0300157A2 (hu)	2003-06-28
DE60018792D1 (de)	2005-04-21
IS6376A (is)	2002-05-10
HUP0300157A3 (en)	2006-01-30
AR026711A1 (es)	2003-02-26
CN1423646A (zh)	2003-06-11
GT200000204A (es)	2002-05-28
IL149581A0 (en)	2002-11-10
TNSN00235A1 (fr)	2002-05-30
MA26848A1 (fr)	2004-12-20
DE60018792T2 (de)	2006-01-26
PL356669A1 (en)	2004-06-28
HK1052701A1 (zh)	2003-09-26
CO5261496A1 (es)	2003-03-31
MXPA02005539A (es)	2002-09-02
EP1233959B1 (de)	2005-03-16
ZA200204285B (en)	2003-05-29
PA8508201A1 (es)	2005-08-04
AP2002002532A0 (en)	2002-06-30

Legal Events

Date	Code	Title	Description
2005-09-15	RER	Ceased as to paragraph 5 lit. 3 law introducing patent treaties

Publication	Publication Date	Title
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ATE245653T1 (de)	2003-08-15	Imidazolverbindungen als phosphodiesterase vii- hemmer
DE50012542D1 (de)	2006-05-18	Verwendung von kationischen verbindungen
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