ATE312098T1 - Thiazinoxazolidinon - Google Patents

Thiazinoxazolidinon

Info

Publication number
ATE312098T1
ATE312098T1 AT01944126T AT01944126T ATE312098T1 AT E312098 T1 ATE312098 T1 AT E312098T1 AT 01944126 T AT01944126 T AT 01944126T AT 01944126 T AT01944126 T AT 01944126T AT E312098 T1 ATE312098 T1 AT E312098T1
Authority
AT
Austria
Prior art keywords
thiazinoxazolidinone
Prior art date
Application number
AT01944126T
Other languages
English (en)
Inventor
Michael R Barbachyn
Gary E Zurenko
Original Assignee
Pharmacia & Upjohn Co Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pharmacia & Upjohn Co Llc filed Critical Pharmacia & Upjohn Co Llc
Application granted granted Critical
Publication of ATE312098T1 publication Critical patent/ATE312098T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
    • C07D263/08—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D263/16—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D263/18—Oxygen atoms
    • C07D263/20—Oxygen atoms attached in position 2
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Medicinal Preparation (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
AT01944126T 2000-06-16 2001-06-14 Thiazinoxazolidinon ATE312098T1 (de)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US21247400P 2000-06-16 2000-06-16
US23659500P 2000-09-29 2000-09-29
US28558701P 2001-04-20 2001-04-20
PCT/US2001/014854 WO2001098297A2 (en) 2000-06-16 2001-06-14 A thiazine oxazolidinone

Publications (1)

Publication Number Publication Date
ATE312098T1 true ATE312098T1 (de) 2005-12-15

Family

ID=27395744

Family Applications (1)

Application Number Title Priority Date Filing Date
AT01944126T ATE312098T1 (de) 2000-06-16 2001-06-14 Thiazinoxazolidinon

Country Status (16)

Country Link
US (1) US6605609B2 (de)
EP (1) EP1294717B1 (de)
JP (1) JP2004501150A (de)
KR (1) KR20030010721A (de)
CN (1) CN1430618A (de)
AR (1) AR028706A1 (de)
AT (1) ATE312098T1 (de)
AU (1) AU2001266567A1 (de)
BR (1) BR0111520A (de)
CA (1) CA2410358A1 (de)
DE (1) DE60115644T2 (de)
ES (1) ES2253392T3 (de)
MX (1) MXPA02012494A (de)
PE (1) PE20020044A1 (de)
TW (1) TW583184B (de)
WO (1) WO2001098297A2 (de)

