ATE314076T1 - Fosinopril-formulierung - Google Patents

Fosinopril-formulierung

Info

Publication number: ATE314076T1
Authority: AT; Austria
Prior art keywords: fosinopril; formulation; fosinoprilat; ace; prodrug
Prior art date: 2002-03-19

Application number

AT03706893T

Other languages

English (en)

Inventor

Reynir Eyjolfsson

Original Assignee

Actavis Group Hf

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2002-03-19

Filing date

2003-03-19

Publication date

2006-01-15

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=36715398&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ATE314076(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

2003-03-19 Application filed by Actavis Group Hf filed Critical Actavis Group Hf

2006-01-15 Application granted granted Critical

2006-01-15 Publication of ATE314076T1 publication Critical patent/ATE314076T1/de

Links

BIDNLKIUORFRQP-XYGFDPSESA-N (2s,4s)-4-cyclohexyl-1-[2-[[(1s)-2-methyl-1-propanoyloxypropoxy]-(4-phenylbutyl)phosphoryl]acetyl]pyrrolidine-2-carboxylic acid Chemical compound C([P@@](=O)(O[C@H](OC(=O)CC)C(C)C)CC(=O)N1[C@@H](C[C@H](C1)C1CCCCC1)C(O)=O)CCCC1=CC=CC=C1 BIDNLKIUORFRQP-XYGFDPSESA-N 0.000 title abstract 3
238000009472 formulation Methods 0.000 title abstract 3
229960002490 fosinopril Drugs 0.000 title abstract 3
239000000203 mixture Substances 0.000 title abstract 3
229940044094 angiotensin-converting-enzyme inhibitor Drugs 0.000 abstract 1
BYNVYIUJKRRNNC-UHFFFAOYSA-N docosanoic acid;propane-1,2,3-triol Chemical compound OCC(O)CO.CCCCCCCCCCCCCCCCCCCCCC(O)=O BYNVYIUJKRRNNC-UHFFFAOYSA-N 0.000 abstract 1
230000002708 enhancing effect Effects 0.000 abstract 1
WOIWWYDXDVSWAZ-RTWAWAEBSA-N fosinoprilat Chemical compound C([C@@H](C[C@H]1C(=O)O)C2CCCCC2)N1C(=O)CP(O)(=O)CCCCC1=CC=CC=C1 WOIWWYDXDVSWAZ-RTWAWAEBSA-N 0.000 abstract 1
229960003018 fosinoprilat Drugs 0.000 abstract 1
239000000314 lubricant Substances 0.000 abstract 1
238000004519 manufacturing process Methods 0.000 abstract 1
239000008194 pharmaceutical composition Substances 0.000 abstract 1
239000000651 prodrug Substances 0.000 abstract 1
229940002612 prodrug Drugs 0.000 abstract 1

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
- A61K31/549—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame having two or more nitrogen atoms in the same ring, e.g. hydrochlorothiazide
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/66—Phosphorus compounds
- A61K31/675—Phosphorus compounds having nitrogen as a ring hetero atom, e.g. pyridoxal phosphate
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
- A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2059—Starch, including chemically or physically modified derivatives; Amylose; Amylopectin; Dextrin

Landscapes

Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
Chemical & Material Sciences (AREA)
General Health & Medical Sciences (AREA)
Animal Behavior & Ethology (AREA)
Medicinal Chemistry (AREA)
Epidemiology (AREA)
Biophysics (AREA)
Molecular Biology (AREA)
Bioinformatics & Cheminformatics (AREA)
General Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Heart & Thoracic Surgery (AREA)
Cardiology (AREA)
Organic Chemistry (AREA)
Engineering & Computer Science (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Medicinal Preparation (AREA)
Medicines Containing Plant Substances (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

AT03706893T 2002-03-19 2003-03-19 Fosinopril-formulierung ATE314076T1 (de)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
IS6315A IS1935B (is)	2002-03-19	2002-03-19	Fósínópríl lyfjasamsetning
PCT/IS2003/000013 WO2003077929A1 (en)	2002-03-19	2003-03-19	Fosinopril formulation

Publications (1)

Publication Number	Publication Date
ATE314076T1 true ATE314076T1 (de)	2006-01-15

Family

ID=36715398

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT03706893T ATE314076T1 (de)	2002-03-19	2003-03-19	Fosinopril-formulierung

Country Status (13)