Families Citing this family (41)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9928568D0 (en) 1999-12-03 2000-02-02 Zeneca Ltd Chemical compounds
US6544555B2 (en) 2000-02-24 2003-04-08 Advancis Pharmaceutical Corp. Antibiotic product, use and formulation thereof
GB0009803D0 (en) 2000-04-25 2000-06-07 Astrazeneca Ab Chemical compounds
PE20020300A1 (es) * 2000-08-22 2002-05-10 Pharmacia Corp Composicion de solucion de un farmaco antibiotico a base de oxazolidinona con mejoramiento de la carga de farmaco
US6696426B2 (en) * 2000-08-22 2004-02-24 Pharmacia Corporation Preservative free ophthalmic oxazolidinone antibiotic drug delivery systems
US20020068078A1 (en) 2000-10-13 2002-06-06 Rudnic Edward M. Antifungal product, use and formulation thereof
US6541014B2 (en) 2000-10-13 2003-04-01 Advancis Pharmaceutical Corp. Antiviral product, use and formulation thereof
NZ528996A (en) 2001-04-20 2006-01-27 Upjohn Co Process to prepare oxazolidinones
EP1379509A1 (de) 2001-04-20 2004-01-14 PHARMACIA & UPJOHN COMPANY Verfahren zur herstellung von oxazolidinone
CA2453182A1 (en) * 2001-07-10 2003-01-23 Meredith L. Greene Crystalline thiazine oxazolidinones
WO2003093247A2 (en) * 2002-04-30 2003-11-13 Orchid Chemicals & Pharmaceuticals Ltd Antibacterial agents
CA2485340C (en) * 2002-05-07 2015-09-29 The State University Of New York At Stony Brook Methods, devices and formulations for targeted endobronchial therapy
TW200403240A (en) * 2002-06-28 2004-03-01 Upjohn Co Difluorothioacetamides of oxazolidinones as antibacterial agents
US6875784B2 (en) * 2002-10-09 2005-04-05 Pharmacia & Upjohn Company Antimibicrobial [3.1.0.] bicyclic oxazolidinone derivatives
AU2004258949B2 (en) 2003-07-21 2011-02-10 Shionogi, Inc. Antibiotic product, use and formulation thereof
JP2006528190A (ja) 2003-07-21 2006-12-14 アドバンシス ファーマスーティカル コーポレイション 抗生物質製剤、その使用法及び作成方法
JP2006528185A (ja) 2003-07-21 2006-12-14 アドバンシス ファーマスーティカル コーポレイション 抗生物質製剤、その使用法及び作成方法
EP1653925A1 (de) 2003-08-11 2006-05-10 Advancis Pharmaceutical Corporation Robustes pellet
WO2005016278A2 (en) 2003-08-12 2005-02-24 Advancis Pharmaceuticals Corporation Antibiotic product, use and formulation thereof
WO2005023184A2 (en) * 2003-08-29 2005-03-17 Advancis Pharmaceuticals Corporation Antibiotic product, use and formulation thereof
US8460710B2 (en) 2003-09-15 2013-06-11 Shionogi, Inc. Antibiotic product, use and formulation thereof
TWI357901B (en) * 2004-03-12 2012-02-11 Lundbeck & Co As H Substituted morpholine and thiomorpholine derivati
WO2005113520A1 (en) * 2004-05-20 2005-12-01 Pharmacia & Upjohn Company Llc Substituted 2,3,5-trifluorphenyl oxazolidinones for use as antibacterial agents
AU2005269981A1 (en) 2004-07-02 2006-02-09 Bonck, John A Tablet for pulsed delivery
US7838532B2 (en) * 2005-05-18 2010-11-23 Mpex Pharmaceuticals, Inc. Aerosolized fluoroquinolones and uses thereof
US8524735B2 (en) 2005-05-18 2013-09-03 Mpex Pharmaceuticals, Inc. Aerosolized fluoroquinolones and uses thereof
CN101282981B (zh) * 2005-08-11 2012-09-26 塔甘塔治疗公司 膦酸化利福霉素及其在预防和治疗骨和关节感染中的用途
US8357394B2 (en) 2005-12-08 2013-01-22 Shionogi Inc. Compositions and methods for improved efficacy of penicillin-type antibiotics
US8778924B2 (en) 2006-12-04 2014-07-15 Shionogi Inc. Modified release amoxicillin products
US8299052B2 (en) * 2006-05-05 2012-10-30 Shionogi Inc. Pharmaceutical compositions and methods for improved bacterial eradication
EP2018864A1 (de) 2007-07-23 2009-01-28 Biomet Deutschland GmbH Pharmazeutische Zusammensetzung, Substrat mit einer pharmazeutischen Zusammensetzung und Verwendung einer pharmazeutischen Zusammensetzung
CA2739897C (en) 2008-10-07 2017-10-03 Mpex Pharmaceuticals, Inc. Aerosol fluoroquinolone formulations for improved pharmacokinetics
CA2739893C (en) 2008-10-07 2016-10-04 Mpex Pharmaceuticals, Inc. Inhalation of levofloxacin for reducing lung inflammation
SI2473170T1 (sl) 2009-09-04 2019-10-30 Horizon Orphan Llc Uporaba aerosoliziranega levofloksacina za zdravljenje cistične fibroze
US10010758B2 (en) * 2015-07-20 2018-07-03 Kinetic Furniture Of Vermont, Llc Exercise chair
CN106770222A (zh) * 2016-11-23 2017-05-31 百奥森（江苏）食品安全科技有限公司 一种食品中甲硝唑的检测试剂盒
CN108239098B (zh) * 2016-12-26 2021-01-12 中国医学科学院药物研究所 含四氢吡啶的苯并噁嗪噁唑烷酮类化合物及其制备方法和用途
CA3059880A1 (en) * 2017-04-14 2018-10-18 Nal Pharmaceutical Group Limited Pre-filled syringe containing moxifloxacin
WO2021184339A1 (en) 2020-03-20 2021-09-23 Merck Sharp & Dohme Corp. Oxazolidinone compound and methods of use thereof as an antibacterial agent
CN111870594B (zh) * 2020-08-27 2022-03-22 首都医科大学附属北京胸科医院 苯乙肼在制备抗偶发分枝杆菌感染的药物中的应用
US20260062394A1 (en) * 2022-08-10 2026-03-05 Merck Sharp & Dohme Llc Processes for preparing oxazolidinone compounds

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5688792A (en) * 1994-08-16 1997-11-18 Pharmacia & Upjohn Company Substituted oxazine and thiazine oxazolidinone antimicrobials
CN1072222C (zh) 1995-09-01 2001-10-03 法玛西雅厄普约翰公司 以c－c键连接于4－8元杂环环的苯基噁唑烷酮
GB9702213D0 (en) 1996-02-24 1997-03-26 Zeneca Ltd Chemical compounds
JP2001524074A (ja) * 1997-03-13 2001-11-27 スミスクライン・ビーチャム・パブリック・リミテッド・カンパニー 金属−β−ラクタマーゼ阻害特性を有するピロリジンおよびチアゾール誘導体
WO2001034128A2 (en) 1999-11-08 2001-05-17 Pharmacia & Upjohn Company Admixture for intravenous administration of linezolid and other antibacterial agents

Also Published As

Publication number Publication date
US6605609B2 (en) 2003-08-12
DE60115644D1 (en) 2006-01-12
PE20020044A1 (es) 2002-01-30
BR0111520A (pt) 2003-03-18
KR20030010721A (ko) 2003-02-05
JP2004501150A (ja) 2004-01-15
US20020156072A1 (en) 2002-10-24
EP1294717A2 (de) 2003-03-26
EP1294717B1 (de) 2005-12-07
AU2001266567A1 (en) 2002-01-02
MXPA02012494A (es) 2003-04-25
AR028706A1 (es) 2003-05-21
CA2410358A1 (en) 2001-12-27
DE60115644T2 (de) 2006-07-06
WO2001098297A2 (en) 2001-12-27
WO2001098297A3 (en) 2002-06-13
ES2253392T3 (es) 2006-06-01
CN1430618A (zh) 2003-07-16
TW583184B (en) 2004-04-11

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Legal Events

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RER Ceased as to paragraph 5 lit. 3 law introducing patent treaties