Country	Link
US (1)	US7045511B2 (de)
EP (1)	EP1531831B1 (de)
AT (1)	ATE314076T1 (de)
AU (1)	AU2003208599A1 (de)
DE (1)	DE60303041T2 (de)
DK (1)	DK1531831T3 (de)
EA (1)	EA008171B1 (de)
ES (1)	ES2256721T3 (de)
IS (1)	IS1935B (de)
NO (1)	NO20044390L (de)
PT (1)	PT1531831E (de)
UA (1)	UA78988C2 (de)
WO (1)	WO2003077929A1 (de)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
ES2322854T3 (es) *	2003-06-26	2009-06-30	Teva Pharmaceutical Industries Limited	Composiciones farmaceuticas estables de derivados del acido 2-aza-biciclo(3.3.0)-octano-3-carboxilico.
US20050095287A1 (en) *	2003-10-29	2005-05-05	Matharu Amol S.	Fosinopril composition
GB2411355B (en) *	2004-02-27	2006-02-22	Niche Generics Ltd	Pharmaceutical composition
MX2007008392A (es) *	2005-02-11	2007-09-06	Aventis Pharma Inc	Esteres de acido propano-fosfinico sustituido.
WO2006100602A2 (en) *	2005-03-22	2006-09-28	Aurobindo Pharma Ltd	Immediate release stable solid oral dosage forms op fosinopril
KR20080112387A (ko) *	2006-04-19	2008-12-24	테바 파마슈티컬 인더스트리즈 리미티드	2-아자-비사이클로[3.3.0]-옥탄-3-카르복실산 유도체의 안정한 약학 조성물
GB0612540D0 (en) *	2006-06-23	2006-08-02	Novartis Ag	Galenical formulations of organic compounds
ATE406173T1 (de) *	2006-07-10	2008-09-15	Teva Pharma	Stabile zubereitung enthaltend eine kombination aus einer feuchtigkeitsempfindlichen aktiven substanz und einer zweiten aktiven substanz und verfahren zur herstellung der zubereitung.
US20140179712A1 (en)	2012-12-21	2014-06-26	Astrazeneca Ab	Pharmaceutical formulation of n-[5-[2-(3,5-dimethoxyphenyl)ethyl]-2h-pyrazol-3-yl]-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamide

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4337201A (en) *	1980-12-04	1982-06-29	E. R. Squibb & Sons, Inc.	Phosphinylalkanoyl substituted prolines
US5006344A (en)	1989-07-10	1991-04-09	E. R. Squibb & Sons, Inc.	Fosinopril tablet formulations
US6521647B2 (en) *	2000-04-04	2003-02-18	Pfizer Inc.	Treatment of renal disorders
CA2330904C (en) *	2001-01-11	2006-10-24	Bernard Charles Sherman	Fosinopril sodium tablet formulation
JP2005508978A (ja) *	2001-11-02	2005-04-07	ファイザー・プロダクツ・インク	Ｐｄｅ９阻害薬によるインスリン抵抗性症候群及び２型糖尿病の治療
ITMI20012366A1 (it) *	2001-11-09	2003-05-09	Farmatron Ltd	Sistemi terapeutici stabilizzati a rilascio immediato e/o modificato per la somministrazione orale di principi attivi e/o eccipienti e/o ali

2002
- 2002-03-19 IS IS6315A patent/IS1935B/is unknown
2003
- 2003-03-19 DE DE60303041T patent/DE60303041T2/de not_active Expired - Lifetime
- 2003-03-19 AT AT03706893T patent/ATE314076T1/de active
- 2003-03-19 EA EA200401218A patent/EA008171B1/ru not_active IP Right Cessation
- 2003-03-19 WO PCT/IS2003/000013 patent/WO2003077929A1/en not_active Ceased
- 2003-03-19 ES ES03706893T patent/ES2256721T3/es not_active Expired - Lifetime
- 2003-03-19 AU AU2003208599A patent/AU2003208599A1/en not_active Abandoned
- 2003-03-19 DK DK03706893T patent/DK1531831T3/da active
- 2003-03-19 US US10/507,918 patent/US7045511B2/en not_active Expired - Fee Related
- 2003-03-19 PT PT03706893T patent/PT1531831E/pt unknown
- 2003-03-19 UA UA20041008392A patent/UA78988C2/uk unknown
- 2003-03-19 EP EP03706893A patent/EP1531831B1/de not_active Expired - Lifetime
2004
- 2004-10-18 NO NO20044390A patent/NO20044390L/no not_active Application Discontinuation

Also Published As

Publication number	Publication date
ES2256721T3 (es)	2006-07-16
US7045511B2 (en)	2006-05-16
EP1531831A1 (de)	2005-05-25
DK1531831T3 (da)	2006-05-15
US20050256086A1 (en)	2005-11-17
IS6315A (is)	2003-09-20
UA78988C2 (en)	2007-05-10
WO2003077929A1 (en)	2003-09-25
NO20044390L (no)	2004-12-15
PT1531831E (pt)	2006-05-31
EA200401218A1 (ru)	2005-12-29
DE60303041T2 (de)	2006-08-24
DE60303041D1 (de)	2006-02-02
IS1935B (is)	2004-06-16
AU2003208599A1 (en)	2003-09-29
EA008171B1 (ru)	2007-04-27
EP1531831B1 (de)	2005-12-28

Legal Events

Date

Code

Title

Description

2006-09-15

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